Récepteur adrénergique
Les récepteurs adrénergiques sont des GPCR activés par les catécholamines, telles que l'adrénaline et la noradrénaline. Ces récepteurs sont classés en sous-types alpha et bêta, chacun jouant un rôle clé dans la régulation du rythme cardiaque, de la pression artérielle et de la réponse de lutte ou de fuite. Les modulateurs des récepteurs adrénergiques sont essentiels dans le traitement des maladies cardiovasculaires, de l'asthme et des troubles anxieux. Chez CymitQuimica, nous offrons une large gamme de modulateurs des récepteurs adrénergiques de haute qualité pour soutenir vos recherches en endocrinologie, pharmacologie cardiovasculaire et réponse au stress.
Sous-catégories appartenant à la catégorie "Récepteur adrénergique"
730 produits trouvés pour "Récepteur adrénergique"
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Ancarolol
CAS :Ancarolol is a blocking agent of beta-adrenergic.Formule :C18H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.39Rec 15/2615 dihydrochloride
CAS :Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.Formule :C26H35Cl2N5O5Degré de pureté :97.04% - 99.76%Couleur et forme :SolidMasse moléculaire :568.49Arbutamine
CAS :Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.
Formule :C18H23NO4Degré de pureté :95.06%Couleur et forme :SolidMasse moléculaire :317.38(S)-(-)-Propranolol hydrochloride
CAS :(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。Formule :C16H22ClNO2Degré de pureté :99.02% - 99.91%Couleur et forme :SolidMasse moléculaire :295.8(S)-Terazosin
CAS :(S)-Terazosin is an active S-enantiomer of Terazosin.Formule :C19H25N5O4Couleur et forme :SolidMasse moléculaire :387.43T-0509
CAS :T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-
Formule :C18H23NO5Degré de pureté :97.52% - 98.43%Couleur et forme :SolidMasse moléculaire :333.38Cyclazosin HCl
CAS :Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formule :C23H28ClN5O4Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :473.95Levobunolol hydrochloride
CAS :Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。Formule :C17H26ClNO3Degré de pureté :98.49% - >99.99%Couleur et forme :SolidMasse moléculaire :327.85L748337
CAS :L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formule :C26H31N3O5SDegré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :497.61ADRA1D receptor antagonist 1 HCl
CAS :ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.Formule :C15H14Cl2N4ODegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :337.2Romifidine
CAS :Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Formule :C9H9BrFN3Couleur et forme :SolidMasse moléculaire :258.09LY377604
CAS :LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.Formule :C31H32N4O4Degré de pureté :99.72% - >99.99%Couleur et forme :SolidMasse moléculaire :524.61SM-2470
CAS :SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.Formule :C23H30ClN5O3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :459.97Falintolol
CAS :Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.
Formule :C12H24N2O2Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :228.33ORM-10921
CAS :ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formule :C18H23NO2Degré de pureté :99.46% - 99.98%Couleur et forme :SolidMasse moléculaire :285.38Imiloxan
CAS :Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formule :C14H16N2O2Degré de pureté :98.13% - 99.8%Couleur et forme :SolidMasse moléculaire :244.29Xamoterol hemifumarate
CAS :Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormule :C36H54N6O14Degré de pureté :99.79%Couleur et forme :White SolidMasse moléculaire :794.37Fipamezole
CAS :Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.Formule :C14H15FN2Degré de pureté :99.32% - 99.97%Couleur et forme :SolidMasse moléculaire :230.28Rezatomidine
CAS :Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.Formule :C13H16N2SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :232.34Bedoradrine
CAS :Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formule :C24H32N2O5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :428.52Bedoradrine sulfate
CAS :Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formule :C24H32N2O5H2O4SDegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :477.56GP2-114
CAS :GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.Formule :C19H24N2O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :344.4Egis-11150
CAS :Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formule :C19H21ClFN5O2Degré de pureté :97.49% - >99.99%Couleur et forme :SolidMasse moléculaire :405.85Amosulalol
CAS :Amosulalol is a combined alpha and beta adrenoceptor antagonist.Formule :C18H24N2O5SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :380.46Ref: TM-T30027
1mg175,00€2mg264,00€5mg404,00€1mL*10mM (DMSO)430,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€CL 316243
CAS :CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formule :C20H18ClNNa2O7Degré de pureté :98.00% - 99.68%Couleur et forme :SolidMasse moléculaire :465.79Midaglizole hydrochloride
CAS :Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formule :C16H19Cl2N3Degré de pureté :99.39% - 99.82%Couleur et forme :SolidMasse moléculaire :324.25Ref: TM-T11015
1mg54,00€5mg119,00€1mL*10mM (DMSO)152,00€10mg188,00€25mg306,00€50mg416,00€100mg532,00€200mg705,00€Soquinolol
CAS :Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a longFormule :C17H26N2O3Degré de pureté :97.48% - 98.63%Couleur et forme :SolidMasse moléculaire :306.4Neldazosin
CAS :Neldazosin is used as a potent α1-adrenoceptor antagonist.Formule :C18H25N5O4Degré de pureté :99.76% - 99.97%Couleur et forme :SolidMasse moléculaire :375.42Oxyfedrine L-form HCl
CAS :Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Formule :C19H24ClNO3Degré de pureté :99.5% - 99.57%Couleur et forme :SolidMasse moléculaire :349.85Ref: TM-T24579
1mg92,00€5mg178,00€1mL*10mM (DMSO)203,00€10mg313,00€25mg485,00€50mg700,00€100mg893,00€200mg1.198,00€JP1302
CAS :JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formule :C24H24N4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :368.47Ecastolol
CAS :Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formule :C26H33N3O6Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :483.56Ref: TM-T11148
1mg349,00€5mg697,00€1mL*10mM (DMSO)880,00€10mg888,00€25mg1.395,00€50mg1.783,00€100mg2.530,00€Nemazoline Free Base
CAS :Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formule :C10H11Cl2N3Degré de pureté :98.06% - 98.83%Couleur et forme :SolidMasse moléculaire :244.12Butofilolol
CAS :Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formule :C17H26FNO3Degré de pureté :98.96% - >99.99%Couleur et forme :SolidMasse moléculaire :311.392Rafabegron
CAS :Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formule :C21H23ClN2O4Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :402.87Pipoxazole
CAS :Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formule :C14H20N4ODegré de pureté :98.58% - 99.53%Couleur et forme :SolidMasse moléculaire :260.33Taprizosin
CAS :Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Formule :C25H26N6O4SDegré de pureté :98.10% - 99.11%Couleur et forme :SolidMasse moléculaire :506.58Milveterol HCl
CAS :Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formule :C25H30ClN3O4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :471.98Dabelotine
CAS :Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.Formule :C15H22N2O2Degré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :262.35(S)-(+)-Niguldipine hydrochloride
CAS :(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formule :C36H40ClN3O6Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :646.17Besipirdine
CAS :Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formule :C16H17N3Degré de pureté :97.15% - 98.85%Couleur et forme :SolidMasse moléculaire :251.33Palatrigine
CAS :Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.Formule :C12H13Cl2N5Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :298.17Bisaramil hydrochloride
CAS :Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.Formule :C17H24Cl2N2O2Degré de pureté :98.64% - 99.48%Couleur et forme :SolidMasse moléculaire :359.29ST 91
CAS :ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formule :C13H20ClN3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :253.77Ref: TM-T23397
5mg49,00€1mL*10mM (DMSO)50,00€10mg72,00€25mg142,00€50mg245,00€100mg354,00€200mg497,00€Vadocaine
CAS :Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formule :C18H28N2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :304.43N-5984
CAS :N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.
Formule :C20H22ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.85Phentolamine Analogue 1
CAS :Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formule :C17H19N3ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :281.35Ref: TM-T12444
1mg81,00€1mL*10mM (DMSO)163,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€RS100329 hydrochloride
CAS :RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.Formule :C20H26ClF3N4O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :462.89Bufuralol
CAS :Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Formule :C16H23NO2Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :261.36L-796568 free base
CAS :L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formule :C31H27F3N4O3S2Couleur et forme :SolidMasse moléculaire :624.7Domesticine, (-)-
CAS :Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.Formule :C19H19NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :325.36GW-597901
CAS :GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.Formule :C25H38N2O6SCouleur et forme :SolidMasse moléculaire :494.64Epinephrine HCl
CAS :Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formule :C9H14ClNO3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :219.67LK 204-545
CAS :LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.Formule :C25H32N4O6Couleur et forme :SolidMasse moléculaire :484.54BU-E 75
CAS :BU-E 75 is an agonist of the histamine H2.Formule :C21H24F2N6Couleur et forme :SolidMasse moléculaire :398.45Celiprolol hydrochloride
CAS :Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formule :C20H33N3O4·HClCouleur et forme :White Crystalline SolidMasse moléculaire :415.96NGD9002
CAS :NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formule :C20H31N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.49(±)-N-Methylcoclaurine
CAS :N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].Formule :C18H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.36Nolomirole HCl
CAS :Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFormule :C19H28ClNO4Degré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :369.88Mefenidil
CAS :Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.Formule :C12H11N3Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :197.24KUC-7322
CAS :Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.Formule :C21H27NO5Couleur et forme :SolidMasse moléculaire :373.44Bunazosin Hydrochloride
CAS :Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formule :C19H28ClN5O3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :409.91Todralazine hydrochloride
CAS :Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Formule :C11H13ClN4O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :268.7Indacaterol xinafoate
CAS :Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Formule :C35H36N2O6Couleur et forme :SolidMasse moléculaire :580.67Indacaterol acetate
CAS :Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Formule :C26H32N2O5Couleur et forme :SolidMasse moléculaire :452.54AR-08
CAS :AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.Formule :C12H12N6Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :240.26Vemtoberant
CAS :Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.Formule :C29H37N3O8S2Couleur et forme :SolidMasse moléculaire :619.75Prenalterol hydrochloride
CAS :Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formule :C12H20ClNO3Couleur et forme :SolidMasse moléculaire :261.75Abediterol
CAS :Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formule :C25H30F2N2O4Couleur et forme :SolidMasse moléculaire :460.51Bufuralol (hydrochloride)
CAS :Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Formule :C16H24ClNO2Couleur et forme :SolidMasse moléculaire :297.82BMS-194449
CAS :BMS-194449 is a full beta 3 agonist.Formule :C24H24F4N2O6SCouleur et forme :SolidMasse moléculaire :544.52RS 17053 hydrochloride
CAS :RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formule :C24H30Cl2N2O2Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :449.41N-5984 Hydrochloride
CAS :N-5984 Hydrochloride is a beta3-AR agonist.Formule :C20H23Cl2NO5Couleur et forme :SolidMasse moléculaire :428.31β3-AR agonist 1
CAS :β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/Formule :C22H28N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.55Vatinoxan hydrochloride
CAS :Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formule :C20H27ClN4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.97L-796568 dihydrochloride
CAS :L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.Formule :C31H29Cl2F3N4O3S2Couleur et forme :SolidMasse moléculaire :697.62Fiduxosin hydrochloride
CAS :Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formule :C30H30ClN5O4SCouleur et forme :SolidMasse moléculaire :592.11Ritodrine
CAS :Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].Formule :C17H21NO3Couleur et forme :SolidMasse moléculaire :287.35Binedaline
CAS :Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formule :C19H23N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.41β3-AR agonist 2
CAS :β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formule :C27H38N4O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.68AGN 192836
CAS :AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formule :C12H13N3O2Couleur et forme :SolidMasse moléculaire :231.25Dibenamine hydrochloride
CAS :Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.Formule :C16H19Cl2NDegré de pureté :96.43%Couleur et forme :Oily Liquid SolidMasse moléculaire :296.23BI-167107
CAS :BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).Formule :C21H26N2O4Couleur et forme :SolidMasse moléculaire :370.44Fiduxosin
CAS :Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormule :C30H29N5O4SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :555.65(-)-Isoproterenol hydrochloride
CAS :(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.Formule :C11H17NO3·CIHCouleur et forme :SolidMasse moléculaire :247.72Pronetalol
CAS :Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].Formule :C15H19NOCouleur et forme :SolidMasse moléculaire :229.32SDZ-NVI-085
CAS :SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formule :C15H21NO2SCouleur et forme :SolidMasse moléculaire :279.4Lidamidine
CAS :Lidamidine (Lidamidinum) is an effective antidiarrheal agent that inhibits intestinal secretion, reduces intestinal transit, and inhibits smooth muscleFormule :C11H16N4ODegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :220.27Ref: TM-T25719
1mg115,00€2mg162,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€Ro-70-0004
CAS :Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formule :C20H24F4N4O3Couleur et forme :SolidMasse moléculaire :444.424-hydroxy Nebivolol hydrochloride
CAS :4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.Formule :C22H25F2NO5HClCouleur et forme :SolidMasse moléculaire :457.9OPC-28326
CAS :OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formule :C26H35N3O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :421.58Ref: TM-T13804
1mg177,00€5mg432,00€1mL*10mM (DMSO)537,00€10mg587,00€25mg892,00€50mg1.198,00€100mg1.575,00€200mg2.133,00€Talibegron hydrochloride
CAS :Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formule :C18H22ClNO4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :351.83α1 adrenoceptor-MO-1
CAS :α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Formule :C20H24ClN5ODegré de pureté :99.20% - 99.29%Couleur et forme :SolidMasse moléculaire :385.89Ref: TM-T10003
1mg188,00€5mg371,00€1mL*10mM (DMSO)442,00€10mg513,00€25mg743,00€50mg1.018,00€100mg1.378,00€200mg1.863,00€Deriglidole
CAS :Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Formule :C16H21N3Degré de pureté :98.12% - 99.03%Couleur et forme :SolidMasse moléculaire :255.36(±)-Prenalterol
CAS :(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formule :C12H19NO3Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :225.280990CL
CAS :0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormule :C21H21N5Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :343.42Ref: TM-T13983
1mg192,00€5mg485,00€1mL*10mM (DMSO)507,00€10mg700,00€25mg1.063,00€50mg1.459,00€100mg1.963,00€CGP-20712
CAS :CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formule :C23H25F3N4O5Degré de pureté :99.40% - 99.58%Couleur et forme :SolidMasse moléculaire :494.46Ref: TM-T30846
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€PF-9404C
CAS :PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.Formule :C16H25N3O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.38Anti-MRSA agent 19
CAS :Anti-MRSA agent 19 (Compound 1) is an antibiotic that exhibits activity against Staphylococcus aureus. It is active against 40 clinical isolates from the CDC, representing diverse bacterial species with various resistance factors, including resistance to vancomycin, aminoglycoside/tetracycline, and oxazolidinone (median MIC=4 μg/mL).Formule :C15H10Cl3NO4Couleur et forme :SolidMasse moléculaire :374.6Carazolol hydrochloride
CAS :Carazolol (BM 51052) hydrochloride is a potent antagonist of β1/β2-adrenoceptors and also serves as a powerful and selective agonist of β3-adrenoceptors. It is utilized in research focusing on hypertension.Formule :C18H23ClN2O2Couleur et forme :SolidMasse moléculaire :334.84LK 11
CAS :LK-11, an alkaloid derivative, inhibits the passive uptake of norepinephrine (NA) by synaptic vesicles in the thalamus, similarly to cocaine.Formule :C15H26N2O3Couleur et forme :SolidMasse moléculaire :282.38
