
Récepteur adrénergique
Les récepteurs adrénergiques sont des GPCR activés par les catécholamines, telles que l'adrénaline et la noradrénaline. Ces récepteurs sont classés en sous-types alpha et bêta, chacun jouant un rôle clé dans la régulation du rythme cardiaque, de la pression artérielle et de la réponse de lutte ou de fuite. Les modulateurs des récepteurs adrénergiques sont essentiels dans le traitement des maladies cardiovasculaires, de l'asthme et des troubles anxieux. Chez CymitQuimica, nous offrons une large gamme de modulateurs des récepteurs adrénergiques de haute qualité pour soutenir vos recherches en endocrinologie, pharmacologie cardiovasculaire et réponse au stress.
Sous-catégories appartenant à la catégorie "Récepteur adrénergique"
645 produits trouvés pour "Récepteur adrénergique"
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Butanserin
CAS :<p>Butanserin is a 5-hydroxytryptamine S2-antagonist.</p>Formule :C24H26FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.48Methyldopa hydrochloride
CAS :<p>L-(-)-α-Methyldopa HCl: alpha-adrenergic agonist, antihypertensive, inhibits DOPA decarboxylase.</p>Formule :C10H14ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.68Afurolol Hydrochloride
CAS :<p>Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.</p>Formule :C15H22ClNO4Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :315.79Ulimorelin
CAS :<p>Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.</p>Formule :C30H39FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :538.65Ronactolol
CAS :<p>Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.</p>Formule :C20H26N2O4Couleur et forme :SolidMasse moléculaire :358.43Levobetaxolol
CAS :<p>Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.</p>Formule :C18H29NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.43Guanfacine
CAS :<p>Guanfacine is a selective agonist of the α2A receptor.</p>Formule :C9H9Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :246.09Arnolol
CAS :<p>Arnolol, a beta blocker, slows heart rate, reduces force of beats, lowers blood pressure, and enhances blood flow.</p>Formule :C14H23NO3Couleur et forme :SolidMasse moléculaire :253.34Lubabegron
CAS :<p>Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.</p>Formule :C29H29N3O3SCouleur et forme :SolidMasse moléculaire :499.62Zolertine HCl
CAS :<p>Zolertine HCl is an antagonist of alpha-Adrenoceptor.</p>Formule :C13H19ClN6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.78Cirazoline (free base)
CAS :<p>Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.</p>Formule :C13H16N2OCouleur et forme :SolidMasse moléculaire :216.28ZD 7114 hydrochloride
CAS :<p>β3-adrenoceptor agonist</p>Formule :C22H31ClN2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.94Protokylol
CAS :<p>Protokylol is a β-adrenergic receptor agonist.</p>Formule :C18H21NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.36Metazosin
CAS :<p>Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.</p>Formule :C18H25N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :375.42Piribedil dihydrochloride
CAS :<p>dopamine agonist</p>Formule :C16H20Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.26Todralazine
CAS :<p>Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.</p>Formule :C11H12N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.24BFE-55
CAS :<p>BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors</p>Formule :C14H19NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.31(RS)-Butyryltimolol
CAS :<p>(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.</p>Formule :C17H30N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.51L-Alprenolol
CAS :<p>L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.</p>Formule :C15H23NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.35Centanafadine
CAS :<p>Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).</p>Formule :C15H15NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :209.29S(-)-Bisoprolol
CAS :<p>S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.</p>Formule :C18H31NO4Couleur et forme :SolidMasse moléculaire :325.44Spirendolol
CAS :<p>Spirendolol is an antagonist of β adrenergic receptor.</p>Formule :C21H31NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.48Epinephrine bitartrate
CAS :<p>L-Epinephrine Bitartrate is alpha- and beta-adrenergic receptor stimulator.</p>Formule :C13H19NO9Degré de pureté :98.6% - 99.07%Couleur et forme :White SolidMasse moléculaire :333.3Epanolol
CAS :<p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>Formule :C20H23N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.41Adrenaline sulfate
CAS :<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Formule :C9H15NO7SCouleur et forme :SolidMasse moléculaire :281.279Broxaterol
CAS :<p>Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.</p>Formule :C9H15BrN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :263.13B-HT 933 dihydrochloride
CAS :<p>Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.</p>Formule :C9H17Cl2N3OCouleur et forme :SolidMasse moléculaire :254.16Levobunolol
CAS :<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Formule :C17H25NO3Couleur et forme :White To Pink PowderMasse moléculaire :291.39Bufetolol
CAS :<p>Bufetolol is an antagonist of beta-adrenoceptor.</p>Formule :C18H29NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.43Alprenolol tartrate, (S)-
CAS :<p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>Formule :C19H29NO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.44Guanoxabenz hydrochloride
CAS :<p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>Formule :C8H9Cl3N4OCouleur et forme :SolidMasse moléculaire :283.54Methyldopate hydrochloride
CAS :<p>Methyldopate HCl is an agent of antihypertensive.</p>Formule :C12H18ClNO4Couleur et forme :SolidMasse moléculaire :275.73UK 1745
CAS :<p>UK 1745 is a novel drug of cardiotonic.</p>Formule :C16H23ClN2O2Couleur et forme :SolidMasse moléculaire :310.82Guanethidine
CAS :<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Formule :C10H22N4Couleur et forme :SolidMasse moléculaire :198.31A 55453
CAS :<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Formule :C25H32N6O3Couleur et forme :SolidMasse moléculaire :464.56RS 79948 hydrochloride
CAS :<p>α2-adrenoreceptor antagonist</p>Formule :C19H29ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.96MK761
CAS :<p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>Formule :C13H19N3O2Couleur et forme :SolidMasse moléculaire :249.31Napamezole
CAS :<p>Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.</p>Formule :C14H16N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :212.29Flestolol sulfate
CAS :<p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>Formule :C15H24FN3O8SCouleur et forme :SolidMasse moléculaire :425.43BMS-466442
CAS :<p>BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.</p>Formule :C31H30N4O5Couleur et forme :SolidMasse moléculaire :538.59Mabuterol hydrochloride
CAS :<p>Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.</p>Formule :C13H19Cl2F3N2OCouleur et forme :SolidMasse moléculaire :347.20Arbutamine hydrochloride
CAS :<p>Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.</p>Formule :C18H24ClNO4Couleur et forme :SolidMasse moléculaire :353.84Fenmetozole
CAS :<p>Fenmetozole is an antagonist of the actions of ethanol.</p>Formule :C10H10Cl2N2OCouleur et forme :SolidMasse moléculaire :245.11CP 59430
CAS :<p>CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.</p>Formule :C21H22N8O3Couleur et forme :SolidMasse moléculaire :434.45Clencyclohexerol
CAS :<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Formule :C14H20Cl2N2O2Couleur et forme :SolidMasse moléculaire :319.23Dapiprazole
CAS :<p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>Formule :C19H27N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :325.45BRL 37344 sodium
CAS :<p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>Formule :C19H22ClNNaO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.83Pronethalol hydrochloride
CAS :<p>β-adrenergic antagonist</p>Formule :C15H20ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.78Naminterol
CAS :<p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>Formule :C19H26N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.42Zenidolol
CAS :<p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>Formule :C17H27NO2Couleur et forme :SolidMasse moléculaire :277.4ONO-2952
CAS :<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Formule :C22H20ClFN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.86(-)-S-Timolol
CAS :<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Formule :C13H26N4O4SCouleur et forme :SolidMasse moléculaire :334.44Trimazosin
CAS :<p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>Formule :C20H29N5O6Couleur et forme :SolidMasse moléculaire :435.47Primidolol
CAS :<p>Primidolol is a beta adrenergic receptor antagonist and antihypertensive agent.</p>Formule :C17H23N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.38Oxyfedrine
CAS :<p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>Formule :C19H23NO3Couleur et forme :SolidMasse moléculaire :313.39Ko-3290
CAS :<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Formule :C19H25N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :343.42Imiloxan hydrochloride
CAS :<p>Imiloxan hydrochloride is an α2-adrenoceptor antagonist.</p>Formule :C14H17ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :280.75Metrenperone
CAS :<p>Metrenperone is used as a S(2)-receptor blocker.</p>Formule :C24H26FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :407.48Zinterol hydrochloride
CAS :<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Formule :C19H27ClN2O4SCouleur et forme :SolidMasse moléculaire :414.95Hexoprenaline
CAS :<p>Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.</p>Formule :C22H32N2O6Couleur et forme :SolidMasse moléculaire :420.5Fenmetozole Tosylate
CAS :<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Formule :C17H18Cl2N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :417.31Agroclavine
CAS :<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Formule :C16H18N2Couleur et forme :SolidMasse moléculaire :238.33ADRA1D receptor antagonist 1 free base
CAS :<p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>Formule :C15H13ClN4OCouleur et forme :SolidMasse moléculaire :300.74(E)-Guanabenz
CAS :<p>(E)-Guanabenz is an oral α2-adrenoceptor agonist, antihypertensive, GADD34 inhibitor, and has neuroprotective properties.</p>Formule :C8H8Cl2N4Couleur et forme :SolidMasse moléculaire :231.08Ro 363 hydrochloride
CAS :<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Formule :C19H26ClNO6Couleur et forme :SolidMasse moléculaire :399.87Pargolol hydrochloride
CAS :<p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>Formule :C16H24ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.82Edivoxetine
CAS :<p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>Formule :C18H26FNO4Couleur et forme :SolidMasse moléculaire :339.4Medroxalol
CAS :<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Formule :C20H24N2O5Couleur et forme :SolidMasse moléculaire :372.42Povafonidine
CAS :<p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>Formule :C11H13N5Couleur et forme :SolidMasse moléculaire :215.25MG 1
CAS :<p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>Formule :C17H25N3O2Degré de pureté :98.98% - >99.99%Couleur et forme :SolidMasse moléculaire :303.4ZK-90055 hydrochloride
CAS :<p>ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.</p>Formule :C16H23ClN2O4Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :342.82Thioproperazine
CAS :<p>Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.</p>Formule :C22H30N4O2S2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :446.63Guanadrel
CAS :<p>Guanadrel is an antihypertensive agent.</p>Formule :C10H19N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :213.28(E)-Alprenoxime
CAS :<p>(E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.</p>Formule :C15H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.35Dexnafenodone Hydrochloride
CAS :<p>Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.</p>Formule :C20H24ClNOCouleur et forme :SolidMasse moléculaire :329.86LY 87130
CAS :<p>LY 87130 is a phenylethanolamine-N-methyltransferase inhibitor.</p>Formule :C12H13NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :171.24Talsupram hydrochloride
CAS :<p>noradrenalin re-uptake inhibitor</p>Formule :C20H26ClNSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.95RS 52367
CAS :<p>RS 52367 is a beta-adrenergic antagonist.</p>Formule :C18H34ClN3O3SCouleur et forme :SolidMasse moléculaire :408S 12024-2
CAS :<p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>Formule :C16H26N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.45Flerobuterol
CAS :<p>Flerobuterol is a potential antidepressant agent related to beta-adrenergic agonists.</p>Formule :C12H18FNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :211.28Befunolol HCl
CAS :<p>Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.</p>Formule :C16H22ClNO4Couleur et forme :SolidMasse moléculaire :327.8Flutonidine
CAS :<p>Flutonidine is an agonist of alpha2-Adrenergic receptor.</p>Formule :C10H12FN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :193.22S-Nitroso-N-acetylcysteine
CAS :<p>S-Nitroso-N-acetylcysteine inhibits proliferation and survival of multiple MM cells. It acts by the S-nitrosylation-dependent inhibition of STAT3 and NF-κB.</p>Formule :C5H8N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :192.19Bremazocine
CAS :<p>Bremazocineis a potent opiate kappa-agonist and centrally acting analgesic.</p>Formule :C20H29NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.45RS 15385-197
CAS :<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Formule :C18H26N2O3SCouleur et forme :SolidMasse moléculaire :350.48Garomefrine HCl
CAS :<p>Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.</p>Formule :C9H14ClFN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.73Cafaminol
CAS :<p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>Formule :C11H17N5O3Couleur et forme :SolidMasse moléculaire :267.28R 47243
CAS :<p>R 47243 is used as a racemic alpha 2 antagonist.</p>Formule :C22H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :395.52Burimamide
CAS :<p>Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.</p>Formule :C9H16N4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :212.32BE 2254
CAS :<p>BE 2254 is an antagonist of central noradrenergic receptor.</p>Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38Dabuzalgron HCl
CAS :<p>Dabuzalgron, an adrenoceptor agonist, is used potentially for the treatment of urinary incontinence.</p>Formule :C12H17Cl2N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :354.25Butidrine
CAS :<p>Butidrine has an Antiarrhythmic activities.</p>Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38Dipiproverine hydrochloride
CAS :<p>Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.</p>Formule :C20H32Cl2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.39JTH-601 free base
CAS :<p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>Formule :C24H35NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54JNJ-7925476 HCl
CAS :<p>JNJ-7925476 HCl inhibits DAT, NET, SERT; ED(50): DAT 2.4, NET 0.09, SERT 0.18 mg/kg in rats.</p>Formule :C20H20ClNCouleur et forme :SolidMasse moléculaire :309.83L-748328
CAS :<p>L-748328 is a potent and selective antagonist of human beta(3)-adrenergic receptor.</p>Formule :C23H27N3O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.61SKF 86466 hydrochloride
CAS :<p>SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.</p>Formule :C11H15Cl2NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.15KUL-7211
CAS :<p>KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.</p>Formule :C19H23NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.39Esprolol hydrochloride
CAS :<p>Esprolol is a β-adrenergic receptor antagonist.</p>Formule :C17H28ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.86Dipiproverine
CAS :<p>Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.</p>Formule :C20H30N2O2Couleur et forme :SolidMasse moléculaire :330.46Dihydroalprenolol, (S)-
CAS :<p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>Formule :C15H25NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :251.36Levomoprolol
CAS :<p>Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.</p>Formule :C13H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.31L-771688 dihydrochloride
CAS :<p>L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.</p>Formule :C28H35Cl2F2N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :630.51Levoprotiline
CAS :<p>Levoprotiline, a fast-acting antidepressant, is the R-enantiomer of Oxaprotiline and successor to maprotiline.</p>Formule :C20H23NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.4SNAP 5089
CAS :<p>α1A-adrenoceptor antagonist</p>Formule :C36H40N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.73Dilevalol
CAS :<p>Dilevalol, an RR-stereoisomer of labetalol, is a beta-blocker with partial beta 2-agonism and minimal alpha 1-blockade.</p>Formule :C19H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.41Delequamine HCl
CAS :<p>Delequamine HCl: potent, selective alpha 2-adrenoceptor blocker; pKi 9.45 in rat cortex, pA2 9.72 in guinea-pig ileum.</p>Formule :C18H27ClN2O3SCouleur et forme :SolidMasse moléculaire :386.94Oxaprotiline
CAS :<p>Oxaprotiline: an antidepressant, norepinephrine inhibitor, and H1 blocker; studied in hospital depression but not marketed.</p>Formule :C20H23NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.4Zometapine
CAS :<p>Zometapine (CI 716) is an antidepressant compound that is a derivative of pyrazole and diazepine.</p>Formule :C14H15ClN4Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :274.75Levoprotiline hydrochloride
CAS :<p>Levoprotiline hydrochloride is an antidepressant.</p>Formule :C20H24ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.86FMS586
CAS :<p>FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.</p>Formule :C24H30N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :390.52Tilisolol HCl
CAS :<p>Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.</p>Formule :C17H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :340.85(S)-Viloxazine Hydrochloride
CAS :<p>(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.</p>Formule :C13H20ClNO3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :273.76Tranterol hydrochloride
CAS :<p>Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.</p>Formule :C13H19Cl2F3N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.2Pamatolol
CAS :<p>Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.</p>Formule :C16H26N2O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :310.39Cicloprolol hydrochloride
CAS :<p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>Formule :C18H30ClNO4Degré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :359.89L-771688
CAS :<p>L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign</p>Formule :C28H33F2N5O5Degré de pureté :94.15%Couleur et forme :SolidMasse moléculaire :557.59Indanidine
CAS :<p>Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the</p>Formule :C11H13N5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :215.25TD-5471 hydrochloride
CAS :<p>TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (</p>Formule :C32H32ClN3O4Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :558.07Napitane
CAS :<p>napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the</p>Formule :C22H25NO2Degré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :335.44Norfenefrine HCl
CAS :<p>Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.</p>Formule :C8H12ClNO2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :189.64KUL-7211 racemate
CAS :<p>KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.</p>Formule :C19H23NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.39Ro 363
CAS :<p>RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.</p>Formule :C19H25NO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.4Labetalone hydrochloride
CAS :<p>Labetalone hydrochloride, a Labetalol impurity, is an orally active alpha and beta-adrenoceptor blocker.</p>Formule :C19H23ClN2O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :362.85Naphazoline
CAS :<p>Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity.</p>Formule :C14H14N2Degré de pureté :99.79%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :210.27Moprolol
CAS :<p>Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].</p>Formule :C13H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.31N-Methyldopamine hydrochloride
CAS :<p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>Formule :C9H14ClNO2Couleur et forme :SolidMasse moléculaire :203.67Ancarolol
CAS :<p>Ancarolol is a blocking agent of beta-adrenergic.</p>Formule :C18H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.39Rec 15/2615 dihydrochloride
CAS :<p>Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.</p>Formule :C26H35Cl2N5O5Degré de pureté :97.04% - 99.76%Couleur et forme :SolidMasse moléculaire :568.49Arbutamine
CAS :<p>Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.</p>Formule :C18H23NO4Degré de pureté :95.06%Couleur et forme :SolidMasse moléculaire :317.38(S)-(-)-Propranolol hydrochloride
CAS :<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>Formule :C16H22ClNO2Degré de pureté :99.02% - 99.91%Couleur et forme :SolidMasse moléculaire :295.8(S)-Terazosin
CAS :<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Formule :C19H25N5O4Couleur et forme :SolidMasse moléculaire :387.43T-0509
CAS :<p>T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-</p>Formule :C18H23NO5Degré de pureté :97.52% - 98.43%Couleur et forme :SolidMasse moléculaire :333.38Cyclazosin HCl
CAS :<p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>Formule :C23H28ClN5O4Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :473.95Levobunolol hydrochloride
CAS :<p>Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。</p>Formule :C17H26ClNO3Degré de pureté :98.49% - >99.99%Couleur et forme :SolidMasse moléculaire :327.85L748337
CAS :<p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>Formule :C26H31N3O5SDegré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :497.61ADRA1D receptor antagonist 1 HCl
CAS :<p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>Formule :C15H14Cl2N4ODegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :337.2Romifidine
CAS :<p>Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.</p>Formule :C9H9BrFN3Couleur et forme :SolidMasse moléculaire :258.09LY377604
CAS :<p>LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.</p>Formule :C31H32N4O4Degré de pureté :99.72% - >99.99%Couleur et forme :SolidMasse moléculaire :524.61SM-2470
CAS :<p>SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.</p>Formule :C23H30ClN5O3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :459.97Falintolol
CAS :<p>Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.</p>Formule :C12H24N2O2Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :228.33Bedoradrine sulfate
CAS :<p>Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formule :C24H32N2O5H2O4SDegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :477.56GP2-114
CAS :<p>GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.</p>Formule :C19H24N2O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :344.4Egis-11150
CAS :<p>Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.</p>Formule :C19H21ClFN5O2Degré de pureté :97.49% - >99.99%Couleur et forme :SolidMasse moléculaire :405.85Amosulalol
CAS :<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formule :C18H24N2O5SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :380.46CL 316243
CAS :<p>CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.</p>Formule :C20H18ClNNa2O7Degré de pureté :98.00% - 99.68%Couleur et forme :SolidMasse moléculaire :465.79Midaglizole hydrochloride
CAS :<p>Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).</p>Formule :C16H19Cl2N3Degré de pureté :99.39% - 99.82%Couleur et forme :SolidMasse moléculaire :324.25Soquinolol
CAS :<p>Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long</p>Formule :C17H26N2O3Degré de pureté :97.48% - 98.63%Couleur et forme :SolidMasse moléculaire :306.4Neldazosin
CAS :<p>Neldazosin is used as a potent α1-adrenoceptor antagonist.</p>Formule :C18H25N5O4Degré de pureté :99.74% - 99.76%Couleur et forme :SolidMasse moléculaire :375.42Oxyfedrine L-form HCl
CAS :<p>Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.</p>Formule :C19H24ClNO3Degré de pureté :99.5% - 99.57%Couleur et forme :SolidMasse moléculaire :349.85JP1302
CAS :<p>JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.</p>Formule :C24H24N4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :368.47Ecastolol
CAS :<p>Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.</p>Formule :C26H33N3O6Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :483.56Nemazoline Free Base
CAS :<p>Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.</p>Formule :C10H11Cl2N3Degré de pureté :98.06% - 98.83%Couleur et forme :SolidMasse moléculaire :244.12Butofilolol
CAS :<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Formule :C17H26FNO3Degré de pureté :98.96% - >99.99%Couleur et forme :SolidMasse moléculaire :311.392Rafabegron
CAS :<p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>Formule :C21H23ClN2O4Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :402.87Pipoxazole
CAS :<p>Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.</p>Formule :C14H20N4ODegré de pureté :98.58% - 99.53%Couleur et forme :SolidMasse moléculaire :260.33Taprizosin
CAS :<p>Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.</p>Formule :C25H26N6O4SDegré de pureté :96.34% - 99.11%Couleur et forme :SolidMasse moléculaire :506.58Milveterol HCl
CAS :<p>Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).</p>Formule :C25H30ClN3O4Degré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :471.98(S)-(+)-Niguldipine hydrochloride
CAS :<p>(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.</p>Formule :C36H40ClN3O6Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :646.17Dabelotine
CAS :<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Formule :C15H22N2O2Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :262.35Besipirdine
CAS :<p>Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.</p>Formule :C16H17N3Degré de pureté :97.15% - 98.85%Couleur et forme :SolidMasse moléculaire :251.33Palatrigine
CAS :<p>Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.</p>Formule :C12H13Cl2N5Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :298.17Bisaramil hydrochloride
CAS :<p>Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.</p>Formule :C17H24Cl2N2O2Degré de pureté :98.64% - 99.48%Couleur et forme :SolidMasse moléculaire :359.29Imiloxan
CAS :<p>Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.</p>Formule :C14H16N2O2Degré de pureté :98.13% - 99.8%Couleur et forme :SolidMasse moléculaire :244.29ST 91
CAS :<p>ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.</p>Formule :C13H20ClN3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :253.77ORM-10921
CAS :<p>ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.</p>Formule :C18H23NO2Degré de pureté :99.46% - 99.85%Couleur et forme :SolidMasse moléculaire :285.38Fipamezole
CAS :<p>Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.</p>Formule :C14H15FN2Degré de pureté :99.32% - >99.99%Couleur et forme :SolidMasse moléculaire :230.28Xamoterol hemifumarate
CAS :<p>Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationship</p>Formule :C36H54N6O14Degré de pureté :99.79%Couleur et forme :White SolidMasse moléculaire :794.37Rezatomidine
CAS :<p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>Formule :C13H16N2SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :232.34Bedoradrine
CAS :<p>Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formule :C24H32N2O5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :428.52Vatinoxan hydrochloride
CAS :<p>Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.</p>Formule :C20H27ClN4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.97Nolomirole HCl
CAS :<p>Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to study</p>Formule :C19H28ClNO4Degré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :369.88Abediterol
CAS :<p>Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.</p>Formule :C25H30F2N2O4Couleur et forme :SolidMasse moléculaire :460.51N-5984
CAS :<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formule :C20H22ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.854-hydroxy Nebivolol hydrochloride
CAS :<p>4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.</p>Formule :C22H25F2NO5HClCouleur et forme :SolidMasse moléculaire :457.9(-)-Isoproterenol hydrochloride
CAS :<p>(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.</p>Formule :C11H17NO3·CIHCouleur et forme :SolidMasse moléculaire :247.72BI-167107
CAS :<p>BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).</p>Formule :C21H26N2O4Couleur et forme :SolidMasse moléculaire :370.44AGN 192836
CAS :<p>AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).</p>Formule :C12H13N3O2Couleur et forme :SolidMasse moléculaire :231.25β3-AR agonist 2
CAS :<p>β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).</p>Formule :C27H38N4O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.68Mefenidil
CAS :<p>Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.</p>Formule :C12H11N3Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :197.24(±)-N-Methylcoclaurine
CAS :<p>N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].</p>Formule :C18H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :299.36Todralazine hydrochloride
CAS :<p>Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.</p>Formule :C11H13ClN4O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :268.7BMS-194449
CAS :<p>BMS-194449 is a full beta 3 agonist.</p>Formule :C24H24F4N2O6SCouleur et forme :SolidMasse moléculaire :544.52Celiprolol hydrochloride
CAS :<p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>Formule :C20H33N3O4·HClCouleur et forme :White Crystalline SolidMasse moléculaire :415.96Bunazosin Hydrochloride
CAS :<p>Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.</p>Formule :C19H28ClN5O3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :409.91BU-E 75
CAS :<p>BU-E 75 is an agonist of the histamine H2.</p>Formule :C21H24F2N6Couleur et forme :SolidMasse moléculaire :398.45β3-AR agonist 1
CAS :<p>β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/</p>Formule :C22H28N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :444.55L-796568 free base
CAS :<p>L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).</p>Formule :C31H27F3N4O3S2Couleur et forme :SolidMasse moléculaire :624.7RS100329 hydrochloride
CAS :<p>RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.</p>Formule :C20H26ClF3N4O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :462.89Bufuralol (hydrochloride)
CAS :<p>Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.</p>Formule :C16H24ClNO2Couleur et forme :SolidMasse moléculaire :297.82LK 204-545
CAS :<p>LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.</p>Formule :C25H32N4O6Couleur et forme :SolidMasse moléculaire :484.54NGD9002
CAS :<p>NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.</p>Formule :C20H31N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.49L-796568 dihydrochloride
CAS :<p>L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.</p>Formule :C31H29Cl2F3N4O3S2Couleur et forme :SolidMasse moléculaire :697.62RS 17053 hydrochloride
CAS :<p>RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.</p>Formule :C24H30Cl2N2O2Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :449.41Ritodrine
CAS :<p>Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].</p>Formule :C17H21NO3Couleur et forme :SolidMasse moléculaire :287.35Binedaline
CAS :<p>Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.</p>Formule :C19H23N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.41Epinephrine HCl
CAS :<p>Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.</p>Formule :C9H14ClNO3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :219.67Dibenamine hydrochloride
CAS :<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Formule :C16H19Cl2NDegré de pureté :96.43%Couleur et forme :Oily Liquid SolidMasse moléculaire :296.23AR-08
CAS :<p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>Formule :C12H12N6Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :240.26Fiduxosin
CAS :<p>Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki</p>Formule :C30H29N5O4SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :555.65
