Récepteur adrénergique
Les récepteurs adrénergiques sont des GPCR activés par les catécholamines, telles que l'adrénaline et la noradrénaline. Ces récepteurs sont classés en sous-types alpha et bêta, chacun jouant un rôle clé dans la régulation du rythme cardiaque, de la pression artérielle et de la réponse de lutte ou de fuite. Les modulateurs des récepteurs adrénergiques sont essentiels dans le traitement des maladies cardiovasculaires, de l'asthme et des troubles anxieux. Chez CymitQuimica, nous offrons une large gamme de modulateurs des récepteurs adrénergiques de haute qualité pour soutenir vos recherches en endocrinologie, pharmacologie cardiovasculaire et réponse au stress.
Sous-catégories appartenant à la catégorie "Récepteur adrénergique"
730 produits trouvés pour "Récepteur adrénergique"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ivabradine-d3 hydrochloride
CAS :Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Formule :C27H37ClN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.07Yohimbic acid, ethyl ester
CAS :Yohimbic acid, ethyl ester is a biochemical with possible effects on reserpine action.Formule :C22H28N2O3Couleur et forme :SolidMasse moléculaire :368.47Synephrine hemitartrate
CAS :Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.Formule :C9H13NO2C4H6O6Couleur et forme :SolidMasse moléculaire :242.26O-Desmethyl Mebeverine alcohol hydrochloride
CAS :O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.Formule :C15H26ClNO2Couleur et forme :SolidMasse moléculaire :287.83Phendioxan
CAS :Phendioxan is a biochemcial.Formule :C25H27NO5Couleur et forme :SolidMasse moléculaire :421.49Cetamolol hydrochloride
CAS :Cetamolol hydrochloride is a biochemical.Formule :C16H27ClN2O4Couleur et forme :SolidMasse moléculaire :346.85SU 4029 dihydrochloride
CAS :SU 4029 dihydrochloride is a bioactive chemical.Formule :C9H21Cl2N3OCouleur et forme :SolidMasse moléculaire :258.19(±)-4-hydroxy Propranolol β-D-Glucuronide
CAS :(±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol , which is a metabolite of propranolol.Formule :C22H29NO9Couleur et forme :SolidMasse moléculaire :451.47Desglymidodrine
CAS :Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Formule :C10H15NO3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :197.23Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Formule :C22H30N2O7SDegré de pureté :97.05% - 98.53%Couleur et forme :SoildMasse moléculaire :466.55Carbazochrome salicylate
CAS :Carbazochrome salicylate can be used as a coagulant.Formule :C17H18N4NaO6Couleur et forme :White Crystalline PowderMasse moléculaire :397.343Bamosiran
CAS :Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.Couleur et forme :SolidCTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formule :C97H131F3I2N20O25S2Couleur et forme :SolidMasse moléculaire :2352.13Benzquinamide
CAS :Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancerFormule :C22H32N2O5Degré de pureté :94.86%Couleur et forme :SolidMasse moléculaire :404.5PNMT-IN-1
PNMT-IN-1 (inhibitor 4) is a selective second generation inhibitor [1] of phenylethanolamine N-methyltransferase (PNMT), exhibiting a Ki value of 1.2 nM and anCouleur et forme :Odour SolidSB-206606
CAS :SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.Formule :C19H22ClNO4Couleur et forme :SolidMasse moléculaire :363.83Chir 2279
CAS :CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).Formule :C34H36N4O4Couleur et forme :SolidMasse moléculaire :564.67Quinazosin hydrochloride
CAS :Quinazosin hydrochloride is an antihypertensive agent.Formule :C17H25Cl2N5O2Couleur et forme :SolidMasse moléculaire :402.32(+)-ORM-10921
CAS :(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.Formule :C18H23NO2Degré de pureté :99.23%Couleur et forme :SoildMasse moléculaire :285.38CTP-347
CAS :CTP-347, a deuterated version of paroxetine, is potentially the best non-hormonal drug in its class for the treatment of hot flashes.Formule :C19H20FNO3Couleur et forme :SolidMasse moléculaire :331.38YM 09538
CAS :YM 09538 is a biochemical.Formule :C18H25ClN2O5SCouleur et forme :SolidMasse moléculaire :416.92Dabelotine, (R)-
CAS :Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formule :C15H22N2O2Couleur et forme :SolidMasse moléculaire :262.35Mapenterol hydrochloride
CAS :Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.Formule :C14H21Cl2F3N2ODegré de pureté :98.11% - 99.98%Couleur et forme :SolidMasse moléculaire :361.23Ref: TM-T40622
1mg49,00€5mg102,00€1mL*10mM (DMSO)107,00€10mg149,00€25mg249,00€50mg358,00€100mg520,00€500mg1.035,00€Moxonidine hydrochloride
CAS :Moxonidine Hydrochloride: selective I1 imidazoline receptor agonist, stronger than α2-AR; lowers blood pressure; central action.Formule :C9H13Cl2N5OCouleur et forme :SolidMasse moléculaire :278.14TH023
TH023 is an inhibitor of the TLR4 signaling pathway, specifically targeting the formation of TLR4 homodimers. In HEK-Blue hTLR4 cells, TH023 suppresses the secretion of embryonic alkaline phosphatase with an IC50 of 0.354 μM and inhibits NO expression in RAW264.7 cells, with an IC50 of 1.61 μM. Additionally, TH023 inhibits the activation of NF-κB and reduces the nuclear translocation of NF-κB p65. The compound demonstrates anti-inflammatory effects in a mouse model of LPS-induced acute sepsis and improves lung injury in mice.Formule :C22H21ClF2N4OCouleur et forme :SolidMasse moléculaire :430.88Phenylethanolamine A
CAS :Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formule :C19H24N2O4Couleur et forme :SolidMasse moléculaire :344.40Sibenadet hydrochloride
CAS :Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.Formule :C22H29ClN2O5S2Couleur et forme :SolidMasse moléculaire :501.06α1A-AR Degrader 9c
CAS :α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Formule :C38H43N11O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :829.82Agaridoxin
CAS :Agaridoxin is a mushroom metabolite.
Formule :C11H14N2O5Couleur et forme :SolidMasse moléculaire :254.242Formoterol O-β-D-Glucuronide
CAS :Formoterol O-β-D-glucuronide is a metabolite of formoterol .Formule :C25H32N2O10Couleur et forme :SolidMasse moléculaire :520.535Idazoxan
CAS :Idazoxan is an alpha2 receptor antagonist that also exhibits activity at imidazoline [I1] and [I2] receptors, playing a role in modulating dopamine release.Formule :C11H12N2O2Masse moléculaire :204.23Bucindolol Formate
Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.Formule :C23H27N3O4Degré de pureté :99.76% - 99.88%Couleur et forme :SolidMasse moléculaire :409.48Nolomirole
CAS :Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.Formule :C19H27NO4Couleur et forme :SolidMasse moléculaire :333.42Oxaprotiline hydrochloride
CAS :Oxaprotiline hydrochloride is an antidepressant.Formule :C20H24ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.86AG-825
CAS :AG-825（Tyrphostin C15） is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (TyrphostinFormule :C19H15N3O3S2Degré de pureté :99.52%Couleur et forme :Yellow SolidMasse moléculaire :397.47Ref: TM-T14138
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg105,00€25mg222,00€50mg371,00€100mg597,00€500mg1.234,00€Carazolol-d7
CAS :Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.Formule :C18H22N2O2Couleur et forme :SolidMasse moléculaire :305.42(±)5(6)-EET
CAS :5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473Ethylnorepinephrine hydrochloride
CAS :Ethylnorepinephrine hydrochloride is a unique bronchodilator.
Formule :C10H16ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.69Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Couleur et forme :Odour Solid5-hydroxy Propranolol
CAS :5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Formule :C16H21NO3Couleur et forme :SolidMasse moléculaire :275.348Phenoxybenzamine
CAS :Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.Formule :C18H22ClNODegré de pureté :98%Couleur et forme :Crystals From Petroleum Ether SolidMasse moléculaire :303.83L-770644 dihydrochloride
CAS :L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formule :C30H38ClN7O4SCouleur et forme :SolidMasse moléculaire :628.19Terazosin dimer impurity dihydrochloride
CAS :Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.Formule :C24H30Cl2N8O4Couleur et forme :SolidMasse moléculaire :565.46(R)-(+)-Atenolol
CAS :(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formule :C14H22N2O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :266.34L-770644
CAS :L-770644 is an agonist of B3 adrenergic receptor.Formule :C30H37N7O4SCouleur et forme :SolidMasse moléculaire :591.72Amitraz
CAS :Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.Formule :C19H23N3Degré de pureté :99.88%Couleur et forme :White/Pale Yellow Crystalline SolidMasse moléculaire :293.41BMS-196085
CAS :BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.Formule :C24H26F2N2O5SCouleur et forme :SolidMasse moléculaire :492.54Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47Ritobegron HCl
CAS :Ritobegron (KUC-7483), a β3-adrenergic agonist, targets human β-AR effectively and is highly selective for rat bladder.Formule :C23H32ClNO5Couleur et forme :SolidMasse moléculaire :437.96Metaraminol
CAS :Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.Formule :C9H13NO2Couleur et forme :SolidMasse moléculaire :167.21
