AChR
Les inhibiteurs des récepteurs de l'acétylcholine (AChR) sont des composés qui bloquent l'activité des récepteurs de l'acétylcholine, essentiels pour la neurotransmission dans les systèmes nerveux central et périphérique. Les AChR jouent un rôle crucial dans la contraction musculaire, la mémoire et les fonctions cognitives. Les inhibiteurs des AChR sont utilisés pour étudier des conditions telles que la myasthénie grave, la maladie d'Alzheimer et d'autres troubles neurologiques. En modulant l'activité des AChR, ces inhibiteurs peuvent aider à démêler les complexités de la signalisation cholinergique dans le cerveau. Chez CymitQuimica, nous fournissons une gamme d'inhibiteurs des AChR pour soutenir vos recherches en neurosciences, pharmacologie et maladies neurodégénératives.
623 produits trouvés pour "AChR"
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5-AAM-2-CP
CAS :5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.Formule :C8H9ClN2ODegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :184.62Tropicamide
CAS :Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for diagnostic use.Formule :C17H20N2O2Degré de pureté :99.78% - 99.94%Couleur et forme :White PowderMasse moléculaire :284.35[Ala2,8,9,11,19,22,24,25,27,28]-VIP
CAS :[Ala2,8,9,11,19,22,24,25,27,28]-VIP can be used for related research in the field of life sciences. Its product number is T36637 and CAS number is 866552-34-3.Formule :C131H219N41O33SCouleur et forme :SolidMasse moléculaire :2928.51nAChR agonist CMPI hydrochloride
CAS :CMPI hydrochloride: Potent α4:α4 nAChR PAM; EC50 0.26 μM for (α4)3(β2)2 response to ACh; may aid nicotine dependence, neuropsychiatric research.Formule :C18H20Cl2N4OCouleur et forme :SolidMasse moléculaire :379.29R-(+)-Cotinine
CAS :R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.Formule :C10H12N2OCouleur et forme :SolidMasse moléculaire :176.22PDE4-IN-4
CAS :PDE4-IN-4 is a compound acting as both a potent M3 antagonist (p IC 50 = 10.2) and a PDE4 inhibitor (p IC 50 = 8.8), designed for inhalation-based treatment ofFormule :C36H37Cl2N3O7SCouleur et forme :SolidMasse moléculaire :726.67Muscarinic toxin 3
CAS :Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57Formule :C319H489N89O97S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7379.35Perlapine
CAS :Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM).Formule :C19H21N3Couleur et forme :SolidMasse moléculaire :291.39Cevimeline hydrochloride hemihydrate
CAS :<p>Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.</p>Formule :C20H38Cl2N2O3S2Degré de pureté :97.00%Couleur et forme :SolidMasse moléculaire :489.553-hydroxy Darifenacin
CAS :3-hydroxy Darifenacin, darifenacin metabolite, blocks M1-5 muscarinic receptors with varying potency (Kis: 2.24-79.43 nM) in CHO cells.Formule :C28H30N2O3Couleur et forme :SolidMasse moléculaire :442.559LtIA-F
LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.Formule :C86H121N25O22S4Couleur et forme :SolidMasse moléculaire :1985.31(S)-Dinotefuran
CAS :(S)-Dinotefuran, a neonicotinoid, more toxic to bees than its R-isomer, targets α8 nAChR.Formule :C7H14N4O3Couleur et forme :SolidMasse moléculaire :202.21MK-0969
CAS :MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.Formule :C24H30F2N4O2Couleur et forme :SolidMasse moléculaire :444.52Imidafenacin Metabolite M4
CAS :Imidafenacin M4 is a CYP3A4-formed metabolite of the muscarinic antagonist imidafenacin.Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.368ANQ-9040
CAS :ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.Formule :C36H58N2O5SCouleur et forme :SolidMasse moléculaire :630.92Octamylamine
CAS :Octamylamine is a bioactive chemical.Formule :C13H29NCouleur et forme :SolidMasse moléculaire :199.3761Epiboxidine hydrochloride
CAS :Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.Formule :C10H15ClN2OCouleur et forme :SolidMasse moléculaire :214.69M1/M4 muscarinic agonist 2
Compound 40 is a selective M1/M4 muscarinic antagonist with an IC50 of 19 nM for M1 receptors and 42 nM for M4 receptors [1].Couleur et forme :Odour SolidFlupyradifurone
CAS :<p>Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.</p>Formule :C12H11ClF2N2O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.68sabcomeline
CAS :Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.Formule :C10H15N3OCouleur et forme :SolidMasse moléculaire :193.25Lupanine hydrochloride
CAS :Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.Formule :C15H25ClN2OCouleur et forme :SolidMasse moléculaire :284.83α-Conotoxin imi
CAS :alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.Formule :C52H78N20O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1351.56Small Cardioactive Peptide B (SCPB)
CAS :SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).Formule :C52H80N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1141.41Navafenterol
CAS :AZD-8871, a potential COPD and asthma treatment, may work well with ICS.Formule :C38H42N6O6S2Couleur et forme :SolidMasse moléculaire :742.91Methylatropine (nitrate)
CAS :Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.Formule :C18H26N2O6Couleur et forme :SolidMasse moléculaire :366.414CDD0102 HCl
CAS :CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.Formule :C8H13ClN4ODegré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :216.67Destomycin A
CAS :Destomycin A, an aminoglycoside antibiotic, exhibits activity against bacterial (Gram-positive and Gram-negative), antifungal, and anthelmintic agents. It inhibits peptide synthesis in Escherichia coli cells and stimulates adenylate cyclase in animal tissues.Formule :C20H37N3O13Couleur et forme :SolidMasse moléculaire :527.52(+)-Coclaurine hydrochloride
CAS :(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.Formule :C17H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.8Fentonium bromide
CAS :<p>Fentonium bromide is a biochemical.</p>Formule :C31H34BrNO4Couleur et forme :SolidMasse moléculaire :564.51nAChR modulator-2
CAS :nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .Formule :C12H8ClN3O2Couleur et forme :SolidMasse moléculaire :261.66α-Conotoxin PIA
CAS :Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nMFormule :C79H125N27O25S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1981.3Ebiratide
CAS :Ebiratide is an analog of ACTH 4-9.Formule :C48H73N11O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :996.23[D-Trp7,9,10]-Substance P
CAS :<p>Substance P analog that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.</p>Formule :C79H105N21O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1588.89Pozanicline hydrochloride
Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.Formule :C11H17ClN2ODegré de pureté :97.13% - 99.81%Couleur et forme :SolidMasse moléculaire :228.72Ref: TM-T16563L
1mg77,00€5mg155,00€10mg220,00€25mg338,00€50mg472,00€100mg632,00€200mg853,00€1mL*10mM (DMSO)134,00€TC-2216
CAS :TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.Formule :C12H17N3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :203.28Oxotremorine
CAS :Oxotremorine acts as an agonist of mAChR, specifically activating the M1 and M3 acetylcholine receptors. In drug discrimination experiments with macaques, it exhibits effects similar to nicotine.Formule :C12H18N2OCouleur et forme :SolidMasse moléculaire :206.28PF-06827443
PF-06827443 is a orally bioavailable, CNS-penetrant M1-selective PAM with minimal agonist activity.Formule :C24H24N2O4Couleur et forme :SolidMasse moléculaire :404.47N,N-Dicyclohexylcarbodiimide
CAS :N,N-Dicyclohexylcarbodiimide (Dicyclohexylcarbodiimide) is a cross-linking agent used in the synthesis of active ester-containing reagents.Formule :C13H22N2Degré de pureté :98.28% - 99.73%Couleur et forme :SolidMasse moléculaire :206.335-Hydroxymethyl tolterodine formate
CAS :5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine and Fesoterodine. It is synthesized by the cytochrome P450 (CYP) isoenzyme CYP2D6 and plasma esterases.Formule :C23H33NO4Couleur et forme :SolidMasse moléculaire :387.515-AMAM-2-CP
CAS :5-AMAM-2-CP, a significant metabolite of Acetamiprid, serves as a global insecticide within the neonicotinoid class and acts as an nAChR agonist [1] [2].Formule :C9H11ClN2OCouleur et forme :SolidMasse moléculaire :198.65(Rac)-5-Carboxy tolterodine
CAS :(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.Formule :C22H29NO3Couleur et forme :SolidMasse moléculaire :355.47Thiothixene
CAS :Thiothixene has a wide range of applications in life science related research.Formule :C23H29N3O2S2Couleur et forme :SolidMasse moléculaire :443.62RuBi-Nicotine
CAS :Nicotinic receptor agonistFormule :C40H44Cl2N8RuDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :808.81M4 mAChR agonist-1
CAS :M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).Formule :C14H18N4OSDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :290.38(R)-Dinotefuran
CAS :(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.Formule :C7H14N4O3Couleur et forme :SolidMasse moléculaire :202.21NNC 11-1607
CAS :NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.Formule :C30H32N6O2S2Couleur et forme :SolidMasse moléculaire :572.74Navafenterol saccharinate
CAS :AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).Formule :C45H47N7O9S3Couleur et forme :SolidMasse moléculaire :926.09α-Conotoxin EI
CAS :Selective antagonist of neuromuscular nicotinic receptors α1β1γδFormule :C83H125N27O27S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2093.37bPiDDB
CAS :<p>bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.</p>Formule :C24H38Br2N2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :514.38DSPE-PEG5000-RVG29
DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.Couleur et forme :Odour SolidHydroxybupropion
CAS :Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formule :C13H18ClNO2Degré de pureté :99.73%Couleur et forme :Off-White SolidMasse moléculaire :255.74Ref: TM-T11588
1mg89,00€5mg204,00€10mg331,00€25mg545,00€50mg777,00€100mg1.063,00€1mL*10mM (DMSO)232,00€Epiboxidine
CAS :Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.Formule :C10H14N2OCouleur et forme :SolidMasse moléculaire :178.23Irsogladine maleate
CAS :Compound PDK0375, with CAS No. 84504-69-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0375 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C9H7Cl2N5Couleur et forme :SolidMasse moléculaire :256.09(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS :<p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>Formule :C22H32ClNO2Couleur et forme :SolidMasse moléculaire :377.95Ebiratide TFA
<p>Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.</p>Formule :C48H73N11O10S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :996.23 (free base)TC-2559 difumarate
CAS :TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.Formule :C20H26N2O9Couleur et forme :SolidMasse moléculaire :438.43Lobeline sulfate
CAS :Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.Formule :C22H29NO6SDegré de pureté :98%Couleur et forme :White PowderMasse moléculaire :435.54Mant-GTPγS
CAS :<p>Mant-GTPγS, an effective GTP analog, displays strong competitive inhibition of adenylyl cyclase (AC). Additionally, it acts as a potent inhibitor of YdeH.</p>Formule :C18H23N6O14P3SCouleur et forme :SolidMasse moléculaire :672.39trans-Cevimeline hydrochloride
CAS :AF 102A hydrochloride is a biochemical.Formule :C10H18ClNOSCouleur et forme :SolidMasse moléculaire :235.77Lu AE51090
CAS :Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.Formule :C24H29N3O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :407.51Desfesoterodine
CAS :<p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>Formule :C22H31NO2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :341.49Bensultap
CAS :Bensultap is an agricultural chemical typically used as a pesticide.Formule :C17H21NO4S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.61Aceclidine (hydrochloride)
CAS :agonist of muscarinic receptorsFormule :C9H16ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :205.68Anabaseine
CAS :Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.Formule :C10H12N2Couleur et forme :SolidMasse moléculaire :160.22G-Protein antagonist peptide
CAS :Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.Formule :C57H64N12O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1093.27Perindoprilat
CAS :Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.Formule :C17H28N2O5Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :340.41Soclenicant
CAS :Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availabilityFormule :C24H26N4O3Degré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :418.49M 8218
CAS :M 8218 is a bioactive chemical.Formule :C20H29NO2Couleur et forme :SolidMasse moléculaire :315.45Muscarine
CAS :Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.Formule :C9H20NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :174.26nAChR modulator-1
CAS :nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .Formule :C12H8ClN3O2Couleur et forme :SolidMasse moléculaire :261.66(±)-Coniine
CAS :(±)-Coniine, a piperidine alkaloid, is a toxin found in poison hemlock.Formule :C8H17NCouleur et forme :SolidMasse moléculaire :127.23Tiquizium
CAS :<p>Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.</p>Formule :C19H24NS2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :330.53N-Ethyl-N-(3-pyridylmethyl)amine
CAS :N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.Formule :C8H12N2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :136.19β2AR/M-receptor agonist-1
CAS :β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFormule :C43H56BrN3O7Couleur et forme :SolidMasse moléculaire :806.82TDI-10229
CAS :TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.Formule :C16H16ClN5Degré de pureté :99.85% - 99.89%Couleur et forme :SoildMasse moléculaire :313.78Ref: TM-T64355
1mg42,00€5mg165,00€10mg235,00€25mg432,00€50mg648,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)177,00€BTMPS
CAS :BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.Formule :C28H52N2O4Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :480.72LAS190792
CAS :LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.Formule :C39H43ClN4O9S2Couleur et forme :SolidMasse moléculaire :811.36TIP 39, Tuberoinfundibular Neuropeptide
CAS :TIP39 is a synthetic neuropeptide agonist for human and rat PTH2 receptors from the hypothalamus.Formule :C202H325N61O54SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4504.2Biperiden Hydrochloride
CAS :Biperiden HCl is an anti-Parkinson's drug, blocks M1 receptors, manages all Parkinson's types, and is FDA-approved. Non-toxic at 0.11 mg/kg to rats' cognition.Formule :C21H30ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.92nAChR agonist 2
CAS :Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,Formule :C11H16N2Couleur et forme :SolidMasse moléculaire :176.263M3/PDE4 modulator-1
M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.Formule :C38H41Cl2N3O8SCouleur et forme :SolidMasse moléculaire :770.72Emraclidine
CAS :Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.Formule :C20H21F3N4ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :390.4Ref: TM-T9694
1mg127,00€2mgÀ demander5mg305,00€10mg494,00€25mg882,00€50mg1.198,00€100mg1.586,00€1mL*10mM (DMSO)338,00€DSPE-PEG2000-RVG29
DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.Couleur et forme :Odour Solid(rel)-Asperparaline A
CAS :<p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>Formule :C20H29N3O3Couleur et forme :SolidMasse moléculaire :359.47Migrastatin
CAS :Migrastatin is a bacterial metabolite that has been found inStreptomyceswith antimuscarinic and anticancer activities.1,2It binds to M1-5muscarinicFormule :C27H39NO7Couleur et forme :SolidMasse moléculaire :489.609Bencycloquidium Bromide
CAS :Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.Formule :C21H32BrNO2Couleur et forme :SolidMasse moléculaire :410.39α-Conotoxin PIA TFA
α-Conotoxin PIA TFA, targeting nicotinic acetylcholine receptor (nAChR) subtypes with α6 and α3 subunits, acts as an antagonist.Formule :C81H126F3N27O27S4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :2095.3Bis-Br-ANT-ATP tetrasodium
Bis-Br-ANT-ATP(tetrasodium) is a fluorescent derivative of adenosine-5'-triphosphate (ATP). It selectively inhibits the adenylyl cyclase toxin CyaA of Bordetella pertussis with a Ki of 12.6 nM. This compound is utilized in research related to whooping cough.Couleur et forme :Odour SolidRivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.Formule :C10H16Cl2N2Degré de pureté :99.4%Couleur et forme :SoildMasse moléculaire :235.15Ref: TM-T12738L1
1mg35,00€5mg74,00€10mg105,00€25mg246,00€50mg444,00€100mg650,00€1mL*10mM (DMSO)116,00€VU6028418
CAS :VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).Couleur et forme :SolidProadrenomedullin (1-20), human
CAS :Endogenous peptide; agonist of MRGPRX2 (EC50=251 nM); noncompetitive inhibitor of nicotinic receptors; reduces catecholamine secretion; antihypertensive.Formule :C112H178N36O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2460.84α-Muricholic acid
CAS :α-Muricholic acid is the most abundant primary bile acid in rodents.Formule :C24H40O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.57ABT-107
CAS :ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Formule :C19H20N4OCouleur et forme :SolidMasse moléculaire :320.396NSC 23766
CAS :NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formule :C24H35N7Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :421.58Metixene hydrochloride hydrate
CAS :Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.Formule :C20H26ClNOSDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :363.95Fipexide hydrochloride
CAS :Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formule :C20H22Cl2N2O4Couleur et forme :SolidMasse moléculaire :425.31Tolterodine
CAS :Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Formule :C22H31NODegré de pureté :99.71%Couleur et forme :White Like Or Light Brown Crystalline PowderMasse moléculaire :325.49YM-58790 hydrochloride
CAS :YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Formule :C27H32ClN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :466.02Palmatine hydroxide
CAS :Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41Cevimeline
CAS :Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Formule :C10H17NOSCouleur et forme :Off-White SolidMasse moléculaire :199.31
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