AChR
Les inhibiteurs des récepteurs de l'acétylcholine (AChR) sont des composés qui bloquent l'activité des récepteurs de l'acétylcholine, essentiels pour la neurotransmission dans les systèmes nerveux central et périphérique. Les AChR jouent un rôle crucial dans la contraction musculaire, la mémoire et les fonctions cognitives. Les inhibiteurs des AChR sont utilisés pour étudier des conditions telles que la myasthénie grave, la maladie d'Alzheimer et d'autres troubles neurologiques. En modulant l'activité des AChR, ces inhibiteurs peuvent aider à démêler les complexités de la signalisation cholinergique dans le cerveau. Chez CymitQuimica, nous fournissons une gamme d'inhibiteurs des AChR pour soutenir vos recherches en neurosciences, pharmacologie et maladies neurodégénératives.
623 produits trouvés pour "AChR"
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YM-58790 hydrochloride
CAS :YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Formule :C27H32ClN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :466.02Palmatine hydroxide
CAS :Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41β2AR/M-receptor agonist-2
CAS :<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formule :C36H49ClN4O7SCouleur et forme :SolidMasse moléculaire :717.31Dexetimide
CAS :Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Formule :C23H26N2O2Couleur et forme :SolidMasse moléculaire :362.46Varenicline Hydrochloride
CAS :Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Formule :C13H14ClN3Degré de pureté :99.854%Couleur et forme :SolidMasse moléculaire :247.72Ref: TM-T23502
1mg38,00€5mg80,00€10mg105,00€25mg192,00€50mg297,00€100mg441,00€200mg646,00€1mL*10mM (DMSO)88,00€Glycerophosphoinositol choline
CAS :Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Formule :C14H32NO12PCouleur et forme :SolidMasse moléculaire :437.38Cevimeline hydrochloride
CAS :Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.Formule :C10H18ClOSCouleur et forme :SolidMasse moléculaire :235.77(±)-Darifenacin
CAS :(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.Formule :C28H30N2O2Couleur et forme :SolidMasse moléculaire :426.55VU0467485
CAS :VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.Formule :C17H17FN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.41Clorprenaline
CAS :Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formule :C11H16ClNODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :213.7SSR180711 hydrochloride
CAS :SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formule :C14H18BrClN2O2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :361.66Pirmenol hydrochloride
CAS :Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μMFormule :C22H31ClN2OCouleur et forme :SolidMasse moléculaire :374.95Tebanicline dihydrochloride
CAS :Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.Formule :C9H13Cl3N2OCouleur et forme :SolidMasse moléculaire :271.57Biperiden
CAS :Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.Formule :C21H29NODegré de pureté :99.65%Couleur et forme :Crystals SolidMasse moléculaire :311.46Ispronicline
CAS :Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitiveFormule :C14H22N2ODegré de pureté :97.70% - 99.16%Couleur et forme :SolidMasse moléculaire :234.34(S)-(+)-Dimethindene maleate
CAS :(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormule :C24H28N2O4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :408.49Sabcomeline hydrochloride
CAS :Sabcomeline is a selective M1 receptor partial agonist.Formule :C10H16ClN3OCouleur et forme :SolidMasse moléculaire :229.71NS3861 fumarate
CAS :NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.Formule :C16H18BrNO4SCouleur et forme :SolidMasse moléculaire :400.29NKH477
CAS :NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Formule :C27H44ClNO8Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :546.09ABT-107
CAS :ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Formule :C19H20N4OCouleur et forme :SolidMasse moléculaire :320.396NSC 23766
CAS :NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formule :C24H35N7Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :421.58DL-Cystine
CAS :DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .Formule :C6H12N2O4S2Couleur et forme :SolidMasse moléculaire :240.3NBTGR
CAS :NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).Formule :C17H18N6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.43Piperidolate hydrochloride
CAS :Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Formule :C21H26ClNO2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :359.89Succinylcholine Chloride Dihydrate
CAS :<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Formule :C14H30N2O4·2Cl·2H2ODegré de pureté :99.87%Couleur et forme :White SolidMasse moléculaire :397.34Tebanicline hydrochloride
CAS :Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Formule :C9H12Cl2N2ODegré de pureté :91.74% - 98.78%Couleur et forme :SolidMasse moléculaire :235.11VU0357017 hydrochloride
CAS :VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formule :C18H28ClN3O3Degré de pureté :99% - 99.97%Couleur et forme :SolidMasse moléculaire :369.89α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formule :C69H107N23O24S4Degré de pureté :94.82% - 97.79%Couleur et forme :SolidMasse moléculaire :1770.99VU0119498
CAS :VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formule :C15H10BrNO2Degré de pureté :97.56%Couleur et forme :SolidMasse moléculaire :316.15Clothianidin
CAS :Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Formule :C6H8ClN5O2SDegré de pureté :99.71% - 99.87%Couleur et forme :Solid PowderMasse moléculaire :249.68VU0152100
CAS :<p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>Formule :C18H19N3O2SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :341.43Nitrobenzylthioinosine
CAS :<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41KH7
CAS :KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formule :C17H15BrN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :419.3VU0467154
CAS :VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Formule :C17H15F3N4O3S2Degré de pureté :99.51% - 99.53%Couleur et forme :SolidMasse moléculaire :444.45Ref: TM-T17244
1mg49,00€2mg66,00€5mg97,00€10mg133,00€25mg250,00€50mg423,00€100mg735,00€200mg998,00€1mL*10mM (DMSO)106,00€NS9283
CAS :<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Formule :C14H8N4ODegré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :248.24ML380
CAS :<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Formule :C23H25F3N4O3SDegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :494.53Varenicline Tartrate
CAS :<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Formule :C13H13N3·C4H6O6Degré de pureté :98.23% - 98.32%Couleur et forme :Tan SolidMasse moléculaire :361.35Cyclodrine hydrochloride
CAS :Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFormule :C19H30ClNO3Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :355.9Isopropamide Iodide
CAS :<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Formule :C23H33IN2ODegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :480.43Mc-Val-Ala-PAB
CAS :<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Formule :C25H34N4O6Degré de pureté :98.34% - 99.24%Couleur et forme :SolidMasse moléculaire :486.56Nitenpyram
CAS :Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.Formule :C11H15ClN4O2Degré de pureté :99.03%Couleur et forme :Light-Yellow CrystalMasse moléculaire :270.72Mecamylamine hydrochloride
CAS :Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formule :C11H22ClNDegré de pureté :99.76% - >99.99%Couleur et forme :White SolidMasse moléculaire :203.75Solifenacin hydrochloride
CAS :Solifenacin Hcl is a muscarinic receptor antagonist.Formule :C23H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.93JHU37152
CAS :JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Formule :C19H20ClFN4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :358.84Encenicline
CAS :Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formule :C16H17ClN2OSDegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :320.84Ref: TM-T7193
1mg73,00€5mg140,00€10mg220,00€25mg369,00€50mg523,00€100mg712,00€200mg938,00€1mL*10mM (DMSO)153,00€Syn-Ake acetate
CAS :Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formule :C19H29N5O3·2(C2H4O2)Degré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :495.58Sofpironium bromide
CAS :Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formule :C22H32BrNO5Degré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :470.4Ref: TM-T28827
1mg74,00€5mg160,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€1mL*10mM (DMSO)165,00€Mecamylamine
CAS :Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formule :C11H21NCouleur et forme :SolidMasse moléculaire :167.29Oxyphencyclimine Hydrochloride
CAS :Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Formule :C20H29ClN2O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :380.91Pempidine
CAS :Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formule :C10H21NDegré de pureté :98.18% - 99.28%Couleur et forme :Colorless - Light Yellow Clear LiquidMasse moléculaire :155.28Propiverine
CAS :Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Formule :C23H29NO3Couleur et forme :SolidMasse moléculaire :367.48NS 1738
CAS :NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formule :C14H9Cl2F3N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :365.13Dinotefuran
CAS :Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formule :C7H14N4O3Degré de pureté :99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :202.21Procyclidine hydrochloride
CAS :Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.Formule :C19H30ClNODegré de pureté :99.24% - 99.88%Couleur et forme :Crystals From Petroleum Ether White PowderMasse moléculaire :323.9Dronedarone
CAS :Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formule :C31H44N2O5SDegré de pureté :98.85% - 99.99%Couleur et forme :SolidMasse moléculaire :556.76EB-3D
CAS :EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Formule :C30H36Br2N4O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :644.4Ref: TM-T7955
1mg92,00€2mg120,00€5mg187,00€10mg274,00€25mg472,00€50mg655,00€100mg924,00€200mg1.225,00€1mL*10mM (DMSO)278,00€Oxyphenonium bromide
CAS :<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Formule :C21H34BrNO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :428.404MC-Val-Cit-PABC-PNP
CAS :MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.Formule :C35H43N7O11Degré de pureté :97.2% - 98.055%Couleur et forme :SolidMasse moléculaire :737.76Propantheline
CAS :Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Formule :C23H30NO3Couleur et forme :SolidMasse moléculaire :368.49Bestim
CAS :Bestim is an immunomodulatory dipeptide that is synthetic.Formule :C16H19N3O5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :333.34Ref: TM-T25146
1mg88,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)182,00€VU0152099
CAS :VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formule :C18H17N3O3SDegré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :355.41Adiphenine
CAS :Adiphenine is an inhibitor of nicotinic receptors.Formule :C20H25NO2Couleur et forme :SolidMasse moléculaire :311.42Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Formule :C12H16N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :207.23Simufilam dihydrochloride
CAS :Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Formule :C15H23Cl2N3ODegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :332.3Ref: TM-T9172
1mg52,00€5mg90,00€10mg143,00€25mg294,00€50mg380,00€100mg497,00€200mg655,00€1mL*10mM (DMSO)101,00€Batefenterol
CAS :Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Formule :C40H42ClN5O7Degré de pureté :97.94% - 98.4%Couleur et forme :SolidMasse moléculaire :740.24suvn-911
CAS :suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Formule :C11H14Cl2N2ODegré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :261.15Ref: TM-T9787
1mg71,00€5mg140,00€10mg215,00€25mg359,00€50mg510,00€100mg695,00€200mg937,00€1mL*10mM (DMSO)182,00€Coluracetam
CAS :Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Formule :C19H23N3O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :341.4Aclidinium bromide
CAS :<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Formule :C26H30NO4S2·BrDegré de pureté :99.53% - 99.69%Couleur et forme :SolidMasse moléculaire :564.55Encenicline hydrochloride
CAS :Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formule :C16H17ClN2OS·HClDegré de pureté :98.34% - 99.85%Couleur et forme :SolidMasse moléculaire :357.3Pempidine HCl
CAS :Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formule :C10H22ClNCouleur et forme :SolidMasse moléculaire :191.74Umeclidinium bromide
CAS :Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Formule :C29H34BrNO2Degré de pureté :98.4% - 99.89%Couleur et forme :SolidMasse moléculaire :508.49Ref: TM-T4997
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg212,00€50mg350,00€100mg525,00€1mL*10mM (DMSO)87,00€PHA 568487 free base
CAS :<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Formule :C16H20N2O3Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :288.34Batefenterol Succinate
CAS :Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formule :C44H48ClN5O11Couleur et forme :SolidMasse moléculaire :858.34VU0238441
CAS :VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formule :C16H9ClF3NO2Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :339.7Benzetimide hydrochloride
CAS :Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Formule :C23H27ClN2O2Degré de pureté :99.32%Couleur et forme :Off-White PowderMasse moléculaire :398.93Oxyphencyclimine
CAS :Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Formule :C20H28N2O3Couleur et forme :SolidMasse moléculaire :344.45(S)-UFR2709
CAS :(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Formule :C13H17NO2Couleur et forme :SolidMasse moléculaire :219.284mAChR-IN-1 hydrochloride
CAS :mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formule :C23H26ClIN2O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :524.82Ref: TM-T5655
1mg40,00€5mg90,00€10mg133,00€25mg227,00€50mg314,00€100mg393,00€200mg520,00€1mL*10mM (DMSO)95,00€Solifenacin
CAS :Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formule :C23H26N2O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :362.46LY2119620
CAS :LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Formule :C19H24ClN5O3SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :437.94Pirmenol
CAS :Pirmenol is a new antiarrhythmic drugFormule :C22H30N2ODegré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :338.49Anisotropine Methylbromide
CAS :Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formule :C17H32BrNO2Degré de pureté :99.73%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :362.35Darifenacin
CAS :Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formule :C28H30N2O2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :426.55Ref: TM-T62320
2mg42,00€5mg62,00€10mg87,00€25mg160,00€50mg250,00€100mg376,00€200mg550,00€1mL*10mM (DMSO)67,00€Ilmetropium iodide
CAS :Ilmetropium iodide is a bronchodilator.Formule :C20H30INO3Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :459.36BNC210
CAS :BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.Formule :C17H23N3O3Degré de pureté :97.05% - >99.99%Couleur et forme :SolidMasse moléculaire :317.38Brompheniramine
CAS :Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formule :C16H19BrN2Couleur et forme :SolidMasse moléculaire :319.24Harman hydrochloride
CAS :Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Formule :C12H11ClN2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :218.68Ursulcholic acid
CAS :Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Formule :C24H40O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.7Nor-benzetimide
CAS :Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formule :C16H20N2O2Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :272.34Ref: TM-T22380
1mg72,00€5mg136,00€10mg197,00€25mg324,00€50mg452,00€100mg607,00€200mg810,00€1mL*10mM (DMSO)135,00€Nitrocaramiphen hydrochloride
CAS :Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formule :C18H27ClN2O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :370.87W-84 dibromide
CAS :<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Formule :C32H44Br2N4O4Degré de pureté :95.56%Couleur et forme :SolidMasse moléculaire :708.52PSEM 89S TFA
CAS :<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Formule :C18H23F3N2O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.38CCMI
CAS :CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Formule :C19H15Cl2N3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :388.25Glycopyrrolate
CAS :Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formule :C19H28BrNO3Degré de pureté :99.41% - 99.64%Couleur et forme :SolidMasse moléculaire :398.33SEN12333
CAS :SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonistFormule :C20H25N3O2Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :339.43Ref: TM-T23348
2mg39,00€5mg57,00€10mg95,00€25mg167,00€50mg269,00€100mg432,00€200mg622,00€1mL*10mM (DMSO)63,00€9-Ethyladenine
CAS :9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formule :C7H9N5Degré de pureté :99.35% - 99.37%Couleur et forme :SolidMasse moléculaire :163.18BQCA
CAS :<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Formule :C18H15NO4Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :309.32PNU-282987 S enantiomer free base
CAS :PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Formule :C14H17ClN2ODegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :264.75Ref: TM-T7695
1mg74,00€5mg170,00€10mg230,00€25mg356,00€50mg487,00€100mg658,00€200mg884,00€1mL*10mM (DMSO)190,00€4BP-TQS
CAS :4BP-TQS is an allosteric agonist of α7 nAChRs.Formule :C18H17BrN2O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :405.31TBPB
CAS :<p>TBPB is an allosteric M1 mAChR agonist.</p>Formule :C25H32N4ODegré de pureté :97.87% - 99.9%Couleur et forme :SolidMasse moléculaire :404.55
