AChR
Les inhibiteurs des récepteurs de l'acétylcholine (AChR) sont des composés qui bloquent l'activité des récepteurs de l'acétylcholine, essentiels pour la neurotransmission dans les systèmes nerveux central et périphérique. Les AChR jouent un rôle crucial dans la contraction musculaire, la mémoire et les fonctions cognitives. Les inhibiteurs des AChR sont utilisés pour étudier des conditions telles que la myasthénie grave, la maladie d'Alzheimer et d'autres troubles neurologiques. En modulant l'activité des AChR, ces inhibiteurs peuvent aider à démêler les complexités de la signalisation cholinergique dans le cerveau. Chez CymitQuimica, nous fournissons une gamme d'inhibiteurs des AChR pour soutenir vos recherches en neurosciences, pharmacologie et maladies neurodégénératives.
575 produits trouvés pour "AChR"
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Orphenadrine Citrate
CAS :<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Formule :C18H23NO·C6H8O7Degré de pureté :98% - 99.58%Couleur et forme :White SolidMasse moléculaire :461.5Ipratropium bromide monohydrate
CAS :<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Formule :C20H32BrNO4Degré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :430.38Gallamine triethiodide
CAS :<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Formule :C30H60I3N3O3Degré de pureté :98.90%Couleur et forme :White Amorphous Powder SolidMasse moléculaire :891.53Nicardipine hydrochloride
CAS :<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formule :C26H30ClN3O6Degré de pureté :99.58% - 99.89%Couleur et forme :Yellow SolidMasse moléculaire :515.99Bambuterol hydrochloride
CAS :<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formule :C18H30ClN3O5Degré de pureté :99.53% - 99.61%Couleur et forme :White SolidMasse moléculaire :403.91Droperidol
CAS :<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formule :C22H22FN3O2Degré de pureté :97.16% - 98%Couleur et forme :SolidMasse moléculaire :379.43DL-trihexyphenidyl hydrochloride
CAS :<p>DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.</p>Formule :C20H32ClNODegré de pureté :99.63% - 99.71%Couleur et forme :SolidMasse moléculaire :337.93Dicyclomine hydrochloride
CAS :<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Formule :C19H36ClNO2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :345.95Nebracetam hydrochloride
CAS :<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Formule :C12H17ClN2ODegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :240.729MK-7622
CAS :<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formule :C25H25N3O2Degré de pureté :99.77% - 99.8%Couleur et forme :SolidMasse moléculaire :399.48Homatropine Methylbromide
CAS :<p>Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.</p>Formule :C17H24BrNO3Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :370.29Acetamiprid
CAS :<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Formule :C10H11ClN4Degré de pureté :99.66%Couleur et forme :White PowderMasse moléculaire :222.67Temephos
CAS :<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Formule :C16H20O6P2S3Degré de pureté :≥95%Couleur et forme :White Crystalline Solid Or LiquidMasse moléculaire :466.47Benztropine mesylate
CAS :<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Methscopolamine
CAS :<p>Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.</p>Formule :C18H24BrNO4Degré de pureté :99.12% - ≥98%Couleur et forme :SolidMasse moléculaire :398.29Valethamate bromide
CAS :<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Formule :C19H32BrNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :386.37Carbetapentane citrate
CAS :<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Formule :C20H31NO3·C6H8O7Degré de pureté :99.46%Couleur et forme :White To Off-White SolidMasse moléculaire :525.59Diphenmanil methylsulfate
CAS :<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Formule :C20H24N·CH3O4SDegré de pureté :98% - 99.27%Couleur et forme :SolidMasse moléculaire :389.51Nefiracetam
CAS :<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formule :C14H18N2O2Degré de pureté :97.37%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :246.3Procainamide hydrochloride
CAS :<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Formule :C13H21N3O·HClDegré de pureté :99.83% - 99.97%Couleur et forme :White To Slightly Yellow PowderMasse moléculaire :271.79Trospium chloride
CAS :<p>Trospium chloride treats urinary incontinence without causing liver damage.</p>Formule :C25H30ClNO3Degré de pureté :99.84% - >99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :427.964Neostigmine methyl sulfate
CAS :<p>Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.</p>Formule :C13H22N2O6SDegré de pureté :99.34% - 99.53%Couleur et forme :Crystalline SolidMasse moléculaire :334.39Dipivefrin hydrochloride
CAS :<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formule :C19H27NO5·HClDegré de pureté :99.22% - 99.92%Couleur et forme :Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMasse moléculaire :387.9Methacholine Chloride
CAS :<p>Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of acetylcholine.</p>Formule :C8H18ClNO2Degré de pureté :99.37% - 99.74%Couleur et forme :White Hygroscopic Crystals With Slight Odor Of Dead FishMasse moléculaire :195.69PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formule :C36H51Cl3N4O7SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :790.24Adiphenine hydrochloride
CAS :<p>Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.</p>Formule :C20H25NO2·HClDegré de pureté :97.76% - 99.53%Couleur et forme :White Or Almost White PowderMasse moléculaire :347.88Benzethonium chloride
CAS :<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Formule :C27H42ClNO2Degré de pureté :99.91%Couleur et forme :White To Off-White Solid Solid Particulate/PowderMasse moléculaire :448.09VU 0365114
CAS :<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Formule :C22H14F3NO3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :397.35Rivastigmine tartrate
CAS :<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Formule :C14H22N2O2·C4H6O6Degré de pureté :98% - 99.66%Couleur et forme :White To Off-White PowderMasse moléculaire :400.43Zelminemab
CAS :<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Degré de pureté :98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Couleur et forme :LiquidPyrantel tartrate
CAS :<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Formule :C15H20N2O6SDegré de pureté :99.96%Couleur et forme :White CrystalsMasse moléculaire :356.39Pirenzepine dihydrochloride
CAS :<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Formule :C19H21N5O2·2HClDegré de pureté :99.48% - 99.62%Couleur et forme :White PowderMasse moléculaire :424.32Promethazine hydrochloride
CAS :<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.88Bethanechol chloride
CAS :<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Formule :C7H17N2O2·ClDegré de pureté :95% - 99.73%Couleur et forme :White CrystallineMasse moléculaire :196.68Deschloroclozapine
CAS :<p>Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.</p>Formule :C18H20N4Degré de pureté :99.61% - 99.98%Couleur et forme :SolidMasse moléculaire :292.38Lysipressin acetate(50-57-7(fb_acetate))
CAS :<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formule :C48H69N13O14S2Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1116.28Fesoterodine fumarate
CAS :<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Formule :C26H37NO3·C4H4O4Degré de pureté :99.16%Couleur et forme :White SolidMasse moléculaire :527.65Vecuronium bromide
CAS :<p>Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle</p>Formule :C34H57BrN2O4Degré de pureté :99.63% - 99.92%Couleur et forme :White PowderMasse moléculaire :637.73Pancuronium dibromide
CAS :<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Formule :C35H60Br2N2O4Degré de pureté :99.86%Couleur et forme :solidMasse moléculaire :732.67Rocuronium bromide
CAS :<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Formule :C32H53BrN2O4Degré de pureté :99.77% - >99.99%Couleur et forme :White Or Off-White PowderMasse moléculaire :609.68TAK-071
CAS :<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Formule :C24H24FN3O3Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :421.46nAChR agonist 1
CAS :<p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>Formule :C20H18ClNO3S2Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :419.94Pyrantel pamoate
CAS :<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Formule :C34H30N2O6SDegré de pureté :99.71%Masse moléculaire :594.699-Cyclopentyladenine
CAS :<p>9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signaling</p>Formule :C10H13N5Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :203.24Clidinium bromide
CAS :<p>Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.</p>Formule :C22H26BrNO3Degré de pureté :98.89% - 99.86%Couleur et forme :White Crystalline SolidMasse moléculaire :432.35Hexamethonium Bromide
CAS :<p>Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.</p>Formule :C12H30Br2N2Degré de pureté :99.76%Couleur et forme :White Crystalline Powder And AgglomeratesMasse moléculaire :362.19Oxybutynin
CAS :<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Formule :C22H31NO3Degré de pureté :97.81% - 99.57%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :357.49Benactyzine hydrochloride
CAS :<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Formule :C20H26ClNO3Degré de pureté :99.03% - 99.94%Couleur et forme :SolidMasse moléculaire :363.88Flavoxate hydrochloride
CAS :<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formule :C24H26ClNO4Degré de pureté :99.78%Couleur et forme :White SolidMasse moléculaire :427.922',5'-Dideoxyadenosine
CAS :<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Formule :C10H13N5O2Degré de pureté :99.55%Couleur et forme :White SolidMasse moléculaire :235.24Fipexide
CAS :<p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>Formule :C20H21ClN2O4Degré de pureté :97.6% - 99.95%Couleur et forme :SolidMasse moléculaire :388.84(Rac)-ABT-202 dihydrochloride
CAS :<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Formule :C9H15Cl2N3Degré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :236.142Carbachol
CAS :<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Formule :C6H15ClN2O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :182.65Tolterodine tartrate
CAS :<p>Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.</p>Formule :C22H31NO·C4H6O6Degré de pureté :99.95%Couleur et forme :White-To-Off-White Crystalline PowderMasse moléculaire :475.58Propantheline bromide
CAS :<p>Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscle</p>Formule :C23H30BrNO3Degré de pureté :98% - ≥98%Masse moléculaire :448.4Primidone
CAS :<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Formule :C12H14N2O2Degré de pureté :99.91%Couleur et forme :Crystals (Ntp 1992)Masse moléculaire :218.25Dequalinium chloride
CAS :<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Formule :C30H40Cl2N4Degré de pureté :99.79% - 99.9%Couleur et forme :SolidMasse moléculaire :527.59Solifenacin succinate
CAS :<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Formule :C23H26N2O2·C4H6O4Degré de pureté :99.85% - 99.98%Couleur et forme :SolidMasse moléculaire :480.56Darifenacin hydrobromide
CAS :<p>Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.</p>Formule :C28H31BrN2O2Degré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :505.45SSR 180
CAS :<p>SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.</p>Formule :C14H17BrN2O2Degré de pureté :98.82%Couleur et forme :SoildMasse moléculaire :325.20Atropine methyl bromide
CAS :<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Formule :C18H26BrNO3Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :384.308Tazomeline
CAS :<p>Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.</p>Formule :C14H23N3S2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :297.48V-11-0711 HCl
<p>V-11-0711 HCl is a selective and highly effective choline kinase α (ChoKα) inhibitor that inhibits the catalytic activity of Chk.</p>Formule :C27H36ClNO3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :458.03(Rac)-Sabcomeline HCl
CAS :<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Formule :C10H16ClN3ODegré de pureté :99.58%Couleur et forme :SoildMasse moléculaire :229.71Cotinine
CAS :<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Formule :C10H12N2ODegré de pureté :98% - 99.89%Couleur et forme :Viscous Oil SolidMasse moléculaire :176.22Ribavirin
CAS :<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Formule :C8H12N4O5Degré de pureté :99.09% - 99.83%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.20Tiotropium bromide
CAS :<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Formule :C19H22BrNO4S2Degré de pureté :96.82% - 99.97%Couleur et forme :White SolidMasse moléculaire :472.42DSPE-PEG1000-RVG29
<p>DSPE-PEG1000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 can specifically bind to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and cross the BBB.</p>Couleur et forme :Odour SolidMK-0969
CAS :<p>MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Formule :C24H30F2N4O2Couleur et forme :SolidMasse moléculaire :444.52nAChR modulator-2
CAS :<p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formule :C12H8ClN3O2Couleur et forme :SolidMasse moléculaire :261.66α-Muricholic acid
CAS :<p>α-Muricholic acid is the most abundant primary bile acid in rodents.</p>Formule :C24H40O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.57α-Conotoxin EI
CAS :<p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>Formule :C83H125N27O27S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2093.37Octamylamine
CAS :<p>Octamylamine is a bioactive chemical.</p>Formule :C13H29NCouleur et forme :SolidMasse moléculaire :199.3761Bencycloquidium Bromide
CAS :<p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>Formule :C21H32BrNO2Couleur et forme :SolidMasse moléculaire :410.39nAChR agonist CMPI hydrochloride
CAS :<p>CMPI hydrochloride: Potent α4:α4 nAChR PAM; EC50 0.26 μM for (α4)3(β2)2 response to ACh; may aid nicotine dependence, neuropsychiatric research.</p>Formule :C18H20Cl2N4OCouleur et forme :SolidMasse moléculaire :379.29(S)-Dinotefuran
CAS :<p>(S)-Dinotefuran, a neonicotinoid, more toxic to bees than its R-isomer, targets α8 nAChR.</p>Formule :C7H14N4O3Couleur et forme :SolidMasse moléculaire :202.21Angiopeptin TFA
CAS :Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formule :C58H73F6N11O14S2Couleur et forme :SolidMasse moléculaire :1326.39[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS :<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Formule :C82H120N20O25Couleur et forme :SolidMasse moléculaire :1785.95LtIA-F
<p>LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.</p>Formule :C86H121N25O22S4Couleur et forme :SolidMasse moléculaire :1985.31α-Conotoxin PIA TFA
<p>α-Conotoxin PIA TFA, targeting nicotinic acetylcholine receptor (nAChR) subtypes with α6 and α3 subunits, acts as an antagonist.</p>Formule :C81H126F3N27O27S4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :2095.3Muscarinic toxin 3
CAS :<p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>Formule :C319H489N89O97S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7379.35DSPE-PEG5000-RVG29
<p>DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.</p>Couleur et forme :Odour Solid(-)-Coclaurine hydrochloride
CAS :<p>(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.</p>Formule :C17H20ClNO3Degré de pureté :99.07%Couleur et forme :SoildMasse moléculaire :321.8Perlapine
CAS :<p>Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM).</p>Formule :C19H21N3Couleur et forme :SolidMasse moléculaire :291.39Atracurium
CAS :<p>Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.</p>Formule :C53H72N2O122Couleur et forme :SolidMasse moléculaire :929.14Anagyrine hydrochloride
CAS :<p>Anagyrine hydrochloride, a quinolizidine from Lupinus albus, targets muscarinic/nicotinic receptors; IC50: 132/2096 µM. It desensitizes nAChR directly.</p>Formule :C15H21ClN2OCouleur et forme :SolidMasse moléculaire :280.798-Aminoadenine
CAS :<p>8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.</p>Formule :C5H6N6Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :150.14rac-Desethyl Oxybutynin (hydrochloride)
CAS :<p>rac-Desethyl oxybutynin, active oxybutynin metabolite, binds to mAChRs; K_i values 3.12-16 nM; lowers rat micturition pressure.</p>Formule :C20H28ClNO3Couleur et forme :SolidMasse moléculaire :365.89TMPH
CAS :<p>TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.</p>Formule :C16H31NO2Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :269.42Guanylyl Imidodiphosphate (lithium salt)
CAS :<p>Guanylyl Imidodiphosphate (lithium salt) is a non-hydrolyzable GTP analog that increases adenylate cyclase activity.</p>Formule :C10H13Li4N6O13P3Couleur et forme :SolidMasse moléculaire :545.93Doxacurium Chloride
CAS :<p>Doxacurium Chloride is a muscarinic acetylcholine receptor M2 antagonist.</p>Formule :C56H78ClN2O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1070.69Epiboxidine hydrochloride
CAS :<p>Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.</p>Formule :C10H15ClN2OCouleur et forme :SolidMasse moléculaire :214.69VU6028418
CAS :<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Couleur et forme :SolidPF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Formule :C36H50Cl2N4O7SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :753.78R-(+)-Cotinine
CAS :<p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>Formule :C10H12N2OCouleur et forme :SolidMasse moléculaire :176.22Cisatracurium besylate
CAS :<p>Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.</p>Formule :C53H72N2O12·2C6H5O3SDegré de pureté :97.89% - 99.85%Couleur et forme :White Or White Powder CategoryMasse moléculaire :1243.48Cyclodrine
CAS :<p>Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.</p>Formule :C19H29NO3Degré de pureté :97.62%Couleur et forme :SoildMasse moléculaire :319.44Angiopeptin
CAS :<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Formule :C54H71N11O10S2Couleur et forme :SolidMasse moléculaire :1098.34Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Formule :C20H18O6Couleur et forme :SolidMasse moléculaire :354.358α-Bungarotoxin
CAS :<p>Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).</p>Formule :C338H529N97O105S11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7984.14Cevimeline hydrochloride hemihydrate
CAS :<p>Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.</p>Formule :C20H38Cl2N2O3S2Degré de pureté :97.00%Couleur et forme :SolidMasse moléculaire :489.55AC1-IN-1
CAS :<p>AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).</p>Formule :C18H18FN5O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :355.37ANQ-9040
CAS :<p>ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.</p>Formule :C36H58N2O5SCouleur et forme :SolidMasse moléculaire :630.92Biperiden Hydrochloride
CAS :<p>Biperiden HCl is an anti-Parkinson's drug, blocks M1 receptors, manages all Parkinson's types, and is FDA-approved. Non-toxic at 0.11 mg/kg to rats' cognition.</p>Formule :C21H30ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.92nAChR agonist 2
CAS :<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Formule :C11H16N2Couleur et forme :SolidMasse moléculaire :176.263Emraclidine
CAS :<p>Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.</p>Formule :C20H21F3N4ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :390.4TIP 39, Tuberoinfundibular Neuropeptide
CAS :<p>TIP39 is a synthetic neuropeptide agonist for human and rat PTH2 receptors from the hypothalamus.</p>Formule :C202H325N61O54SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4504.2Lupanine hydrochloride
CAS :<p>Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.</p>Formule :C15H25ClN2OCouleur et forme :SolidMasse moléculaire :284.83Pozanicline hydrochloride
<p>Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.</p>Formule :C11H17ClN2ODegré de pureté :97.13% - 99.81%Couleur et forme :SolidMasse moléculaire :228.72PDE4-IN-4
CAS :<p>PDE4-IN-4 is a compound acting as both a potent M3 antagonist (p IC 50 = 10.2) and a PDE4 inhibitor (p IC 50 = 8.8), designed for inhalation-based treatment of</p>Formule :C36H37Cl2N3O7SCouleur et forme :SolidMasse moléculaire :726.67Methylatropine (nitrate)
CAS :<p>Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>Formule :C18H26N2O6Couleur et forme :SolidMasse moléculaire :366.414nAChR modulator-1
CAS :<p>nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formule :C12H8ClN3O2Couleur et forme :SolidMasse moléculaire :261.66Heliosupine N-oxide
<p>Heliosupine N-oxide is a useful organic compound for research related to life sciences and the catalog number is T125058.</p>Formule :C20H31NO8Couleur et forme :SolidMasse moléculaire :413.467Small Cardioactive Peptide B (SCPB)
CAS :<p>SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).</p>Formule :C52H80N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1141.41Epiboxidine
CAS :<p>Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.</p>Formule :C10H14N2OCouleur et forme :SolidMasse moléculaire :178.23M 8218
CAS :<p>M 8218 is a bioactive chemical.</p>Formule :C20H29NO2Couleur et forme :SolidMasse moléculaire :315.45Desfesoterodine
CAS :<p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>Formule :C22H31NO2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :341.49α-Conotoxin AuIB
CAS :<p>Selective antagonist of α3β4 nicotinic acetylcholine receptors.</p>Formule :C65H89N17O21S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1572.76Flupyradifurone
CAS :<p>Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.</p>Formule :C12H11ClF2N2O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.68α-Conotoxin imi
CAS :<p>alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.</p>Formule :C52H78N20O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1351.56Tiquizium
CAS :<p>Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.</p>Formule :C19H24NS2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :330.53CVN417
<p>CVN417 is an orally active antagonist of nAChR containing the α6 subunit, modulating phasic dopaminergic neurotransmission in an impulse-dependent fashion.</p>Couleur et forme :Odour SolidPerindoprilat
CAS :<p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>Formule :C17H28N2O5Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :340.41Dicloromezotiaz
CAS :<p>Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.</p>Formule :C19H12Cl3N3O2SCouleur et forme :SolidMasse moléculaire :452.74[D-Trp7,9,10]-Substance P
CAS :<p>Substance P analog that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.</p>Formule :C79H105N21O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1588.89SIB 1553A
CAS :<p>SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.</p>Formule :C13H19NOSDegré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :237.36(+)-Coclaurine hydrochloride
CAS :<p>(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.</p>Formule :C17H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.8Destomycin A
CAS :<p>Destomycin A, an aminoglycoside antibiotic, exhibits activity against bacterial (Gram-positive and Gram-negative), antifungal, and anthelmintic agents. It inhibits peptide synthesis in Escherichia coli cells and stimulates adenylate cyclase in animal tissues.</p>Formule :C20H37N3O13Couleur et forme :SolidMasse moléculaire :527.52CDD0102 HCl
CAS :<p>CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.</p>Formule :C8H13ClN4ODegré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :216.67Mant-GTPγS
CAS :<p>Mant-GTPγS, an effective GTP analog, displays strong competitive inhibition of adenylyl cyclase (AC). Additionally, it acts as a potent inhibitor of YdeH.</p>Formule :C18H23N6O14P3SCouleur et forme :SolidMasse moléculaire :672.39Navafenterol saccharinate
CAS :<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Formule :C45H47N7O9S3Couleur et forme :SolidMasse moléculaire :926.09Thiothixene
CAS :<p>Thiothixene has a wide range of applications in life science related research.</p>Formule :C23H29N3O2S2Couleur et forme :SolidMasse moléculaire :443.62Fentonium bromide
CAS :<p>Fentonium bromide is a biochemical.</p>Formule :C31H34BrNO4Couleur et forme :SolidMasse moléculaire :564.51(S)-UFR2709 hydrochloride
CAS :<p>(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in rats, studies nicotine addiction.</p>Formule :C13H18ClNO2Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :255.74PF-06827443
<p>PF-06827443 is a orally bioavailable, CNS-penetrant M1-selective PAM with minimal agonist activity.</p>Formule :C24H24N2O4Couleur et forme :SolidMasse moléculaire :404.475-Hydroxymethyl tolterodine formate
CAS :<p>5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine and Fesoterodine. It is synthesized by the cytochrome P450 (CYP) isoenzyme CYP2D6 and plasma esterases.</p>Formule :C23H33NO4Couleur et forme :SolidMasse moléculaire :387.51(Rac)-5-Carboxy tolterodine
CAS :<p>(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.</p>Formule :C22H29NO3Couleur et forme :SolidMasse moléculaire :355.47RuBi-Nicotine
CAS :<p>Nicotinic receptor agonist</p>Formule :C40H44Cl2N8RuDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :808.81(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS :<p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>Formule :C22H32ClNO2Couleur et forme :SolidMasse moléculaire :377.95NNC 11-1607
CAS :<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Formule :C30H32N6O2S2Couleur et forme :SolidMasse moléculaire :572.74N,N-Dicyclohexylcarbodiimide
CAS :<p>N,N-Dicyclohexylcarbodiimide (Dicyclohexylcarbodiimide) is a cross-linking agent used in the synthesis of active ester-containing reagents.</p>Formule :C13H22N2Degré de pureté :98.28% - 99.73%Couleur et forme :SolidMasse moléculaire :206.33bPiDDB
CAS :<p>bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.</p>Formule :C24H38Br2N2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :514.38TC-2216
CAS :<p>TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.</p>Formule :C12H17N3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :203.28Irsogladine maleate
CAS :<p>Compound PDK0375, with CAS No. 84504-69-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0375 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C9H7Cl2N5Couleur et forme :SolidMasse moléculaire :256.09trans-Cevimeline hydrochloride
CAS :<p>AF 102A hydrochloride is a biochemical.</p>Formule :C10H18ClNOSCouleur et forme :SolidMasse moléculaire :235.77Lobeline sulfate
CAS :<p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>Formule :C22H29NO6SDegré de pureté :98%Couleur et forme :White PowderMasse moléculaire :435.54Hydroxybupropion
CAS :<p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>Formule :C13H18ClNO2Degré de pureté :99.73%Couleur et forme :Off-White SolidMasse moléculaire :255.74Oxotremorine
CAS :<p>Oxotremorine acts as an agonist of mAChR, specifically activating the M1 and M3 acetylcholine receptors. In drug discrimination experiments with macaques, it exhibits effects similar to nicotine.</p>Formule :C12H18N2OCouleur et forme :SolidMasse moléculaire :206.28Methyllycaconitine citrate
CAS :<p>Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.</p>Formule :C43H58N2O17Degré de pureté :98.03% - 98.91%Couleur et forme :SolidMasse moléculaire :874.92G-Protein antagonist peptide
CAS :<p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>Formule :C57H64N12O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1093.27M4 mAChR agonist-1
CAS :<p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).</p>Formule :C14H18N4OSDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :290.38Muscarine
CAS :<p>Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Formule :C9H20NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :174.26M3/PDE4 modulator-1
<p>M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.</p>Formule :C38H41Cl2N3O8SCouleur et forme :SolidMasse moléculaire :770.725-AMAM-2-CP
CAS :<p>5-AMAM-2-CP, a significant metabolite of Acetamiprid, serves as a global insecticide within the neonicotinoid class and acts as an nAChR agonist [1] [2].</p>Formule :C9H11ClN2OCouleur et forme :SolidMasse moléculaire :198.65(R)-Dinotefuran
CAS :<p>(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.</p>Formule :C7H14N4O3Couleur et forme :SolidMasse moléculaire :202.21Ebiratide TFA
<p>Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.</p>Formule :C48H73N11O10S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :996.23 (free base)TDI-10229
CAS :<p>TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.</p>Formule :C16H16ClN5Degré de pureté :99.85% - 99.89%Couleur et forme :SoildMasse moléculaire :313.78BTMPS
CAS :<p>BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.</p>Formule :C28H52N2O4Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :480.72Anabaseine
CAS :<p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>Formule :C10H12N2Couleur et forme :SolidMasse moléculaire :160.22N-Ethyl-N-(3-pyridylmethyl)amine
CAS :<p>N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.</p>Formule :C8H12N2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :136.19Soclenicant
CAS :<p>Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availability</p>Formule :C24H26N4O3Degré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :418.49Rivanicline 2HCl
<p>Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.</p>Formule :C10H16Cl2N2Degré de pureté :99.4%Couleur et forme :SoildMasse moléculaire :235.15Proadrenomedullin (1-20), human
CAS :<p>Endogenous peptide; agonist of MRGPRX2 (EC50=251 nM); noncompetitive inhibitor of nicotinic receptors; reduces catecholamine secretion; antihypertensive.</p>Formule :C112H178N36O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2460.84TC-2559 difumarate
CAS :<p>TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.</p>Formule :C20H26N2O9Couleur et forme :SolidMasse moléculaire :438.43Bensultap
CAS :<p>Bensultap is an agricultural chemical typically used as a pesticide.</p>Formule :C17H21NO4S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.61Ebiratide
CAS :<p>Ebiratide is an analog of ACTH 4-9.</p>Formule :C48H73N11O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :996.23GeX-2
CAS :<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Formule :C103H169N43O27Couleur et forme :SolidMasse moléculaire :2441.72Aceclidine (hydrochloride)
CAS :<p>agonist of muscarinic receptors</p>Formule :C9H16ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :205.68Tropicamide
CAS :<p>Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for diagnostic use.</p>Formule :C17H20N2O2Degré de pureté :99.78% - 99.94%Couleur et forme :White PowderMasse moléculaire :284.35Navafenterol
CAS :<p>AZD-8871, a potential COPD and asthma treatment, may work well with ICS.</p>Formule :C38H42N6O6S2Couleur et forme :SolidMasse moléculaire :742.91α-Conotoxin PIA
CAS :<p>Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM</p>Formule :C79H125N27O25S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1981.3(-)-OPC-51803
CAS :<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Formule :C26H32ClN3O2Degré de pureté :98.73% - 99.59%Couleur et forme :SoildMasse moléculaire :454(rel)-Asperparaline A
CAS :<p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>Formule :C20H29N3O3Couleur et forme :SolidMasse moléculaire :359.47sabcomeline
CAS :<p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>Formule :C10H15N3OCouleur et forme :SolidMasse moléculaire :193.25DSPE-PEG2000-RVG29
<p>DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.</p>Couleur et forme :Odour SolidLu AE51090
CAS :<p>Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.</p>Formule :C24H29N3O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :407.515-AAM-2-CP
CAS :<p>5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.</p>Formule :C8H9ClN2ODegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :184.62(R)-(+)-Anatabine
CAS :<p>(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.</p>Formule :C10H12N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :160.22(Rac)-Sabcomeline
CAS :<p>(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.</p>Formule :C10H15N3ODegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :193.25LAS190792
CAS :<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Formule :C39H43ClN4O9S2Couleur et forme :SolidMasse moléculaire :811.36Br-PBTC
CAS :<p>Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.</p>Formule :C14H15BrN2OSCouleur et forme :SolidMasse moléculaire :339.25β2AR/M-receptor agonist-1
CAS :<p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>Formule :C43H56BrN3O7Couleur et forme :SolidMasse moléculaire :806.82Dexetimide
CAS :<p>Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.</p>Formule :C23H26N2O2Couleur et forme :SolidMasse moléculaire :362.46Metixene hydrochloride hydrate
CAS :<p>Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.</p>Formule :C20H26ClNOSDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :363.95Fipexide hydrochloride
CAS :<p>Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.</p>Formule :C20H22Cl2N2O4Couleur et forme :SolidMasse moléculaire :425.31NKH477
CAS :<p>NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.</p>Formule :C27H44ClNO8Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :546.09Tolterodine
CAS :<p>Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.</p>Formule :C22H31NODegré de pureté :99.71%Couleur et forme :White Like Or Light Brown Crystalline PowderMasse moléculaire :325.49YM-58790 hydrochloride
CAS :<p>YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).</p>Formule :C27H32ClN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :466.02Palmatine hydroxide
CAS :<p>Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.</p>Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41Cevimeline
CAS :<p>Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.</p>Formule :C10H17NOSCouleur et forme :Off-White SolidMasse moléculaire :199.31Pirmenol hydrochloride
CAS :<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Formule :C22H31ClN2OCouleur et forme :SolidMasse moléculaire :374.95Varenicline Hydrochloride
CAS :<p>Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).</p>Formule :C13H14ClN3Degré de pureté :99.854%Couleur et forme :SolidMasse moléculaire :247.72Cevimeline hydrochloride
CAS :<p>Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.</p>Formule :C10H18ClOSCouleur et forme :SolidMasse moléculaire :235.77Glycerophosphoinositol choline
CAS :<p>Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.</p>Formule :C14H32NO12PCouleur et forme :SolidMasse moléculaire :437.38Ispronicline
CAS :<p>Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive</p>Formule :C14H22N2ODegré de pureté :97.70% - 99.16%Couleur et forme :SolidMasse moléculaire :234.34Sabcomeline hydrochloride
CAS :<p>Sabcomeline is a selective M1 receptor partial agonist.</p>Formule :C10H16ClN3OCouleur et forme :SolidMasse moléculaire :229.71(±)-Darifenacin
CAS :<p>(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.</p>Formule :C28H30N2O2Couleur et forme :SolidMasse moléculaire :426.55VU0467485
CAS :<p>VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.</p>Formule :C17H17FN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.41Clorprenaline
CAS :<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Formule :C11H16ClNODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :213.7ABT-107
CAS :<p>ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.</p>Formule :C19H20N4OCouleur et forme :SolidMasse moléculaire :320.396
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