AChR
Les inhibiteurs des récepteurs de l'acétylcholine (AChR) sont des composés qui bloquent l'activité des récepteurs de l'acétylcholine, essentiels pour la neurotransmission dans les systèmes nerveux central et périphérique. Les AChR jouent un rôle crucial dans la contraction musculaire, la mémoire et les fonctions cognitives. Les inhibiteurs des AChR sont utilisés pour étudier des conditions telles que la myasthénie grave, la maladie d'Alzheimer et d'autres troubles neurologiques. En modulant l'activité des AChR, ces inhibiteurs peuvent aider à démêler les complexités de la signalisation cholinergique dans le cerveau. Chez CymitQuimica, nous fournissons une gamme d'inhibiteurs des AChR pour soutenir vos recherches en neurosciences, pharmacologie et maladies neurodégénératives.
575 produits trouvés pour "AChR"
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Pirmenol hydrochloride
CAS :<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Formule :C22H31ClN2OCouleur et forme :SolidMasse moléculaire :374.95N6-Methyladenosine 5'-monophosphate disodium salt
CAS :<p>N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.</p>Formule :C11H14N5Na2O7PDegré de pureté :99.36% - 99.36%Couleur et forme :SolidMasse moléculaire :405.21DL-Cystine
CAS :<p>DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .</p>Formule :C6H12N2O4S2Couleur et forme :SolidMasse moléculaire :240.3Solifenacin D5 hydrochloride
CAS :<p>Solifenacin D5 HCl: deuterium-labeled M1, M2, M3 muscarinic receptor antagonist with pKi 7.6, 6.9, 8.0.</p>Formule :C23H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.96Tolterodine
CAS :<p>Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.</p>Formule :C22H31NODegré de pureté :99.71%Couleur et forme :White Like Or Light Brown Crystalline PowderMasse moléculaire :325.49NKH477
CAS :<p>NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.</p>Formule :C27H44ClNO8Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :546.09NSC 23766
CAS :<p>NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.</p>Formule :C24H35N7Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :421.58Telenzepine dihydrochloride
CAS :<p>muscarinic M1 receptor antagonist</p>Formule :C19H23ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.93Fipexide hydrochloride
CAS :<p>Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.</p>Formule :C20H22Cl2N2O4Couleur et forme :SolidMasse moléculaire :425.31SSR180711 hydrochloride
CAS :<p>SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.</p>Formule :C14H18BrClN2O2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :361.66Clorprenaline
CAS :<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Formule :C11H16ClNODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :213.7Cevimeline hydrochloride
CAS :<p>Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.</p>Formule :C10H18ClOSCouleur et forme :SolidMasse moléculaire :235.77Cevimeline
CAS :<p>Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.</p>Formule :C10H17NOSCouleur et forme :Off-White SolidMasse moléculaire :199.31Nanofin
CAS :<p>Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.</p>Formule :C7H15NDegré de pureté :97.38% - 99.818%Couleur et forme :Clear Colorless To Slightly Yellow LiquidMasse moléculaire :113.2Encenicline hydrochloride
CAS :<p>Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).</p>Formule :C16H17ClN2OS·HClDegré de pureté :98.34% - 99.85%Couleur et forme :SolidMasse moléculaire :357.3PHA 568487 free base
CAS :<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Formule :C16H20N2O3Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :288.34Tacrine hydrochloride (hydrate)
CAS :<p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>Formule :C13H14N2·XHCl·XH2ODegré de pureté :99.01% - 99.89%Couleur et forme :SolidMasse moléculaire :234.72NS3861
CAS :<p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>Formule :C12H14BrNSDegré de pureté :99.853%Couleur et forme :SolidMasse moléculaire :284.22Thiacloprid
CAS :<p>Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.</p>Formule :C10H9ClN4SDegré de pureté :98.66% - 99.95%Couleur et forme :Yellowish Crystalline PowderMasse moléculaire :252.72Cyclopentolate Hydrochloride
CAS :<p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>Formule :C17H26ClNO3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :327.85A-867744
CAS :<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Formule :C20H19ClN2O3SDegré de pureté :95.66%Couleur et forme :SolidMasse moléculaire :402.89PSEM 89S TFA
CAS :<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Formule :C18H23F3N2O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.38Mivacurium dichloride
CAS :<p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>Formule :C58H80Cl2N2O14Degré de pureté :99.2% - 99.48%Couleur et forme :Off-White SolidMasse moléculaire :1100.17Fesoterodine
CAS :<p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>Formule :C26H37NO3Degré de pureté :97.1%Couleur et forme :SolidMasse moléculaire :411.58DMAB-anabaseine dihydrochloride
CAS :<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Formule :C19H23Cl2N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :364.31Ethyl (triphenylphosphoranylidene) acetate
CAS :<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Formule :C22H21O2PDegré de pureté :97.985%Couleur et forme :White Or Slight Yellow PowderMasse moléculaire :348.37NS9283
CAS :<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Formule :C14H8N4ODegré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :248.24mAChR-IN-1 hydrochloride
CAS :<p>mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.</p>Formule :C23H26ClIN2O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :524.82Umeclidinium bromide
CAS :<p>Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.</p>Formule :C29H34BrNO2Degré de pureté :98.4% - 99.89%Couleur et forme :SolidMasse moléculaire :508.49ST034307
CAS :<p>ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).</p>Formule :C10H4Cl4O2Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :297.95(-)-(S)-B-973B
CAS :<p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>Formule :C24H26F2N6ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :452.5Pozanicline dihydrochloride
CAS :<p>Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)</p>Formule :C11H18Cl2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.18Cyclodrine hydrochloride
CAS :<p>Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of</p>Formule :C19H30ClNO3Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :355.9NS 1738
CAS :<p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>Formule :C14H9Cl2F3N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :365.13BNC210
CAS :<p>BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.</p>Formule :C17H23N3O3Degré de pureté :97.05% - >99.99%Couleur et forme :SolidMasse moléculaire :317.38Harman hydrochloride
CAS :<p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>Formule :C12H11ClN2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :218.68Nitenpyram
CAS :<p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>Formule :C11H15ClN4O2Degré de pureté :99.03%Couleur et forme :Light-Yellow CrystalMasse moléculaire :270.72PHA 543613 hydrochloride
CAS :<p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>Formule :C15H18ClN3O2Couleur et forme :SolidMasse moléculaire :307.78VU0238441
CAS :<p>VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.</p>Formule :C16H9ClF3NO2Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :339.7Solifenacin
CAS :Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formule :C23H26N2O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :362.46Anisotropine Methylbromide
CAS :<p>Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.</p>Formule :C17H32BrNO2Degré de pureté :99.73%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :362.35Dronedarone
CAS :<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formule :C31H44N2O5SDegré de pureté :98.85% - 99.58%Couleur et forme :SolidMasse moléculaire :556.76Pempidine
CAS :<p>Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.</p>Formule :C10H21NDegré de pureté :98.18% - 99.28%Couleur et forme :Colorless - Light Yellow Clear LiquidMasse moléculaire :155.28Dinotefuran
CAS :<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Formule :C7H14N4O3Degré de pureté :99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :202.21Sofpironium bromide
CAS :<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Formule :C22H32BrNO5Degré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :470.4Varenicline Tartrate
CAS :<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Formule :C13H13N3·C4H6O6Degré de pureté :98.23% - 98.32%Couleur et forme :Tan SolidMasse moléculaire :361.35JHU37152
CAS :<p>JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.</p>Formule :C19H20ClFN4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :358.84Clothianidin
CAS :<p>Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.</p>Formule :C6H8ClN5O2SDegré de pureté :99.71% - 99.87%Couleur et forme :Solid PowderMasse moléculaire :249.68Syn-Ake acetate
CAS :<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Formule :C19H29N5O3·2(C2H4O2)Degré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :495.58α-Conotoxin MII acetate
<p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>Formule :C69H107N23O24S4Degré de pureté :94.82% - 97.79%Couleur et forme :SolidMasse moléculaire :1770.99VU0357017 hydrochloride
CAS :<p>VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.</p>Formule :C18H28ClN3O3Degré de pureté :99% - 99.97%Couleur et forme :SolidMasse moléculaire :369.89Piperidolate hydrochloride
CAS :<p>Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.</p>Formule :C21H26ClNO2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :359.89KH7
CAS :<p>KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.</p>Formule :C17H15BrN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :419.3Batefenterol
CAS :<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formule :C40H42ClN5O7Degré de pureté :97.94% - 98.4%Couleur et forme :SolidMasse moléculaire :740.24Dicyclomine
CAS :<p>Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.</p>Formule :C19H35NO2Couleur et forme :SolidMasse moléculaire :309.49Tebanicline hydrochloride
CAS :<p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>Formule :C9H12Cl2N2ODegré de pureté :91.74% - 98.71%Couleur et forme :SolidMasse moléculaire :235.11TBPB
CAS :<p>TBPB is an allosteric M1 mAChR agonist.</p>Formule :C25H32N4ODegré de pureté :97.87% - 99.9%Couleur et forme :SolidMasse moléculaire :404.559-Ethyladenine
CAS :<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Formule :C7H9N5Degré de pureté :99.35% - 99.41%Couleur et forme :SolidMasse moléculaire :163.18suvn-911
CAS :<p>suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.</p>Formule :C11H14Cl2N2ODegré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :261.15Atracurium besylate
CAS :<p>Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.</p>Formule :C65H82N2O18S2Degré de pureté :98.94% - 99.71%Couleur et forme :SolidMasse moléculaire :1243.49A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Formule :C17H21ClN4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :316.834BP-TQS
CAS :<p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>Formule :C18H17BrN2O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :405.31Imidafenacin
CAS :<p>Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.</p>Formule :C20H21N3ODegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :319.4Brompheniramine
CAS :<p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>Formule :C16H19BrN2Couleur et forme :SolidMasse moléculaire :319.24Varenicline dihydrochloride
CAS :<p>Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.</p>Formule :C13H15Cl2N3Degré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :284.18SEN12333
CAS :<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Formule :C20H25N3O2Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :339.43Ilmetropium iodide
CAS :<p>Ilmetropium iodide is a bronchodilator.</p>Formule :C20H30INO3Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :459.36Ursulcholic acid
CAS :<p>Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.</p>Formule :C24H40O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.7Pirmenol
CAS :<p>Pirmenol is a new antiarrhythmic drug</p>Formule :C22H30N2ODegré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :338.49Darifenacin
CAS :<p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>Formule :C28H30N2O2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :426.55LY2119620
CAS :<p>LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.</p>Formule :C19H24ClN5O3SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :437.94Benzetimide hydrochloride
CAS :<p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>Formule :C23H27ClN2O2Degré de pureté :99.32%Couleur et forme :Off-White PowderMasse moléculaire :398.93Oxyphencyclimine
CAS :<p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>Formule :C20H28N2O3Couleur et forme :SolidMasse moléculaire :344.45Aclidinium bromide
CAS :<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Formule :C26H30NO4S2·BrDegré de pureté :99.53% - 99.69%Couleur et forme :SolidMasse moléculaire :564.55Coluracetam
CAS :<p>Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.</p>Formule :C19H23N3O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :341.4Mecamylamine hydrochloride
CAS :<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Formule :C11H22ClNDegré de pureté :99.76% - >99.99%Couleur et forme :White SolidMasse moléculaire :203.75Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Formule :C12H16N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :207.23BQCA
CAS :<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Formule :C18H15NO4Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :309.32Oxyphencyclimine Hydrochloride
CAS :<p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>Formule :C20H29ClN2O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :380.91Propantheline
CAS :<p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>Formule :C23H30NO3Couleur et forme :SolidMasse moléculaire :368.49Encenicline
CAS :<p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>Formule :C16H17ClN2OSDegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :320.84Propiverine
CAS :<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Formule :C23H29NO3Couleur et forme :SolidMasse moléculaire :367.48JHU37160
CAS :JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Formule :C19H20ClFN4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :358.84OXOMEMAZINE
CAS :<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Formule :C18H22N2O2SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :330.44Mecamylamine
CAS :<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Formule :C11H21NCouleur et forme :SolidMasse moléculaire :167.29Methylbenactyzium Bromide
CAS :<p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>Formule :C21H28BrNO3Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :422.36Solifenacin hydrochloride
CAS :<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Formule :C23H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.93Donepezil Hydrochloride
CAS :<p>Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).</p>Formule :C24H29NO3·HClDegré de pureté :99.55% - 99.8%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :415.96Isopropamide Iodide
CAS :<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Formule :C23H33IN2ODegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :480.43SQ22536
CAS :<p>SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.</p>Formule :C9H11N5ODegré de pureté :99.18%Couleur et forme :Off-White SolidMasse moléculaire :205.22ML380
CAS :<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Formule :C23H25F3N4O3SDegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :494.53VU0467154
CAS :<p>VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.</p>Formule :C17H15F3N4O3S2Degré de pureté :98.28% - 99.51%Couleur et forme :SolidMasse moléculaire :444.45VU0152100
CAS :<p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>Formule :C18H19N3O2SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :341.43Ipratropium Bromide
CAS :<p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>Formule :C20H30BrNO3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :412.37VU0119498
CAS :<p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>Formule :C15H10BrNO2Degré de pureté :97.56%Couleur et forme :SolidMasse moléculaire :316.15Succinylcholine Chloride Dihydrate
CAS :<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Formule :C14H30N2O4·2Cl·2H2ODegré de pureté :99.87%Couleur et forme :White SolidMasse moléculaire :397.34VU10010
CAS :<p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>Formule :C17H16ClN3OSDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :345.85Procyclidine hydrochloride
CAS :<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Formule :C19H30ClNODegré de pureté :99.24% - 99.88%Couleur et forme :Crystals From Petroleum Ether White PowderMasse moléculaire :323.9Oxotremorine sesquifumarate
CAS :<p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>Formule :C12H18N2OC4H4O4Degré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :380.39TQS
CAS :<p>TQS (4-Naphthalen-1-yl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide) is a positive allosteric modulator of α7 nACh receptors.</p>Formule :C22H20N2O2SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :376.47MC-Val-Cit-PAB
CAS :<p>MC-Val-Cit-PAB: cathepsin-cleavable ADC linker used in FDA-approved brentuximab vedotin.</p>Formule :C28H40N6O7Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :572.65Revefenacin
CAS :<p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>Formule :C35H43N5O4Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :597.75Nitrocaramiphen hydrochloride
CAS :<p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>Formule :C18H27ClN2O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :370.87Piperidolate
CAS :<p>Piperidolate inhibits intestinal cramp induced by acetylcholine</p>Formule :C21H25NO2Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :323.43PNU-282987 S enantiomer free base
CAS :<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Formule :C14H17ClN2ODegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :264.75VU 0238429
CAS :<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Formule :C17H12F3NO4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :351.28Glycopyrrolate
CAS :<p>Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.</p>Formule :C19H28BrNO3Degré de pureté :99.41% - 99.64%Couleur et forme :SolidMasse moléculaire :398.33CCMI
CAS :<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Formule :C19H15Cl2N3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :388.25W-84 dibromide
CAS :<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Formule :C32H44Br2N4O4Degré de pureté :95.56%Couleur et forme :SolidMasse moléculaire :708.52Prifinium bromide
CAS :<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Formule :C22H28BrNDegré de pureté :97.99%Couleur et forme :SolidMasse moléculaire :386.37Nor-benzetimide
CAS :<p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>Formule :C16H20N2O2Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :272.34PNU-120596
CAS :<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Formule :C13H14ClN3O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :311.72MC-Val-Cit-PABC-PNP
CAS :<p>MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.</p>Formule :C35H43N7O11Degré de pureté :97.2% - 98.055%Couleur et forme :SolidMasse moléculaire :737.76Blarcamesine
CAS :<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Formule :C19H23NODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :281.39(S)-UFR2709
CAS :<p>(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.</p>Formule :C13H17NO2Couleur et forme :SolidMasse moléculaire :219.284Mc-Val-Ala-PAB
CAS :<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Formule :C25H34N4O6Degré de pureté :98.34% - 99.24%Couleur et forme :SolidMasse moléculaire :486.56PHA 568487
CAS :<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Formule :C20H24N2O7Couleur et forme :SolidMasse moléculaire :404.419VU0152099
CAS :<p>VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).</p>Formule :C18H17N3O3SDegré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :355.41Bestim
CAS :<p>Bestim is an immunomodulatory dipeptide that is synthetic.</p>Formule :C16H19N3O5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :333.34Oxyphenonium bromide
CAS :<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Formule :C21H34BrNO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :428.404Nitrobenzylthioinosine
CAS :<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41Monepantel
CAS :<p>Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.</p>Formule :C20H13F6N3O2SDegré de pureté :99.83%Couleur et forme :White PowderMasse moléculaire :473.39Velufenacin
CAS :<p>Velufenacin is an antagonist of muscarinic receptor[1].</p>Formule :C19H20ClFN2O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :362.83Pentoxyverine
CAS :<p>Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.</p>Formule :C20H31NO3Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :333.47Xanomeline tartrate
CAS :<p>Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。</p>Formule :C18H29N3O7SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :431.5AF-710B
CAS :<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Formule :C20H27N3OSDegré de pureté :98.62% - 99.89%Couleur et forme :SolidMasse moléculaire :357.51Mepenzolate Bromide
CAS :<p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>Formule :C21H26BrNO3Degré de pureté :95.73% - 99.21%Couleur et forme :SolidMasse moléculaire :420.34Pipecuronium bromide
CAS :<p>Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.</p>Formule :C35H62Br2N4O4Degré de pureté :>99.99%Couleur et forme :PowderMasse moléculaire :762.7Varenicline
CAS :<p>Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.</p>Formule :C13H13N3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :211.26Atropine hydrobromide
CAS :<p>Atropine hydrobromide is a biochemical.</p>Formule :C17H24BrNO3Couleur et forme :SolidMasse moléculaire :370.28Anatabine dicitrate
<p>Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.</p>Formule :C22H28N2O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :544.46Pyrantel
CAS :<p>Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.</p>Formule :C11H14N2SDegré de pureté :98%Couleur et forme :Crystals From Methanol Yellowish Crystalline PowderMasse moléculaire :206.31Flavoxate
CAS :<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Formule :C24H25NO4Couleur et forme :SolidMasse moléculaire :391.46(±)-Atropine-d3 (N-methyl-d3)
CAS :(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Formule :C17H20D3NO3Masse moléculaire :292.39Oxantel
CAS :<p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>Formule :C13H16N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :216.28Aprofene
CAS :<p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>Formule :C21H27NO2Couleur et forme :SolidMasse moléculaire :325.44Catestatin
CAS :Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Formule :C107H173N37O26SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2425.84Dianicline dihydrochloride
CAS :<p>Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.</p>Formule :C13H16N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :216.28Biperiden lactate
CAS :<p>Biperiden lactate is a biochemical.</p>Formule :C24H35NO4Couleur et forme :SolidMasse moléculaire :401.54VU0029767
CAS :<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Formule :C21H21N3O3Couleur et forme :SolidMasse moléculaire :363.41Azacyclonol hydrochloride
CAS :<p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>Formule :C18H22ClNOCouleur et forme :Off White Crystalline PowderMasse moléculaire :303.83Diphenidol
CAS :<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Formule :C21H27NOCouleur et forme :Needles From Petroleum Ether SolidMasse moléculaire :309.45Sulindac sulfide
CAS :<p>Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.</p>Formule :C20H17FO2SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :340.41N-0861 racemate
CAS :<p>N-0861 racemate is the racemate of N-0861.</p>Formule :C13H17N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :243.31Sulfoxaflor
CAS :<p>Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.</p>Formule :C10H10F3N3OSDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :277.27Sch412348
CAS :<p>Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.</p>Formule :C22H21F2N9ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.46SR 16584
CAS :<p>α3β4 nAChR antagonist</p>Formule :C17H22N2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :270.37Tarafenacin
CAS :<p>Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.</p>Formule :C21H20F4N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.39Meseclazone
CAS :<p>Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.</p>Formule :C11H10ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.654-DAMP
CAS :<p>4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.</p>Formule :C21H26INO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.34mAChr-in-1
CAS :<p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>Formule :C23H25IN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :488.36Darenzepine
CAS :<p>Darenzepine is a muscarinic receptor inhibitor.</p>Formule :C21H21N3O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :347.41UB 165 fumarate
CAS :<p>UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.</p>Formule :C17H19ClN2O4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :350.8CDD0102
CAS :<p>CDD0102 is a potent agonist of M1 Muscarinic receptor.</p>Formule :C8H12N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :180.215-Iodo-A-85380 dihydrochloride
CAS :<p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>Formule :C9H13Cl2IN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.02Dimethyl-W84 (dibromide)
CAS :<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Formule :C34H48Br2N4O4Couleur et forme :SolidMasse moléculaire :736.59LY 2087101
CAS :<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Formule :C15H11FN2OS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.39AR-R 17779 hydrochloride
CAS :<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Formule :C9H15ClN2O2Couleur et forme :SolidMasse moléculaire :218.68Elucaine
CAS :<p>Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.</p>Formule :C19H23NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.39(R,R)-Glycopyrrolate
CAS :<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Formule :C19H28BrNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.34SIB 1508Y maleate
CAS :<p>neuronal nicotinic ACh receptor agonist</p>Formule :C16H18N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.33LRE1
CAS :<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Formule :C12H13ClN4SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :280.78Terodiline
CAS :<p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>Formule :C20H27NDegré de pureté :98.20% - 99.59%Couleur et forme :SolidMasse moléculaire :281.44Methacholine bromide
CAS :<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Formule :C8H18BrNO2Couleur et forme :SolidMasse moléculaire :240.141Nuvenzepine
CAS :<p>Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.</p>Formule :C19H20N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.39DA 4626
CAS :<p>DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.</p>Formule :C14H18N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :242.32Telenzepine
CAS :<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Formule :C19H22N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :370.47AC260584
CAS :AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Formule :C20H29FN2O2Couleur et forme :SolidMasse moléculaire :348.45Neramexane Mesylate
CAS :<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Formule :C12H27NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.41Chlorisondamine diiodide
CAS :<p>long lasting nicotinic antagonist</p>Formule :C14H20Cl4I2N2Couleur et forme :SolidMasse moléculaire :611.94ML381
CAS :<p>ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.</p>Formule :C21H21N3O4Couleur et forme :SolidMasse moléculaire :379.41ML169
CAS :<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Formule :C21H17BrFN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.34Zamifenacin
CAS :<p>Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.</p>Formule :C27H29NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :415.52BNC375
CAS :<p>BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).</p>Formule :C19H23ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.92(R,R)-Reboxetine mesylate
CAS :<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Formule :C20H27NO6SCouleur et forme :SolidMasse moléculaire :409.5M1 ligand 1
CAS :<p>Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.</p>Formule :C20H21NO2Couleur et forme :SolidMasse moléculaire :307.39Benzatropine
CAS :<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Formule :C21H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.43Muscarine iodide
CAS :<p>Muscarinic acetylcholine receptor agonist</p>Formule :C9H20INO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :301.17Tridihexethyl chloride
CAS :<p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>Formule :C21H36ClNOCouleur et forme :SolidMasse moléculaire :353.97TC 2559 difumarate
CAS :<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Formule :C12H18N2OC4H404Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :380.39TC299423
CAS :<p>TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.</p>Formule :C11H15N3Couleur et forme :SolidMasse moléculaire :189.26SM-21 maleate
CAS :<p>Increases release of acetylcholine,σ2 antagonist</p>Formule :C22H28ClNO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.91TC 1698 dihydrochloride
CAS :<p>nicotinic α7 receptor agonist</p>Formule :C13H18N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :202.3Beperidium iodide
CAS :<p>Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).</p>Formule :C23H34IN3O3Couleur et forme :SolidMasse moléculaire :527.44WIN 62,577
CAS :<p>WIN 62,577 is a allosteric antagonist of mAChR.</p>Formule :C29H31N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :437.58Benzamide Derivative 1
CAS :<p>Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.</p>Formule :C22H34ClN3O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :423.98Alvameline
CAS :<p>Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.</p>Formule :C9H15N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :193.25Muscarine chloride
CAS :<p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Formule :C9H20ClNO2Couleur et forme :SolidMasse moléculaire :209.71Quifenadine
CAS :<p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>Formule :C20H23NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.4DAU 5884 hydrochloride
CAS :<p>muscarinic M3 receptor antagonist</p>Formule :C17H22ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.83Nelonicline
CAS :<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Formule :C17H19N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.42BTM-1086
CAS :<p>BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.</p>Formule :C21H25N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :367.51CP-601932
CAS :<p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>Formule :C12H12F3NCouleur et forme :SolidMasse moléculaire :227.23Eucatropine
CAS :<p>Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.</p>Formule :C17H25NO3Couleur et forme :SolidMasse moléculaire :291.39Thiochrome
CAS :<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Formule :C12H14N4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.33VU0090157
CAS :<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Formule :C19H21N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.39S-(+)-Mecamylamine hydrochloride
CAS :<p>Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.</p>Formule :C11H22ClNCouleur et forme :SolidMasse moléculaire :203.75T761-0184
CAS :<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Formule :C16H20FN3OCouleur et forme :SolidMasse moléculaire :289.35Revatropate
CAS :<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Formule :C19H27NO4SCouleur et forme :SolidMasse moléculaire :365.49Rispenzepine
CAS :<p>Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.</p>Formule :C19H20N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.39
