AChR
Les inhibiteurs des récepteurs de l'acétylcholine (AChR) sont des composés qui bloquent l'activité des récepteurs de l'acétylcholine, essentiels pour la neurotransmission dans les systèmes nerveux central et périphérique. Les AChR jouent un rôle crucial dans la contraction musculaire, la mémoire et les fonctions cognitives. Les inhibiteurs des AChR sont utilisés pour étudier des conditions telles que la myasthénie grave, la maladie d'Alzheimer et d'autres troubles neurologiques. En modulant l'activité des AChR, ces inhibiteurs peuvent aider à démêler les complexités de la signalisation cholinergique dans le cerveau. Chez CymitQuimica, nous fournissons une gamme d'inhibiteurs des AChR pour soutenir vos recherches en neurosciences, pharmacologie et maladies neurodégénératives.
575 produits trouvés pour "AChR"
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Atropine methyl bromide
CAS :<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Formule :C18H26BrNO3Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :384.308Nicardipine hydrochloride
CAS :<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formule :C26H30ClN3O6Degré de pureté :99.58% - 99.89%Couleur et forme :Yellow SolidMasse moléculaire :515.99Deschloroclozapine
CAS :<p>Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.</p>Formule :C18H20N4Degré de pureté :99.61% - 99.98%Couleur et forme :SolidMasse moléculaire :292.38Temephos
CAS :<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Formule :C16H20O6P2S3Degré de pureté :≥95%Couleur et forme :White Crystalline Solid Or LiquidMasse moléculaire :466.47Cotinine
CAS :<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Formule :C10H12N2ODegré de pureté :98% - 99.89%Couleur et forme :Viscous Oil SolidMasse moléculaire :176.22Bambuterol hydrochloride
CAS :<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formule :C18H30ClN3O5Degré de pureté :99.53% - 99.61%Couleur et forme :White SolidMasse moléculaire :403.91Lysipressin acetate(50-57-7(fb_acetate))
CAS :<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formule :C48H69N13O14S2Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1116.28Dequalinium chloride
CAS :<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Formule :C30H40Cl2N4Degré de pureté :99.79% - 99.9%Couleur et forme :SolidMasse moléculaire :527.59Ipratropium bromide monohydrate
CAS :<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Formule :C20H32BrNO4Degré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :430.38Gallamine triethiodide
CAS :<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Formule :C30H60I3N3O3Degré de pureté :98.90%Couleur et forme :White Amorphous Powder SolidMasse moléculaire :891.53Droperidol
CAS :<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formule :C22H22FN3O2Degré de pureté :97.16% - 98%Couleur et forme :SolidMasse moléculaire :379.43Tiotropium bromide
CAS :<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Formule :C19H22BrNO4S2Degré de pureté :96.82% - 99.97%Couleur et forme :White SolidMasse moléculaire :472.42Orphenadrine Citrate
CAS :<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Formule :C18H23NO·C6H8O7Degré de pureté :98% - 99.58%Couleur et forme :White SolidMasse moléculaire :461.5Benztropine mesylate
CAS :<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Adiphenine hydrochloride
CAS :<p>Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.</p>Formule :C20H25NO2·HClDegré de pureté :97.76% - 99.53%Couleur et forme :White Or Almost White PowderMasse moléculaire :347.88DL-trihexyphenidyl hydrochloride
CAS :<p>DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.</p>Formule :C20H32ClNODegré de pureté :99.63% - 99.71%Couleur et forme :SolidMasse moléculaire :337.93Pyrantel pamoate
CAS :<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Formule :C34H30N2O6SDegré de pureté :99.71%Masse moléculaire :594.69Rivastigmine tartrate
CAS :<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Formule :C14H22N2O2·C4H6O6Degré de pureté :98% - 99.66%Couleur et forme :White To Off-White PowderMasse moléculaire :400.43(Rac)-Sabcomeline HCl
CAS :<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Formule :C10H16ClN3ODegré de pureté :99.58%Couleur et forme :SoildMasse moléculaire :229.71Promethazine hydrochloride
CAS :<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.889-Cyclopentyladenine
CAS :<p>9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signaling</p>Formule :C10H13N5Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :203.24Fesoterodine fumarate
CAS :<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Formule :C26H37NO3·C4H4O4Degré de pureté :99.16%Couleur et forme :White SolidMasse moléculaire :527.65Zelminemab
CAS :<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Degré de pureté :98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Couleur et forme :LiquidPrimidone
CAS :<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Formule :C12H14N2O2Degré de pureté :99.91%Couleur et forme :Crystals (Ntp 1992)Masse moléculaire :218.25MK-7622
CAS :<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formule :C25H25N3O2Degré de pureté :99.77% - 99.8%Couleur et forme :SolidMasse moléculaire :399.48Methscopolamine
CAS :<p>Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.</p>Formule :C18H24BrNO4Degré de pureté :99.12% - ≥98%Couleur et forme :SolidMasse moléculaire :398.29Ribavirin
CAS :<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Formule :C8H12N4O5Degré de pureté :99.09% - 99.83%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.20(Rac)-ABT-202 dihydrochloride
CAS :<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Formule :C9H15Cl2N3Degré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :236.142Procainamide hydrochloride
CAS :<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Formule :C13H21N3O·HClDegré de pureté :99.83% - 99.97%Couleur et forme :White To Slightly Yellow PowderMasse moléculaire :271.79PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formule :C36H51Cl3N4O7SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :790.24Acetamiprid
CAS :<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Formule :C10H11ClN4Degré de pureté :99.66%Couleur et forme :White PowderMasse moléculaire :222.67Rocuronium bromide
CAS :<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Formule :C32H53BrN2O4Degré de pureté :99.77% - >99.99%Couleur et forme :White Or Off-White PowderMasse moléculaire :609.68TAK-071
CAS :<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Formule :C24H24FN3O3Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :421.46Carbachol
CAS :<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Formule :C6H15ClN2O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :182.65Benzethonium chloride
CAS :<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Formule :C27H42ClNO2Degré de pureté :99.91%Couleur et forme :White To Off-White Solid Solid Particulate/PowderMasse moléculaire :448.09Pyrantel tartrate
CAS :<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Formule :C15H20N2O6SDegré de pureté :99.96%Couleur et forme :White CrystalsMasse moléculaire :356.39Dicyclomine hydrochloride
CAS :<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Formule :C19H36ClNO2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :345.95VU 0365114
CAS :<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Formule :C22H14F3NO3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :397.35Bethanechol chloride
CAS :<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Formule :C7H17N2O2·ClDegré de pureté :95% - 99.73%Couleur et forme :White CrystallineMasse moléculaire :196.68Benactyzine hydrochloride
CAS :<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Formule :C20H26ClNO3Degré de pureté :99.03% - 99.94%Couleur et forme :SolidMasse moléculaire :363.88Solifenacin succinate
CAS :<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Formule :C23H26N2O2·C4H6O4Degré de pureté :99.85% - 99.98%Couleur et forme :SolidMasse moléculaire :480.56Diphenmanil methylsulfate
CAS :<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Formule :C20H24N·CH3O4SDegré de pureté :98% - 99.27%Couleur et forme :SolidMasse moléculaire :389.51Pirenzepine dihydrochloride
CAS :<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Formule :C19H21N5O2·2HClDegré de pureté :99.48% - 99.62%Couleur et forme :White PowderMasse moléculaire :424.32Neostigmine methyl sulfate
CAS :<p>Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.</p>Formule :C13H22N2O6SDegré de pureté :99.34% - 99.53%Couleur et forme :Crystalline SolidMasse moléculaire :334.39Pancuronium dibromide
CAS :<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Formule :C35H60Br2N2O4Degré de pureté :99.86%Couleur et forme :solidMasse moléculaire :732.67Nefiracetam
CAS :<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formule :C14H18N2O2Degré de pureté :97.37%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :246.3Nebracetam hydrochloride
CAS :<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Formule :C12H17ClN2ODegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :240.729Carbetapentane citrate
CAS :<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Formule :C20H31NO3·C6H8O7Degré de pureté :99.46%Couleur et forme :White To Off-White SolidMasse moléculaire :525.59Valethamate bromide
CAS :<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Formule :C19H32BrNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :386.372',5'-Dideoxyadenosine
CAS :<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Formule :C10H13N5O2Degré de pureté :99.55%Couleur et forme :White SolidMasse moléculaire :235.24
