
DPP-4
Les inhibiteurs de DPP-4 sont des composés qui inhibent la Dipeptidyl Peptidase-4, une enzyme impliquée dans l'inactivation des hormones incrétines, qui régulent le métabolisme du glucose. En inhibant la DPP-4, ces composés prolongent l'action des hormones incrétines, augmentant la sécrétion d'insuline et réduisant les niveaux de glucose dans le sang. Les inhibiteurs de DPP-4 sont largement utilisés dans le traitement du diabète de type 2 et dans les recherches axées sur les troubles métaboliques. Chez CymitQuimica, nous proposons des inhibiteurs de DPP-4 pour soutenir vos recherches en endocrinologie, gestion du diabète et maladies métaboliques.
23 produits trouvés pour "DPP-4"
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Denagliptin
CAS :Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study ofFormule :C20H18F3N3ODegré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :373.37Saxagliptin hydrate
CAS :Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).Formule :C18H25N3O2·H2ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :333.43Retagliptin Phosphate
CAS :Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Formule :C19H21F6N4O7PDegré de pureté :98.70%Couleur et forme :SolidMasse moléculaire :562.36Ref: TM-T12710
1mg34,00€2mg42,00€5mg60,00€10mg87,00€25mg161,00€50mg245,00€100mgÀ demander1mL*10mM (DMSO)79,00€DPP-IV-IN-2
CAS :DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Formule :C18H26N4O5Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :378.423-Pyridylacetic acid hydrochloride
CAS :3-Pyridylacetic acid HCl (3-PAA) is a strong acid, reactive with amines/alcohols/acids, and an organic catalyst.Formule :C7H8ClNO2Degré de pureté :99.31% - 99.95%Couleur et forme :White To Beige Crystalline PowderMasse moléculaire :173.6DPP4/CD26 Protein, Mouse, Recombinant (hFc)
DPP4/CD26 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.Degré de pureté :99% - > 95 % as determined by SDS-PAGE.Couleur et forme :Lyophilized PowderMasse moléculaire :112.9 kDa (predicted)DPP4/CD26 Protein, Mouse, Recombinant (His)
DPP4/CD26 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.Couleur et forme :Lyophilized PowderMasse moléculaire :85.9 kDa (predicted)Alogliptin Benzoate
CAS :Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.Formule :C25H27N5O4Degré de pureté :99.94% - >99.99%Couleur et forme :White PowderMasse moléculaire :461.51Diprotin A
CAS :Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formule :C17H31N3O4Degré de pureté :99.29%Couleur et forme :White PowderMasse moléculaire :341.45Saxagliptin
CAS :Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.Formule :C18H25N3O2Degré de pureté :99.17% - 99.95%Couleur et forme :SolidMasse moléculaire :315.41Alogliptin
CAS :Alogliptin (SYR-322)(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of <10 nM, exhibits greater than 10, 000-fold selectivity over DPP-8 and DPP-9Formule :C18H21N5O2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :339.39Ref: TM-T6192
2mg34,00€5mg49,00€10mg60,00€25mg81,00€50mg92,00€100mg129,00€200mg178,00€1mL*10mM (DMSO)50,00€Omarigliptin
CAS :Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.Formule :C17H20F2N4O3SDegré de pureté :99.68% - 99.77%Couleur et forme :SolidMasse moléculaire :398.43Ref: TM-T2316
1mg38,00€2mg50,00€5mg80,00€10mg117,00€25mg200,00€50mg333,00€100mg477,00€500mg1.063,00€1mL*10mM (DMSO)131,00€Trelagliptin succinate
CAS :Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Formule :C22H26FN5O6Degré de pureté :99.27% - 99.92%Couleur et forme :SolidMasse moléculaire :475.47Anagliptin
CAS :Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.Formule :C19H25N7O2Degré de pureté :97.59% - 99.98%Couleur et forme :SolidMasse moléculaire :383.45Ref: TM-T7133
1mg47,00€5mg92,00€10mg137,00€25mg224,00€50mg331,00€100mg502,00€200mg715,00€1mL*10mM (DMSO)97,00€Picolamine
CAS :Picolamine acts as a potential inhibitor of DPP-4.Formule :C6H8N2Degré de pureté :98.3%Couleur et forme :Light Yellow LiquidMasse moléculaire :108.14Teneligliptin
CAS :Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formule :C22H30N6OSDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :426.58Cofrogliptin
CAS :Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).Formule :C18H19F5N4O3SCouleur et forme :SolidMasse moléculaire :466.43Gemigliptin Tartrate(911637-19-9 free base)
CAS :Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).Formule :C22H25F8N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :639.45Gosogliptin
CAS :Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.Formule :C17H24F2N6ODegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :366.41Imigliptin
CAS :Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.Formule :C21H24N6ODegré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :376.46
