Récepteur de la mélatonine
Los receptores de ácido lisofosfatídico (LPA) son un grupo de GPCR que responden al LPA, un lípido bioactivo involucrado en la proliferación, migración y supervivencia celular. La señalización de LPA juega un papel crucial en varios procesos fisiológicos, incluyendo la cicatrización de heridas, el desarrollo vascular y la metástasis del cáncer. La modulación de la actividad de los receptores de LPA se está explorando para aplicaciones terapéuticas en el cáncer, la fibrosis y las enfermedades inflamatorias. En CymitQuimica, ofrecemos una gama de moduladores de receptores de LPA de alta calidad para apoyar su investigación en señalización celular, oncología y trastornos inflamatorios.
26 produits trouvés pour "Récepteur de la mélatonine"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Agomelatine
CAS :Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Formule :C15H17NO2Degré de pureté :99.92%Couleur et forme :White SolidMasse moléculaire :243.3Ramelteon
CAS :Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.Formule :C16H21NO2Degré de pureté :97.21% - 99.92%Couleur et forme :Crystalline SolidMasse moléculaire :259.34Ref: TM-T1463
2mg44,00€5mg65,00€10mg88,00€25mg136,00€50mg202,00€100mg325,00€500mg512,00€1mL*10mM (DMSO)71,00€Luzindole
CAS :Luzindole (N-0774) is a selective melatonin receptor antagonist.Formule :C19H20N2ODegré de pureté :98.53%Couleur et forme :Off-White Amorphous SolidMasse moléculaire :292.37Ref: TM-T15795
1mg49,00€2mg66,00€5mg92,00€10mg138,00€25mg245,00€50mg349,00€100mg512,00€200mg730,00€1mL*10mM (DMSO)147,00€UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Couleur et forme :Odour Solid4-P-PDOT
CAS :4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.Formule :C19H21NODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :279.38Melatonin-Tamoxifen Conjugate
Melatonin-Tamoxifen Conjugate (compound 16c) is an anticancer drug conjugate made of Melatonin and Tamoxifen, serving as an effective antagonist of ERα (IC50 = 863 nM). In cells expressing the hMT1 receptor, it binds to MLT receptors (Ki = 3.1 nM) and exhibits the ability to promote β-arrestin activation (EC50 = 914 nM) and ERK activation (EC50 = 98 nM). The IC50 values for Melatonin-Tamoxifen Conjugate in MCF-7, MDA-MB-231, and HT-1080 cell lines are 6.8 μM, 6.4 μM, and 1.7 μM, respectively.Formule :C47H58N4O4Couleur et forme :SolidMasse moléculaire :742.99Ramelteon-d5
CAS :Ramelteon-d5 is a deuterated compound of Ramelteon.Formule :C16H16D5NO2Couleur et forme :SolidMasse moléculaire :264.37ACH-000143
CAS :ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formule :C13H16ClN3O3Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :297.74Ref: TM-T9193
1mg52,00€5mg116,00€10mg182,00€25mg320,00€50mg449,00€100mg615,00€200mg830,00€1mL*10mM (DMSO)128,00€Tasimelteon
CAS :Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formule :C15H19NO2Degré de pureté :98.93% - 99.93%Couleur et forme :SolidMasse moléculaire :245.32N-ACETYLTRYPTAMINE
CAS :N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Formule :C12H14N2ODegré de pureté :98.79%Couleur et forme :PowderMasse moléculaire :202.25Melatonin
CAS :<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Formule :C13H16N2O2Degré de pureté :98% - 99.89%Couleur et forme :Pale Yellow Leaflets From Benzene SolidMasse moléculaire :232.28S26131
CAS :S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormule :C31H34N2O4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :498.61UCM 608
CAS :UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formule :C19H20N2O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :308.37DH-97
CAS :DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Formule :C22H26N2OCouleur et forme :SolidMasse moléculaire :334.45Cgp 52608
CAS :CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.Formule :C8H12N4OS2Couleur et forme :SolidMasse moléculaire :244.34GR 196429
CAS :GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.Formule :C14H18N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :246.3S-22153
CAS :S22153 is an antagonist of melatonin receptor.Formule :C14H17NOSCouleur et forme :SolidMasse moléculaire :247.36Melatonin receptor agonist 1
CAS :Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formule :C15H19N3O2Couleur et forme :SolidMasse moléculaire :273.33S20928
CAS :S20928 is an antagonist of melatonin receptor.Formule :C17H19NOCouleur et forme :SolidMasse moléculaire :253.34
