Récepteur de l'histamine
Les récepteurs de l'histamine sont des GPCR qui médiatisent les effets de l'histamine, une amine biogène impliquée dans les réponses immunitaires, la sécrétion d'acide gastrique et la neurotransmission. Il existe quatre sous-types de récepteurs de l'histamine (H1, H2, H3 et H4), chacun jouant des rôles distincts dans les réactions allergiques, la fonction gastrique et l'activité du système nerveux central. Les antagonistes des récepteurs de l'histamine sont largement utilisés dans le traitement des allergies, des ulcères gastriques et du mal des transports. Chez CymitQuimica, nous offrons une sélection complète de modulateurs de récepteurs de l'histamine de haute qualité pour soutenir vos recherches en immunologie, gastroentérologie et neuropharmacologie.
358 produits trouvés pour "Récepteur de l'histamine"
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Dimenhydrinate
CAS :<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Formule :C24H28ClN5O3Degré de pureté :99.57% - 99.77%Couleur et forme :Crystals Physical Description Crystalline White Powder (Ntp 1992)Masse moléculaire :469.96Pimethixene
CAS :<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Histamine
CAS :<p>Histamine (Ergamine) is an amine derived by the enzymatic decarboxylation of histamine. Histamine is a potent stimulant of gastric secretion of central action. High-Quality, Low-Cost!</p>Formule :C5H9N3Degré de pureté :96.63% - >99.99%Couleur et forme :Needles From Chloroform SolidMasse moléculaire :111.15Levodropropizine
CAS :<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Formule :C13H20N2O2Degré de pureté :99.87% - 99.93%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.31Astemizole
CAS :<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Formule :C28H31FN4ODegré de pureté :98.24% - 99.67%Couleur et forme :White Crystals SolidMasse moléculaire :458.57Chloropyramine hydrochloride
CAS :<p>Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.</p>Formule :C16H20ClN3·HClDegré de pureté :99.45% - 99.8%Couleur et forme :SolidMasse moléculaire :326.26Azacyclonol
CAS :<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Formule :C18H21NODegré de pureté :99.46%Couleur et forme :Solid PowderMasse moléculaire :267.37Lafutidine
CAS :<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Formule :C22H29N3O4SDegré de pureté :98.55%Couleur et forme :Yellowish White Crystalline PowderMasse moléculaire :431.55Amodiaquine dihydrochloride dihydrate
CAS :<p>Amodiaquine dihydrochloride dihydrate (Amodiaquin hydrochloride) is an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory effects</p>Formule :C20H28Cl3N3O3Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :464.82Antazoline hydrochloride
CAS :<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Formule :C17H19N3·HClDegré de pureté :98% - 99.53%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :301.82Brompheniramine maleate
CAS :<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Fexofenadine hydrochloride
CAS :<p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>Formule :C32H40ClNO4Degré de pureté :>99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :538.12Perphenazine
CAS :<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.99%Couleur et forme :SolidMasse moléculaire :403.97Fenspiride hydrochloride
CAS :<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formule :C15H20N2O2·HClDegré de pureté :99.64% - 99.92%Couleur et forme :SolidMasse moléculaire :296.79Tripelennamine hydrochloride
CAS :<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Formule :C16H21N3·HClDegré de pureté :99.54% - 99.81%Couleur et forme :White SolidMasse moléculaire :291.82Benztropine mesylate
CAS :<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Famotidine
CAS :<p>Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.</p>Formule :C8H15N7O2S3Degré de pureté :98.93% - 99.91%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :337.45Rupatadine Fumarate
CAS :<p>Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.</p>Formule :C26H26ClN3·C4H4O4Degré de pureté :99.86%Couleur et forme :White Or Almost-White PowderMasse moléculaire :532.03Ketotifen fumarate
CAS :<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Formule :C23H23NO5SDegré de pureté :99.25% - 99.73%Couleur et forme :SolidMasse moléculaire :425.50Chlorprothixene hydrochloride
CAS :<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Formule :C18H18ClNS·HClDegré de pureté :99.76%Couleur et forme :White PowderMasse moléculaire :352.32Diphenylpyraline hydrochloride
CAS :<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Formule :C19H23NO·HClDegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :317.85Azatadine dimaleate
CAS :<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Formule :C28H30N2O8Degré de pureté :99.7% - >99.99%Couleur et forme :PowderMasse moléculaire :522.55Mepyramine maleate
CAS :<p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>Formule :C21H27N3O5Degré de pureté :99.51% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :401.47Dexchlorpheniramine Maleate
CAS :<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86Cyproheptadine hydrochloride sesquihydrate
CAS :<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Formule :C21H24ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88Cimetidine
CAS :<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Formule :C10H16N6SDegré de pureté :99.82%Couleur et forme :Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Masse moléculaire :252.34Mifentidine
CAS :<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Formule :C13H16N4Degré de pureté :98.34% - 99.73%Couleur et forme :SolidMasse moléculaire :228.29Promethazine hydrochloride
CAS :<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.88Doxylamine succinate
CAS :<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formule :C21H28N2O5Degré de pureté :99.61%Couleur et forme :5 1 (Ntp 1992)Masse moléculaire :388.46Mebhydrolin napadisylate
CAS :<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Formule :C19H20N2C10H8O6S2Degré de pureté :99.35% - 99.96%Couleur et forme :White Or Almost White CrystallineMasse moléculaire :420.52Mizolastine
CAS :<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Formule :C24H25FN6ODegré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :432.49Terfenadine
CAS :<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Formule :C32H41NO2Degré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :471.67Doxepin hydrochloride
CAS :<p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>Formule :C19H22ClNODegré de pureté :99.65% - 99.91%Couleur et forme :White To Off-White PowderMasse moléculaire :315.84Triprolidine hydrochloride monohydrate
CAS :<p>Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.</p>Formule :C19H25ClN2ODegré de pureté :99.68% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :332.87Talastine
CAS :<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Formule :C19H21N3ODegré de pureté :98.50% - 99.44%Couleur et forme :SolidMasse moléculaire :307.39Pheniramine maleate
CAS :<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Formule :C16H20N2·C4H4O4Degré de pureté :99.85%Couleur et forme :Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CMasse moléculaire :356.42Cetirizine dihydrochloride
CAS :<p>Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.</p>Formule :C21H27Cl3N2O3Degré de pureté :99.4% - 99.97%Couleur et forme :SolidMasse moléculaire :461.81Hydroxyzine Pamoate
CAS :<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Formule :C44H43ClN2O8Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :763.27Ranitidine Hydrochloride
CAS :<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Formule :C13H23ClN4O3SDegré de pureté :99.30% - 99.49%Couleur et forme :SolidMasse moléculaire :350.86Carbinoxamine Maleate Salt
CAS :<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Formule :C20H23ClN2O5Degré de pureté :99.97%Couleur et forme :Off-White SolidMasse moléculaire :406.86Cinnarizine
CAS :<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Formule :C26H28N2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :368.51Meclizine dihydrochloride
CAS :<p>Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation</p>Formule :C25H27ClN2·2HClDegré de pureté :98.05% - 99.79%Couleur et forme :White Slightly Yellowish Crystalline PowderMasse moléculaire :463.87Levocetirizine
CAS :<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Formule :C21H25ClN2O3Degré de pureté :98% - 99.9%Couleur et forme :White PowderMasse moléculaire :388.89JNJ-39758979
CAS :<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formule :C11H19N5Degré de pureté :98.33% - 99.62%Couleur et forme :SolidMasse moléculaire :221.3Orphenadrine hydrochloride
CAS :<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Formule :C18H23NO·HClDegré de pureté :99.88%Couleur et forme :Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Masse moléculaire :305.85MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Formule :C24H26F3N3O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :477.48Pemirolast potassium
CAS :<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Formule :C10H7KN6ODegré de pureté :98.91% - 99.63%Couleur et forme :Crystals From Dimethylformamide Crystalline SolidMasse moléculaire :266.31Clemastine fumarate
CAS :<p>Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.</p>Formule :C25H30ClNO5Degré de pureté :99.52% - >99.99%Couleur et forme :Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderMasse moléculaire :459.97Roxatidine Acetate hydrochloride
CAS :<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Formule :C19H29ClN2O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :384.9Loratadine
CAS :<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Formule :C22H23ClN2O2Degré de pureté :99.71% - 99.98%Couleur et forme :White PowderMasse moléculaire :382.88
