Récepteur de l'histamine
Les récepteurs de l'histamine sont des GPCR qui médiatisent les effets de l'histamine, une amine biogène impliquée dans les réponses immunitaires, la sécrétion d'acide gastrique et la neurotransmission. Il existe quatre sous-types de récepteurs de l'histamine (H1, H2, H3 et H4), chacun jouant des rôles distincts dans les réactions allergiques, la fonction gastrique et l'activité du système nerveux central. Les antagonistes des récepteurs de l'histamine sont largement utilisés dans le traitement des allergies, des ulcères gastriques et du mal des transports. Chez CymitQuimica, nous offrons une sélection complète de modulateurs de récepteurs de l'histamine de haute qualité pour soutenir vos recherches en immunologie, gastroentérologie et neuropharmacologie.
385 produits trouvés pour "Récepteur de l'histamine"
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Cyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88Cetirizine dihydrochloride
CAS :Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formule :C21H27Cl3N2O3Degré de pureté :99.4% - 99.97%Couleur et forme :SolidMasse moléculaire :461.81Mepyramine maleate
CAS :Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Formule :C21H27N3O5Degré de pureté :99.51% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :401.47Promethazine hydrochloride
CAS :Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.88Mifentidine
CAS :Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Formule :C13H16N4Degré de pureté :98.34% - 99.73%Couleur et forme :SolidMasse moléculaire :228.29Amitriptyline hydrochloride
CAS :Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormule :C20H24ClNDegré de pureté :97% - 99.94%Couleur et forme :Crystals White To Off-White PowderMasse moléculaire :313.86Pimethixene
CAS :Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Ref: TM-T12489
2mg33,00€5mg48,00€10mg62,00€25mg101,00€50mg149,00€100mg215,00€200mg320,00€1mL*10mM (DMSO)50,00€Loratadine
CAS :Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.Formule :C22H23ClN2O2Degré de pureté :99.71% - 99.98%Couleur et forme :White PowderMasse moléculaire :382.88Pheniramine maleate
CAS :Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formule :C16H20N2·C4H4O4Degré de pureté :99.85%Couleur et forme :Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CMasse moléculaire :356.42Chlorpheniramine maleate
CAS :Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formule :C20H23ClN2O4Degré de pureté :99.64% - 99.98%Couleur et forme :Odorless White Crystalline Solid Or White Powder With A Bitter TasteMasse moléculaire :390.87KSK67
CAS :KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with KiFormule :C22H27N3O2Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :365.47Betahistine mesylate
CAS :Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.Formule :C8H12N2·2(CH4O3S)Degré de pureté :98% - 99.85%Couleur et forme :CoaMasse moléculaire :328.4Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFormule :C7H13N3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :171.2Samelisant
CAS :Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Formule :C21H31N3O3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :373.49Ref: TM-T9770
1mg105,00€2mg158,00€5mg260,00€10mg416,00€25mg687,00€50mg964,00€100mg1.288,00€500mg2.602,00€1mL*10mM (DMSO)268,00€Methapyrilene hydrochloride
CAS :Methapyrilene hydrochloride is a biochemical.Formule :C14H20ClN3SCouleur et forme :Liquid Solution) 5 5 (Ntp 1992)Masse moléculaire :297.85Tecastemizole
CAS :Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formule :C19H21FN4Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :324.4Ref: TM-T26253
1mg54,00€5mg118,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mg1.161,00€1mL*10mM (DMSO)131,00€KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Formule :C26H28N4O3Degré de pureté :97.51%Couleur et forme :SoildMasse moléculaire :444.53Cetirizine D8 dihydrochloride
CAS :Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Formule :C21H26Cl2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.4Donetidine
CAS :Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formule :C20H25N5O3SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :415.51Histamine H4 receptor antagonist-1
CAS :Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Formule :C30H38N8O2Couleur et forme :SolidMasse moléculaire :542.68Sufotidine
CAS :Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.Formule :C20H31N5O3SDegré de pureté :99.03% - 99.92%Couleur et forme :SolidMasse moléculaire :421.56Thioperamide maleate
CAS :Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formule :C19H28N4O4SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :408.52Conessine hydrobromide
CAS :Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Formule :C24H41BrN2Couleur et forme :SolidMasse moléculaire :437.51Diphenhydramine hydrochloride
CAS :DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.Formule :C17H22ClNODegré de pureté :99.84%Couleur et forme :Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Masse moléculaire :291.82Dalcotidine
CAS :Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.Formule :C18H29N3O2Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :319.44Ref: TM-T31195
1mg63,00€5mg140,00€10mg200,00€25mg324,00€50mg470,00€100mg662,00€200mg893,00€1mL*10mM (DMSO)140,00€Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormule :C26H27N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.51Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Couleur et forme :Odour SolidOxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.Formule :C20H23N5O5SDegré de pureté :97.34%Couleur et forme :SoildMasse moléculaire :445.49Bodilisant
CAS :Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Formule :C27H34BF2N3OCouleur et forme :SolidMasse moléculaire :465.4Nizatidine
CAS :Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Formule :C12H21N5O2S2Degré de pureté :98.39% - 99.43%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :331.46Cetirizine Impurity C
CAS :Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formule :C21H25ClN2O3Couleur et forme :SolidMasse moléculaire :388.89Vapitadine
CAS :Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formule :C17H20N4ODegré de pureté :99.77% - 99.86%Couleur et forme :SoildMasse moléculaire :296.37Cetirizine Impurity C dihydrochloride
CAS :Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formule :C21H27Cl3N2O3Couleur et forme :SolidMasse moléculaire :461.81H4R antagonist 3
CAS :H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFormule :C19H21ClN4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :372.924-Methylhistamine
CAS :4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFormule :C6H11N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :125.17Methimepip dihydrobromide
CAS :Methimepip dihydrobromide is a selective H3R agonist.Formule :C10H19Br2N3Couleur et forme :SolidMasse moléculaire :341.091Alcaftadine carboxylic acid
CAS :Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Formule :C19H21N3O2Couleur et forme :SolidMasse moléculaire :323.39Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS
Couleur et forme :Odour SolidDexchlorpheniramine free base
CAS :Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Formule :C16H19ClN2Degré de pureté :98%Couleur et forme :Oily Liquid SolidMasse moléculaire :274.79JNJ-10181457 (hydrochloride)
CAS :JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormule :C20H30Cl2N2OCouleur et forme :SolidMasse moléculaire :385.37Levocarnitine propionate hydrochloride
CAS :Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formule :C10H20ClNO4Degré de pureté :90% - 99.77%Couleur et forme :SolidMasse moléculaire :253.72(S)-Azelastine hydrochloride
CAS :(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formule :C22H25Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.363-hydroxy Desloratidine
CAS :3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Formule :C19H19ClN2OCouleur et forme :SolidMasse moléculaire :326.82(+)-Dropropizine
CAS :(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Formule :C13H20N2O2Degré de pureté :>99.99%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.31Cetirizine Impurity D
CAS :Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Formule :C30H28Cl2N2Couleur et forme :SolidMasse moléculaire :487.46Cetirizine methyl ester
CAS :Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Formule :C22H27ClN2O3Couleur et forme :SolidMasse moléculaire :402.91AM-0466
CAS :AM-0466 has a wide range of applications in life science related research.Formule :C27H19F3N4O4SCouleur et forme :SolidMasse moléculaire :552.52Oxmetidine
CAS :Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Formule :C19H21N5O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :399.47Ref: TM-T68122
1mg358,00€5mg848,00€10mg1.153,00€25mg1.693,00€50mg2.313,00€100mg3.115,00€500mg6.255,00€Alimemazine D6
CAS :Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.48Antazoline phosphate
CAS :Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formule :C17H22N3O4PDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :363.35
