Récepteur de l'histamine
Les récepteurs de l'histamine sont des GPCR qui médiatisent les effets de l'histamine, une amine biogène impliquée dans les réponses immunitaires, la sécrétion d'acide gastrique et la neurotransmission. Il existe quatre sous-types de récepteurs de l'histamine (H1, H2, H3 et H4), chacun jouant des rôles distincts dans les réactions allergiques, la fonction gastrique et l'activité du système nerveux central. Les antagonistes des récepteurs de l'histamine sont largement utilisés dans le traitement des allergies, des ulcères gastriques et du mal des transports. Chez CymitQuimica, nous offrons une sélection complète de modulateurs de récepteurs de l'histamine de haute qualité pour soutenir vos recherches en immunologie, gastroentérologie et neuropharmacologie.
385 produits trouvés pour "Récepteur de l'histamine"
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Hydroxyzine D8
CAS :Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formule :C21H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.95Alimemazine D6
CAS :Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.481-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS :MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formule :C6H9ClN2O2Couleur et forme :SolidMasse moléculaire :176.601Tiotidine
CAS :Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formule :C10H16N8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.42Acrivastine D7
CAS :Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.Formule :C22H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.48Fexofenadine-d6
CAS :Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formule :C32H39NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.69Emedastine Difumarate
CAS :Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formule :C25H34N4O9Couleur et forme :SolidMasse moléculaire :534.56Diphenylpyraline
CAS :Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Formule :C19H23NOCouleur et forme :SolidMasse moléculaire :281.39Gizzerosine
CAS :Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.Formule :C11H20N4O2Couleur et forme :SolidMasse moléculaire :240.3WZ4141
CAS :WZ4141 is an intermediate in compound synthesis.Formule :C16H13N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.29Doxepin D3 Hydrochloride
CAS :Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 andFormule :C19H22ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.86Cetirizine D8
CAS :Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formule :C21H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.94Cetirizine D4
CAS :Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formule :C21H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.91Clobenpropit dihydrobromide
CAS :Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)Formule :C14H19Br2ClN4SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :470.7Antazoline
CAS :Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formule :C17H19N3Degré de pureté :≥95%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :265.35Betahistine EP Impurity C
CAS :Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formule :C15H19N3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :241.33Fenspiride
CAS :Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.Formule :C15H20N2O2Couleur et forme :SolidMasse moléculaire :260.33Emedastine
CAS :Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.Formule :C17H26N4ODegré de pureté :97.1% - 97.76%Couleur et forme :OilMasse moléculaire :302.41Ref: TM-T3979
1mg34,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg109,00€25mg177,00€50mg264,00€100mg394,00€500mg883,00€Fexofenadine hydrochloride
CAS :Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Formule :C32H39NO4·HClDegré de pureté :99.39% - ≥95%Couleur et forme :SolidMasse moléculaire :538.13Psoralenoside
CAS :Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formule :C17H18O9Degré de pureté :99.03% - 99.49%Couleur et forme :SolidMasse moléculaire :366.32Ref: TM-TN1008
1mg90,00€2mg132,00€5mg215,00€1mL*10mM (DMSO)222,00€10mg344,00€25mg568,00€50mg800,00€100mg1.063,00€Conessine
CAS :Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.Formule :C24H40N2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :356.59Chlorpheniramine
CAS :Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.Formule :C16H19ClN2Couleur et forme :SolidMasse moléculaire :274.79Pemirolast
CAS :Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formule :C10H8N6OCouleur et forme :SolidMasse moléculaire :228.21Hydroxyzine
CAS :Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formule :C21H27ClN2O2Degré de pureté :99.54% - ≥95%Couleur et forme :Oil SolidMasse moléculaire :374.9Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3SCH-37370
CAS :SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formule :C21H21ClN2ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :352.86Ref: TM-T19686
1mg48,00€5mg89,00€1mL*10mM (DMSO)90,00€10mg115,00€25mg195,00€50mg290,00€100mg393,00€200mg520,00€H4 Receptor antagonist 1
CAS :H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formule :C16H17ClN4ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :316.79GSK189254A
CAS :GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formule :C21H25N3O2Degré de pureté :98.71% - 99.858%Couleur et forme :SolidMasse moléculaire :351.44Ref: TM-TQ0066
1mg50,00€1mL*10mM (DMSO)64,00€5mg84,00€10mg114,00€25mg205,00€50mg333,00€100mg477,00€200mg690,00€S 38093
CAS :S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formule :C17H24N2O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :288.38Ref: TM-T4099
2mg35,00€5mg50,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg124,00€50mg198,00€100mg316,00€200mg442,00€Bilastine
CAS :Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFormule :C28H37N3O3Degré de pureté :99.86% - >99.99%Couleur et forme :SolidMasse moléculaire :463.61Triprolidine hydrochloride
CAS :Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formule :C19H23ClN2Couleur et forme :SolidMasse moléculaire :314.852Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Niaprazine
CAS :Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Decloxizine
CAS :Decloxizine is a H1 receptor antagonistFormule :C21H28N2O2Degré de pureté :99.53%Couleur et forme :White Or Similar To White PowderMasse moléculaire :340.46Clobenpropit 2HBr
CAS :Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formule :C14H17ClN4SCouleur et forme :SolidMasse moléculaire :308.83Lodoxamide
CAS :Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formule :C11H6ClN3O6Degré de pureté :99.13% - 99.96%Couleur et forme :SolidMasse moléculaire :311.63Osthole
CAS :Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Formule :C15H16O3Degré de pureté :99.93% - 99.96%Couleur et forme :Fine White PowderMasse moléculaire :244.29HTMT dimaleate
CAS :HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formule :C27H33F3N4O9Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :614.57Triprolidine
CAS :Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formule :C19H22N2Couleur et forme :SolidMasse moléculaire :278.39Acitazanolast
CAS :Acitazanolast (WP-871) is an anti-allergic drug candidate.Formule :C9H7N5O3Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :233.182-Pyridylethylamine dihydrochloride
CAS :2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formule :C7H12Cl2N2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :195.09Betahistine
CAS :Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formule :C8H12N2Degré de pureté :99.87% - 99.87%Couleur et forme :Yellowish Liquid Liquid LiquidMasse moléculaire :136.19Dioxopromethazine
CAS :Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formule :C17H20N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :316.42Buclizine
CAS :Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formule :C28H33ClN2Couleur et forme :SolidMasse moléculaire :433.03Desloratadine
CAS :Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.Formule :C19H19ClN2Degré de pureté :99.79% - >99.99%Couleur et forme :SolidMasse moléculaire :310.82C-Type Natriuretic Peptide (CNP) (1-22), human
CAS :C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formule :C93H157N27O28S3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :2197.6Ref: TM-TP1187
500µg84,00€1mg113,00€5mg391,00€10mg623,00€25mg895,00€50mg1.198,00€100mg1.611,00€200mg2.152,00€Fexofenadine
CAS :Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formule :C32H39NO4Degré de pureté :99.35%Couleur et forme :White To Off-White SolidMasse moléculaire :501.66Tiaramide hydrochloride
CAS :Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formule :C15H19Cl2N3O3SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :392.3Ref: TM-T28972
1mg66,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg177,00€25mg299,00€50mg447,00€100mg623,00€200mg882,00€JNJ-5207852 dihydrochloride
CAS :JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormule :C20H34Cl2N2ODegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :389.4
