Récepteur opioïde
Les récepteurs opioïdes sont un groupe de récepteurs couplés aux protéines G qui médiatisent les effets des opioïdes endogènes et exogènes. Ces récepteurs jouent un rôle central dans la modulation de la douleur, la régulation de l'humeur et les comportements addictifs. Les agonistes et antagonistes des récepteurs opioïdes sont largement utilisés dans la gestion de la douleur et le traitement des dépendances, ainsi que dans la recherche sur les troubles neurologiques et psychiatriques. Chez CymitQuimica, nous offrons une sélection complète de modulateurs des récepteurs opioïdes de haute qualité pour soutenir vos recherches en neurobiologie, gestion de la douleur et thérapie contre les addictions.
297 produits trouvés pour "Récepteur opioïde"
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Moguisteine
CAS :<p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>Formule :C16H21NO5SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :339.41Trimebutine maleate
CAS :<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Formule :C26H33NO9Degré de pureté :99.76% - 99.98%Couleur et forme :White SolidMasse moléculaire :503.55Meptazinol hydrochloride
CAS :<p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>Formule :C15H23NO·HClDegré de pureté :99.75%Couleur et forme :White SolidMasse moléculaire :269.81Matrine
CAS :<p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>Formule :C15H24N2ODegré de pureté :97.16% - >99.99%Couleur et forme :SolidMasse moléculaire :248.36CP 866087
CAS :<p>CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.</p>Formule :C24H30N2O3SDegré de pureté :99.22% - 99.74%Couleur et forme :SolidMasse moléculaire :426.57Naltrexone hydrochloride
CAS :<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Formule :C20H24ClNO4Degré de pureté :98.72% - 99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :377.862Loperamide hydrochloride
CAS :<p>Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.</p>Formule :C29H34Cl2N2O2Degré de pureté :99.91% - >99.99%Couleur et forme :Crystals Practically Insoluble In WaterMasse moléculaire :513.50Alvimopan
CAS :<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Formule :C25H32N2O4Degré de pureté :99.47% - 99.78%Couleur et forme :SolidMasse moléculaire :424.53Samidorphan HCl
CAS :<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formule :C21H27ClN2O4Degré de pureté :96.79% - 97.85%Couleur et forme :SoildMasse moléculaire :406.9BTRX-335140
CAS :<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Formule :C25H32FN5O2Degré de pureté :98% - 99.89%Couleur et forme :SolidMasse moléculaire :453.55Apitegromab
CAS :<p>Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including</p>Degré de pureté :95% - 97.59% (SDS-PAGE); 99.78% (SEC-HPLC)Couleur et forme :LiquidSinomenine hydrochloride
CAS :<p>Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.</p>Formule :C19H24ClNO4Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :365.851LY2940094
CAS :<p>LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.</p>Formule :C22H23ClF2N4O2SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :480.96ZT 52656A hydrochloride
CAS :<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Formule :C19H26ClF3N2ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :390.87Nocistatin
CAS :<p>Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.</p>Formule :C32H56N10O12Couleur et forme :SolidMasse moléculaire :772.85SB 205607 dihydrobromide
CAS :<p>non-peptide δ1 opioid receptor agonist</p>Formule :C23H24N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.45Valorphin
CAS :<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Formule :C44H61N9O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :892.01β-Endorphin (1-27) (human)
CAS :<p>β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,</p>Formule :C139H217N33O40SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3022.47CSD-CH2(1,8)-NH2
<p>CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.</p>Formule :C76H125N25O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1693.09Adrenorphin
CAS :<p>Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formule :C44H69N15O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :984.18N-Phenethylnoroxymorphone
CAS :<p>N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.</p>Formule :C24H25NO4Couleur et forme :SolidMasse moléculaire :391.46AT-121 hydrochloride
CAS :<p>AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.</p>Formule :C24H39ClN4O3SDegré de pureté :97.28% - >99.99%Couleur et forme :SolidMasse moléculaire :499.11(S,S)-J-113397
CAS :<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Formule :C24H37N3O2Couleur et forme :SolidMasse moléculaire :399.57Leumorphin, human
CAS :<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Formule :C150H224N42O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3351.64Dynorphin B (1-9)
CAS :<p>Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selective</p>Formule :C54H78N16O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1143.3HINT1-IN-1
<p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>Formule :C23H24N8O5Couleur et forme :SolidMasse moléculaire :492.49DPDPE
CAS :<p>DPDPE is selective δ-opioid receptor agonist peptide.</p>Formule :C30H39N5O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :645.79Frakefamide TFA
<p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>Formule :C32H35F4N5O7Couleur et forme :SolidMasse moléculaire :677.64Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Formule :C44H59N11O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :901.43Helianorphin-19
<p>Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.</p>Couleur et forme :Liquidβ-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Formule :C141H221N33O42SDegré de pureté :96.52%Couleur et forme :SolidMasse moléculaire :3082.52Trimebutine
CAS :<p>Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid</p>Formule :C22H29NO5Degré de pureté :98.13% - 99.49%Couleur et forme :SolidMasse moléculaire :387.47CTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Formule :C52H71N11O13S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Formule :C84H142N32O23Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :1968.23β-Endorphin (6-31), human
CAS :<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Formule :C131H218N34O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2909.38LY255582
CAS :<p>LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,</p>Formule :C22H35NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.52Neuropeptide AF (human)
CAS :<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Formule :C90H132N26O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1978.17Naldemedine
CAS :<p>Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.</p>Formule :C32H34N4O6Couleur et forme :SolidMasse moléculaire :570.64(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS :<p>E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioid</p>Formule :C50H81N15O9Couleur et forme :SolidMasse moléculaire :1036.27BPR1M97
CAS :<p>BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.</p>Formule :C18H18Cl2N2ODegré de pureté :98.78% - 99.95%Couleur et forme :SolidMasse moléculaire :349.25Ac-RYYRIK-NH2
CAS :<p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>Formule :C44H70N14O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :939.12Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Degré de pureté :99.89%Couleur et forme :Soildβ-Endorphin, equine
CAS :<p>Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.</p>Formule :C154H248N42O44SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3423.94difelikefalin acetate(1024828-77-0 Free base)
CAS :<p>is a ketone and a building block.</p>Formule :C38H57N7O8Degré de pureté :96.94%Couleur et forme :SolidMasse moléculaire :739.9[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Formule :C31H43N5O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.65[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formule :C63H103FN22O17Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :1459.63Axelopran
CAS :<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Formule :C26H39N3O4Couleur et forme :SolidMasse moléculaire :457.61β-Lipotropin (60-65)
CAS :<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Formule :C33H47N9O8SCouleur et forme :SolidMasse moléculaire :729.85Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Formule :C46H66N10O12S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :1015.21KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Formule :C38H38N2O5Couleur et forme :SolidMasse moléculaire :602.72Clocinnamox mesylate
CAS :<p>Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).</p>Formule :C30H33ClN2O7SCouleur et forme :SolidMasse moléculaire :601.11DALDA TFA
<p>DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.</p>Formule :C30H45N9O5·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :611.74 (free base)Dynorphin B (1-13) (TFA)
<p>Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .</p>Formule :C76H116N21F3O19Couleur et forme :SolidMasse moléculaire :1684.86KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Formule :C21H25N3Couleur et forme :SolidMasse moléculaire :319.44β-Endorphin, equine TFA
<p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>Formule :C156H249F3N42O46SCouleur et forme :SolidMasse moléculaire :3537.96Akuammicine
CAS :<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Formule :C20H22N2O2Couleur et forme :SolidMasse moléculaire :322.408Nociceptin(1-7)
CAS :<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formule :C31H41N7O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :655.709[(pF)Phe4]Nociceptin(1-13)NH2
CAS :<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Formule :C61H99FN22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1399.6Ac-RYYRWK-NH2 TFA
CAS :<p>Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.</p>Formule :C51H70F3N15O11Couleur et forme :SolidMasse moléculaire :1126.21ICI 174,864
CAS :<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Formule :C38H53N5O7Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :691.87PL-017
CAS :<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Formule :C29H37N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :535.64[Met5]-Enkephalin, amide
CAS :<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Formule :C27H36N6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.68MT-7716 hydrochloride
CAS :<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Formule :C27H29ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477N-Acetyl-α-Endorphin
CAS :N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formule :C79H122N18O27SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1787.98PIPE-3297
<p>PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.</p>Formule :C23H30N2OMasse moléculaire :350.23581[Nphe1]Nociceptin(1-13)NH2
CAS :<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Formule :C61H100N22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1381.6SNC 80
CAS :<p>SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.</p>Formule :C28H39N3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :449.63[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS :'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'Formule :C76H128N24O15Couleur et forme :SolidMasse moléculaire :1617.98CJ-15208
CAS :<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formule :C34H35N5O4Couleur et forme :SolidMasse moléculaire :577.67U-54494A hydrochloride
CAS :<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Formule :C18H25Cl3N2OCouleur et forme :SolidMasse moléculaire :391.76Ac-RYYRWK-NH2
CAS :<p>Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.</p>Formule :C49H69N15O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1012.17Gluten Exorphin B5
CAS :<p>Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.</p>Formule :C30H38N6O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.66Herkinorin
CAS :<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formule :C28H30O8Couleur et forme :SolidMasse moléculaire :494.53Dermorphin
CAS :<p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>Formule :C40H50N8O10Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :802.87[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Formule :C63H101F3N22O17Couleur et forme :SolidMasse moléculaire :1495.61Dynorphin B (1-13)
CAS :Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Formule :C74H115N21O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.84β-Endorphin (rat)
CAS :<p>β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.</p>Formule :C157H254N42O44SCouleur et forme :SolidMasse moléculaire :3466.07CTAP
CAS :<p>Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.</p>Formule :C51H69N13O11S2Degré de pureté :98%Couleur et forme :White Solid/PowderMasse moléculaire :1104.32Orphanin FQ(1-11)
CAS :<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formule :C49H75N15O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1098.2Ro 64-6198
CAS :<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Formule :C26H31N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54β-Naltrexamine dihydrochloride
CAS :<p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>Formule :C20H28Cl2N2O3Degré de pureté :95.98%Couleur et forme :SoildMasse moléculaire :415.35Biphalin TFA
CAS :<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Formule :C46H56N10O10·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :909.00 (free base)CTOP
CAS :<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Formule :C50H67N11O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1062.28Cebranopadol hemicitrate
CAS :<p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>Couleur et forme :Solid[DPro10] Dynorphin A (1-11)acetate,porcine
<p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>Formule :C65H107N21O15Degré de pureté :99.05%Couleur et forme :SoildMasse moléculaire :1422.7Nociceptin (1-13), amide
CAS :<p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>Formule :C61H100N22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1381.59UFP-101
CAS :<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formule :C82H138N32O21Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1908.19[Arg14,Lys15]Nociceptin
CAS :<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Formule :C82H137N31O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1909.18N-Desmethyl Loperamide
CAS :<p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>Formule :C28H31ClN2O2Couleur et forme :SolidMasse moléculaire :463.01MT-7716 free base
CAS :<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Formule :C27H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.54Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Couleur et forme :Odour SolidBAM-22P
CAS :<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Formule :C130H184N38O31S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2839.22TAN67
CAS :<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Formule :C23H26Br2N2OCouleur et forme :SolidMasse moléculaire :506.282Boc-ypgflt(O-tbu)
CAS :<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Formule :C44H64N6O11Couleur et forme :SolidMasse moléculaire :853.01N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Formule :C36H40N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Formule :C32H45N5OCouleur et forme :SolidMasse moléculaire :515.73(Rac)-SNC80
CAS :<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Formule :C28H39N3O2Couleur et forme :SolidMasse moléculaire :449.63DAMGO (TFA)
CAS :<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Formule :C28H36F3N5O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.61Deltorphin
CAS :<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Formule :C44H62N10O10S2Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :955.15AP-238
CAS :<p>AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.</p>Formule :C18H26N2OCouleur et forme :SolidMasse moléculaire :286.41
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