Récepteur opioïde
Les récepteurs opioïdes sont un groupe de récepteurs couplés aux protéines G qui médiatisent les effets des opioïdes endogènes et exogènes. Ces récepteurs jouent un rôle central dans la modulation de la douleur, la régulation de l'humeur et les comportements addictifs. Les agonistes et antagonistes des récepteurs opioïdes sont largement utilisés dans la gestion de la douleur et le traitement des dépendances, ainsi que dans la recherche sur les troubles neurologiques et psychiatriques. Chez CymitQuimica, nous offrons une sélection complète de modulateurs des récepteurs opioïdes de haute qualité pour soutenir vos recherches en neurobiologie, gestion de la douleur et thérapie contre les addictions.
297 produits trouvés pour "Récepteur opioïde"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Leumorphin, human
CAS :<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Formule :C150H224N42O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3351.64Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Formule :C46H66N10O12S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :1015.21CJ-15208
CAS :<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formule :C34H35N5O4Couleur et forme :SolidMasse moléculaire :577.67N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Formule :C36H40N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :652.74N-Acetyl-α-Endorphin
CAS :N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formule :C79H122N18O27SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1787.98Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Formule :C32H45N5OCouleur et forme :SolidMasse moléculaire :515.73Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Degré de pureté :99.89%Couleur et forme :SoildCTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Formule :C52H71N11O13S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Formule :C84H142N32O23Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS :<p>is a ketone and a building block.</p>Formule :C38H57N7O8Degré de pureté :96.94%Couleur et forme :SolidMasse moléculaire :739.9[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formule :C63H103FN22O17Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :1459.63[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Formule :C31H43N5O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.65β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Formule :C141H221N33O42SDegré de pureté :96.52%Couleur et forme :SolidMasse moléculaire :3082.52β-Endorphin (6-31), human
CAS :<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Formule :C131H218N34O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2909.38Deltorphin
CAS :<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Formule :C44H62N10O10S2Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :955.15Porcine dynorphin A(1-13)
CAS :Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.Formule :C75H126N24O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1603.95Loperamide phenyl
CAS :<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Formule :C35H37ClN2O2Couleur et forme :SolidMasse moléculaire :553.14Endomorphin 2 TFA
CAS :<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Formule :C34H38F3N5O7Couleur et forme :SolidMasse moléculaire :685.69BMS-986121
CAS :<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Formule :C15H9Cl2N3O2SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :366.22[Leu5]-Enkephalin
CAS :<p>[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM</p>Formule :C28H37N5O7Degré de pureté :99.87% - 99.88%Couleur et forme :SolidMasse moléculaire :555.62Alvimopan dihydrate (LY246736 dihydrate)
CAS :<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Formule :C25H36N2O6Couleur et forme :SolidMasse moléculaire :460.56Asimadoline
CAS :<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Formule :C27H30N2O2Couleur et forme :SolidMasse moléculaire :414.54BAN ORL 24 dihydrochloride
CAS :<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Formule :C27H37Cl2N3O2Degré de pureté :95.03%Couleur et forme :SolidMasse moléculaire :506.51Dermorphin TFA
CAS :<p>Dermorphin TFA is a new class of opioids-like peptides</p>Formule :C42H51F3N8O12Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :916.89Deltorphin I
CAS :<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Formule :C37H52N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :768.86Sec-O-Glucosylhamaudol
CAS :<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Formule :C21H26O10Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :438.43BRL 52537 hydrochloride
CAS :<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Formule :C18H25Cl3N2ODegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :391.76DPDPE TFA (88373-73-3 free base)
CAS :<p>DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.</p>Formule :C32H40F3N5O9S2Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :759.81Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Formule :C31H41N7O9Degré de pureté :98.92%Couleur et forme :SoildMasse moléculaire :655.7Aticaprant
CAS :<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Formule :C26H27FN2O2Degré de pureté :99.53% - 99.93%Couleur et forme :SolidMasse moléculaire :418.5BMS986187
CAS :<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Formule :C31H34O4Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :470.6Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Formule :C46H74N14O11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :999.17[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Formule :C29H37F3N6O8SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :686.7LY2940094 tartrate
CAS :<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Formule :C26H29ClF2N4O8SCouleur et forme :SolidMasse moléculaire :631.04MCOPPB triHydrochloride
CAS :<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Formule :C26H43Cl3N4Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :518.01Salvinorin A
CAS :<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Formule :C23H28O8Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :432.46Naloxegol oxalate
CAS :<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Formule :C36H55NO15Degré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :741.83Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formule :C51H73N15O11Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :1072.22Nalmefene hydrochloride
CAS :<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Formule :C21H26ClNO3Degré de pureté :98% - 99.85%Couleur et forme :SolidMasse moléculaire :375.89Difelikefalin acetate
CAS :<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Formule :C38H57N7O8Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :739.9AR-M 1000390 hydrochloride
CAS :<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Formule :C23H29ClN2ODegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :384.94Tyr-Gly-Gly-Phe-Met-OH
CAS :<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formule :C27H35N5O7SDegré de pureté :≥95%Couleur et forme :White Lyophilised SolidMasse moléculaire :573.66b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formule :C25H31N3O7Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :485.53Endomorphin 2
CAS :<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Formule :C32H37N5O5Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :571.67Methylnaltrexone bromide
CAS :Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formule :C21H26BrNO4Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :436.35EST73502 HCl
CAS :<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formule :C19H27ClF2N2O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :388.88JTC-801
CAS :<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formule :C26H25N3O2·HClDegré de pureté :99.27% - 99.59%Couleur et forme :SolidMasse moléculaire :447.96BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Formule :C132H188N38O33S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :2899.27BMS-986122
CAS :<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Formule :C16H15BrClNO3S2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :448.78ADL-5859
CAS :<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Formule :C24H28N2O3·HClDegré de pureté :98.78% - 99.11%Couleur et forme :SolidMasse moléculaire :428.95N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.66Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formule :C51H79N15O16Degré de pureté :95.54%Couleur et forme :SolidMasse moléculaire :1158.26Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Formule :C101H159N31O25Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :2207.58(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Formule :C33H46N6O10Degré de pureté :94.17%Couleur et forme :SoildMasse moléculaire :686.75Sinomenine
CAS :<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formule :C19H23NO4Degré de pureté :99.02% - 99.73%Couleur et forme :White PowderMasse moléculaire :329.39Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Formule :C77H130N24O17Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :1664Alvimopan monohydrate
CAS :<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formule :C25H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.55Endomorphin 1
CAS :<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Formule :C34H38N6O5Degré de pureté :95.92%Couleur et forme :Solid (Solid Powder )Masse moléculaire :610.7Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Formule :C76H119N21O19Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :1630.89ADL-5747 (HCl)
CAS :<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formule :C24H29ClN2O3Couleur et forme :SolidMasse moléculaire :428.95Asimadoline hydrochloride
CAS :<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Formule :C27H31ClN2O2Degré de pureté :98.94% - 99.32%Couleur et forme :SolidMasse moléculaire :451.01PZM21
CAS :<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formule :C19H27N3O2SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :361.5MCOPPB
CAS :<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formule :C26H40N4Couleur et forme :SolidMasse moléculaire :408.62DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Formule :C28H36F3N5O8Degré de pureté :98.67% - 99.76%Couleur et forme :SolidMasse moléculaire :627.6BW-180C
CAS :<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Formule :C29H39N5O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :569.65GR 89696 free base
CAS :<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Formule :C19H25Cl2N3O3Couleur et forme :SolidMasse moléculaire :414.33EST73502 hydrochloride
CAS :<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Formule :C19H27ClF2N2O2Couleur et forme :SolidMasse moléculaire :388.88CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Formule :C53H70F3N13O13S2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :1218.33BMS986188
CAS :<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Formule :C30H31BrO4Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :535.47Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Formule :C63H101F3N22O17Degré de pureté :97.64%Couleur et forme :SolidMasse moléculaire :1495.61Corydaline
CAS :<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Formule :C22H27NO4Degré de pureté :98.97% - 99.86%Couleur et forme :SolidMasse moléculaire :369.45Deltorphin 2
CAS :<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formule :C38H54N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :782.88Naloxegol (NKTR-118)
CAS :<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Formule :C34H53NO11Couleur et forme :SolidMasse moléculaire :651.78Bisacodyl
CAS :<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Formule :C22H19NO4Degré de pureté :99.45% - 99.78%Couleur et forme :Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMasse moléculaire :361.39GR103545
CAS :<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Formule :C23H29Cl2N3O7Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :530.4Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Formule :C59H95N19O14Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1294.53Gluten Exorphin C
CAS :<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Formule :C29H45N5O8Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :591.7Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formule :C51H68N12O13Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :1057.16LY2795050
CAS :<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Formule :C23H22ClN3O2Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :407.89N-Desmethylclozapine
CAS :<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8DAMGO
CAS :<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formule :C26H35N5O6Degré de pureté :98.83% - 99.92%Couleur et forme :SolidMasse moléculaire :513.59Leuphasyl TFA
CAS :<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Formule :C31H40F3N5O9Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :683.67Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formule :C50H72N15O15SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1326.26[D-Ala2]leucine-enkephalin
CAS :<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formule :C29H39N5O7Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :569.65Nociceptin
CAS :<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Formule :C79H129N27O22Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :1809.04[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Formule :C30H42N6O8Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :614.69GRT2932Q
CAS :<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Formule :C25H26ClN3OCouleur et forme :SolidMasse moléculaire :419.95BW 373U86
CAS :<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Formule :C27H37N3O2Couleur et forme :SolidMasse moléculaire :435.6TIPP
CAS :<p>TIPP is an agent of delta opioid antagonist.</p>Formule :C37H38N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :634.72ICI 154,129
CAS :<p>Selective δ opioid antagonist</p>Formule :C34H46N4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :638.82JTC-801 free base
CAS :<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Formule :C26H25N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.5ML 190
CAS :<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Formule :C27H32N6O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :488.58Diallyl G
CAS :<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Formule :C38H53N5O8Couleur et forme :SolidMasse moléculaire :707.86Loperamide oxide
CAS :<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Formule :C29H33ClN2O3Couleur et forme :SolidMasse moléculaire :493.04GSK1521498 free base
CAS :<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Formule :C24H20F2N4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :402.44CR-665 Acetate
CAS :<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Formule :C38H53N9O6Couleur et forme :SolidMasse moléculaire :731.899LY 164929
CAS :<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Formule :C28H41N5O4Couleur et forme :SolidMasse moléculaire :511.66ADL-5859 HCl
CAS :<p>ADL-5859 is a delta-opioid receptor agonist.</p>Formule :C24H28N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49GSK1521498 free base (hydrochloride)
CAS :<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Formule :C24H21ClF2N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.9SR8993
CAS :<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Formule :C25H37FN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.59
![[(pF)Phe4]Nociceptin(1-13)NH2 acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1885L1.webp&w=3840&q=75)
![[D-Ala2]leucine-enkephalin acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1367L.webp&w=3840&q=75)
![[Leu5]-Enkephalin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT7173.webp&w=3840&q=75)
![[Met5]-Enkephalin, amide TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1254.webp&w=3840&q=75)
![[D-Ala2]leucine-enkephalin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1367.webp&w=3840&q=75)
![[Leu5]-Enkephalin, amide acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1113L.webp&w=3840&q=75)
