Récepteur opioïde
Les récepteurs opioïdes sont un groupe de récepteurs couplés aux protéines G qui médiatisent les effets des opioïdes endogènes et exogènes. Ces récepteurs jouent un rôle central dans la modulation de la douleur, la régulation de l'humeur et les comportements addictifs. Les agonistes et antagonistes des récepteurs opioïdes sont largement utilisés dans la gestion de la douleur et le traitement des dépendances, ainsi que dans la recherche sur les troubles neurologiques et psychiatriques. Chez CymitQuimica, nous offrons une sélection complète de modulateurs des récepteurs opioïdes de haute qualité pour soutenir vos recherches en neurobiologie, gestion de la douleur et thérapie contre les addictions.
297 produits trouvés pour "Récepteur opioïde"
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LY2940094
CAS :<p>LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.</p>Formule :C22H23ClF2N4O2SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :480.96Sinomenine hydrochloride
CAS :<p>Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.</p>Formule :C19H24ClNO4Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :365.851Apitegromab
CAS :<p>Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including</p>Degré de pureté :95% - 97.59% (SDS-PAGE); 99.78% (SEC-HPLC)Couleur et forme :LiquidSamidorphan HCl
CAS :<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formule :C21H27ClN2O4Degré de pureté :96.79% - 97.85%Couleur et forme :SoildMasse moléculaire :406.9Naltrexone hydrochloride
CAS :<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Formule :C20H24ClNO4Degré de pureté :98.72% - 99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :377.862Meptazinol hydrochloride
CAS :<p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>Formule :C15H23NO·HClDegré de pureté :99.75%Couleur et forme :White SolidMasse moléculaire :269.81BTRX-335140
CAS :<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Formule :C25H32FN5O2Degré de pureté :98% - 99.89%Couleur et forme :SolidMasse moléculaire :453.55Moguisteine
CAS :<p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>Formule :C16H21NO5SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :339.41Matrine
CAS :<p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>Formule :C15H24N2ODegré de pureté :97.16% - >99.99%Couleur et forme :SolidMasse moléculaire :248.36Trimebutine maleate
CAS :<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Formule :C26H33NO9Degré de pureté :99.76% - 99.98%Couleur et forme :White SolidMasse moléculaire :503.55Loperamide hydrochloride
CAS :<p>Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.</p>Formule :C29H34Cl2N2O2Degré de pureté :99.91% - >99.99%Couleur et forme :Crystals Practically Insoluble In WaterMasse moléculaire :513.50Alvimopan
CAS :<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Formule :C25H32N2O4Degré de pureté :99.47% - 99.78%Couleur et forme :SolidMasse moléculaire :424.53ZT 52656A hydrochloride
CAS :<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Formule :C19H26ClF3N2ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :390.87CP 866087
CAS :<p>CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.</p>Formule :C24H30N2O3SDegré de pureté :99.22% - 99.74%Couleur et forme :SolidMasse moléculaire :426.57KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Formule :C21H25N3Couleur et forme :SolidMasse moléculaire :319.44DPDPE
CAS :<p>DPDPE is selective δ-opioid receptor agonist peptide.</p>Formule :C30H39N5O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :645.79UFP-101
CAS :<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formule :C82H138N32O21Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1908.19Dermorphin
CAS :<p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>Formule :C40H50N8O10Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :802.87SNC 80
CAS :<p>SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.</p>Formule :C28H39N3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :449.63[DPro10] Dynorphin A (1-11)acetate,porcine
<p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>Formule :C65H107N21O15Degré de pureté :99.05%Couleur et forme :SoildMasse moléculaire :1422.7Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Couleur et forme :Odour SolidDuP 747 HCl
CAS :<p>DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.</p>Formule :C24H29Cl3N2O2Degré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :483.86β-Endorphin, equine TFA
<p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>Formule :C156H249F3N42O46SCouleur et forme :SolidMasse moléculaire :3537.96Frakefamide TFA
<p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>Formule :C32H35F4N5O7Couleur et forme :SolidMasse moléculaire :677.644-Hydroxy-1-(2-phenylethyl)piperidine
CAS :<p>4-Hydroxy-1-(2-phenylethyl)piperidine is a synthetic ligand for muscarinic acetylcholine receptors (mAChR) or non-opioid intracellular sigma-1 receptors (σ1 receptors). It serves as a metabolite of the opioid compounds furanylfentanyl and 4-fluoroisobutyryl fentanyl (FIBF).</p>Formule :C13H19NOCouleur et forme :SolidMasse moléculaire :205.3U-48520
CAS :<p>U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.</p>Formule :C16H23ClN2OCouleur et forme :SolidMasse moléculaire :294.82ICI 174,864
CAS :<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Formule :C38H53N5O7Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :691.87DBPR116
CAS :<p>DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.</p>Formule :C19H18FNO3SCouleur et forme :SolidMasse moléculaire :359.42AH 7959
CAS :<p>AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.</p>Formule :C19H26Cl2N2OCouleur et forme :SolidMasse moléculaire :369.33Biphalin TFA
CAS :<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Formule :C46H56N10O10·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :909.00 (free base)Ac-RYYRIK-NH2
CAS :<p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>Formule :C44H70N14O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :939.12Orphine
CAS :<p>Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.</p>Formule :C20H23N3OCouleur et forme :SolidMasse moléculaire :321.42AH 7563
CAS :<p>AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.</p>Formule :C16H24N2OCouleur et forme :SolidMasse moléculaire :260.38Corynantheidine
CAS :<p>Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.</p>Formule :C22H28N2O3Couleur et forme :SolidMasse moléculaire :368.47Axelopran
CAS :<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Formule :C26H39N3O4Couleur et forme :SolidMasse moléculaire :457.61DAMGO (TFA)
CAS :<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Formule :C28H36F3N5O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :627.61Fluorphine
CAS :<p>Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.</p>Formule :C20H22FN3OCouleur et forme :SolidMasse moléculaire :339.41KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Formule :C38H38N2O5Couleur et forme :SolidMasse moléculaire :602.72HINT1-IN-1
<p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>Formule :C23H24N8O5Couleur et forme :SolidMasse moléculaire :492.49Akuammicine
CAS :<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Formule :C20H22N2O2Couleur et forme :SolidMasse moléculaire :322.408Nociceptin(1-7)
CAS :<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formule :C31H41N7O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :655.709[(pF)Phe4]Nociceptin(1-13)NH2
CAS :<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Formule :C61H99FN22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1399.6Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Formule :C44H59N11O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :901.43KOR agonist 3
<p>KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.</p>Formule :C24H24N2O3Couleur et forme :SolidMasse moléculaire :388.46PL-017
CAS :<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Formule :C29H37N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :535.64(-)-9-Hydroxycorynantheidine
CAS :<p>(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.</p>Formule :C22H28N2O4Couleur et forme :SolidMasse moléculaire :384.47Ro 64-6198
CAS :<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Formule :C26H31N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54Orphanin FQ(1-11)
CAS :<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formule :C49H75N15O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1098.2Piperidylthiambutene hydrochloride
CAS :<p>Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.</p>Formule :C17H22ClNS2Couleur et forme :SolidMasse moléculaire :339.95[Nphe1]Nociceptin(1-13)NH2
CAS :<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Formule :C61H100N22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1381.6U-54494A hydrochloride
CAS :<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Formule :C18H25Cl3N2OCouleur et forme :SolidMasse moléculaire :391.76AH 8529
CAS :<p>AH 8529 is an orally active opioid compound with analgesic properties.</p>Formule :C16H23ClN2OCouleur et forme :SolidMasse moléculaire :294.82Gluten Exorphin B5
CAS :<p>Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.</p>Formule :C30H38N6O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.66Herkinorin
CAS :<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formule :C28H30O8Couleur et forme :SolidMasse moléculaire :494.53AH 8532
CAS :<p>AH 8532 is an opioid compound with analgesic effects and is effective in inhibiting the quinone-induced writhing response in mice, with an oral ED50 of 16 mg/kg.</p>Formule :C16H23ClN2OCouleur et forme :SolidMasse moléculaire :294.82Dynorphin B (1-13)
CAS :Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Formule :C74H115N21O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.84Neuropeptide AF (human)
CAS :<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Formule :C90H132N26O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1978.17CTAP
CAS :<p>Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.</p>Formule :C51H69N13O11S2Degré de pureté :98%Couleur et forme :White Solid/PowderMasse moléculaire :1104.32R-6890
CAS :<p>R-6890 is an opioid compound with analgesic properties.</p>Formule :C21H24ClN3OCouleur et forme :SolidMasse moléculaire :369.89β-Naltrexamine dihydrochloride
CAS :<p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>Formule :C20H28Cl2N2O3Degré de pureté :95.98%Couleur et forme :SoildMasse moléculaire :415.35N-Phenethylnoroxymorphone
CAS :<p>N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.</p>Formule :C24H25NO4Couleur et forme :SolidMasse moléculaire :391.46CTOP
CAS :<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Formule :C50H67N11O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1062.28Cebranopadol hemicitrate
CAS :<p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>Couleur et forme :SolidAP-238
CAS :<p>AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.</p>Formule :C18H26N2OCouleur et forme :SolidMasse moléculaire :286.41MT-7716 free base
CAS :<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Formule :C27H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.54LY255582
CAS :<p>LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,</p>Formule :C22H35NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.52BAM-22P
CAS :<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Formule :C130H184N38O31S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2839.22TAN67
CAS :<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Formule :C23H26Br2N2OCouleur et forme :SolidMasse moléculaire :506.282Boc-ypgflt(O-tbu)
CAS :<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Formule :C44H64N6O11Couleur et forme :SolidMasse moléculaire :853.01Trimebutine
CAS :<p>Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid</p>Formule :C22H29NO5Degré de pureté :98.13% - 99.49%Couleur et forme :SolidMasse moléculaire :387.47(Rac)-SNC80
CAS :<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Formule :C28H39N3O2Couleur et forme :SolidMasse moléculaire :449.63Ac-RYYRWK-NH2
CAS :<p>Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.</p>Formule :C49H69N15O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1012.17Naldemedine
CAS :<p>Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.</p>Formule :C32H34N4O6Couleur et forme :SolidMasse moléculaire :570.64AT-121 hydrochloride
CAS :<p>AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.</p>Formule :C24H39ClN4O3SDegré de pureté :97.28% - >99.99%Couleur et forme :SolidMasse moléculaire :499.11[Arg14,Lys15]Nociceptin
CAS :<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Formule :C82H137N31O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1909.18N-Desmethyl Loperamide
CAS :<p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>Formule :C28H31ClN2O2Couleur et forme :SolidMasse moléculaire :463.01β-Endorphin, equine
CAS :<p>Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.</p>Formule :C154H248N42O44SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3423.94MT-7716 hydrochloride
CAS :<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Formule :C27H29ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477(S,S)-J-113397
CAS :<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Formule :C24H37N3O2Couleur et forme :SolidMasse moléculaire :399.57Clocinnamox mesylate
CAS :<p>Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).</p>Formule :C30H33ClN2O7SCouleur et forme :SolidMasse moléculaire :601.11Adrenorphin
CAS :<p>Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formule :C44H69N15O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :984.18[Met5]-Enkephalin, amide
CAS :<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Formule :C27H36N6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :572.68Valorphin
CAS :<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Formule :C44H61N9O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :892.01(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS :<p>E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioid</p>Formule :C50H81N15O9Couleur et forme :SolidMasse moléculaire :1036.27[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Formule :C63H101F3N22O17Couleur et forme :SolidMasse moléculaire :1495.61Nocistatin
CAS :<p>Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.</p>Formule :C32H56N10O12Couleur et forme :SolidMasse moléculaire :772.85Helianorphin-19
<p>Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.</p>Couleur et forme :Liquidβ-Lipotropin (60-65)
CAS :<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Formule :C33H47N9O8SCouleur et forme :SolidMasse moléculaire :729.85[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS :<p>'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'</p>Formule :C76H128N24O15Couleur et forme :SolidMasse moléculaire :1617.98β-Endorphin (rat)
CAS :<p>β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.</p>Formule :C157H254N42O44SCouleur et forme :SolidMasse moléculaire :3466.07Dynorphin B (1-13) (TFA)
<p>Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .</p>Formule :C76H116N21F3O19Couleur et forme :SolidMasse moléculaire :1684.86Ac-RYYRWK-NH2 TFA
CAS :<p>Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.</p>Formule :C51H70F3N15O11Couleur et forme :SolidMasse moléculaire :1126.21Nociceptin (1-13), amide
CAS :<p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>Formule :C61H100N22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1381.59BPR1M97
CAS :<p>BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.</p>Formule :C18H18Cl2N2ODegré de pureté :98.78% - 99.95%Couleur et forme :SolidMasse moléculaire :349.25PIPE-3297
<p>PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.</p>Formule :C23H30N2OMasse moléculaire :350.23581β-Endorphin (1-27) (human)
CAS :<p>β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,</p>Formule :C139H217N33O40SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3022.47SB 205607 dihydrobromide
CAS :<p>non-peptide δ1 opioid receptor agonist</p>Formule :C23H24N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.45Dynorphin B (1-9)
CAS :<p>Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selective</p>Formule :C54H78N16O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1143.3DALDA TFA
<p>DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.</p>Formule :C30H45N9O5·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :611.74 (free base)CSD-CH2(1,8)-NH2
<p>CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.</p>Formule :C76H125N25O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1693.09Leumorphin, human
CAS :<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Formule :C150H224N42O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3351.64Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Formule :C46H66N10O12S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :1015.21CJ-15208
CAS :<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formule :C34H35N5O4Couleur et forme :SolidMasse moléculaire :577.67N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Formule :C36H40N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :652.74N-Acetyl-α-Endorphin
CAS :N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formule :C79H122N18O27SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1787.98Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Formule :C32H45N5OCouleur et forme :SolidMasse moléculaire :515.73Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Degré de pureté :99.89%Couleur et forme :SoildCTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Formule :C52H71N11O13S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Formule :C84H142N32O23Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS :<p>is a ketone and a building block.</p>Formule :C38H57N7O8Degré de pureté :96.94%Couleur et forme :SolidMasse moléculaire :739.9[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formule :C63H103FN22O17Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :1459.63[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Formule :C31H43N5O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.65β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Formule :C141H221N33O42SDegré de pureté :96.52%Couleur et forme :SolidMasse moléculaire :3082.52β-Endorphin (6-31), human
CAS :<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Formule :C131H218N34O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2909.38Deltorphin
CAS :<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Formule :C44H62N10O10S2Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :955.15Porcine dynorphin A(1-13)
CAS :<p>Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.</p>Formule :C75H126N24O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1603.95Loperamide phenyl
CAS :<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Formule :C35H37ClN2O2Couleur et forme :SolidMasse moléculaire :553.14Endomorphin 2 TFA
CAS :<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Formule :C34H38F3N5O7Couleur et forme :SolidMasse moléculaire :685.69BMS-986121
CAS :<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Formule :C15H9Cl2N3O2SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :366.22[Leu5]-Enkephalin
CAS :<p>[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM</p>Formule :C28H37N5O7Degré de pureté :99.87% - 99.88%Couleur et forme :SolidMasse moléculaire :555.62Alvimopan dihydrate (LY246736 dihydrate)
CAS :<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Formule :C25H36N2O6Couleur et forme :SolidMasse moléculaire :460.56Asimadoline
CAS :<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Formule :C27H30N2O2Couleur et forme :SolidMasse moléculaire :414.54BAN ORL 24 dihydrochloride
CAS :<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Formule :C27H37Cl2N3O2Degré de pureté :95.03%Couleur et forme :SolidMasse moléculaire :506.51Dermorphin TFA
CAS :<p>Dermorphin TFA is a new class of opioids-like peptides</p>Formule :C42H51F3N8O12Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :916.89Deltorphin I
CAS :<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Formule :C37H52N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :768.86Sec-O-Glucosylhamaudol
CAS :<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Formule :C21H26O10Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :438.43BRL 52537 hydrochloride
CAS :<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Formule :C18H25Cl3N2ODegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :391.76DPDPE TFA (88373-73-3 free base)
CAS :<p>DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.</p>Formule :C32H40F3N5O9S2Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :759.81Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Formule :C31H41N7O9Degré de pureté :98.92%Couleur et forme :SoildMasse moléculaire :655.7Aticaprant
CAS :<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Formule :C26H27FN2O2Degré de pureté :99.53% - 99.93%Couleur et forme :SolidMasse moléculaire :418.5BMS986187
CAS :<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Formule :C31H34O4Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :470.6Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Formule :C46H74N14O11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :999.17[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Formule :C29H37F3N6O8SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :686.7LY2940094 tartrate
CAS :<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Formule :C26H29ClF2N4O8SCouleur et forme :SolidMasse moléculaire :631.04MCOPPB triHydrochloride
CAS :<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Formule :C26H43Cl3N4Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :518.01Salvinorin A
CAS :<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Formule :C23H28O8Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :432.46Naloxegol oxalate
CAS :<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Formule :C36H55NO15Degré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :741.83Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formule :C51H73N15O11Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :1072.22Nalmefene hydrochloride
CAS :<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Formule :C21H26ClNO3Degré de pureté :98% - 99.85%Couleur et forme :SolidMasse moléculaire :375.89Difelikefalin acetate
CAS :<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Formule :C38H57N7O8Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :739.9AR-M 1000390 hydrochloride
CAS :<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Formule :C23H29ClN2ODegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :384.94Tyr-Gly-Gly-Phe-Met-OH
CAS :<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formule :C27H35N5O7SDegré de pureté :≥95%Couleur et forme :White Lyophilised SolidMasse moléculaire :573.66b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formule :C25H31N3O7Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :485.53Endomorphin 2
CAS :<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Formule :C32H37N5O5Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :571.67Methylnaltrexone bromide
CAS :<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Formule :C21H26BrNO4Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :436.35EST73502 HCl
CAS :<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formule :C19H27ClF2N2O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :388.88JTC-801
CAS :<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formule :C26H25N3O2·HClDegré de pureté :99.27% - 99.59%Couleur et forme :SolidMasse moléculaire :447.96BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Formule :C132H188N38O33S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :2899.27BMS-986122
CAS :<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Formule :C16H15BrClNO3S2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :448.78ADL-5859
CAS :<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Formule :C24H28N2O3·HClDegré de pureté :98.78% - 99.11%Couleur et forme :SolidMasse moléculaire :428.95N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.66Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formule :C51H79N15O16Degré de pureté :95.54%Couleur et forme :SolidMasse moléculaire :1158.26Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Formule :C101H159N31O25Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :2207.58(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Formule :C33H46N6O10Degré de pureté :94.17%Couleur et forme :SoildMasse moléculaire :686.75Sinomenine
CAS :<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formule :C19H23NO4Degré de pureté :99.02% - 99.73%Couleur et forme :White PowderMasse moléculaire :329.39Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Formule :C77H130N24O17Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :1664Alvimopan monohydrate
CAS :<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formule :C25H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :442.55Endomorphin 1
CAS :<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Formule :C34H38N6O5Degré de pureté :95.92%Couleur et forme :Solid (Solid Powder )Masse moléculaire :610.7Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Formule :C76H119N21O19Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :1630.89ADL-5747 (HCl)
CAS :<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formule :C24H29ClN2O3Couleur et forme :SolidMasse moléculaire :428.95Asimadoline hydrochloride
CAS :<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Formule :C27H31ClN2O2Degré de pureté :98.94% - 99.32%Couleur et forme :SolidMasse moléculaire :451.01PZM21
CAS :<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formule :C19H27N3O2SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :361.5MCOPPB
CAS :<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formule :C26H40N4Couleur et forme :SolidMasse moléculaire :408.62DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Formule :C28H36F3N5O8Degré de pureté :98.67% - 99.76%Couleur et forme :SolidMasse moléculaire :627.6BW-180C
CAS :<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Formule :C29H39N5O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :569.65GR 89696 free base
CAS :<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Formule :C19H25Cl2N3O3Couleur et forme :SolidMasse moléculaire :414.33EST73502 hydrochloride
CAS :<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Formule :C19H27ClF2N2O2Couleur et forme :SolidMasse moléculaire :388.88CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Formule :C53H70F3N13O13S2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :1218.33BMS986188
CAS :<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Formule :C30H31BrO4Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :535.47Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Formule :C63H101F3N22O17Degré de pureté :97.64%Couleur et forme :SolidMasse moléculaire :1495.61Corydaline
CAS :<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Formule :C22H27NO4Degré de pureté :98.97% - 99.86%Couleur et forme :SolidMasse moléculaire :369.45Deltorphin 2
CAS :<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formule :C38H54N8O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :782.88Naloxegol (NKTR-118)
CAS :<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Formule :C34H53NO11Couleur et forme :SolidMasse moléculaire :651.78Bisacodyl
CAS :<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Formule :C22H19NO4Degré de pureté :99.45% - 99.78%Couleur et forme :Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMasse moléculaire :361.39GR103545
CAS :<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Formule :C23H29Cl2N3O7Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :530.4Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Formule :C59H95N19O14Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1294.53Gluten Exorphin C
CAS :<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Formule :C29H45N5O8Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :591.7Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formule :C51H68N12O13Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :1057.16LY2795050
CAS :<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Formule :C23H22ClN3O2Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :407.89N-Desmethylclozapine
CAS :<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8DAMGO
CAS :<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formule :C26H35N5O6Degré de pureté :98.83% - 99.92%Couleur et forme :SolidMasse moléculaire :513.59Leuphasyl TFA
CAS :<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Formule :C31H40F3N5O9Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :683.67Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formule :C50H72N15O15SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1326.26[D-Ala2]leucine-enkephalin
CAS :<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formule :C29H39N5O7Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :569.65Nociceptin
CAS :<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Formule :C79H129N27O22Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :1809.04[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Formule :C30H42N6O8Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :614.69GRT2932Q
CAS :<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Formule :C25H26ClN3OCouleur et forme :SolidMasse moléculaire :419.95BW 373U86
CAS :<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Formule :C27H37N3O2Couleur et forme :SolidMasse moléculaire :435.6TIPP
CAS :<p>TIPP is an agent of delta opioid antagonist.</p>Formule :C37H38N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :634.72ICI 154,129
CAS :<p>Selective δ opioid antagonist</p>Formule :C34H46N4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :638.82JTC-801 free base
CAS :<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Formule :C26H25N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.5ML 190
CAS :<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Formule :C27H32N6O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :488.58Diallyl G
CAS :<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Formule :C38H53N5O8Couleur et forme :SolidMasse moléculaire :707.86Loperamide oxide
CAS :<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Formule :C29H33ClN2O3Couleur et forme :SolidMasse moléculaire :493.04GSK1521498 free base
CAS :<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Formule :C24H20F2N4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :402.44CR-665 Acetate
CAS :<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Formule :C38H53N9O6Couleur et forme :SolidMasse moléculaire :731.899LY 164929
CAS :<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Formule :C28H41N5O4Couleur et forme :SolidMasse moléculaire :511.66ADL-5859 HCl
CAS :<p>ADL-5859 is a delta-opioid receptor agonist.</p>Formule :C24H28N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49GSK1521498 free base (hydrochloride)
CAS :<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Formule :C24H21ClF2N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.9SR8993
CAS :<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Formule :C25H37FN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.59
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