Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
249 produits trouvés pour "Récepteur d'adénosine"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formule :C21H26NO10PDegré de pureté :97.04%Couleur et forme :SoildMasse moléculaire :483.41N6-Ethyladenosine
CAS :N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Formule :C12H17N5O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :295.29Acefylline
CAS :Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Formule :C9H10N4O4Degré de pureté :99.57%Couleur et forme :White Crystalline SolidMasse moléculaire :238.2DPTN dihydrochloride
CAS :DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formule :C22H20Cl2N4OSDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :459.39Ticlopidine hydrochloride
CAS :Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formule :C14H15Cl2NSDegré de pureté :99.85% - >99.99%Couleur et forme :White PowderMasse moléculaire :300.25AB928
CAS :AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Formule :C23H22N8ODegré de pureté :98.09% - >99.99%Couleur et forme :SolidMasse moléculaire :426.47Ref: TM-T14078
1mg52,00€5mg117,00€10mg187,00€25mg369,00€50mg437,00€100mg628,00€1mL*10mM (DMSO)127,00€Pamabrom
CAS :Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.Formule :C11H18BrN5O3Degré de pureté :99.84% - >99.99%Couleur et forme :CoaMasse moléculaire :348.2Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Formule :C24H29ClF3N5O5SDegré de pureté :97.91%Couleur et forme :SoildMasse moléculaire :592.03Adenosine 5'-monophosphate monohydrate
CAS :Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.
Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24Aminophylline
CAS :Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43Theophylline monohydrate
CAS :Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Adenosine A1 receptor activator T62
CAS :Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8Ref: TM-T14127
1mg64,00€5mg126,00€10mg180,00€25mg290,00€50mg396,00€100mg537,00€200mg712,00€1mL*10mM (DMSO)187,00€YT 146
CAS :YT 146 is a biochemical.Formule :C18H25N5O4Degré de pureté :98.81% - 99.25%Couleur et forme :SolidMasse moléculaire :375.42Doxofylline
CAS :Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formule :C11H14N4O4Degré de pureté :99.958% - >99.99%Couleur et forme :SolidMasse moléculaire :266.25N6-Cyclohexyladenosine
CAS :N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formule :C16H23N5O4Degré de pureté :99.92% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38Theophylline
CAS :Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFormule :C7H8N4O2Degré de pureté :99.65% - 99.98%Couleur et forme :White Solid PowderMasse moléculaire :180.16CGS 15943
CAS :CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formule :C13H8ClN5ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :285.69Ref: TM-T14944
2mg34,00€5mg50,00€10mg82,00€25mg147,00€50mg222,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)55,00€Pentoxifylline
CAS :Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.Formule :C13H18N4O3Degré de pureté :99.26% - 99.93%Couleur et forme :SolidMasse moléculaire :278.31Diphylline
CAS :Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Formule :C10H14N4O4Degré de pureté :98.54%Couleur et forme :Crystals From Alcohol SolidMasse moléculaire :254.24Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78FSCPX
CAS :FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Formule :C23H27FN4O6SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :506.55Ref: TM-T39039
1mg82,00€5mg180,00€10mg271,00€25mg460,00€50mg617,00€100mg825,00€200mg1.108,00€1mL*10mM (DMSO)86,00€LUF7690
CAS :LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection andFormule :C25H24FN5O6SCouleur et forme :SolidMasse moléculaire :541.55A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Formule :C56H71N15O12S2Couleur et forme :SolidMasse moléculaire :1210.39A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Formule :C23H25IN4Couleur et forme :SolidMasse moléculaire :484.38PSB 0777 ammonium salt
CAS :adenosine A2A receptor full agonistFormule :C18H24N6O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.55ABT-702
CAS :ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Formule :C22H19BrN6ODegré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :463.338-Chloro caffeine
CAS :8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64MRS-1706
CAS :MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formule :C27H29N5O5Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :503.55Ref: TM-T16136
1mg34,00€5mg74,00€10mg113,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)84,00€3F6-9G5
3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.Degré de pureté :>95%Couleur et forme :Odour LiquidMasse moléculaire :146.66 kDaDanshenol B
Danshenol B is a natural product that can be used as a reference standard.Formule :C22H26O4Couleur et forme :SolidMasse moléculaire :354.446A-286501
CAS :A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Formule :C11H14BrN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.17Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Formule :C86H115FN16O21Couleur et forme :SolidMasse moléculaire :1727.93Theophyllol
CAS :Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.Formule :C9H10N4Na2O4Couleur et forme :SolidMasse moléculaire :284.18N6-Benzyl-5'-ethylcarboxamido adenosine
CAS :N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formule :C19H22N6O4Couleur et forme :SolidMasse moléculaire :398.42GW-328267
CAS :GW-328267 is an agonist of the adenosine A2 receptor.Formule :C21H26N10O4Couleur et forme :SolidMasse moléculaire :482.5Xanthine amine congener trihydrochloride
CAS :Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formule :C21H29ClN6O4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :464.95Norisoboldine hydrochloride
CAS :Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Formule :C25H31F3N6O8Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :600.55Adenosine receptor antagonist 1
CAS :A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Formule :C22H15ClFN7OCouleur et forme :SolidMasse moléculaire :447.86A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67LUF6096
CAS :LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormule :C22H21Cl2N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :414.33AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.Formule :C21H25N5Couleur et forme :SolidMasse moléculaire :347.211Xanthine amine congener dihydrochloride
CAS :XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Formule :C21H30Cl2N6O4Couleur et forme :SolidMasse moléculaire :501.41LAS101057
CAS :LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formule :C18H14FN5ODegré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :335.34GR79236
CAS :GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formule :C15H21N5O5Couleur et forme :SolidMasse moléculaire :351.36(Rac)-Mirabegron-d5
CAS :(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Formule :C21H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54MRS-3777 hemioxalate
CAS :MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.
Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39Theophylline-d6
CAS :Theophylline-d6, an internal standard for theophylline quantification in GC/LC-MS, relaxes bronchial muscles and treats asthma/COPD.Formule :C7H2D6N4O2Couleur et forme :SolidMasse moléculaire :186.2Norisoboldine
CAS :Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formule :C18H19NO4Degré de pureté :98.12% - 99.7%Couleur et forme :SolidMasse moléculaire :313.35SCH442416
CAS :SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formule :C20H19N7O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :389.41Ref: TM-T23336
1mg46,00€5mg88,00€10mg132,00€25mg266,00€50mg409,00€100mg573,00€200mg807,00€1mL*10mM (DMSO)92,00€Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38ZM241385
CAS :ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Formule :C16H15N7O2Degré de pureté :97.02% - 99.69%Couleur et forme :SolidMasse moléculaire :337.34ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.42% - 98.98%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg58,00€2mg82,00€5mg113,00€10mg177,00€25mg333,00€50mg502,00€100mg710,00€500mg1.494,00€1mL*10mM (DMSO)133,00€Regadenoson hydrate
CAS :Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.Formule :C15H20N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.372-Chloroadenosine
CAS :2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormule :C10H12ClN5O4Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :301.69Preladenant
CAS :Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormule :C25H29N9O3Degré de pureté :98.02% - 99.68%Couleur et forme :SolidMasse moléculaire :503.56Xanthine amine congener hydrochloride
CAS :Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.Formule :C21H29ClN6O4Couleur et forme :SolidMasse moléculaire :464.95Inosine
CAS :Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!Formule :C10H12N4O5Degré de pureté :99.51% - 99.89%Couleur et forme :SolidMasse moléculaire :268.238-Cyclopentyl-1,3-dimethylxanthine
CAS :8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formule :C12H16N4O2Degré de pureté :98.58% - 99.9%Couleur et forme :SolidMasse moléculaire :248.28Nitrobenzylthioinosine
CAS :Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41Tecadenoson
CAS :Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33Binodenoson
CAS :Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formule :C17H25N7O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :391.42Ref: TM-T9516
1mg94,00€5mg222,00€10mg334,00€25mg557,00€50mg745,00€100mg1.044,00€1mL*10mM (DMSO)245,00€CHEMBL241987
CAS :CHEMBL241987 targets the Adenosine receptor A3 (human)Formule :C16H11N3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :261.28CGS 21680 Hydrochloride
CAS :CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formule :C23H29N7O6·HClDegré de pureté :96.74% - 99.53%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T6441
1mg38,00€2mg50,00€5mg81,00€10mg109,00€25mg215,00€50mg389,00€100mg575,00€1mL*10mM (DMSO)95,00€Enprofylline
CAS :Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Ref: TM-T21389
2mg42,00€5mg62,00€10mg88,00€25mg141,00€50mg215,00€100mg318,00€200mg442,00€1mL*10mM (DMSO)59,00€Capadenoson
CAS :Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.57%Couleur et forme :SolidMasse moléculaire :520.03SCH 58261
CAS :SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formule :C18H15N7ODegré de pureté :99.07% - 99.75%Couleur et forme :SolidMasse moléculaire :345.36Ref: TM-T6979
1mg38,00€2mg49,00€5mg80,00€10mg118,00€25mg213,00€50mg344,00€100mg550,00€1mL*10mM (DMSO)81,00€A2B receptor antagonist 2
CAS :A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28Fostamatinib
CAS :Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.Formule :C23H26FN6O9PDegré de pureté :93.08% - 99.38%Couleur et forme :SolidMasse moléculaire :580.46Ref: TM-T6115
1mg40,00€2mg54,00€5mg84,00€10mg112,00€25mg198,00€50mg318,00€100mg520,00€500mg1.134,00€1mL*10mM (DMSO)96,00€Tozadenant
CAS :Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5Alloxazine
CAS :Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formule :C10H6N4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :214.18Taminadenant mesylate
CAS :Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formule :C11H12BrN7O3SCouleur et forme :SolidMasse moléculaire :402.227CPI-444
CAS :CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formule :C20H21N7O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :407.43Ref: TM-T7183
2mg34,00€5mg52,00€10mg73,00€25mg128,00€50mg197,00€100mg295,00€200mg442,00€1mL*10mM (DMSO)52,00€MIPS521
CAS :MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.8Ref: TM-T9330
1mg35,00€2mg50,00€5mg74,00€10mg105,00€25mg178,00€50mg313,00€100mg485,00€1mL*10mM (DMSO)82,00€DPCPX
CAS :DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39CCPA
CAS :CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFormule :C15H20ClN5O4Degré de pureté :99.1%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8Adenosine amine congener
CAS :Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formule :C28H32N8O6Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :576.6Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
2mg35,00€5mg51,00€10mg80,00€25mg131,00€50mg210,00€100mg313,00€200mg445,00€1mL*10mM (DMSO)215,00€PD 117519
CAS :PD 117519 (CI947) is an agonist of adenosine receptorFormule :C19H21N5O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :383.4SDZ WAG 994
CAS :SDZ WAG 994 is an A1 adenosine receptor agonist.Formule :C17H25N5O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :363.41Ref: TM-T23347
1mg63,00€5mg114,00€10mg172,00€25mg299,00€50mg432,00€100mg587,00€200mg792,00€1mL*10mM (DMSO)120,00€Namodenoson
CAS :Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formule :C18H18ClIN6O4Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :544.735-Iodotubercidin
CAS :5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Formule :C11H13IN4O4Degré de pureté :99.88% - 99.98%Couleur et forme :Tan SolidMasse moléculaire :392.15Ref: TM-T6745
1mg43,00€5mg96,00€10mg137,00€25mg268,00€50mg429,00€100mg685,00€200mg888,00€1mL*10mM (DMSO)92,00€Taminadenant
CAS :Taminadenant is an adenosine receptor antagonist.Formule :C10H8BrN7Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :306.12Ref: TM-T16980
2mg34,00€5mg49,00€10mg84,00€25mg114,00€50mg166,00€100mg236,00€200mg353,00€1mL*10mM (DMSO)54,00€N6,N6-Dimethyladenosine
CAS :N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.Formule :C12H17N5O4Degré de pureté :98.79%Couleur et forme :White PowderMasse moléculaire :295.29AZD4635
CAS :AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formule :C15H11ClFN5Degré de pureté :99.15% - 99.90%Couleur et forme :SolidMasse moléculaire :315.73Ref: TM-T4265
1mg37,00€2mg52,00€5mg79,00€10mg116,00€25mg188,00€50mg296,00€100mg457,00€500mg1.008,00€1mL*10mM (DMSO)87,00€1-Ethyl-6-aminouracil
CAS :1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormule :C6H9N3O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :155.15BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg84,00€5mg161,00€10mg235,00€25mg420,00€50mg605,00€100mg842,00€200mg1.134,00€1mL*10mM (DMSO)172,00€Regadenoson
CAS :Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.35Ref: TM-T2671
2mg44,00€5mg62,00€10mg96,00€25mg170,00€50mg259,00€100mg394,00€500mg887,00€1mL*10mM (DMSO)69,00€Reversine
CAS :Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).Formule :C21H27N7ODegré de pureté :98% - 99.45%Couleur et forme :SolidMasse moléculaire :393.49Ref: TM-T1825
1mg35,00€2mg50,00€5mg66,00€10mg84,00€25mg156,00€50mg212,00€100mg371,00€1mL*10mM (DMSO)66,00€Swertisin
CAS :Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Formule :C22H22O10Degré de pureté :99.74% - 99.89%Couleur et forme :SolidMasse moléculaire :446.40Adenosine receptor antagonist 4
CAS :Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formule :C10H13N3Degré de pureté :99.63% - 99.65%Couleur et forme :Off-White PowderMasse moléculaire :175.23Istradefylline
CAS :Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formule :C20H24N4O4Degré de pureté :98.18% - 99.95%Couleur et forme :SolidMasse moléculaire :384.43VPC171
CAS :VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formule :C18H12F3NOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :347.35Ref: TM-T29112
1mg49,00€5mg96,00€10mg124,00€25mg222,00€50mg309,00€100mg439,00€200mg592,00€1mL*10mM (DMSO)88,00€Piclidenoson
CAS :Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Formule :C18H19IN6O4Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :510.29Ref: TM-T7188
2mg39,00€5mg58,00€10mg94,00€25mg173,00€50mg281,00€100mg439,00€200mg628,00€1mL*10mM (DMSO)66,00€5'-N-Ethylcarboxamidoadenosine
CAS :NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formule :C12H16N6O4Degré de pureté :98.95% - ≥95%Couleur et forme :PowderMasse moléculaire :308.29Proxyphylline
CAS :Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Formule :C10H14N4O3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :238.24Rolofylline
CAS :Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46
