Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
242 produits trouvés pour "Récepteur d'adénosine"
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Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formule :C24H29ClF3N5O5SDegré de pureté :96.56%Couleur et forme :SoildMasse moléculaire :592.03Pamabrom
CAS :<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formule :C11H18BrN5O3Degré de pureté :99.84% - >99.99%Couleur et forme :CoaMasse moléculaire :348.2Adenosine 5'-monophosphate monohydrate
CAS :<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24Ticlopidine hydrochloride
CAS :<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formule :C14H15Cl2NSDegré de pureté :99.85% - >99.99%Couleur et forme :White PowderMasse moléculaire :300.25Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Formule :C21H26NO10PDegré de pureté :95.63%Couleur et forme :SoildMasse moléculaire :483.41AB928
CAS :<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formule :C23H22N8ODegré de pureté :98.09% - >99.99%Couleur et forme :SolidMasse moléculaire :426.47Pentoxifylline
CAS :<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Formule :C13H18N4O3Degré de pureté :99.26% - 99.93%Couleur et forme :SolidMasse moléculaire :278.31Diphylline
CAS :<p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>Formule :C10H14N4O4Degré de pureté :98.54%Couleur et forme :Crystals From Alcohol SolidMasse moléculaire :254.24Doxofylline
CAS :<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formule :C11H14N4O4Degré de pureté :99.958% - >99.99%Couleur et forme :SolidMasse moléculaire :266.25Theophylline
CAS :<p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>Formule :C7H8N4O2Degré de pureté :99.65% - 99.98%Couleur et forme :White Solid PowderMasse moléculaire :180.16DPTN dihydrochloride
CAS :<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formule :C22H20Cl2N4OSDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :459.39Adenosine A1 receptor activator T62
CAS :<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8YT 146
CAS :<p>YT 146 is a biochemical.</p>Formule :C18H25N5O4Degré de pureté :98.81% - 99.25%Couleur et forme :SolidMasse moléculaire :375.42Theophylline monohydrate
CAS :<p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>Formule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Aminophylline
CAS :<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43N6-Ethyladenosine
CAS :<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formule :C12H17N5O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :295.29Acefylline
CAS :<p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>Formule :C9H10N4O4Degré de pureté :99.57%Couleur et forme :White Crystalline SolidMasse moléculaire :238.2CGS 15943
CAS :<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Formule :C13H8ClN5ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :285.69N6-Cyclohexyladenosine
CAS :<p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>Formule :C16H23N5O4Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38A3AR agonist 2
<p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68hA3AR agonist 2
<p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78Xanthine amine congener dihydrochloride
CAS :<p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>Formule :C21H30Cl2N6O4Couleur et forme :SolidMasse moléculaire :501.41Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formule :C86H115FN16O21Couleur et forme :SolidMasse moléculaire :1727.93LUF6096
CAS :<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formule :C22H21Cl2N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :414.33ABT-702
CAS :<p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>Formule :C22H19BrN6ODegré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :463.33Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formule :C25H31F3N6O8Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :600.558-Chloro caffeine
CAS :<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Formule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Formule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Formule :C21H25N5Couleur et forme :SolidMasse moléculaire :347.211PSB 0777 ammonium salt
CAS :<p>adenosine A2A receptor full agonist</p>Formule :C18H24N6O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.55MRS-1706
CAS :<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Formule :C27H29N5O5Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :503.55N6-Benzyl-5'-ethylcarboxamido adenosine
CAS :<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Formule :C19H22N6O4Couleur et forme :SolidMasse moléculaire :398.42Norisoboldine hydrochloride
CAS :<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81FSCPX
CAS :<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formule :C23H27FN4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.55Xanthine amine congener trihydrochloride
CAS :<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Formule :C21H29ClN6O4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :464.95Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Formule :C22H26O4Couleur et forme :SolidMasse moléculaire :354.4463F6-9G5
<p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>Degré de pureté :>95%Couleur et forme :Odour LiquidTheophyllol
CAS :<p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>Formule :C9H10N4Na2O4Couleur et forme :SolidMasse moléculaire :284.18Adenosine receptor antagonist 1
CAS :<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Formule :C22H15ClFN7OCouleur et forme :SolidMasse moléculaire :447.86LUF7690
CAS :<p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>Formule :C25H24FN5O6SCouleur et forme :SolidMasse moléculaire :541.55A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Formule :C23H25IN4Couleur et forme :SolidMasse moléculaire :484.38A-286501
CAS :<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Formule :C11H14BrN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.17GW-328267
CAS :<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Formule :C21H26N10O4Couleur et forme :SolidMasse moléculaire :482.5A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Formule :C56H71N15O12S2Couleur et forme :SolidMasse moléculaire :1210.39LAS101057
CAS :<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Formule :C18H14FN5ODegré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :335.34(Rac)-Mirabegron-d5
CAS :<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Formule :C21H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54GR79236
CAS :<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Formule :C15H21N5O5Couleur et forme :SolidMasse moléculaire :351.36MRS-3777 hemioxalate
CAS :<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39
