Récepteur GNRH
Les récepteurs de la gonadolibérine (GnRH) sont des GPCR qui se lient à la GnRH, une hormone responsable de la régulation de la libération de l'hormone lutéinisante (LH) et de l'hormone folliculo-stimulante (FSH) par l'hypophyse. Ces récepteurs sont cruciaux pour la fonction reproductrice et sont ciblés dans les thérapies pour des conditions telles que le cancer de la prostate, l'endométriose et l'infertilité. Les agonistes et antagonistes des récepteurs de la GnRH sont également utilisés dans les technologies de procréation assistée. Chez CymitQuimica, nous offrons une gamme complète de modulateurs de récepteurs de la GnRH de haute qualité pour soutenir vos recherches en santé reproductive, endocrinologie et hormonothérapie.
69 produits trouvés pour "Récepteur GNRH"
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Degarelix acetate(214766-78-6 free base)
CAS :<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formule :C84H107ClN18O18Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :1692.34Abarelix
CAS :<p>Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.</p>Formule :C72H95ClN14O14Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1416.06Alarelin Acetate
CAS :<p>Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.</p>Formule :C56H78N16O12Degré de pureté :99.81% - >99.99%Couleur et forme :White PowderMasse moléculaire :1167.34(R)-Elagolix
CAS :<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Formule :C32H30F5N3O5Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :631.59Kisspeptin-54(human)
CAS :<p>Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.</p>Formule :C258H401N79O78Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5857.49Phoenixin-14
CAS :<p>Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/</p>Formule :C75H110N18O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1583.78Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Formule :C75H110N18O20·xC2HF3O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :1583.78 (free base)Linzagolix choline
CAS :<p>Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.</p>Formule :C27H28F3N3O8SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :611.59Surfagon
CAS :<p>Surfagon is an effective LHRH agonist.</p>Formule :C56H78N16O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1167.34LGnRH-III, lamprey
CAS :<p>GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.</p>Formule :C59H74N18O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1259.33MI 1544
CAS :<p>MI 1544 is a LHRH antagonist.</p>Formule :C71H94ClN17O13Couleur et forme :SolidMasse moléculaire :1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS :<p>LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.</p>Formule :C60H73N15O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1212.31Goserelin acetate(65807-02-5 Free base)
<p>Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>Degré de pureté :99.77%Couleur et forme :Odour SolidBim 21009
CAS :<p>Bim 21009 is an inhibitor of gonadorelin.</p>Formule :C74H92ClN17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1463.08Prolactin Releasing Peptide (1-31), human
CAS :<p>Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).</p>Formule :C160H252N56O42SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3664.15[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS :<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Formule :C67H84N16O13Couleur et forme :SolidMasse moléculaire :1321.48Fsh receptor-binding inhibitor fragment(bi-10)
CAS :<p>FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.</p>Formule :C42H67N13O19Couleur et forme :SolidMasse moléculaire :1058.06Zebrafish Kisspeptin-1
CAS :<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Formule :C58H84N16O15Couleur et forme :SolidMasse moléculaire :1245.39GnRH Associated Peptide (1-24), human
CAS :<p>GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.</p>Formule :C117H190N32O43Couleur et forme :SolidMasse moléculaire :2732.95LH-RH (7-10)
CAS :<p>LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.</p>Formule :C19H36N8O4Couleur et forme :SolidMasse moléculaire :440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS :<p>Analog of LHRH, stimulates LH and FSH release, controls reproduction.</p>Formule :C59H84N18O14Couleur et forme :SolidMasse moléculaire :1269.41Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Formule :C258H401N79O78·C2HF3O2Couleur et forme :SolidMasse moléculaire :5971.45sGnRH-A
CAS :<p>sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.</p>Formule :C64H83N17O12Couleur et forme :SolidMasse moléculaire :1282.45Kisspeptin 13
CAS :<p>Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.</p>Formule :C78H107N21O18Couleur et forme :SolidMasse moléculaire :1626.81Azaline B
CAS :<p>Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.</p>Formule :C80H102ClN23O12Couleur et forme :SolidMasse moléculaire :1613.27A 76154
CAS :<p>A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).</p>Formule :C70H93FN12O12Couleur et forme :SolidMasse moléculaire :1313.584Wy 43657
CAS :<p>Wy 43657 is a gonadorelin antagonist.</p>Formule :C71H86N14O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1343.554APTAA-LHRH
CAS :<p>APTAA-LHRH is a gonadorelin antagonist.</p>Formule :C69H91Cl2N17O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1453.47RS 18286
CAS :<p>RS 18286 is a LHRH antagonist.</p>Formule :C74H101Cl2N17O14Couleur et forme :SolidMasse moléculaire :1523.6Azaline
CAS :<p>Azaline is a gonadorelin antagonist.</p>Formule :C74H106ClN23O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1545.26LHRH, Ala(6)-
CAS :<p>LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.</p>Formule :C56H77N17O13Couleur et forme :SolidMasse moléculaire :1196.32Avorelin
CAS :<p>Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.</p>Formule :C65H85N17O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1296.48LHRH
CAS :<p>Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and has</p>Formule :C55H74N16O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1183.27AG 045572
CAS :<p>AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is</p>Formule :C30H37NO5Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :491.62Lecirelin
CAS :<p>Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.</p>Formule :C59H84N16O12Couleur et forme :SolidMasse moléculaire :1209.4Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formule :C66H87N17O14Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :1342.5Buserelin Acetate (57982-77-1 free base)
CAS :<p>Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).</p>Formule :C62H90N16O15Degré de pureté :99.31% - 99.78%Couleur et forme :SolidMasse moléculaire :1299.48Triptorelin acetate(57773-63-4 free base)
CAS :<p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>Formule :C66H86N18O15Degré de pureté :99.90%Couleur et forme :White PowderMasse moléculaire :1371.53Cetrorelix diacetate
CAS :<p>Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.</p>Formule :C74H100ClN17O18Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :1551.17Lecirelin acetate(61012-19-9 free base)
<p>Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts</p>Formule :C61H88N16O14Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :1269.45Nafarelin acetate(76932-56-4 free base)
CAS :<p>Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.</p>Formule :C68H87N17O15Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :1382.55Elagolix sodium
CAS :<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formule :C32H29F5N3NaO5Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :653.57Histrelin acetate
CAS :<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Formule :C68H90N18O14Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1383.55Relugolix
CAS :<p>Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with</p>Formule :C29H27F2N7O5SDegré de pureté :98.64% - 99.97%Couleur et forme :SolidMasse moléculaire :623.63Linzagolix
CAS :<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Formule :C22H15F3N2O7SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :508.42Fluorogestone acetate
CAS :<p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>Formule :C23H31FO5Degré de pureté :99.47%Couleur et forme :CoaMasse moléculaire :406.49Goserelin acetate
CAS :<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Formule :C61H88N18O16Degré de pureté :99.77% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :1329.46Fertirelin
CAS :<p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>Formule :C55H76N16O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1153.29Ganirelix Acetate
CAS :<p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>Formule :C82H117ClN18O15Degré de pureté :96.05%Couleur et forme :SolidMasse moléculaire :1630.4Sufugolix
CAS :<p>Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.</p>Formule :C36H31F2N5O4SDegré de pureté :97.78%Couleur et forme :SolidMasse moléculaire :667.72LGnRH-III, lamprey acetate(147859-97-0 free base)
<p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>Formule :C61H78N18O16Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :1319.38Cetrorelix Acetate
CAS :<p>Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.</p>Formule :C70H92ClN17O14·xC2H4O2Degré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :1491.11NBI-42902
CAS :<p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>Formule :C27H24F3N3O3Couleur et forme :SolidMasse moléculaire :495.49BAY 1214784
CAS :<p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>Formule :C29H26ClF4N3O5S2Couleur et forme :SolidMasse moléculaire :672.11Argtide
CAS :<p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>Formule :C80H104ClN21O14Couleur et forme :SolidMasse moléculaire :1619.27Opigolix
CAS :<p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>Formule :C25H19F3N4O5SDegré de pureté :98.60% - 98.97%Couleur et forme :SolidMasse moléculaire :544.5BAY-298
CAS :<p>BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.</p>Formule :C27H21ClFN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.93[D-Ala6]-LH-RH
CAS :<p>[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].</p>Formule :C56H77N17O13Couleur et forme :SolidMasse moléculaire :1196.32T 98475
CAS :<p>gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active</p>Formule :C37H37F2N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :657.77BAY-784
CAS :<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Formule :C29H26ClF4N3O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :672.11DCOIT
CAS :<p>DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].</p>Formule :C11H17Cl2NOSCouleur et forme :SolidMasse moléculaire :282.22Abarelix acetate
CAS :<p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>Formule :C72H95ClN14O14·xC2H4O2Couleur et forme :SolidMasse moléculaire :1476.14BAY-899
CAS :<p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>Formule :C25H19F2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.45Acyline
CAS :<p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>Formule :C80H102ClN15O14Couleur et forme :SolidMasse moléculaire :1533.21Merigolix
CAS :<p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>Formule :C36H35F7N4O6Couleur et forme :SolidMasse moléculaire :752.68GnRH-R antagonist 1
CAS :<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Formule :C31H28F5N7O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :721.65GnRH antagonist 2
CAS :<p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>Formule :C28H27F2N9O5Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :607.57(R)-BAY-899
<p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>Formule :C25H19F2N5O2Couleur et forme :SolidMasse moléculaire :459.45Dimethandrolone Undecanoate
CAS :<p>Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.</p>Formule :C31H50O3Degré de pureté :99.65% - >99.99%Couleur et forme :SolidMasse moléculaire :470.73
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