Autres inhibiteurs
Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.
36478 produits trouvés pour "Autres inhibiteurs"
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Mepixetil
Mepixetil is a potent angiotensin II receptor antagonist[1].Formule :C12H18N2O3Couleur et forme :SolidMasse moléculaire :238.282-n-Heptyl-4-quinolinol
CAS :<p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>Formule :C16H21NOCouleur et forme :SolidMasse moléculaire :243.34Pefcalcitol
CAS :Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.Formule :C26H34F5NO4Couleur et forme :SolidMasse moléculaire :519.54Pralatrexate, (R)-
CAS :Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.Formule :C23H23N7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.47RSK4-IN-1
CAS :RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.Formule :C19H20F2N4O3Couleur et forme :SolidMasse moléculaire :390.38AZ14145845
AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.Formule :C32H35N9OCouleur et forme :SolidMasse moléculaire :561.68PPO-IN-1
PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35C20 Sphingomyelin (d18:1/20:1)
CAS :C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).Formule :C43H85N2O6PCouleur et forme :SolidMasse moléculaire :757.119VEGFR-2-IN-26
CAS :VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.Formule :C24H19F3N6O2Couleur et forme :SolidMasse moléculaire :480.44Fusarochromanone
CAS :Fusarochromanone (FC-101) is a mycotoxin produced by Fusarium oxysporum with potent antiangiogenic, anticancer and antimalarial activities.Formule :C15H20N2O4Degré de pureté :95.31% - 96%Couleur et forme :SolidMasse moléculaire :292.33LMD-A
CAS :LMD-A, also known as CCR8 antagonist LMD-A, is a CCR8 antagonist.Formule :C27H32N4O4SCouleur et forme :SolidMasse moléculaire :508.63Seldomycin factor 2
CAS :<p>Seldomycin factor 2 (XK 88-2) is an aminoglycoside antibiotic with broad-spectrum antibacterial activity.</p>Formule :C12H26N4O5Couleur et forme :SolidMasse moléculaire :306.359(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formule :C24H24N4O6Couleur et forme :SolidMasse moléculaire :464.47CI-1029
CAS :CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.Formule :C28H37NO4SCouleur et forme :SolidMasse moléculaire :483.66PI3K-IN-27
CAS :PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.Formule :C30H26F2N6O2SCouleur et forme :SolidMasse moléculaire :572.63P7170
CAS :<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Formule :C21H16F3N9Couleur et forme :SolidMasse moléculaire :451.42Zetomipzomib
CAS :KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) & LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.Formule :C30H42N4O8Couleur et forme :SolidMasse moléculaire :586.68FTO-IN-1 TFA
FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.Formule :C20H17Cl2F3N4O4Couleur et forme :SolidMasse moléculaire :505.27KHK-IN-6
CAS :KHK-IN-6 (compound 33) acts as a KHK inhibitor with an IC50 of 0.6nM.Formule :C23H24F3N5O2SCouleur et forme :SolidMasse moléculaire :491.53NTPDase-IN-3
CAS :NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.Formule :C22H24ClN3OS2Couleur et forme :SolidMasse moléculaire :446.03Cremeomycin
CAS :Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.Formule :C8H6N2O4Couleur et forme :SolidMasse moléculaire :194.144Ataprost
CAS :Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.Formule :C21H32O4Couleur et forme :SolidMasse moléculaire :348.48Monamycin H2
CAS :Monamycin H2 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.Formule :C34H56ClN7O8Masse moléculaire :726.30PPARα agonist 1
PPARα agonist 1 is a complete and potent PPARα agonist.Formule :C27H34O4Couleur et forme :SolidMasse moléculaire :422.561-Hydroxy-2-nonyn-4-one
CAS :<p>1-Hydroxy-2-nonyn-4-one is an antibiotic with activity against yeasts, filamentous fungi, tumors, and shows weak efficacy against both Gram-positive and Gram-negative bacteria.</p>Formule :C9H14O2Couleur et forme :SolidMasse moléculaire :154.206Kurasoin A
CAS :Kurasoin A is an inhibitor of the enzyme farnesyltransferase.Formule :C16H16O3Couleur et forme :SolidMasse moléculaire :256.296Griseolutein A
CAS :Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C17H14N2O6Couleur et forme :SolidMasse moléculaire :342.303AB 5046A
CAS :AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.Formule :C10H14O4Couleur et forme :SolidMasse moléculaire :198.22Vindeburnol
CAS :<p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35Pelagiomicin C
CAS :Pelagiomicin C exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C17H15N3O5Couleur et forme :SolidMasse moléculaire :341.318Mesulergine
CAS :<p>Mesulergine is metabolized into dopaminergic agonists.</p>Formule :C18H26N4O2SCouleur et forme :SolidMasse moléculaire :362.49RDN2150
CAS :<p>RDN2150 (Compound 25), a ZAP-70 inhibitor with an IC50 of 14.6 nM, covalently binds to the C346 residue of ZAP-70, suppressing the expression of CD25 and CD69</p>Formule :C28H29ClN8O4Couleur et forme :SolidMasse moléculaire :577.03Formadicin A
CAS :<p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>Formule :C30H34N4O16Couleur et forme :SolidMasse moléculaire :706.608PDE4-IN-6
PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.Formule :C25H20FNO5SCouleur et forme :SolidMasse moléculaire :465.49Saprisartan potassium
CAS :<p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>Formule :C25H21BrF3KN4O4SCouleur et forme :SolidMasse moléculaire :649.52PF-06305591 dihydrate
PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADMEFormule :C15H26N4O3Couleur et forme :SolidMasse moléculaire :310.3920-Deoxynarasin
CAS :20-Deoxynarasin exhibits activity against Gram-positive bacteria, mycoplasma, coccidia, and viruses, and it also promotes growth.Formule :C43H72O10Couleur et forme :SolidMasse moléculaire :749.03BAY-850 HCl
BAY-850 is a selective probe targeting Atad2A's bromine domain, displacing acetylated H4 peptides and detaching ATAD2 from chromatin at 1μm.Formule :C38H48Cl5N5O3Couleur et forme :SolidMasse moléculaire :800.08Antimalarial agent 3
Antimalarial agent 3 has a potent IC50 of 0.035 μM against Plasmodium and high selectivity for mammalian cells.Formule :C15H16BrN3O2Couleur et forme :SolidMasse moléculaire :350.21Glucosylceramide synthase-IN-3
Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.Formule :C21H20FN3O3Couleur et forme :SolidMasse moléculaire :381.4Halomicin B
CAS :<p>Halomicin B is an ansamycin-type antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Formule :C43H58N2O12Couleur et forme :SolidMasse moléculaire :794.927BMS-824
CAS :BMS-824: potent HCV NS5A inhibitor, IC50 ~5 nM, therapeutic index >10,000, specific to HCV.Formule :C27H25F3N4O5Couleur et forme :SolidMasse moléculaire :542.51FTO-IN-6
CAS :FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).Formule :C14H12N4O6Couleur et forme :SolidMasse moléculaire :332.27LGB-321 HCl
CAS :LGB-321: potent, selective PIM kinase inhibitor, active against PIM2, halts diverse blood cancers' growth, orally effective in mice.Formule :C23H23ClF3N5O2Couleur et forme :SolidMasse moléculaire :493.91Ep vinyl quinidine
CAS :3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.Formule :C20H24N2O2Couleur et forme :SolidMasse moléculaire :324.42Hydroxyakalone
CAS :Hydroxyakalone is an inhibitor of the enzyme xanthine oxidase (XOD, EC 1.2.3.2) and has an IC50 of 4.6 μM for XOD.Formule :C5H5N5O2Couleur et forme :SolidMasse moléculaire :167.126Antibiotic LL Z1640-2
CAS :Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.Formule :C19H22O7Couleur et forme :SolidMasse moléculaire :362.38AL-GDa62
<p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>Formule :C24H28FN3OCouleur et forme :SolidMasse moléculaire :393.5Pradimicin B
CAS :Pradimicin B is an antibiotic with potent antifungal and anti-yeast activities.Formule :C35H36N2O14Couleur et forme :SolidMasse moléculaire :708.665MPO-IN-8
CAS :<p>MPO-IN-8, an orally active myeloperoxidase (MPO) inhibitor, effectively inhibits the production of hypochlorous acid in neutrophils and the release of extracellular traps (NETosis). In mice exhibiting gouty arthritis, it reduces swelling, decreases peroxidase activity, and lowers IL-1β levels.</p>Formule :C12H9N3O2Couleur et forme :SolidMasse moléculaire :227.22EcGUS-IN-1
CAS :<p>EcGUS-IN-1 (Compound E-9) is a non-competitive inhibitor of β-glucuronidase, featuring an IC50 value of 2.68 μM and a Ki value of 1.64 μM. This compound effectively mitigates gastrointestinal adverse events (GIAE) associated with Escherichia coli infections by inhibiting the activity of E. coli β-glucuronidase.</p>Formule :C15H11F3N4SCouleur et forme :SolidMasse moléculaire :336.33Ranakinin
CAS :Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.Formule :C62H95N17O15SCouleur et forme :SolidMasse moléculaire :1350.59Encephalitic alphavirus-IN-1
Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.Formule :C27H25FN6O2Couleur et forme :SolidMasse moléculaire :484.52FCE-27262
CAS :FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.Formule :C23H31N3O3Couleur et forme :SolidMasse moléculaire :397.51MC4355
MC4355 is a dual inhibitor of EZH2 and histone deacetylase (HDAC).Formule :C30H36N4O5Couleur et forme :SolidMasse moléculaire :532.63Ingenol 3-monobenzoate
CAS :<p>Ingenol 3-monobenzoate (Ingenol 3-benzoate) acts as an aversive inducing agent. It binds to and activates protein kinase C (PKC) with a Ki of 0.14 nM. This activation inhibits the gene expression of phosphoenolpyruvate carboxykinase, thereby suppressing gluconeogenesis and increasing blood cortisol levels, which results in food aversion.</p>Formule :C27H32O6Couleur et forme :SolidMasse moléculaire :452.54MDL-43291
CAS :MDL-43291 is a leukotriene receptor antagonist.Formule :C25H42O4SCouleur et forme :SolidMasse moléculaire :438.66Piloquinone
CAS :Piloquinone is a type of phenanthrene compound that exhibits mild inhibitory effects on mycobacteria and protozoa.Formule :C21H20O5Couleur et forme :SolidMasse moléculaire :352.38TP3011
CAS :TP3011 is a potent topoisomerase I inhibitor equipotent as SN38 and is an active metabolite of CH-0793076.Formule :C26H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.51AZD-3409
CAS :AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.Formule :C34H41FN4O4S2Couleur et forme :SolidMasse moléculaire :652.84NCI-006
CAS :<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Formule :C31H24F2N4O4S3Couleur et forme :SolidMasse moléculaire :650.74Enpp-1-IN-11
Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.Formule :C15H15N5O3SCouleur et forme :SolidMasse moléculaire :345.38UAWJ9-36-1
CAS :UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49ASP-8731
CAS :ASP8731 is a selective inhibitor of BACH1 that prevents inflammation and vascular occlusion, and induces fetal hemoglobin in sickle cell disease.Formule :C20H21N5O4Couleur et forme :SolidMasse moléculaire :395.41PCSK9-IN-16
CAS :<p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>Formule :C16H20N6O2S3Couleur et forme :SolidMasse moléculaire :424.56M-89 MLL inhibitor
CAS :M-89, a potent Menin-MLL blocker: Kd 1.4 nM, IC50 25 nM for MV4;11 cells, 55 nM for MOLM-13, >100x selective over HL-60.Formule :C37H47N5O4SCouleur et forme :SolidMasse moléculaire :657.87Nothramicin
CAS :Nothramicin is an anthracycline antibiotic that exhibits antimycobacterial activity.Formule :C30H37NO11Couleur et forme :SolidMasse moléculaire :587.615(R)-ONO-2952
(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.Formule :C22H20ClFN2O2Couleur et forme :SolidMasse moléculaire :398.865,6-Dihydro-4-methoxy-2H-pyran-2-one
CAS :<p>5,6-Dihydro-4-methoxy-2H-pyran-2-one is produced by the Penicillium italicum strain MRC 1360.</p>Formule :C6H8O3Masse moléculaire :128.13GW311616 hydrochloride
CAS :GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formule :C19H32ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.99Hypercalin B
CAS :<p>Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.</p>Formule :C33H42O5Couleur et forme :SolidMasse moléculaire :518.684MMP408
CAS :<p>MMP408 acts as an inhibitor of MMP-12.</p>Formule :C19H20N2O7SCouleur et forme :SolidMasse moléculaire :420.44ART615
<p>ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).</p>Formule :C21H21F3N4O2Couleur et forme :SolidMasse moléculaire :418.41WAY-855
CAS :WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.Formule :C9H11NO4Couleur et forme :SolidMasse moléculaire :197.19LXR antagonist 2
<p>LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).</p>Formule :C34H40N2O5SCouleur et forme :SolidMasse moléculaire :588.76TEI-9063
CAS :TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.Formule :C23H38O4Couleur et forme :SolidMasse moléculaire :378.55Oncopterin
CAS :Oncopterin is found in urine from patients with solid and blood cancers.Formule :C12H18N6O3Couleur et forme :SolidMasse moléculaire :294.31S39625
CAS :S39625 is a stable, potent topoisomerase I inhibitor with anticancer properties, resistant to efflux transporters, inducing gamma-H2AX at nanomolar levels.Formule :C25H22N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.45Anticancer agent 80
Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).Formule :C19H12BrNO5Couleur et forme :SolidMasse moléculaire :414.21SARS-CoV-2-IN-24
SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.Formule :C27H30N4O5Couleur et forme :SolidMasse moléculaire :490.55Transthyretin-IN-1
Transthyretin-IN-1 inhibits TTR fibril formation, aiding Alzheimer’s research.Formule :C10H9Br2NO4Couleur et forme :SolidMasse moléculaire :366.99Sucistil
Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].Formule :C9H15NO4SCouleur et forme :SolidMasse moléculaire :233.28CPX-351
CAS :<p>CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.</p>Formule :C36H42N4O15Degré de pureté :98.95% - 99.763%Couleur et forme :SolidMasse moléculaire :770.74Guraxetan
Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.Formule :C20H34N4O9Couleur et forme :SolidMasse moléculaire :474.51Eurocidin E
CAS :Eurocidin E is an antibiotic that inhibits degranulation and histamine release from rat mast cells.Formule :C40H61NO14Couleur et forme :SolidMasse moléculaire :779.911L 731735
CAS :L 731735 is a farnesyltransferase inhibitor.Formule :C19H40N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.61Oiligodendrocyte differentiation promoter 1
CAS :Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .Formule :C25H25Cl2NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :490.38MPro N3
CAS :Mpro inhibitor blocks MHV-A29, HCoV-229E, FOPV (IC50: 2.7–8.8 μM), and SARS-CoV-2 (IC50: 16.8 μM) in plaque assays.Formule :C35H48N6O8Couleur et forme :SolidMasse moléculaire :680.79Glucoallosamidin A
CAS :Glucoallosamidin A is a glycoside antibiotic that inhibits chitinase activity. It effectively suppresses the chitinase enzyme in Candida albicans [ATCC 10231], exhibiting an IC50 of 3.4 μg/mL.Formule :C26H44N4O14Couleur et forme :SolidMasse moléculaire :636.646Balanol
CAS :Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.Formule :C28H26N2O10Couleur et forme :SolidMasse moléculaire :550.51VU6028418
<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Couleur et forme :LiquidAnti-inflammatory agent 16
Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.Formule :C21H23N5O3Couleur et forme :SolidMasse moléculaire :393.44Keap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.Formule :C26H25F3N2O9SCouleur et forme :SolidMasse moléculaire :598.543'-O-Decarbamoylirumamycin
CAS :3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.Formule :C40H64O11Couleur et forme :SolidMasse moléculaire :720.93Flavipucine
CAS :Flavipucine (Flavipucin) is a glutarimide antibiotic found in the Aspergillus flavipes F-2090/7 strain. It exhibits antibacterial activity against Bacillus subtilis, possesses antiprotozoal properties, and demonstrates cytotoxic effects on various cancer cells.Formule :C12H15NO4Couleur et forme :SolidMasse moléculaire :237.252SphK2-IN-1
CAS :<p>SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.</p>Formule :C23H22ClF3N8OCouleur et forme :SolidMasse moléculaire :518.92L-744832
CAS :<p>L-744832, also known as L-744,832, is a potent Farnesyltransferase inhibitor with potential anticancer activity.</p>Formule :C26H45N3O6S2Couleur et forme :SolidMasse moléculaire :559.78Anti-Trypanosoma cruzi agent-1
<p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49Mevidalen HBA
CAS :<p>Mevidalen (LY3154207), a potent D1 positive allosteric modulator, is in clinical trials for Lewy body dementia.</p>Formule :C31H35Cl2NO6Couleur et forme :SolidMasse moléculaire :588.52Trk-IN-8
<p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>Formule :C18H16F2N6O2Couleur et forme :SolidMasse moléculaire :386.36S-1033
CAS :<p>S-1033 is an FP receptor agonist.</p>Formule :C20H33NaO4Couleur et forme :SolidMasse moléculaire :360.4698Artemisiane E
CAS :Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .Formule :C20H22O5Couleur et forme :SolidMasse moléculaire :342.39LLS30
CAS :<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Formule :C34H33Cl4N5O3Couleur et forme :SolidMasse moléculaire :701.47P-gp inhibitor 2
CAS :Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formule :C29H26N2O6Couleur et forme :SolidMasse moléculaire :498.53STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formule :C17H12N4O4Couleur et forme :SolidMasse moléculaire :336.3DC1SMe
CAS :<p>DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.</p>Formule :C35H30ClN5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :684.23Pyrrolomycin E
CAS :<p>Pyrrolomycin E is a pyrrole-based antibiotic with activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Formule :C10H5Cl3N2O3Couleur et forme :SolidMasse moléculaire :307.517Avorelin acetate
CAS :Avorelin acetate is a luteinizing hormone releasing hormone (LH-RH) agonist.Formule :C67H89N17O14Couleur et forme :SolidMasse moléculaire :1356.55Jietacin A
CAS :<p>Jietacin A exhibits nematocidal activity, capable of killing Burs helenchus Lignicolus at a concentration of 0.25 μg/mL.</p>Formule :C18H34N2O2Couleur et forme :SolidMasse moléculaire :310.475Monensin C
CAS :Monensin C is an oxygenated heterocyclic polyether antibiotic. It exhibits activity against bacteria, mycobacteria, fungi, and protozoa, though it is less effective against Gram-negative bacteria. Additionally, it shows inhibitory effects on HeLa cells.Formule :C37H64O11Couleur et forme :SolidMasse moléculaire :684.898ITK inhibitor 6
CAS :ITK inhibitor 6 selectively targets ITK, BTK, JAK3, EGFR, LCK, blocks PLCγ1 and ERK1/2 phosphorylation, and inhibits cell proliferation.Formule :C28H24F2N4O2Couleur et forme :SolidMasse moléculaire :486.51Tuvatidine
CAS :Tuvatidine is a histamine 2 receptor antagonist.Formule :C10H17N9O2S3Couleur et forme :SolidMasse moléculaire :391.5SLN124
<p>SLN124, a GalNAc-siRNA targeting TMPRSS6, may normalize iron balance by restoring ferroregulation.</p>Couleur et forme :SolidCLR01 sodium
CAS :CLR01 is a tweezer reducing α-synuclein in MSA, inhibits SOD1 in ALS, blocks Ebola/Zika, stabilizes proteins, and lessens mutant p53 toxicity.Formule :C42H30Na2O8P2Couleur et forme :SolidMasse moléculaire :770.6211mPGES-1-IN-1
MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.Formule :C21H14N4O2SCouleur et forme :SolidMasse moléculaire :386.43XN methyl pyrazole
<p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>Formule :C22H24N2O4Couleur et forme :SolidMasse moléculaire :380.44DI-404
CAS :DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.Formule :C35H45ClN6O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :713.29AS1940477
CAS :<p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>Formule :C24H22FN5O2Couleur et forme :SolidMasse moléculaire :431.46TrxR-IN-2
TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.Formule :C22H22N4O4Couleur et forme :SolidMasse moléculaire :406.43TCMDC-135051 TFA (2413716-15-9 free base)
TCMDC-135051 TFA is a highly selective and potent inhibitor of protein kinase PfCLK3.Formule :C31H34F3N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :585.61TCMDC-136230
TCMDC-136230 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystallisation.Formule :C24H34N4O2SCouleur et forme :SolidMasse moléculaire :442.62Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).Formule :C18H17N3O4S2Couleur et forme :SolidMasse moléculaire :403.48SX 3202
CAS :<p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>Formule :C17H11BrFN3O4Couleur et forme :SolidMasse moléculaire :420.19AX15910
AX15910 is a potent inhibitor of BRD4 and ERK5.Formule :C32H38N6O3Couleur et forme :SolidMasse moléculaire :554.7Antimalarial agent 9
<p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>Formule :C28H32BrN3O2Couleur et forme :SolidMasse moléculaire :522.48ATX inhibitor 12
<p>Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.</p>Formule :C30H34FN5O2Couleur et forme :SolidMasse moléculaire :515.62Heme Oxygenase-1-IN-3
CAS :<p>Heme Oxygenase-1-IN-3 (compound 4) serves as a potent and selective inhibitor of heme oxygenase-1 (HO-1) with a dissociation constant (Kd) of 141 nM, making it suitable for use in cancer and neurodegenerative disease research.</p>Formule :C22H18BrFN4O2SCouleur et forme :SolidMasse moléculaire :501.37AGN-204396
CAS :AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).Formule :C32H44FN3O4Couleur et forme :SolidMasse moléculaire :553.71Erabulenol A
CAS :<p>Erabulenol A is a cholesterol ester transfer protein (CETP) inhibitor, extracted from Penicillumsp.</p>Formule :C20H20O6Couleur et forme :SolidMasse moléculaire :356.369ODN 21158
CAS :<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Couleur et forme :SolidHypoglycemic agent 1
CAS :Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.Formule :C25H24FN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.49Lobaric acid
CAS :<p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48Fumaryl-DL-alanine
CAS :Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.Formule :C7H9NO5Couleur et forme :SolidMasse moléculaire :187.15UNC9426
CAS :<p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>Formule :C32H34F6N6ODegré de pureté :98.051%Couleur et forme :SolidMasse moléculaire :632.642KOS-1584
CAS :KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.Formule :C27H39NO5SCouleur et forme :SolidMasse moléculaire :489.67GSK3527497 HCl
CAS :<p>GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.</p>Formule :C17H17Cl2FN4O4SCouleur et forme :SolidMasse moléculaire :463.3054Pyloricidin A2
CAS :Pyloricidin A2 is an antibiotic effective against Helicobacter pylori, produced by Bacillus species HC-70. It exhibits strong anti-Helicobacter pylori activity but shows no activity against other bacteria and yeast.Formule :C32H53N5O10Couleur et forme :SolidMasse moléculaire :667.79Calphostin I
CAS :Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.Formule :C44H38O15Couleur et forme :SolidMasse moléculaire :806.76SP inhibitor 1
<p>SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.</p>Formule :C36H38N2O2Couleur et forme :SolidMasse moléculaire :530.7SGK1-IN-3
SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.Formule :C23H20Cl2N6O3SCouleur et forme :SolidMasse moléculaire :531.41Vimirogant hydrochloride
Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), >1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.Formule :C27H36ClF3N4O3SCouleur et forme :SolidMasse moléculaire :588.21487Trypanothione synthetase-IN-4
Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).Formule :C29H52INO2Couleur et forme :SolidMasse moléculaire :573.63B-3852
CAS :B-3852 is a Bradykinin inhibitor.Formule :C55H74F3N15O11Couleur et forme :SolidMasse moléculaire :1178.27Lunacalcipol
CAS :Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.Formule :C28H42O4SCouleur et forme :SolidMasse moléculaire :474.7Nanaomycin B
CAS :<p>Nanaomycin B is an antibiotic with activity against Gram-positive bacteria, mycobacteria, mycoplasma, and fungi.</p>Formule :C16H16O7Couleur et forme :SolidMasse moléculaire :320.294JBIR-22
CAS :<p>JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.</p>Formule :C23H33NO6Couleur et forme :SolidMasse moléculaire :419.511,6-Dihydroxy-2-chlorophenazine
CAS :<p>1,6-Dihydroxy-2-chlorophenazine exhibits weak antifungal and anti-yeast activity.</p>Formule :C12H7ClN2O2Couleur et forme :SolidMasse moléculaire :246.65Human carbonic anhydrase II-IN-1
Compound S-13: Potent hCA II inhibitor, Kis 4.4, 9.2, 480.2, 14.7 nM for hCA II, I, IV, IX. Used in glaucoma research.Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5Topoisomerase I/II inhibitor 2
<p>Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.</p>Formule :C19H16N2O4Couleur et forme :SolidMasse moléculaire :336.34Antiangiogenic agent 3
Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.Formule :C19H20O7Couleur et forme :SolidMasse moléculaire :360.36Cytosaminomycin B
CAS :<p>Cytosaminomycin B exhibits activity against Eimeria Tenella coccidia.</p>Formule :C26H37N5O8Couleur et forme :SolidMasse moléculaire :547.601Trk-IN-7
<p>Trk-IN-7 inhibits TRKA/B/C (IC50: 0.25-10 nM) & EML4-ALK (<15 nM), also targets various ALK mutations (IC50: 5-50 nM).</p>Formule :C18H17FN6O2Couleur et forme :SolidMasse moléculaire :368.36MMG-11 quarterhydrate
<p>MMG-11 quarterhydrate, a potent hTLR2 antagonist, inhibits TLR2/1 and TLR2/6 with IC50s of 1.7μM and 5.7μM; low toxicity.</p>Formule :C15H16O8Couleur et forme :SolidMasse moléculaire :310.78Tembotrione
CAS :<p>Tembotrione is a chemical compound that may reduce the productivity of carrots. It possesses activity that degrades the quality of carrot stems. Additionally, Tembotrione can be used in studies focusing on the overall productivity of carrot cultivation.</p>Formule :C17H16ClF3O6SCouleur et forme :SolidMasse moléculaire :440.82Vitamin A Propionate
CAS :<p>Vitamin A Propionate, an ester derivative of vitamin A, exhibits varying effects on growth, serum biochemistry, and hematological indices in foal nutrition studies depending on the dosage administered. Both excessively high and low doses lead to adverse impacts. These effects are correlated with the concentrations of vitamin A in the plasma, liver, and kidneys.</p>Formule :C23H34O2Couleur et forme :SolidMasse moléculaire :342.51trans-Doxercalciferol
CAS :trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.Formule :C28H44O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.65RIPK1-IN-26
CAS :<p>RIPK1-IN-26 is a potent inhibitor of Receptor-Interacting Serine/Threonine Kinase 1 (RIPK1), exhibiting anti-necrotic properties in cells. This compound demonstrates good metabolic stability and binding specificity in mice. RIPK1-IN-26 holds potential for development as a PET imaging probe and in the research of neurodegenerative diseases.</p>Formule :C15H20FNO2Couleur et forme :SolidMasse moléculaire :265.32ABCA1 inducer 1
CAS :<p>ABCA1 inducer 1, a non-lipid inducer of ABCA1, enhances ABCA1 expression in E3/4FAD mice expressing human APOE 3/4, augments the lipidation of apolipoprotein (APOE), and reverses various Alzheimer's disease (AD) phenotypes without increasing triglycerides.</p>Formule :C24H24Cl2N2O7S2Couleur et forme :SolidMasse moléculaire :587.49P-gp modulator 3
P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.Formule :C31H37N3O5Couleur et forme :SolidMasse moléculaire :531.64Hynapene A
CAS :Hynapene A exhibits an inhibitory minimum inhibitory concentration (MIC) of 123 μM against Eimeria tenella.Formule :C18H28O5Couleur et forme :SolidMasse moléculaire :324.412MRS2279
CAS :Selective, high affinity competitive antagonist of the P2Y1 receptorFormule :C13H18ClN5O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :469.71GPX100 HCl
CAS :GPX-100, a non-cardiotoxic doxorubicin analog, intercalates DNA and inhibits replication, repair, and protein synthesis.Formule :C27H32ClNO10Couleur et forme :SolidMasse moléculaire :566Sannamycin K
CAS :<p>Sannamycin K is an aminoglycoside antibiotic with weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C13H26N4O4Couleur et forme :SolidMasse moléculaire :302.3712(S)-HEPE
CAS :<p>12(S)-HEPE, made from EPA by 12-LO, is an anti-inflammatory ω-3 derivative affecting leukotriene formation.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45Azonafide-PEABA
CAS :<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formule :C32H33N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :551.64Odiparcil
CAS :Odiparcil is an orally active beta-d-thioxyloside analog.Formule :C15H16O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.35Tribenuron
CAS :<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Formule :C14H15N5O6SCouleur et forme :SolidMasse moléculaire :381.36PD-1/PD-L1-IN-16
PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.Formule :C34H30N4O4Couleur et forme :SolidMasse moléculaire :558.63Hydroxyethyl disulfide
CAS :Hydroxyethyl disulfide can counteract the inhibitory effects of showdomycin on methotrexate-resistant thymidylate synthase and is protected from deactivation by its substrate, deoxyuridine monophosphate, thus preserving the antibiotic's activity.Formule :C4H10O2S2Couleur et forme :SolidMasse moléculaire :154.254-Chloropyridine
CAS :4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.Formule :C5H4ClNCouleur et forme :SolidMasse moléculaire :113.55Epithienamycin C
CAS :<p>Epithienamycin C is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C13H18N2O5SCouleur et forme :SolidMasse moléculaire :314.357Quorum Sensing-IN-1
Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.Formule :C13H10N2O2S2Couleur et forme :SolidMasse moléculaire :290.36ZK-Thiazolidinone
CAS :ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.Formule :C23H26F3N5O2SCouleur et forme :SolidMasse moléculaire :493.55Antimalarial agent 2
Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.Formule :C27H25N3O5Couleur et forme :SolidMasse moléculaire :471.5SAR107375
CAS :SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].Formule :C24H30ClN5O5S2Couleur et forme :SolidMasse moléculaire :568.11RSV-IN-5
CAS :<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Formule :C28H37N7O2Couleur et forme :SolidMasse moléculaire :503.64O-Demethylpaulomycin A
CAS :O-Demethylpaulomycin A is an antibiotic known for its antibacterial properties. It is particularly effective against Gram-positive bacteria, including Staphylococcus aureus.Formule :C33H44N2O17SCouleur et forme :SolidMasse moléculaire :772.771Rimegepant sulfate hydrate
CAS :<p>Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.</p>Formule :C56H64F4N12O13SCouleur et forme :SolidMasse moléculaire :1221.2526Hydranthomycin
CAS :Hydranthomycin is an antibiotic with moderate antifungal activity, exhibiting a minimum inhibitory concentration (MIC) of 25 μg/mL against the rice blast fungus. Additionally, it inhibits the growth of Chlorella (tiny naked algae) and possesses herbicidal properties.Formule :C20H20O5Couleur et forme :SolidMasse moléculaire :340.37AZ0108
CAS :AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.Formule :C24H20F4N6O2Couleur et forme :SolidMasse moléculaire :500.45Chitinovorin C
CAS :Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.Formule :C15H20N4O8SCouleur et forme :SolidMasse moléculaire :416.406Clavalanine
CAS :Clavalanine (Ro 22-5417) is capable of inhibiting various bacteria and fungi.Formule :C8H12N2O4Couleur et forme :SolidMasse moléculaire :200.192Epithienamycin D
CAS :Epithienamycin D is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C13H16N2O5SCouleur et forme :SolidMasse moléculaire :312.342Deoxyfrenolicin
CAS :Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.Formule :C18H18O6Couleur et forme :SolidMasse moléculaire :330.332Theophylline EP impurity C
CAS :Theophylline EP impurity C, an alkaloid with anti-bronchospasm activity, is employed to assess the purity and quality of compounds. This substance also holds potential clinical value in the management of asthma and chronic obstructive pulmonary disease (COPD).Formule :C7H10N4O3Couleur et forme :SolidMasse moléculaire :198.18Propizepine
CAS :Propizepine is a tricyclic antidepressant compound.Formule :C17H20N4OCouleur et forme :SolidMasse moléculaire :296.37Nonsteroidal aromatase inhibitor 1
Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.Formule :C22H16N4O2Couleur et forme :SolidMasse moléculaire :368.3916(R)-Iloprost
CAS :<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49UTPγS trisodium salt
CAS :P2Y2 and P2Y4 receptor agonistFormule :C9H12N2Na3O14P3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :566.15CGP 22979
CAS :CGP 22979 is a renal selective vasodilator prodrug.Formule :C16H24N4O4Couleur et forme :SolidMasse moléculaire :336.39Terfluranol
CAS :Terfluranol, a benzyl derivative, is utilized as an antitumor medication.Formule :C17H17F3O2Couleur et forme :SolidMasse moléculaire :310.31L-690330 hydrate
L-690330 hydrate inhibits IMPase; Ki: 0.30 μM (human), 0.42 μM (bovine cortex); 0.27 μM (recom. human), 0.19 μM (bovine).Formule :C8H14O9P2Couleur et forme :SolidMasse moléculaire :316.14PEN-866
CAS :PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.Formule :C49H49N7O9Couleur et forme :SolidMasse moléculaire :879.95hTrkA-IN-2
<p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>Formule :C24H22F3N5O3Couleur et forme :SolidMasse moléculaire :485.46MSX-3 free acid
CAS :MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.Formule :C21H23N4O7PCouleur et forme :SolidMasse moléculaire :474.40Oral antiplatelet agent 1
CAS :Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.Formule :C23H24N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.53Epicorazine A
CAS :Epicorazine A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, showing an MIC of 25 μg/mL.Formule :C18H16N2O6S2Couleur et forme :SolidMasse moléculaire :420.459Teprosulvose
CAS :Teprosulvose is a radiosensitizer used in veterinary medicine.Formule :C27H52O10SCouleur et forme :SolidMasse moléculaire :568.76DJT06001
CAS :DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.Formule :C21H20ClN3O5SCouleur et forme :SolidMasse moléculaire :461.92Anticancer agent 28
Anticancer agent 28 is 50x more potent than Oridonin, IC50 of 0.09 μM against K562; effective in H22 mouse tumors.Formule :C28H33NO6Couleur et forme :SolidMasse moléculaire :479.56
