Autres inhibiteurs
Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.
35951 produits trouvés pour "Autres inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
SHR0687
CAS :SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.Formule :C39H60N8O5Couleur et forme :SolidMasse moléculaire :720.94SOAT-IN-1
CAS :SOAT-IN-1 (compound 40) is a potent and selective inhibitor targeting the sodium-dependent organic anion transporter (SOAT), exhibiting IC50 values of 1.6 µM for SOAT and 14.3 µM for NTCP.Formule :C20H16ClN3O6SCouleur et forme :SolidMasse moléculaire :461.884-Nitrochalcone
CAS :4-Nitrochalcone (2-(4-Nitrobenzylidene)acetophenone) inhibits proteasomes and suppresses TNFα-induced NF-κB activity.Formule :C15H11NO3Couleur et forme :SolidMasse moléculaire :253.25Hydroxymycotrienin B
CAS :Hydroxymycotrienin B is an ansamycin antibiotic that exhibits activity against human neck tumor cell lines, showing stronger inhibitory effects on human papillomavirus (HPV) gene-positive neck tumor cells, such as HeLa, CaSKi, and SiHa, compared to HPV gene-negative cells.
Formule :C36H48N2O9Couleur et forme :SolidMasse moléculaire :652.774LY2934747
CAS :LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.Formule :C10H13NO4Couleur et forme :SolidMasse moléculaire :211.21HR-546
CAS :HR-546 is a prostaglandin E2 and prostaglandin F2alpha antagonist.Formule :C26H44O6Couleur et forme :SolidMasse moléculaire :452.62ALK5-IN-7
CAS :ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.Formule :C26H28N4O3SCouleur et forme :SolidMasse moléculaire :476.59THR-β agonist 5
CAS :THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].Formule :C22H23N5O2Couleur et forme :SolidMasse moléculaire :389.4522-HDHA
CAS :22-HDHA is an oxidation product of docosahexaenoic acid .Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.49DC1SMe
CAS :DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.Formule :C35H30ClN5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :684.23O-Demethylpaulomycin A
CAS :O-Demethylpaulomycin A is an antibiotic known for its antibacterial properties. It is particularly effective against Gram-positive bacteria, including Staphylococcus aureus.Formule :C33H44N2O17SCouleur et forme :SolidMasse moléculaire :772.771Haloquinone
CAS :Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.Formule :C17H12O5Couleur et forme :SolidMasse moléculaire :296.274Avorelin acetate
CAS :Avorelin acetate is a luteinizing hormone releasing hormone (LH-RH) agonist.Formule :C67H89N17O14Couleur et forme :SolidMasse moléculaire :1356.55Evategrel
CAS :Evategrel is an inhibitor of platelet aggregation.Formule :C21H26ClNO7SCouleur et forme :SolidMasse moléculaire :471.95Tofogliflozin
CAS :Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44Lucilactaene
CAS :Lucilactaene exhibits potent antimalarial activity and functions as a P53-transfected tumor cell cycle inhibitor. It effectively halts the cell cycle progression of H1299/TSP53 cells at the G1 phase.Formule :C22H27NO6Couleur et forme :SolidMasse moléculaire :401.45Dermostatin B
CAS :Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.Formule :C41H66O11Couleur et forme :SolidMasse moléculaire :734.956Pochonin D
CAS :Pochonin D is an inhibitor of heat shock protein 90 (Hsp90) with antiviral and anti-inflammatory properties. It disrupts Hsp90, affecting the stability, folding, and assembly of viral proteins, thereby diminishing viral replication. Additionally, Pochonin D reduces the infiltration of inflammatory cells and decreases the secretion of inflammatory cytokines such as TNF-α and IL-1β, alleviating inflammatory responses. This compound shows potential for research in human rhinovirus (HRV) infections and cancer.
Formule :C18H19ClO5Couleur et forme :SolidMasse moléculaire :350.793AS1940477
CAS :AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.Formule :C24H22FN5O2Couleur et forme :SolidMasse moléculaire :431.46Cinatrin A
CAS :Cinatrin A exhibits inhibitory activity against phospholipase A2 (phospholipaseA2).Formule :C18H26O8Couleur et forme :SolidMasse moléculaire :370.394Nonsteroidal aromatase inhibitor 1
Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.Formule :C22H16N4O2Couleur et forme :SolidMasse moléculaire :368.39PBX-7011
CAS :PBX-7011, an active camptothecin derivative, binds to the DDX5 protein in cells and induces cell death through DDX5 protein degradation [1].Formule :C24H21N3O6Couleur et forme :SolidMasse moléculaire :447.44Teprosulvose
CAS :Teprosulvose is a radiosensitizer used in veterinary medicine.Formule :C27H52O10SCouleur et forme :SolidMasse moléculaire :568.76ZK159222
CAS :ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.Formule :C32H48O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.72Enpp-1-IN-11
Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.Formule :C15H15N5O3SCouleur et forme :SolidMasse moléculaire :345.38Antimalarial agent 9
Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.Formule :C28H32BrN3O2Couleur et forme :SolidMasse moléculaire :522.48Belatacept
CAS :Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.Couleur et forme :LiquidCalphostin A
CAS :Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.Formule :C44H38O12Couleur et forme :SolidMasse moléculaire :758.77AL-6556
CAS :AL-6556 is a prostaglandin DP receptor agonist.Formule :C20H33ClO5Couleur et forme :SolidMasse moléculaire :388.93Piloquinone
CAS :Piloquinone is a type of phenanthrene compound that exhibits mild inhibitory effects on mycobacteria and protozoa.Formule :C21H20O5Couleur et forme :SolidMasse moléculaire :352.38CGS 22652
CAS :CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.Formule :C22H29ClN2O4SCouleur et forme :SolidMasse moléculaire :452.99Carmegliptin dihydrochloride
CAS :Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.Formule :C20H30Cl2FN3O3Couleur et forme :SolidMasse moléculaire :450.384"-Demethylgentamicin C2
CAS :4"-Demethylgentamicin C2 exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C19H39N5O7Couleur et forme :SolidMasse moléculaire :449.54eIF4A3-IN-4
eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).Formule :C24H20N2O5Couleur et forme :SolidMasse moléculaire :416.43Glasmacinal
CAS :Glasmacinal is a non-antibacterial macrolide compound with anti-inflammatory activities.Formule :C37H62N2O10Couleur et forme :SolidMasse moléculaire :694.90ORP-101
CAS :ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.Formule :C60H84N2O8Couleur et forme :SolidMasse moléculaire :961.32GSK 932121
CAS :GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.Formule :C20H15ClF3NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.79MK-7445
CAS :MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.Formule :C21H13Cl2N7OCouleur et forme :SolidMasse moléculaire :450.28eIF4A-IN-3
CAS :eIF4A-IN-3 (Compound 71E) is an inhibitor of the eukaryotic translation initiation factor 4A (eIF4A). This compound can be utilized as a cytotoxic payload for antibody-drug conjugates (ADCs).Formule :C34H37N3O7Couleur et forme :SolidMasse moléculaire :599.67Hexedine
CAS :Hexedine is a biochemical.Formule :C22H45N3Couleur et forme :SolidMasse moléculaire :351.61P2X receptor-1
P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.Formule :C14H14ClN3O3S2Couleur et forme :SolidMasse moléculaire :371.86Plm IV inhibitor-2
CAS :"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."Formule :C39H54N4O4Couleur et forme :SolidMasse moléculaire :642.872-Acetoxyacorenone
CAS :2-Acetoxyacorenone (compound 8) is a sesquiterpenoid compound that can be isolated from the rhizomes of Acorus tatarinowii. It exhibits potential inhibition activity against AChE and β-BACE1, making it useful for Alzheimer's disease research.Formule :C17H26O3Couleur et forme :SolidMasse moléculaire :278.39Kurasoin A
CAS :Kurasoin A is an inhibitor of the enzyme farnesyltransferase.Formule :C16H16O3Couleur et forme :SolidMasse moléculaire :256.296Hazimycin 6
CAS :Hazimycin 6 exhibits weak activity against gram-negative bacteria, yeast, and dermatophytes.Formule :C20H18N4O4Couleur et forme :SolidMasse moléculaire :378.381TA-316
CAS :Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.Formule :C28H25BrN4O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.56Griseolutein A
CAS :Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C17H14N2O6Couleur et forme :SolidMasse moléculaire :342.303BRD-9526
CAS :BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formule :C26H31Cl2N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.51Piptamine
CAS :Piptamine exhibits a broad antibacterial spectrum, with inhibitory MIC (μg/mL) values against various microorganisms as follows: Staphylococcus aureus (0.78-6.25), Enterococcus faecalis (1.56), Bacillus subtilis (1.00), Escherichia coli (12.5), and Candida albicans (6.25).Formule :C20H35N3Couleur et forme :SolidMasse moléculaire :317.51AGN-795
CAS :AGN-795 is a biochemical.Formule :C14H20N2Couleur et forme :SolidMasse moléculaire :216.328Antioxidant agent-3
Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.Formule :C18H14O8Couleur et forme :SolidMasse moléculaire :358.3GZN39838
CAS :GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.Formule :C22H30O6Couleur et forme :SolidMasse moléculaire :390.47Demycarosyl platenomycin
CAS :Demycarosylplatenomycin (DM-PLM) is an antibiotic that exhibits mild activity against Gram-positive bacteria.Formule :C31H51NO11Masse moléculaire :613.74Calphostin I
CAS :Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.Formule :C44H38O15Couleur et forme :SolidMasse moléculaire :806.76Cilobamine (free base)
CAS :Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.Formule :C17H23Cl2NOCouleur et forme :SolidMasse moléculaire :328.28P7170
CAS :P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.Formule :C21H16F3N9Couleur et forme :SolidMasse moléculaire :451.42Pelagiomicin C
CAS :Pelagiomicin C exhibits activity against both Gram-positive and Gram-negative bacteria.Formule :C17H15N3O5Couleur et forme :SolidMasse moléculaire :341.318PI3Kβ-IN-1
CAS :PI3Kβ-IN-1 is a selective, orally active PI3Kβ inhibitor (IC50: 2 nM).Formule :C25H14F2N8Couleur et forme :SolidMasse moléculaire :464.43LXR antagonist 2
LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).
Formule :C34H40N2O5SCouleur et forme :SolidMasse moléculaire :588.76U 80215
CAS :U 80215 is an enzyme-competitive inhibitor.Formule :C42H60N8O6SCouleur et forme :SolidMasse moléculaire :805.04Deoxyfrenolicin
CAS :Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.Formule :C18H18O6Couleur et forme :SolidMasse moléculaire :330.332Antitumor agent-65
CAS :Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.Formule :C18H17NO10Couleur et forme :SolidMasse moléculaire :407.332,3-dinor-11β-Prostaglandin F2α
CAS :2,3-dinor-11β-Prostaglandin F2α (2,3-dinor-11β-PGF2α) was recovered from the urine of both normal monkeys and humans when infused with radiolabeled PGD2, whereFormule :C18H30O5Couleur et forme :SolidMasse moléculaire :326.43ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formule :C29H33ClF2N6O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :683.06Rosiptor acetate
CAS :Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.Formule :C22H39NO4Degré de pureté :98%Couleur et forme :Solid PowderMasse moléculaire :381.55L 767679
CAS :L 767679 is an antagonist of the fibrinogen receptors.Formule :C20H24N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :384.43Topoisomerase I/II inhibitor 2
Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.Formule :C19H16N2O4Couleur et forme :SolidMasse moléculaire :336.34D18
CAS :D18: Dual agonist for TLR7/8, boosts PD-L1, aids tumor sensitivity to PD-1/PD-L1 inhibitors, and is a cytotoxin for ADC HE-S2.Formule :C21H28N6Couleur et forme :SolidMasse moléculaire :364.4916(R)-Iloprost
CAS :Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49Feigrisolide C
CAS :Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.Formule :C21H36O7Couleur et forme :SolidMasse moléculaire :400.506Annonin VI
CAS :Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.Formule :C37H66O7Couleur et forme :SolidMasse moléculaire :622.92Tonantzitlolone
CAS :Tonantzitlolone activates TRPC1/4/5 channels, PKCα/θ, inhibits IRS1/PI3K/AKT, and triggers HSF1 to induce glucose dependence.Formule :C26H40O7Couleur et forme :SolidMasse moléculaire :464.59NRX-2663
CAS :NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).Formule :C20H13F3N2O5Couleur et forme :SolidMasse moléculaire :418.32SSR-182289A (Free)
CAS :SSR-182289A (Free) is a thrombin inhibitor.Formule :C30H33F2N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.68UH 301
CAS :UH 301 is a 5-HT1A receptor antagonist.Formule :C16H24FNOCouleur et forme :SolidMasse moléculaire :265.37iMDK quarterhydrate
iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.Formule :C21H15FN2O3SCouleur et forme :SolidMasse moléculaire :380.91Pentenocin A
CAS :Pentenocin A exhibits a relatively weak inhibitory effect on IL-1 and β-glucuronidase (ICE) activity.Formule :C7H10O5Couleur et forme :SolidMasse moléculaire :174.151Hypoglycemic agent 1
CAS :Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.Formule :C25H24FN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.49PD-1/PD-L1-IN-16
PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.Formule :C34H30N4O4Couleur et forme :SolidMasse moléculaire :558.63TRPC4/5-IN-1
TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.Formule :C21H21N3OCouleur et forme :SolidMasse moléculaire :331.41ZIKV-IN-4
ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.Formule :C33H37NO4Couleur et forme :SolidMasse moléculaire :511.65MEIS-IN-3
MEIS-IN-3 is a potent inhibitor of MEIS.Formule :C25H26N2O4Couleur et forme :SolidMasse moléculaire :418.48Mutatochrome
CAS :Mutatochrome (Citroxanthin) is a compound found in plants.Formule :C40H56OCouleur et forme :SolidMasse moléculaire :552.872Juglomycin B
CAS :Juglomycin B exhibits broad-spectrum antibacterial and antimycobacterial properties and is capable of inhibiting Ehrlich ascites carcinoma in mice.
Formule :C14H10O6Couleur et forme :SolidMasse moléculaire :274.226Mopivabil
Mopivabil is the angiotensin II receptor antagonist[1].Formule :C14H20O3Couleur et forme :SolidMasse moléculaire :236.31SARS-CoV-2-IN-8
SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).Formule :C35H38N6O3Couleur et forme :SolidMasse moléculaire :590.71Epicochlioquinone A
CAS :Epicochlioquinone A inhibits rat liver microsomal ACAT with an IC50 of 1.7 μM and inhibits plasma lecithin-cholesterol acyltransferase (LCAT) with an IC50 of 15.8 μM. At a dosage of 75 mg/kg, it can reduce cholesterol absorption in rats by 50%.Formule :C30H44O8Couleur et forme :SolidMasse moléculaire :532.666GW311616 hydrochloride
CAS :GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formule :C19H32ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.99Dinordrin
CAS :Dinordrin is an implantation inhibitor and hormone.Formule :C27H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.57Isoleucyl tRNA synthetase-IN-2
CAS :Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).Formule :C22H33N5O8SCouleur et forme :SolidMasse moléculaire :527.59AKR1C3-IN-5
AKR1C3-IN-5 inhibits AKR1C3, key in prostate/breast cancers, with MCF-7 cell IC50 of 9.6 μM.Formule :C34H44N2O7Couleur et forme :SolidMasse moléculaire :592.72ER272
CAS :ER272 is a natural PKC activator, inducing hippocampal neurogenesis.Formule :C24H34O6Couleur et forme :SolidMasse moléculaire :418.52AMG-222 tosylate
CAS :AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.Formule :C39H47N9O6SCouleur et forme :SolidMasse moléculaire :769.91BW A868C
CAS :BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formule :C25H37N3O5Couleur et forme :SolidMasse moléculaire :459.58GW-597901 cinnamate
CAS :GW-597901 cinnamate is a long-acting beta(2)-agonist.Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80SENP2-IN-1
CAS :SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.Formule :C32H29N3O5S2Couleur et forme :SolidMasse moléculaire :599.72Crotocin
CAS :Crotocin exhibits bactericidal activity against Cryptococcus neoformans, Candida albicans, and Saccharomyces cerevisiae (brewer’s yeast), but it can be inactivated by blood.Formule :C19H24O5Couleur et forme :SolidMasse moléculaire :332.391Polyoxin L
CAS :Polyoxin L is a nucleoside-type antifungal antibiotic that is notably effective against rice sheath blight.Formule :C16H23N5O12Masse moléculaire :477.38Revamilast sodium
CAS :Revamilast sodium, also known as GRC4039 sodium, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritisFormule :C18H8Cl2F2N3NaO4Couleur et forme :SolidMasse moléculaire :462.17Antiviral agent 7
Antiviral agent 7 is a peptide-based coating that kills viruses.Formule :C29H31F2N3O6Couleur et forme :SolidMasse moléculaire :555.57PGDM
CAS :PGD2 is involved in allergy, asthma, sleep, temperature regulation, inhibits clotting, and relaxes blood vessels; PGDM, its metabolite, is a biomarker.Formule :C16H24O7Couleur et forme :SolidMasse moléculaire :328.36A 74273
CAS :A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.Formule :C44H74N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :787.08Protease-Activated Receptor-1 antagonist 1
Compound 13 is a PAR-1 antagonist with a 3 nM IC50, useful for thrombosis and heart disease research.Formule :C25H24F2N2O3Couleur et forme :SolidMasse moléculaire :438.47GS-9160
CAS :GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.Formule :C20H18FN3O4SCouleur et forme :SolidMasse moléculaire :415.44Topoisomerase I inhibitor 8
CAS :Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.Formule :C24H21FN2O4Couleur et forme :SolidMasse moléculaire :420.43FK-906 HCl
CAS :FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.Formule :C40H64ClN7O7Couleur et forme :SolidMasse moléculaire :790.44PD-1/PD-L1-IN-30
CAS :PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53Epicillin
CAS :Epicillin possesses antibacterial activity.Formule :C16H21N3O4SCouleur et forme :SolidMasse moléculaire :351.4215(S),6(S)-DiHETE
CAS :5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47O-Desmethyl Midostaurin
CAS :O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.Formule :C34H28N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.61Purine phosphoribosyltransferase-IN-2
Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.Formule :C11H15N5Na4O10P2Couleur et forme :SolidMasse moléculaire :531.17Pparδ agonist 5
Pparδ agonist 5 is a selective, orally active PPARδ agonist with an EC50 of 0.335 μM and better selectivity than GW0742.Formule :C23H21F3N2O2SCouleur et forme :SolidMasse moléculaire :446.49IDX-320
CAS :IDX-320 is an HCV protease inhibitor.Formule :C37H43F3N6O7S2Couleur et forme :SolidMasse moléculaire :804.9TCMDC-125431
TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.Formule :C25H27N3O2SCouleur et forme :SolidMasse moléculaire :433.57Monamycin D1
CAS :Monamycin D1 is a lipopeptide antibiotic with activity against Gram-positive bacteria.Formule :C34H57N7O8Masse moléculaire :691.86G12Si-1
G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.Formule :C29H32ClN5O3Couleur et forme :SolidMasse moléculaire :534.05DJT06001
CAS :DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.Formule :C21H20ClN3O5SCouleur et forme :SolidMasse moléculaire :461.92Hsp90-IN-16
Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.Formule :C30H26FN3O6Couleur et forme :SolidMasse moléculaire :543.54Nevirapine dimer
CAS :Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).Formule :C30H26N8O2Couleur et forme :SolidMasse moléculaire :530.58PKCiota-IN-1
CAS :PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).Formule :C25H22FN5OCouleur et forme :SolidMasse moléculaire :427.47PPO-IN-1
PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35Chitinase-IN-5
Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.Formule :C20H21ClFN7Couleur et forme :SolidMasse moléculaire :413.88J-104132
CAS :J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.Formule :C31H33NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.60PDE4-IN-14
CAS :PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, includingFormule :C19H20F2N4O3SCouleur et forme :SolidMasse moléculaire :422.45G-4120
CAS :G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.Formule :C26H36N8O11SCouleur et forme :SolidMasse moléculaire :668.68MK-8970
MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.Formule :C25H29FN6O8Couleur et forme :SolidMasse moléculaire :560.54Anticancer agent 28
Anticancer agent 28 is 50x more potent than Oridonin, IC50 of 0.09 μM against K562; effective in H22 mouse tumors.Formule :C28H33NO6Couleur et forme :SolidMasse moléculaire :479.56STING agonist-20
CAS :STING agonist-20: potent, aids in XMT-2056 synthesis, used as a cancer vaccine adjuvant.Formule :C36H39N11O8Couleur et forme :SolidMasse moléculaire :753.76RN941
CAS :RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.Formule :C34H34FN7O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :639.68KFA1982
CAS :KFA1982 is a novel and potent factor Xa inhibitor.Formule :C28H34ClN3O9S2Couleur et forme :SolidMasse moléculaire :656.17Methysergide maleate
CAS :Methysergide prevents migraines/cluster headaches; treats serotonin syndrome, carcinoid-induced diarrhea; risk of fibrosis limits use.Formule :C25H31N3O6Degré de pureté :98%Couleur et forme :White To Off-WhiteMasse moléculaire :469.54Retelliptine
CAS :Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Formule :C25H32N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :404.55ER Thermo Yellow
CAS :ER Thermo Yellow is a high-sensitivity (3.9%/°C) fluorescent probe designed for temperature visualization specifically targeting the endoplasmic reticulum.Formule :C27H20BClF5N3O3Masse moléculaire :575.72Antibacterial agent 70
Antibacterial agent 70 is a new dihydropyrimidinone-imidazole hybrid antimicrobial agent (MIC: 0.5 μg/ml).Formule :C25H32ClN7O6SCouleur et forme :SolidMasse moléculaire :594.08Hcyb1
Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.Formule :C24H20N4OCouleur et forme :SolidMasse moléculaire :380.44TY 11223
CAS :TY 11223: stable homoisocarbacyclin analog, potently inhibits platelet aggregation with lasting effect and selective activity.Formule :C24H34O5Couleur et forme :SolidMasse moléculaire :402.52KF 20274
CAS :KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.Formule :C21H29N5OCouleur et forme :SolidMasse moléculaire :367.49PARP10/15-IN-1
PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].Formule :C13H10N2O3SCouleur et forme :SolidMasse moléculaire :274.3L 739749
CAS :L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.Formule :C24H41N3O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.73TRPV1 antagonist 3
TRPV1 antagonist 3 (7q) strongly blocks TRPV1 at 2.66 nM IC50, is selective, 60% bioavailable, and crosses the blood-brain barrier.Formule :C23H25N3OSCouleur et forme :SolidMasse moléculaire :391.53Oncopterin
CAS :Oncopterin is found in urine from patients with solid and blood cancers.Formule :C12H18N6O3Couleur et forme :SolidMasse moléculaire :294.31Sucistil
Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].Formule :C9H15NO4SCouleur et forme :SolidMasse moléculaire :233.289-O-Demethyltrigonostemone
CAS :9-O-Demethyltrigonostemone is a natural IDO1 inhibitor, cytotoxic and antiplasmodial agent from the Roots of Strophioblachia fimbricalyx.Formule :C19H20O4Couleur et forme :SolidMasse moléculaire :312.36Antibiotic MA 144M2
CAS :Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.Formule :C42H55NO16Couleur et forme :SolidMasse moléculaire :829.88Fleephilone
CAS :Fleephilone is a fungal metabolite isolated from Trichoderma harzianum. It acts as an HIV REV/RRE binding inhibitor, hindering the interaction between REV protein and RRE RNA with an IC50 of 7.6 μM.Formule :C24H27NO7Couleur et forme :SolidMasse moléculaire :441.474Cilobamine mesylate
CAS :Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.Formule :C18H27Cl2NO4SCouleur et forme :SolidMasse moléculaire :424.38D6808
D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.Formule :C30H25F3N6O2Couleur et forme :SolidMasse moléculaire :558.55FTO-IN-6
CAS :FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).Formule :C14H12N4O6Couleur et forme :SolidMasse moléculaire :332.27Cenicriviroc Sulfone
CAS :Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.Formule :C41H52N4O5SCouleur et forme :SolidMasse moléculaire :712.94Lactoquinomycin B
CAS :Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.Formule :C24H27NO9Couleur et forme :SolidMasse moléculaire :473.473Lp-PLA2-IN-10
Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.Formule :C21H15F5N4O4Couleur et forme :SolidMasse moléculaire :482.36Luffariellolide
CAS :Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.Formule :C25H38O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.57Esorubicin
CAS :Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.Formule :C27H29NO10Couleur et forme :SolidMasse moléculaire :527.52VEGFR-2-IN-5 hydrochloride
VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.Formule :C19H25ClN8Couleur et forme :SolidMasse moléculaire :400.91Dup-714
CAS :Dup-714 is a thrombin inhibitor.Formule :C21H33BN6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.33TAM&Met-IN-1
CAS :TAM&Met-IN-1 inhibits AXL, MER, TYRO3 with IC50s 6.1, 13.2, 21.6 nM, respectively, for cancer research.Formule :C29H27F2N7O5Couleur et forme :SolidMasse moléculaire :591.57Monamycin H2
CAS :Monamycin H2 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.Formule :C34H56ClN7O8Masse moléculaire :726.30Griseorhodin G
CAS :Griseorhodin G is a quinone antibiotic with antitumor activity.Formule :C25H18O12Masse moléculaire :510.40AG-7404
CAS :AG-7404: strong protease inhibitor, fights poliovirus, EC50 0.080-0.674 μM, effective on V-073-resistant strains.Formule :C26H29N5O7Couleur et forme :SolidMasse moléculaire :523.54Dictyopanine A
CAS :Dictyopanine A exhibits a relatively narrow antibacterial spectrum, demonstrating moderate antimicrobial activity only against certain filamentous fungi and Gram-positive bacteria.Formule :C25H34O5Couleur et forme :SolidMasse moléculaire :414.53ONO-AE1-259 lysine
CAS :ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)Formule :C28H49ClN2O6Couleur et forme :SolidMasse moléculaire :545.15KR-67607
CAS :KR-67607, or NTX-101, is a novel 11β-HSD1 inhibitor that protects against eye injury by reducing cortisol and preserving eye structures.Formule :C24H29Cl2F3N4O4SCouleur et forme :SolidMasse moléculaire :597.484α-PDD
CAS :4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.Formule :C40H64O8Couleur et forme :SolidMasse moléculaire :672.93Vindeburnol
CAS :Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35Arterolane maleate
CAS :Arterolane, an adenosine triphosphatase inhibitor, is used potentially for the treatment of malaria.Formule :C26H40N2O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.612Irinotecan Carboxylate Sodium Salt
CAS :Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.Formule :C33H39N4NaO7Couleur et forme :SolidMasse moléculaire :626.68Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).Formule :C18H17N3O4S2Couleur et forme :SolidMasse moléculaire :403.48Metocurine chloride
CAS :Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.Formule :C40H48Cl2N2O6Couleur et forme :SolidMasse moléculaire :723.72BMS-520
CAS :BMS-520: potent oral S1P1 agonist, effective in rat arthritis and mouse multiple sclerosis model.Formule :C23H17F3N4O4Couleur et forme :SolidMasse moléculaire :470.4SSTR4 agonist 4
CAS :SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.Formule :C19H26N4OCouleur et forme :SolidMasse moléculaire :326.44JBJ-08-178-01
CAS :JBJ-08-178-01, a mutant-selective tyrosine kinase inhibitor, targets (HER2) human epidermal growth factor receptor 2 and exhibits antitumoral activity. This compound not only diminishes HER2's kinase activity and protein levels through the induction of proteasomal degradation of the receptor but also shows promise in non-small-cell lung cancer research.Formule :C31H30N8O3Couleur et forme :SolidMasse moléculaire :562.62GR-112000
CAS :GR-112000 is a peptide-based tachykinin NK2 receptor antagonist.Formule :C30H36N6O3Couleur et forme :SolidMasse moléculaire :528.65Dihydrobisdechlorogeodin
CAS :Dihydrobisdechlorogeodin, produced by the fungus strain [FO-4712] of the genus Acremonium, serves as a herbicide.Formule :C17H16O7Couleur et forme :SolidMasse moléculaire :332.31Naltalimide
CAS :Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.Formule :C28H28N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.53PF-446687
CAS :PF-446687 is a highly selective MC4 receptor (MC4R) agonist.Formule :C28H37ClF2N2O2Couleur et forme :SolidMasse moléculaire :507.06PRN694
CAS :PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.Formule :C28H35F2N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :543.67Human carbonic anhydrase II-IN-2
Compound R-13, a potent inhibitor of hCA I/II/IV/IX with K i s of 60.7, 320.7, 2298, and 35.2 nM.Formule :C20H25N3O4SCouleur et forme :SolidMasse moléculaire :403.5YKL-05-093
CAS :YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.Formule :C35H40N6O4Couleur et forme :SolidMasse moléculaire :608.73Hypercalin B
CAS :Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.
Formule :C33H42O5Couleur et forme :SolidMasse moléculaire :518.684Antibiotic MA 144M1
CAS :Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.Formule :C42H55NO15Couleur et forme :SolidMasse moléculaire :813.88Diospyrin
CAS :Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.Formule :C22H14O6Couleur et forme :SolidMasse moléculaire :374.34Kallikrein-IN-1
CAS :Kallikrein-IN-1 (Formula A) is an inhibitor of the kinin-releasing enzyme Kallikrein.Formule :C28H26FN5O4Couleur et forme :SolidMasse moléculaire :515.54TT15
CAS :TT15 is an agonist of the GLP-1R.Formule :C51H44Cl2N4O6Couleur et forme :SolidMasse moléculaire :879.82Enprostil
CAS :Enprostil: synthetic PGE2 analog, reduces gastric acid, protects mucosa, lowers post-meal gastrin, treats ulcers effectively and safely.Formule :C23H28O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.46Polyozellin
CAS :Polyozellin is a prolyl endopeptidase inhibitor with properties effective against inflammation, cancer, and diseases related to oxidative stress.Formule :C22H14O10Couleur et forme :SolidMasse moléculaire :438.341FR-900482
CAS :FR-900482 exhibits high sensitivity to Thermoactinomyces calidolactis strain C 953 and demonstrates activity against cell lines such as P388, B16, EL4, FM3A, L1210, BHK-21, among others.Formule :C14H15N3O6Couleur et forme :SolidMasse moléculaire :321.29PLAP-IN-1
CAS :PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.Formule :C25H21Cl2N3O5Couleur et forme :SoildMasse moléculaire :514.36Antitrypanosomal agent 5
Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).Formule :C30H30N6O4SCouleur et forme :SolidMasse moléculaire :570.66AZ-PFKFB3-67 quarterhydrate
AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).Formule :C26H27N5O4Couleur et forme :SolidMasse moléculaire :460.01Lp-PLA2-IN-6
CAS :Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45Axl-IN-3
Axl-IN-3 is a selective, potent and orally active inhibitor of AXL kinase (IC50: 41.5 nM) and has a low inhibitory effect on other kinases.Formule :C24H25ClN6O2Couleur et forme :SolidMasse moléculaire :464.95Topoisomerase II inhibitor 6
Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.Formule :C19H18N4O2Couleur et forme :SolidMasse moléculaire :334.37Hit 1
Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.Formule :C22H24N4O3S2Couleur et forme :SolidMasse moléculaire :456.58AL 6598
CAS :AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.Formule :C23H39ClO5Couleur et forme :SolidMasse moléculaire :431.01Anticancer agent 62
CAS :Anticancer agent 62 inhibits HepG2, Bel-7402, MCF-7 growth with IC50: 0.019, 0.060, 0.016 μM respectively, and halts tumors.Formule :C20H19ClN3Na2O8PSCouleur et forme :SolidMasse moléculaire :573.85Cilengitide hydrochloride
CAS :Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formule :C27H41ClN8O7Couleur et forme :SolidMasse moléculaire :625.12RMI-18341
CAS :RMI-18341 is a Testosterone 5 alpha reductase inhibitor.Formule :C22H34N2O2Couleur et forme :SolidMasse moléculaire :358.52KCL-440
CAS :RS 57639 is a bioactive chemical.Formule :C18H18N2O2Couleur et forme :SolidMasse moléculaire :294.35SOS1-IN-6
CAS :SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).Formule :C26H28F3N3O2Couleur et forme :SolidMasse moléculaire :471.51Anticancer agent 12
Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3
