Autres inhibiteurs
Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.
37827 produits trouvés pour "Autres inhibiteurs"
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K252d
CAS :<p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>Formule :C26H23N3O5Couleur et forme :SolidMasse moléculaire :457.48TTK inhibitor 3
CAS :<p>TTK inhibitor 3 is a potent and selective TTK (an essential spindle assembly checkpoint enzyme) inhibitor with an IC 50 value of 3.0 nM.</p>Formule :C42H49N9O3Couleur et forme :SolidMasse moléculaire :727.9HR-546
CAS :<p>HR-546 is a prostaglandin E2 and prostaglandin F2alpha antagonist.</p>Formule :C26H44O6Couleur et forme :SolidMasse moléculaire :452.62Dehydelone
CAS :<p>Dehydelone(KOS-1584, R-1645, SK-10088) is a microtubule stabilizer that may be used in the treatment of non-small cell lung cancer.</p>Formule :C27H39NO5SCouleur et forme :SolidMasse moléculaire :489.67JTE 151A
CAS :<p>JTE-151 is a novel RORγ inverse agonist.</p>Formule :C26H30ClN3O5Couleur et forme :SolidMasse moléculaire :499.99NNC-11-1585
CAS :<p>NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.</p>Formule :C18H19N3OSCouleur et forme :SolidMasse moléculaire :325.43SphK1-IN-1
<p>SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.</p>Formule :C22H22N6O2Couleur et forme :SolidMasse moléculaire :402.45STAT3-IN-7
CAS :<p>STAT3-IN-7, an orally active aryl sulfonamido azetidine compound, serves as a STAT3 inhibitor with anticancer activities.</p>Formule :C30H26F5N5O4SCouleur et forme :SolidMasse moléculaire :647.62ACT-281959
CAS :<p>ACT-281959, a prodrug of ACT-246475, is a potent P2Y12 antagonist, better than Clopidogrel, effective orally, and in human trials.</p>Formule :C38H55N6O14PCouleur et forme :SolidMasse moléculaire :850.85MraY-IN-1
<p>MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.</p>Formule :C35H46N3O5Couleur et forme :SolidMasse moléculaire :588.76P-gp modulator 3
<p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>Formule :C31H37N3O5Couleur et forme :SolidMasse moléculaire :531.64Trk-IN-7
<p>Trk-IN-7 inhibits TRKA/B/C (IC50: 0.25-10 nM) & EML4-ALK (<15 nM), also targets various ALK mutations (IC50: 5-50 nM).</p>Formule :C18H17FN6O2Couleur et forme :SolidMasse moléculaire :368.36DAD
<p>DAD is an ion channel blocker (blocks voltage-gated potassium channels) and is a third generation photoelectric switch that responds to visible light.</p>Formule :C26H40N6OCouleur et forme :SolidMasse moléculaire :452.64NVP-CFC218
CAS :<p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>Formule :C37H45ClN4O4Couleur et forme :SolidMasse moléculaire :645.23Nolpitantium Free Base
CAS :<p>Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.</p>Formule :C37H45Cl2N2O2Couleur et forme :SolidMasse moléculaire :620.67Indinavir monohydrate
CAS :<p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>Formule :C36H49N5O5Couleur et forme :SolidMasse moléculaire :631.82SHR902275
CAS :<p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>Formule :C26H23F3N4O4Couleur et forme :SolidMasse moléculaire :512.48Esorubicin
CAS :<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formule :C27H29NO10Couleur et forme :SolidMasse moléculaire :527.52TP-030-1
CAS :<p>TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.</p>Formule :C23H22N4O3Couleur et forme :SolidMasse moléculaire :402.45AS2575959
CAS :<p>AS2575959 is a novel GPR40 agonist, exhibiting glucose metabolism improvement and synergistic effect with sitagliptin on insulin and incretin secretion.</p>Formule :C32H35NaO7Couleur et forme :SolidMasse moléculaire :554.6148rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formule :C25H24Cl2FN3O3Couleur et forme :SolidMasse moléculaire :504.38PD-1/PD-L1-IN-13
<p>PD-1/PD-L1-IN-13 is a potent immune checkpoint PD-1/PD-L1 inhibitor with an IC50 value of 10.2 nM for PD-1/PD- L1 interaction.PD-1/PD-L1-IN-13 promotes CD8+ T-</p>Formule :C36H34ClF2N3O9Couleur et forme :SolidMasse moléculaire :726.12Tilpisertib fosmecarbil
CAS :<p>Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.</p>Formule :C35H36ClN8O7PCouleur et forme :SolidMasse moléculaire :747.14P7170
CAS :<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Formule :C21H16F3N9Couleur et forme :SolidMasse moléculaire :451.42Plm IV inhibitor-2
CAS :<p>"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."</p>Formule :C39H54N4O4Couleur et forme :SolidMasse moléculaire :642.87DD04107
CAS :<p>DD04107 inhibits α-CGRP release, targets Synaptotagmin 1 in sensory neurons.</p>Formule :C48H88N14O12SCouleur et forme :SolidMasse moléculaire :1085.36(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formule :C24H24N4O6Couleur et forme :SolidMasse moléculaire :464.47Retezorogant
CAS :<p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>Formule :C23H33ClN2O3Couleur et forme :SolidMasse moléculaire :420.97IT-066 HCl
CAS :<p>IT-066 HCl is a histamine H2 receptor antagonist.</p>Formule :C19H25ClN4O3Couleur et forme :SolidMasse moléculaire :392.88Camptothecin-20(S)-O-propionate
CAS :<p>CZ-48 is a DNA topoisomerase inhibitor.</p>Formule :C23H20N2O5Couleur et forme :SolidMasse moléculaire :404.42Leustroducsin B
CAS :<p>Leustroducsin B is a novel colony-stimulating factor (CSF) inducer extracted from Streptomyces platensis SANK 60191.</p>Formule :C34H56NO10PCouleur et forme :SolidMasse moléculaire :669.78YKL-05-093
CAS :<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formule :C35H40N6O4Couleur et forme :SolidMasse moléculaire :608.73Gougerotin
CAS :<p>Gougerotin is an inhibitor of protein synthesis.</p>Formule :C16H25N7O8Couleur et forme :SolidMasse moléculaire :443.41Adiaft
CAS :<p>Adiaftis a bioactive chemical.</p>Formule :C10H11IN2O4Couleur et forme :SolidMasse moléculaire :350.11MRS2179 tetrasodium hydrate
<p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>Formule :C11H15N5Na4O10P2Couleur et forme :SolidMasse moléculaire :576.21BGC-638
CAS :<p>BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.</p>Formule :C32H33N5O9Couleur et forme :SolidMasse moléculaire :631.63Sekdel sequence
CAS :Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.Formule :C29H49N7O14Couleur et forme :SolidMasse moléculaire :719.74PPO-IN-1
<p>PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).</p>Formule :C18H10F3N3O4SCouleur et forme :SolidMasse moléculaire :421.35Isoleucyl tRNA synthetase-IN-2
CAS :<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formule :C22H33N5O8SCouleur et forme :SolidMasse moléculaire :527.59Mopivabil
<p>Mopivabil is the angiotensin II receptor antagonist[1].</p>Formule :C14H20O3Couleur et forme :SolidMasse moléculaire :236.31PI3K-IN-26
CAS :<p>PI3K-IN-26 is an effective PI3K inhibitor. PI3K-IN-26 inhibits the proliferation of SU-DHL-6 cells, IC50= 36 nM.</p>Formule :C21H18N6OSCouleur et forme :SolidMasse moléculaire :402.47Antibacterial agent 69
<p>Antibacterial agent 69 is a novel structural antimicrobial modulator that can be used against lethal multidrug-resistant bacterial infections (MIC: 2.978 μM).</p>Formule :C24H19N3O4SCouleur et forme :SolidMasse moléculaire :445.49Cilobamine (free base)
CAS :<p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>Formule :C17H23Cl2NOCouleur et forme :SolidMasse moléculaire :328.28Piceid 6″-O-azelaic acid ester
<p>Piceid 6″-O-azelaic acid ester exhibited strong intracellular tyrosinase inhibition and decolorization activity.</p>Formule :C24H36O10Couleur et forme :SolidMasse moléculaire :484.54Kri 1314
CAS :Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.Formule :C38H51N5O7Couleur et forme :SolidMasse moléculaire :689.84C-di-IMP
CAS :<p>Cyclic-di-IMP (C-di-IMP), a STING agonist, serves as a research tool in tumor studies.</p>Formule :C20H22N8O14P2Couleur et forme :SolidMasse moléculaire :660.38MMG-11 quarterhydrate
<p>MMG-11 quarterhydrate, a potent hTLR2 antagonist, inhibits TLR2/1 and TLR2/6 with IC50s of 1.7μM and 5.7μM; low toxicity.</p>Formule :C15H16O8Couleur et forme :SolidMasse moléculaire :310.78LPA5 antagonist 2
<p>LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.</p>Formule :C26H25FN2O4SCouleur et forme :SolidMasse moléculaire :480.55Glycotriosyl glutamine
CAS :<p>Glycotriosyl glutamine is a nephritogenoside analog.</p>Formule :C23H40N2O18Couleur et forme :SolidMasse moléculaire :632.57(S)-Butaprost free acid
CAS :<p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>Formule :C23H38O5Couleur et forme :SolidMasse moléculaire :394.54Lasonolide A
CAS :<p>Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.</p>Formule :C41H60O9Couleur et forme :SolidMasse moléculaire :696.91PTP1B-IN-21
<p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>Formule :C22H22O11Couleur et forme :SolidMasse moléculaire :462.4PARP10/15-IN-1
<p>PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].</p>Formule :C13H10N2O3SCouleur et forme :SolidMasse moléculaire :274.3KF 20274
CAS :<p>KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.</p>Formule :C21H29N5OCouleur et forme :SolidMasse moléculaire :367.49Namitecan
CAS :Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Formule :C23H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.44FTI 276 TFA
CAS :FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).Formule :C23H28F3N3O5S2Couleur et forme :SolidMasse moléculaire :547.61Thielavin B
CAS :<p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>Formule :C31H34O10Couleur et forme :SolidMasse moléculaire :566.6Atiratecan
CAS :<p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>Formule :C31H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :586.64Unoprostone
CAS :<p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>Formule :C22H38O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.53GNE-616
CAS :<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formule :C24H23F4N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :537.53Oral antiplatelet agent 1
CAS :<p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>Formule :C23H24N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.53hTrkA-IN-2
<p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>Formule :C24H22F3N5O3Couleur et forme :SolidMasse moléculaire :485.46PEN-866
CAS :<p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>Formule :C49H49N7O9Couleur et forme :SolidMasse moléculaire :879.95AVE 0991
CAS :<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Formule :C29H32N4O5S2Degré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :580.72Azonafide-PEABA
CAS :<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formule :C32H33N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :551.6420-HEDE
CAS :20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.Formule :C20H36O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.50Ro-51
CAS :<p>dual P2X3 and P2X2/3 antagonist</p>Formule :C17H23IN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.29Exicorilant
CAS :<p>Exicorilant is a selective oral GR antagonist (Ki: 7 nM) that may reduce obesity, glucose intolerance, & dyslipidemia.</p>Formule :C26H23F4N7O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :589.56BAY-091
CAS :<p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>Formule :C26H21FN4O2Degré de pureté :97.66% - 99.23%Couleur et forme :SoildMasse moléculaire :440.47BMS-751324
CAS :<p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>Formule :C32H35N6O10PCouleur et forme :SolidMasse moléculaire :694.63ATR-IN-7
CAS :<p>ATR-IN-7 is a potent inhibitor of ATR.</p>Formule :C21H22FN7OCouleur et forme :SolidMasse moléculaire :407.44AZD-3409
CAS :<p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>Formule :C34H41FN4O4S2Couleur et forme :SolidMasse moléculaire :652.84NA 382
CAS :<p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>Formule :C31H28N4O6Couleur et forme :SolidMasse moléculaire :552.58Basroparib
CAS :<p>Basroparib is an inhibitor of ribose polymerase (PARP) and has shown antitumour effects.</p>Formule :C18H21F2N7O3Couleur et forme :SolidMasse moléculaire :421.4Anticancer agent 79
<p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>Formule :C20H12F3NO5Couleur et forme :SolidMasse moléculaire :403.31MDL-43291
CAS :<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formule :C25H42O4SCouleur et forme :SolidMasse moléculaire :438.66MDL-100173
CAS :<p>MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.</p>Formule :C24H26N2O4SCouleur et forme :SolidMasse moléculaire :438.54TLN-232
CAS :<p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>Formule :C36H49N9O7S2Couleur et forme :SolidMasse moléculaire :783.96Plagiochilin A
CAS :<p>Plagiochilin A Inhibits Cytokinetic Abscission and Induces Cell Death</p>Formule :C15H14O7Couleur et forme :SolidMasse moléculaire :306.27BMS-961955
CAS :<p>BMS-961955 is an allosteric inhibitor of the hepatitis C virus NS5B polymerase.</p>Formule :C37H43FN4O4SCouleur et forme :SolidMasse moléculaire :658.83Ac-ATS010-KE
CAS :<p>Ac-ATS010-KE is a novel Selective, irreversible, and Rapid Cell-Permeable Inhibitor of Human Caspase-3.</p>Formule :C43H41F5N6O12SCouleur et forme :SolidMasse moléculaire :960.88N-methyl Leukotriene C4
CAS :<p>N-methyl LTC4 is a stable synthetic analog of LTC4 and a selective CysLT2 agonist, useful in studying leukotriene pharmacology.</p>Formule :C31H49N3O9SCouleur et forme :SolidMasse moléculaire :639.8AL-6556
CAS :<p>AL-6556 is a prostaglandin DP receptor agonist.</p>Formule :C20H33ClO5Couleur et forme :SolidMasse moléculaire :388.93PF-06815345 hydrochloride
CAS :<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Formule :C27H30Cl2FN9O4Couleur et forme :SolidMasse moléculaire :634.49H 218-54
CAS :<p>H 218-54 is a renin inhibitor.</p>Formule :C37H56N2O5SCouleur et forme :SolidMasse moléculaire :640.92DC41SMe
CAS :<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Formule :C38H36ClN5O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :726.31Novokinin
CAS :<p>Angiotensin AT2 receptor agonist</p>Formule :C39H61N11O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :795.972,4-Diaminoanisole
CAS :<p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>Formule :C7H10N2OCouleur et forme :SolidMasse moléculaire :138.175-Fluoroorotic acid monohydrate
CAS :5-Fluoroorotic acid (monohydrate) (5-Fluorouracil-6-carboxylic acid Mono(hydrate); 5-FOA) is employed to detect the expression of the URA3 gene in yeast molecular genetic constructs. Yeast possessing an active URA3 gene (which encodes orotidine-5'-monophosphate decarboxylase) convert 5-FOA into 5-fluorodeoxyuridine, a substance toxic to cells. Yeast strains with mutations in the URA3 gene that confer resistance can grow in the presence of 5-FOA if uracil is added to the medium.Formule :C5H5FN2O5Couleur et forme :SolidMasse moléculaire :192.10Porphine
CAS :<p>Porphine (Porphyrin), the parent compound of the porphyrin family, plays a crucial role within biological systems.</p>Formule :C20H14N4Couleur et forme :SolidMasse moléculaire :310.352,3-Dimethoxy-4-(methylthio)benzeneethanamine
CAS :2,3-Dimethoxy-4-(methylthio)benzeneethanamine (compound 22) is an analog of methoxybenzothiazine, employed in researching pharmacological agents that model human psychiatric disorders.Formule :C11H17NO2SCouleur et forme :SolidMasse moléculaire :227.32UCN-02
CAS :<p>UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.</p>Formule :C28H26N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.53TA-316
CAS :<p>Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.</p>Formule :C28H25BrN4O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :641.56Mycinamicin Ⅳ
CAS :Monamycin IV is an ester peptide antibiotic active against Gram-positive bacteria.Formule :C37H61NO11Couleur et forme :SolidMasse moléculaire :695.88TP3011
CAS :<p>TP3011 is a potent topoisomerase I inhibitor equipotent as SN38 and is an active metabolite of CH-0793076.</p>Formule :C26H26N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.51ER Thermo Yellow
CAS :<p>ER Thermo Yellow is a high-sensitivity (3.9%/°C) fluorescent probe designed for temperature visualization specifically targeting the endoplasmic reticulum.</p>Formule :C27H20BClF5N3O3Masse moléculaire :575.72Griseorhodin G
CAS :<p>Griseorhodin G is a quinone antibiotic with antitumor activity.</p>Formule :C25H18O12Masse moléculaire :510.40Maltophilin
CAS :<p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>Formule :C29H38N2O6Masse moléculaire :510.62Polyoxin J
CAS :<p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>Formule :C17H25N5O12Masse moléculaire :491.41Glaucarubin
CAS :<p>Glaucarubin is a bitter lactone naturally found in the fruits of Simaruba glauca. It is employed as an anti-amebic agent in research focused on amebiasis. The compound exhibits good tolerability, with a median lethal dose (LD50) of 1,600 mg/kg in mice and 6,400 mg/kg in rats.</p>Formule :C25H36O10Masse moléculaire :496.55Dihydropergillin
CAS :<p>Dihydropergillin is produced by the Aspergillus terreus strain (ATCC 38849) and has the ability to inhibit plant growth.</p>Formule :C15H18O4Masse moléculaire :262.30Papyracon D
CAS :<p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>Formule :C14H18O5Masse moléculaire :266.296-Hydroxytetrangulol
CAS :<p>6-Hydroxytetrangulol is an inducer of CPP32 protease found in Streptomyces.</p>Formule :C19H12O5Couleur et forme :SolidMasse moléculaire :320.30Saframycin Mx2
CAS :<p>Saframycin Mx2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C29H38N4O8Couleur et forme :SolidMasse moléculaire :570.634Hypercalin B
CAS :<p>Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.</p>Formule :C33H42O5Couleur et forme :SolidMasse moléculaire :518.684Monamycin I
CAS :Monamycin I is an ester peptide antibiotic with activity against Gram-positive bacteria.Formule :C35H58ClN7O8Couleur et forme :SolidMasse moléculaire :740.33Coriolin B
CAS :<p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>Formule :C23H36O6Couleur et forme :SolidMasse moléculaire :408.528Kynapcin-28
CAS :<p>Kynapcin-28 is a non-competitive inhibitor of prolyl endopeptidase (PEP) with an IC50 of 76.80 μM and exhibits weak inhibitory effects on other serine proteases.</p>Formule :C19H12O10Couleur et forme :SolidMasse moléculaire :400.293Deoxyradicinin
CAS :<p>Deoxyradicinin is a biosynthetic precursor of Radicinin. It can inhibit Xylella fastidiosa and Liberibacter crescens, with a minimum inhibitory concentration (MIC) of 3.5 μg/mL against Liberibacter crescens. Deoxyradicinin is applicable for research on controlling plant diseases caused by these pathogens.</p>Formule :C12H12O4Couleur et forme :SolidMasse moléculaire :220.221Cremeomycin
CAS :<p>Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.</p>Formule :C8H6N2O4Couleur et forme :SolidMasse moléculaire :194.144Diatretyne Ⅰ
CAS :Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.Formule :C8H5NO3Couleur et forme :SolidMasse moléculaire :163.133HKT-IN-1
CAS :<p>3HKT-IN-1 (Compound 17122279) is an inhibitor of Anopheles gambiae 3-hydroxykynurenine transaminase (3HKT) and is utilized in malaria research.</p>Formule :C12H11BrN2O3Couleur et forme :SolidMasse moléculaire :311.131Gilvusmycin
CAS :<p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>Formule :C38H34N6O8Couleur et forme :SolidMasse moléculaire :702.712UNC9426
CAS :<p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>Formule :C32H34F6N6ODegré de pureté :98.051%Couleur et forme :SolidMasse moléculaire :632.642Inosamycin A
CAS :<p>Inosamycin A is a broad-spectrum antibiotic.</p>Formule :C23H45N5O14Couleur et forme :SolidMasse moléculaire :615.628Disorazol A
CAS :<p>Disorazol A1 is a tubulin inhibitor with antifungal properties. It functions by inhibiting tubulin polymerization and disrupting microtubule formation, thereby blocking mitosis and arresting the cell cycle at the G2/M phase, which induces apoptosis. Disorazol A1 also inhibits L929 mouse fibroblasts with an IC50 value of 3 pm and causes accumulation of p53 protein in the nucleus. Disorazol A1 holds potential for cancer research.</p>Formule :C43H54N2O10Couleur et forme :SolidMasse moléculaire :758.896Cystothiazole A
CAS :<p>Cystothiazole A exhibits antifungal properties, effectively inhibiting Candida albicans, Saccharomyces cerevisiae, and Aspergillus fumigatus with minimum inhibitory concentrations (MIC) of 0.4 μg/mL, 0.1 μg/mL, and 1.6 μg/mL, respectively. It also demonstrates inhibitory activity against human tumor cells such as HPT-116 and K562, with MIC values of 130 ng/mL and 110 ng/mL. However, it shows no antibacterial activity.</p>Formule :C20H26N2O4S2Couleur et forme :SolidMasse moléculaire :422.561Pterulinic acid
CAS :<p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>Formule :C15H11ClO4Couleur et forme :SolidMasse moléculaire :290.70Rhamnitol
CAS :<p>Rhamnitol, the reduction product of L-rhamnose, can be observed during the metabolism of rhamnose in the body. Rhamnitol is promising for use in assessing intestinal permeability and studying carbohydrate metabolism.</p>Formule :C6H14O5Couleur et forme :SolidMasse moléculaire :166.17Cytosaminomycin B
CAS :<p>Cytosaminomycin B exhibits activity against Eimeria Tenella coccidia.</p>Formule :C26H37N5O8Couleur et forme :SolidMasse moléculaire :547.601Nanaomycin B
CAS :<p>Nanaomycin B is an antibiotic with activity against Gram-positive bacteria, mycobacteria, mycoplasma, and fungi.</p>Formule :C16H16O7Couleur et forme :SolidMasse moléculaire :320.294Feudomycin B
CAS :<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Formule :C28H31NO10Couleur et forme :SolidMasse moléculaire :541.546Haliangicin B
CAS :<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Formule :C22H32O5Couleur et forme :SolidMasse moléculaire :376.49Epelmycin D
CAS :<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.599Danavorexton
CAS :Danavorexton is an orexin receptor agonist.Formule :C21H32N2O5SCouleur et forme :SolidMasse moléculaire :424.55Pluracidomycin C2
CAS :<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C11H15NO9S2Couleur et forme :SolidMasse moléculaire :369.37Haliangicin A
CAS :<p>Haliangicin A exhibits antifungal activity against filamentous fungi and also affects oomycetes, though it does not possess antibacterial properties.</p>Formule :C22H32O5Couleur et forme :SolidMasse moléculaire :376.492-n-Heptyl-4-quinolinol
CAS :<p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>Formule :C16H21NOCouleur et forme :SolidMasse moléculaire :243.34Chitinovorin C
CAS :<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Formule :C15H20N4O8SCouleur et forme :SolidMasse moléculaire :416.4064-Nitrochalcone
CAS :<p>4-Nitrochalcone (2-(4-Nitrobenzylidene)acetophenone) inhibits proteasomes and suppresses TNFα-induced NF-κB activity.</p>Formule :C15H11NO3Couleur et forme :SolidMasse moléculaire :253.25Seldomycin factor 2
CAS :<p>Seldomycin factor 2 (XK 88-2) is an aminoglycoside antibiotic with broad-spectrum antibacterial activity.</p>Formule :C12H26N4O5Couleur et forme :SolidMasse moléculaire :306.359Gilvocarcin E
CAS :<p>Gilvocarcin E exhibits activity against Gram-positive bacteria and is capable of inhibiting Sarcoma 180 and P388 leukemia cells.</p>Formule :C27H28O9Couleur et forme :SolidMasse moléculaire :496.506Napyradiomycin C2
CAS :<p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>Formule :C25H27Cl3O5Couleur et forme :SolidMasse moléculaire :513.838Miyakamide B1
CAS :<p>Miyakamide B1 is an antibiotic with insecticidal properties, capable of inhibiting the growth of brine shrimp. It displays moderate activity against Xanthomonas bacteria and inhibits P388 cells with an IC50 of 8.8 μg/mL.</p>Formule :C31H32N4O4Couleur et forme :SolidMasse moléculaire :524.61Nanaomycin E
CAS :<p>Nanaomycin E is an antibiotic with activity against Gram-positive bacteria and fungi.</p>Formule :C16H14O7Couleur et forme :SolidMasse moléculaire :318.278Fosfazinomycin B
CAS :<p>Fosfazinomycin B exhibits activity against plant pathogenic fungi such as the rice blast pathogen (Xanthomonas oryzae).</p>Formule :C10H23N6O6PCouleur et forme :SolidMasse moléculaire :354.32-Hydroxygentamicin A3
CAS :<p>2-Hydroxygentamicin A3 is an aminoglycoside antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Formule :C18H36N4O11Couleur et forme :SolidMasse moléculaire :484.499Phellinsin
CAS :<p>Phellinsin selectively inhibits the activity of chitin synthase I and II, with IC50 values of 76 and 28 μg/mL, respectively. It also exhibits antimicrobial effects against pathogens such as anthracnose, rice blast fungus, Aspergillus fumigatus, and Trichophyton mentagrophytes, with a MIC ranging from 12.5 to 50 μg/mL.</p>Formule :C18H14O8Couleur et forme :SolidMasse moléculaire :358.30Epoxyquinomicin A
CAS :<p>Epoxyquinomicin A is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus with MIC values of 3-12.5 µg/mL. Additionally, it shows cytotoxicity in cancer cells L1210, B16, and S180, with an IC50 of 2-8 µg/mL. Furthermore, Epoxyquinomicin A demonstrates anti-inflammatory effects in collagen-induced arthritis.</p>Formule :C14H10ClNO6Couleur et forme :SolidMasse moléculaire :323.685Polyoxin E
CAS :<p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>Formule :C17H23N5O13Couleur et forme :SolidMasse moléculaire :505.39C20 Sphingomyelin (d18:1/20:1)
CAS :<p>C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).</p>Formule :C43H85N2O6PCouleur et forme :SolidMasse moléculaire :757.119Pluracidomycin C1
CAS :<p>Pluracidomycin C1 is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria and also possesses β-lactamase inhibitory properties.</p>Formule :C10H13NO10S2Couleur et forme :SolidMasse moléculaire :371.341Citrinin hydrate
CAS :<p>Citrinin hydrate is an inhibitor of human rhinovirus (HRV) 3C protease, with an IC50 of 1.0 mM.</p>Formule :C13H16O6Couleur et forme :SolidMasse moléculaire :268.263Leucomycin V
CAS :<p>Leucomycin V is a macrolide antibiotic. Leucomycin A9 exhibits strong activity against Gram-positive bacteria and also affects spirochetes, rickettsiae, and chlamydiae.</p>Formule :C35H59NO13Couleur et forme :SolidMasse moléculaire :701.842Pradimicin B
CAS :<p>Pradimicin B is an antibiotic with potent antifungal and anti-yeast activities.</p>Formule :C35H36N2O14Couleur et forme :SolidMasse moléculaire :708.6651-Deamino-1-hydroxysagamicin
CAS :<p>1-Deamino-1-hydroxysagamicin (AntibioticSUM-3) is an aminoglycoside antibiotic that is effective against both Gram-positive and Gram-negative bacteria.</p>Formule :C20H40N4O8Couleur et forme :SolidMasse moléculaire :464.554Phenazostatin B
CAS :<p>Phenazostatin B is a phenazine derivative known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. It inhibits glutamate toxicity in N18-RE-105 cells, with an EC50 of 0.33 μg/mL.</p>Formule :C32H26N4O4Couleur et forme :SolidMasse moléculaire :530.57Nemotin
CAS :<p>Nemotin exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while its effectiveness against Gram-negative bacteria is present but relatively weaker.</p>Formule :C11H8O2Couleur et forme :SolidMasse moléculaire :172.18Cuevaene A
CAS :<p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>Formule :C21H22O5Couleur et forme :SolidMasse moléculaire :354.396Chloroquinocin
CAS :<p>Chloroquinocin exhibits moderate activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA).</p>Formule :C17H15ClO5Couleur et forme :SolidMasse moléculaire :334.751Epelmycin C
CAS :<p>Epelmycin C exhibits antibacterial activity against both Gram-positive and Gram-negative bacteria, as well as antifungal activity against Candida albicans. It also shows activity against leukemia L1210.</p>Formule :C36H45NO14Couleur et forme :SolidMasse moléculaire :715.741Amidomycin
CAS :<p>Amidomycin is an antibiotic that primarily targets yeast.</p>Formule :C40H68N4O12Couleur et forme :SolidMasse moléculaire :796.993'-GMP
CAS :<p>3'-GMP is a nucleotide that can be isolated from the tubers of Helianthus tuberosus L. (Jerusalem artichoke).</p>Formule :C10H14N5O8PCouleur et forme :SolidMasse moléculaire :363.221Epicorazine A
CAS :<p>Epicorazine A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, showing an MIC of 25 μg/mL.</p>Formule :C18H16N2O6S2Couleur et forme :SolidMasse moléculaire :420.4595-Hydroxy-3,4,7-triphenyl-2,6-benzofurandione
CAS :<p>5-Hydroxy-3,4,7-triphenyl-2,6-benzofurandione is an inhibitor of xanthine oxidase (XO) found in the fungus Peniophora sanguinea.</p>Formule :C26H16O4Couleur et forme :SolidMasse moléculaire :392.40PARP1-IN-5
<p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>Formule :C25H24N2O5SCouleur et forme :SolidMasse moléculaire :464.53LY2934747
CAS :<p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>Formule :C10H13NO4Couleur et forme :SolidMasse moléculaire :211.21Leucomycin A9
CAS :<p>Leucomycin A9 is a macrolide antibiotic known for its potent activity against Gram-positive bacteria. It is also effective against spirochetes, rickettsiae, and chlamydiae.</p>Formule :C37H61NO14Couleur et forme :SolidMasse moléculaire :743.8785α-reductase-IN-1
CAS :<p>5α-reductase-IN-1 is a potent inhibitor of the enzyme 5α-reductase.</p>Formule :C31H37NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :503.63Antitumor agent-75
<p>Antitumor agent-75 is a novel and potent antitumor agent.</p>Formule :C26H23FN6Couleur et forme :SolidMasse moléculaire :438.5α-Prumycin hydrochloride
CAS :<p>α-Prumycin hydrochloride is a carbohydrate antibiotic with antifungal properties and weak antibacterial activity.</p>Formule :C8H19Cl2N3O4Couleur et forme :SolidMasse moléculaire :292.16Domitroban
CAS :<p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>Formule :C20H27NO4SCouleur et forme :SolidMasse moléculaire :377.5AZD-3199 dihydrobromide
CAS :<p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>Formule :C32H44Br2N4O4SCouleur et forme :SolidMasse moléculaire :740.59Vicanicin
CAS :<p>Vicanicin is an aryl phenol ether compound found in lichens. It inhibits the expression of Hsp70, modulates intracellular redox-sensitive mechanisms, increases reactive oxygen species (ROS) in cancer cells, alters the Bax/Bcl-2 ratio, activates caspase-3, and induces apoptosis. Vicanicin suppresses cell growth and promotes apoptosis in androgen-sensitive (LNCaP) and androgen-insensitive (DU-145) human prostate cancer cells. It holds potential for prostate cancer research.</p>Formule :C18H16Cl2O5Couleur et forme :SolidMasse moléculaire :383.223PDE5-IN-8
CAS :<p>PDE5-IN-8 (compound 2) is an inhibitor of PDEs.</p>Formule :C22H20ClN3O2Couleur et forme :SolidMasse moléculaire :393.87Xylarianaphthol-1
CAS :<p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>Formule :C16H20BrFN2O2Couleur et forme :SolidMasse moléculaire :371.24Pentacosafluorotridecanoic Acid
CAS :<p>Pentacosafluorotridecanoic Acid (PFTrDA) is a perfluoroalkyl substance (PFAS) that exhibits various biological impacts across different species. In zebrafish embryos, exposure to PFTrDA induces yolk sac edema and increases mRNA expression of thyroid hormone synthesis genes, including tshβ, at concentrations of 0.1 and 0.3 mg/L. At a dosage of 10 mg/kg, PFTrDA reduces serum testosterone and luteinizing hormone levels, as well as palmitic acid, linoleic acid, and oleic acid levels in the testicular interstitial cells of late adolescent rats. In humans, maternal plasma levels of PFTrDA during pregnancy are positively correlated with the development of eczema in female infants (but not male infants), and PFTrDA levels are higher in the livers of cancerous humans compared to non-cancerous ones. Additionally, PFTrDA is found in marine mammals.</p>Formule :C13HF25O2Couleur et forme :SolidMasse moléculaire :664.11Bagremycin B
CAS :<p>Bagremycin B is produced by the bacterium Streptomyces strain Tu 4128. It exhibits weak activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>Formule :C17H15NO4Couleur et forme :SolidMasse moléculaire :297.305EcGUS-IN-1
CAS :<p>EcGUS-IN-1 (Compound E-9) is a non-competitive inhibitor of β-glucuronidase, featuring an IC50 value of 2.68 μM and a Ki value of 1.64 μM. This compound effectively mitigates gastrointestinal adverse events (GIAE) associated with Escherichia coli infections by inhibiting the activity of E. coli β-glucuronidase.</p>Formule :C15H11F3N4SCouleur et forme :SolidMasse moléculaire :336.33Ingenol 3-monobenzoate
CAS :<p>Ingenol 3-monobenzoate (Ingenol 3-benzoate) acts as an aversive inducing agent. It binds to and activates protein kinase C (PKC) with a Ki of 0.14 nM. This activation inhibits the gene expression of phosphoenolpyruvate carboxykinase, thereby suppressing gluconeogenesis and increasing blood cortisol levels, which results in food aversion.</p>Formule :C27H32O6Couleur et forme :SolidMasse moléculaire :452.54Damavaricin D
CAS :<p>Damavaricin D exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Formule :C38H49NO12Couleur et forme :SolidMasse moléculaire :711.795MMP408
CAS :<p>MMP408 acts as an inhibitor of MMP-12.</p>Formule :C19H20N2O7SCouleur et forme :SolidMasse moléculaire :420.44PD-1/PD-L1-IN-30
CAS :<p>PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.</p>Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53Gentamicin C2
CAS :<p>Gentamicin C2 is an aminoglycoside antibiotic.</p>Formule :C20H41N5O7Couleur et forme :SolidMasse moléculaire :463.569GLS1 Inhibitor-5
<p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>Couleur et forme :SolidOdiparcil
CAS :<p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>Formule :C15H16O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.35NTPDase-IN-1
<p>NTPDase-IN-1 selectively inhibits NTPDases 1, 2, 8 with IC50 of 0.05, 0.23, 0.54 μM. Non-competitive, K m 21 μM, used in cancer, immune, infection research.</p>Formule :C18H25N3OS2Couleur et forme :SolidMasse moléculaire :363.54Ep vinyl quinidine
CAS :<p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>Formule :C20H24N2O2Couleur et forme :SolidMasse moléculaire :324.42RSV-IN-5
CAS :<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Formule :C28H37N7O2Couleur et forme :SolidMasse moléculaire :503.64ML-SI1
CAS :<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formule :C23H26Cl2N2O3Couleur et forme :SolidMasse moléculaire :449.37AD5075
CAS :<p>AD5075 is a bioactive chemical.</p>Formule :C22H20N2O5SCouleur et forme :SolidMasse moléculaire :424.47Antibiotic LL Z1640-2
CAS :<p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>Formule :C19H22O7Couleur et forme :SolidMasse moléculaire :362.38PF-446687
CAS :<p>PF-446687 is a highly selective MC4 receptor (MC4R) agonist.</p>Formule :C28H37ClF2N2O2Couleur et forme :SolidMasse moléculaire :507.06Unoprostone isopropyl
CAS :<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Formule :C25H44O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.61TCMDC-125431
<p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>Formule :C25H27N3O2SCouleur et forme :SolidMasse moléculaire :433.57PSMA-1007
CAS :<p>PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.</p>Formule :C49H55FN8O16Couleur et forme :SolidMasse moléculaire :1030.01Amdinocillin methylacetate
CAS :<p>Amdinocillin methylacetate is a Synthetic penicillin.</p>Formule :C18H27N3O4SCouleur et forme :SolidMasse moléculaire :381.49SGLT1/2-IN-1
CAS :<p>SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.</p>Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48Lobaric acid
CAS :<p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>Formule :C25H28O8Couleur et forme :SolidMasse moléculaire :456.48Hit 1
<p>Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.</p>Formule :C22H24N4O3S2Couleur et forme :SolidMasse moléculaire :456.58ZINC000104379474
<p>ZINC000104379474 is a compound that targets SARS-CoV-2 endoribonuclease.</p>Formule :C27H33N3O10Couleur et forme :SolidMasse moléculaire :559.57CYP1B1-IN-2
<p>CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].</p>Formule :C20H11F3O2Couleur et forme :SolidMasse moléculaire :340.3AN-12-H5
CAS :<p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>Formule :C24H23N3O4S3Couleur et forme :SolidMasse moléculaire :513.65Cilobamine mesylate
CAS :<p>Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.</p>Formule :C18H27Cl2NO4SCouleur et forme :SolidMasse moléculaire :424.38RMG8-8
<p>RMG8-8 shows the excellent efficacy against C. neoformans (1.56 μg/mL).</p>Formule :C41H78N8O5Couleur et forme :SolidMasse moléculaire :763.11GSK340
<p>GSK340 is a BET inhibitor.</p>Formule :C26H31N3O2Couleur et forme :SolidMasse moléculaire :417.55Dinalbuphine sebacate
CAS :<p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>Formule :C52H68N2O10Couleur et forme :SolidMasse moléculaire :881.1Pyridoxatin
CAS :<p>Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.</p>Formule :C15H21NO3Couleur et forme :SolidMasse moléculaire :263.33Pyrromycin
CAS :<p>Pyrromycin is a monosaccharide anthracycline which can be used to inhibit cellular RNA synthesis.</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.60Epoxyquinomicin B
CAS :<p>Epoxyquinomicin B is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus, with a minimum inhibitory concentration (MIC) of 6.25-12.5 µg/mL. It also shows cytotoxicity in cancer cells L1210, with an IC50 of 16.3 µg/mL. Additionally, Epoxyquinomicin B demonstrates anti-inflammatory effects on collagen-induced arthritis.</p>Formule :C14H11NO6Couleur et forme :SolidMasse moléculaire :289.24
