Autres inhibiteurs
Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.
37853 produits trouvés pour "Autres inhibiteurs"
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Gentamicin C1
CAS :<p>Gentamicin C1 is a broad-spectrum aminoglycoside antibiotic with antibacterial activity.</p>Formule :C21H43N5O7Couleur et forme :SolidMasse moléculaire :477.595MV061194
CAS :<p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>Formule :C28H37N5O4SCouleur et forme :SolidMasse moléculaire :539.693'-GMP
CAS :<p>3'-GMP is a nucleotide that can be isolated from the tubers of Helianthus tuberosus L. (Jerusalem artichoke).</p>Formule :C10H14N5O8PCouleur et forme :SolidMasse moléculaire :363.221AKR1C3-IN-8
<p>AKR1C3-IN-8 (Compound 5) is an effective and selective AKR1C3 inhibitor (IC50=0.069 μM). AKR1C3-IN-8 has antitumor activity.</p>Formule :C23H20N4O3Couleur et forme :SolidMasse moléculaire :400.43Novokinin
CAS :<p>Angiotensin AT2 receptor agonist</p>Formule :C39H61N11O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :795.97Guraxetan
<p>Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.</p>Formule :C20H34N4O9Couleur et forme :SolidMasse moléculaire :474.51EP-7041 HCl
CAS :<p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>Formule :C19H27ClN4O4Couleur et forme :SolidMasse moléculaire :410.89BMS-681
CAS :<p>BMS-681 is a CCR2 antagonist blocking chemokine binding, aiding control of inflammatory and neurodegenerative diseases.</p>Formule :C26H36F3N5OCouleur et forme :SolidMasse moléculaire :491.59SSR-182289A (Free)
CAS :SSR-182289A (Free) is a thrombin inhibitor.Formule :C30H33F2N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.68Anticancer agent 27
<p>Anticancer agent 27 is a promising candidate for the treatment of cancer and deserves further development.</p>Formule :C28H31NO6Couleur et forme :SolidMasse moléculaire :477.55Methysergide maleate
CAS :<p>Methysergide prevents migraines/cluster headaches; treats serotonin syndrome, carcinoid-induced diarrhea; risk of fibrosis limits use.</p>Formule :C25H31N3O6Degré de pureté :98%Couleur et forme :White To Off-WhiteMasse moléculaire :469.54Papyracon D
CAS :<p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>Formule :C14H18O5Masse moléculaire :266.29Epicorazine A
CAS :<p>Epicorazine A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, showing an MIC of 25 μg/mL.</p>Formule :C18H16N2O6S2Couleur et forme :SolidMasse moléculaire :420.459Inosamycin A
CAS :<p>Inosamycin A is a broad-spectrum antibiotic.</p>Formule :C23H45N5O14Couleur et forme :SolidMasse moléculaire :615.628Endophenazine D
CAS :<p>Endophenazine D is a phenazine-class antibiotic.</p>Formule :C15H12N2O4Couleur et forme :SolidMasse moléculaire :284.27TTK inhibitor 3
CAS :<p>TTK inhibitor 3 is a potent and selective TTK (an essential spindle assembly checkpoint enzyme) inhibitor with an IC 50 value of 3.0 nM.</p>Formule :C42H49N9O3Couleur et forme :SolidMasse moléculaire :727.9Hetrombopag olamine
CAS :<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Formule :C29H36N6O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :580.63Monorden diacetate
CAS :<p>Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.</p>Formule :C22H21ClO8Couleur et forme :SolidMasse moléculaire :448.85RK-582
CAS :<p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>Formule :C27H35FN6O3Couleur et forme :SolidMasse moléculaire :510.6Odiparcil
CAS :<p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>Formule :C15H16O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :324.35GW-597901 cinnamate
CAS :<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80RIP1 kinase inhibitor 1
CAS :<p>RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.</p>Formule :C24H20ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.9GSK 932121
CAS :<p>GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.</p>Formule :C20H15ClF3NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.79OP-2507
CAS :<p>OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.</p>Formule :C25H41NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :419.6Peridinin
CAS :<p>Peridinin is an exceptionally potent and membrane-embedded inhibitor of bilayer lipid peroxidation.</p>Formule :C39H50O7Couleur et forme :SolidMasse moléculaire :630.81O4
CAS :<p>O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.</p>Formule :C24H15NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.387-Hydroxyguanine
CAS :<p>7-Hydroxyguanine is an antibiotic that inhibits the growth of L1210 leukemia cells.</p>Formule :C5H5N5O2Couleur et forme :SolidMasse moléculaire :167.126Napyradiomycin A2
CAS :<p>Napyradiomycin A2 is an antibiotic that exhibits activity against Gram-positive bacteria and mycobacteria.</p>Formule :C25H30Cl2O6Couleur et forme :SolidMasse moléculaire :497.408Formadicin B
CAS :<p>Formadicin B exhibits significant activity against various species of Pseudomonas, Proteus, and Alcaligenes.</p>Formule :C30H34N4O15Couleur et forme :SolidMasse moléculaire :690.61DAD dichloride
<p>DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.</p>Formule :C26H42Cl2N6OCouleur et forme :SolidMasse moléculaire :525.56ZBH-1205
CAS :<p>ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.</p>Formule :C29H31N3O8Couleur et forme :SolidMasse moléculaire :549.57MSX-3 free acid
CAS :<p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>Formule :C21H23N4O7PCouleur et forme :SolidMasse moléculaire :474.40PF-5177624
CAS :<p>PF-5177624 is a selective and potent PDK1 inhibitor inducing anti-tumor activity in breast cancer cells.</p>Formule :C25H25FN8O2Couleur et forme :SolidMasse moléculaire :488.52TRK-IN-12
CAS :<p>TRK-IN-12 (9e), a macrocyclic TRK inhibitor (G595R IC50=13.1 nM), outperforms LOXO-101 in Ba/F3-NTRK1 cells.</p>Formule :C18H19ClFN5O3SCouleur et forme :SolidMasse moléculaire :439.89(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formule :C24H24N4O6Couleur et forme :SolidMasse moléculaire :464.47Keap1-Nrf2-IN-1 TFA
<p>Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.</p>Formule :C26H25F3N2O9SCouleur et forme :SolidMasse moléculaire :598.54Elacestrant S enantiomer
<p>Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.</p>Formule :C30H38N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.63Bacithrocin D
CAS :<p>Bacithrocin D (Thiolstatin D) inhibits various proteases and has the capability to prolong clotting time. It exhibits IC50 values of 124, 9, 0.85, and 0.01 μM against thrombin, factor Xa, trypsin, and papain, respectively.</p>Formule :C17H25N5O3Couleur et forme :SolidMasse moléculaire :347.412Clavamycin A
CAS :<p>Clavamycin A displays notable antifungal activity against Candida species, with its effects being antagonized by dipeptides or tripeptides, although not by amino acids. It lacks antibacterial properties and does not inhibit β-lactamase.</p>Formule :C16H22N4O9Couleur et forme :SolidMasse moléculaire :414.367FTO-IN-4
CAS :<p>FTO-IN-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (FTO).</p>Formule :C22H16Cl2N6O6Couleur et forme :SolidMasse moléculaire :531.31AL 6598
CAS :<p>AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.</p>Formule :C23H39ClO5Couleur et forme :SolidMasse moléculaire :431.01Rezatapopt
CAS :<p>Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.</p>Formule :C28H31F4N5O2Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :545.57AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Formule :C32H38N6O3Couleur et forme :SolidMasse moléculaire :554.7Antibiotic MA 144M1
CAS :<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formule :C42H55NO15Couleur et forme :SolidMasse moléculaire :813.885(S),6(R)-DiHETE
CAS :<p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47ML-SI1
CAS :<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formule :C23H26Cl2N2O3Couleur et forme :SolidMasse moléculaire :449.37CN-716 HCl
CAS :<p>cn-716 is a novel Zika virus (ZIKV) NS2B-NS3pro protease inhibitor.</p>Formule :C22H33BCl2N6O4Couleur et forme :SolidMasse moléculaire :527.25KR-67607
CAS :<p>KR-67607, or NTX-101, is a novel 11β-HSD1 inhibitor that protects against eye injury by reducing cortisol and preserving eye structures.</p>Formule :C24H29Cl2F3N4O4SCouleur et forme :SolidMasse moléculaire :597.48BRD7929
CAS :<p>BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.</p>Formule :C33H38N4O2Couleur et forme :SolidMasse moléculaire :522.68Fumaryl-DL-alanine
CAS :<p>Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.</p>Formule :C7H9NO5Couleur et forme :SolidMasse moléculaire :187.15Lp-PLA2-IN-6
CAS :<p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45CYP2C9/CYP2C19-IN-1
<p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formule :C27H28N2O6SCouleur et forme :SolidMasse moléculaire :508.59Glasmacinal
CAS :Glasmacinal is a non-antibacterial macrolide compound with anti-inflammatory activities.Formule :C37H62N2O10Couleur et forme :SolidMasse moléculaire :694.90Asperenone
CAS :<p>Asperenone is a 15-lipoxygenase (15-LOX) inhibitor with an IC50 of 0.3 mM. Additionally, it acts as a platelet aggregation inhibitor with an IC50 of 0.23 mM. Asperenone also exhibits antifungal properties, inhibiting the growth of pathogenic fungi Ophiostoma crassivaginatum and O. piliferum, and may be utilized in research related to cardiovascular diseases and anti-infective treatments.</p>Formule :C20H22OCouleur et forme :SolidMasse moléculaire :278.388Leucomycin A7
CAS :<p>Leucomycin A7 is a component of the leucomycin complex, isolated from *Streptomyces kitasatoensis*. It possesses antibacterial activity, effectively inhibiting the growth of gram-positive bacteria, while its inhibitory effect on gram-negative bacteria is comparatively weaker.</p>Formule :C38H63NO14Couleur et forme :SolidMasse moléculaire :757.905GNE-203
CAS :<p>GNE-203 is a Met inhibitor.</p>Formule :C30H29Cl2F3N8O3Couleur et forme :SolidMasse moléculaire :677.50Antitumor agent-187
CAS :<p>Antitumor agent-187 (compound I) is an isoflavone derivative with antitumor activity. It exhibits IC50 values of 5.23 μM and 2.63 μM against A2780 and SKOV3 cell lines, respectively.</p>Formule :C24H26N2O7Couleur et forme :SolidMasse moléculaire :454.47nNOS-IN-25
CAS :nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.Formule :C21H22N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.43PDE4-IN-6
<p>PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.</p>Formule :C25H20FNO5SCouleur et forme :SolidMasse moléculaire :465.49Griseolic acid C
CAS :<p>Griseolic acid C (Dihydrodeoxygriseolic acid) is an antibiotic found in the Streptomyces griseoaurantiacus SANK43894 strain. This compound is a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase [EC 3.1.4.17], with an IC50 of 0.12 μM (enzyme sourced from rat brain tissue).</p>Formule :C14H15N5O7Couleur et forme :SolidMasse moléculaire :365.298A 74273
CAS :<p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>Formule :C44H74N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :787.08Salfredin C1
CAS :<p>Salfredin C1 is an inhibitor of aldose reductase.</p>Formule :C13H11NO6Couleur et forme :SolidMasse moléculaire :277.229Saframycin D
CAS :<p>Saframycin D exhibits activity against Gram-positive bacteria and shows weaker potency against mycobacteria.</p>Formule :C28H31N3O9Couleur et forme :SolidMasse moléculaire :553.56NI-Pano
<p>NI-Pano (CH-03) is a novel hypoxia-activated KDAC inhibitor capable of O2-dependent release of the compound panobinostat.</p>Formule :C26H28N6O4Couleur et forme :SolidMasse moléculaire :488.54VEGFR-2-IN-16
<p>VEGFR-2-IN-16 (Compound 15b) is a potent inhibitor of VEGFR-2 (IC50: 86.36 nM) that exhibits antitumour effects.</p>Formule :C21H13Cl2N3O2Couleur et forme :SolidMasse moléculaire :410.25Eilatine
CAS :<p>Eilatine is a novel marine alkaloid inhibits in vitro proliferation of progenitor cells in chronic myeloid leukemia patients.</p>Formule :C24H12N4Couleur et forme :SolidMasse moléculaire :356.38CS-003 HCl
CAS :<p>CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.</p>Formule :C34H39Cl3N2O6SCouleur et forme :SolidMasse moléculaire :710.1CVS-1578
CAS :<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formule :C20H30N6O5SCouleur et forme :SolidMasse moléculaire :466.55AT-IAP
CAS :AT-IAP is an effective dual antagonist of XIAP and cIAP1.Formule :C29H40FN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :509.66PCSK9-IN-17
CAS :<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Formule :C16H19N5OSCouleur et forme :SolidMasse moléculaire :329.42Pentenocin A
CAS :<p>Pentenocin A exhibits a relatively weak inhibitory effect on IL-1 and β-glucuronidase (ICE) activity.</p>Formule :C7H10O5Couleur et forme :SolidMasse moléculaire :174.151AL-6556
CAS :<p>AL-6556 is a prostaglandin DP receptor agonist.</p>Formule :C20H33ClO5Couleur et forme :SolidMasse moléculaire :388.93Antiproliferative agent-3
<p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>Formule :C11H12N2O5SCouleur et forme :SolidMasse moléculaire :284.29Haliangicin B
CAS :<p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>Formule :C22H32O5Couleur et forme :SolidMasse moléculaire :376.49KF-19418
CAS :<p>KF-19418 is a follicle stimulant that directly activates follicles in vitro and promotes hair growth in vivo.</p>Formule :C21H14N4OCouleur et forme :SolidMasse moléculaire :338.36Benadrostin
CAS :<p>Benadrostin is a Poly(ADP-ribose) synthetase inhibitor with an IC50 of 35μM.</p>Formule :C8H5NO4Couleur et forme :SolidMasse moléculaire :179.13Glucopiericidin B
CAS :<p>Glucopiericidin B exhibits antibacterial activity.</p>Formule :C31H47NO9Couleur et forme :SolidMasse moléculaire :577.706Carpetimycin A
CAS :<p>Carpetimycin A exhibits potent activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. It also acts as a strong inhibitor of β-lactamase.</p>Formule :C14H18N2O6SCouleur et forme :SolidMasse moléculaire :342.368Hydroxymycotrienin A
CAS :<p>Hydroxymycotrienin A is an ansamycin antibiotic with the ability to inhibit human neck tumor cell lines. Its inhibitory effect is more pronounced on HPV-positive neck tumor cells (such as HeLa, CaSKi, and SiHa) compared to HPV-negative cells.</p>Formule :C36H48N2O9Couleur et forme :SolidMasse moléculaire :652.774AVE-1330A free acid
CAS :<p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>Formule :C7H11N3O6SCouleur et forme :SolidMasse moléculaire :265.24SAR107375
CAS :<p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>Formule :C24H30ClN5O5S2Couleur et forme :SolidMasse moléculaire :568.11BDZ-h
CAS :<p>BDZ-h inhibits both closed/open states of all 4 homomeric & 2 GluA2R-complex AMPA receptors.</p>Formule :C21H21N5O3SCouleur et forme :SolidMasse moléculaire :423.49AT1R antagonist 2
<p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>Formule :C29H37N5O4S2Couleur et forme :SolidMasse moléculaire :583.77Enprostil
CAS :<p>Enprostil: synthetic PGE2 analog, reduces gastric acid, protects mucosa, lowers post-meal gastrin, treats ulcers effectively and safely.</p>Formule :C23H28O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.46Dihydroabikoviromycin
CAS :<p>Dihydroabikoviromycin is a secondary metabolite of Streptomyces anulatus and acts as a polyketide synthase inhibitor.</p>Formule :C10H13NOCouleur et forme :SolidMasse moléculaire :163.216PrCP-7414
CAS :<p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>Formule :C31H33Cl2N5O2Couleur et forme :SolidMasse moléculaire :578.53TSWV-IN-1
<p>TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.</p>Formule :C26H31FO4S2Couleur et forme :SolidMasse moléculaire :490.65CH-38083
CAS :<p>CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.</p>Formule :C18H24ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :337.84AB 5046A
CAS :<p>AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.</p>Formule :C10H14O4Couleur et forme :SolidMasse moléculaire :198.22BW A868C
CAS :BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formule :C25H37N3O5Couleur et forme :SolidMasse moléculaire :459.58Dicetrorelix pamoate
CAS :<p>Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.</p>Formule :C163H200Cl2N34O34Couleur et forme :SolidMasse moléculaire :3250.49Retelliptine
CAS :Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Formule :C25H32N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :404.55CXN37378
CAS :<p>CXN37378, aka NAP, is a potent MOR-selective antagonist with no official name yet, termed per MedKoo Nomenclature.</p>Formule :C27H31N3O4Couleur et forme :SolidMasse moléculaire :461.55Eurocidin E
CAS :<p>Eurocidin E is an antibiotic that inhibits degranulation and histamine release from rat mast cells.</p>Formule :C40H61NO14Couleur et forme :SolidMasse moléculaire :779.911PPARγ agonist 1
<p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>Formule :C34H39NO3Couleur et forme :SolidMasse moléculaire :509.68GSK1820795A
CAS :<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formule :C35H34N8Couleur et forme :SolidMasse moléculaire :566.7Tofogliflozin
CAS :Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formule :C22H26O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.44Collinone
CAS :<p>Collinone is a recombinant polyketide antibiotic with antimicrobial activity against Gram-positive bacteria and exhibits cytotoxicity.</p>Formule :C27H18O12Couleur et forme :SolidMasse moléculaire :534.425PDE5-IN-8
CAS :<p>PDE5-IN-8 (compound 2) is an inhibitor of PDEs.</p>Formule :C22H20ClN3O2Couleur et forme :SolidMasse moléculaire :393.87Idraparinux Na
CAS :<p>Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa Inhibitor</p>Formule :C38H55Na9O49S7Couleur et forme :SolidMasse moléculaire :1727.14Citreamicin γ
CAS :<p>Citreamicin γ demonstrates activity against aerobic and anaerobic Gram-positive bacteria.</p>Formule :C33H25NO12Couleur et forme :SolidMasse moléculaire :627.551Glucoallosamidin A
CAS :<p>Glucoallosamidin A is a glycoside antibiotic that inhibits chitinase activity. It effectively suppresses the chitinase enzyme in Candida albicans [ATCC 10231], exhibiting an IC50 of 3.4 μg/mL.</p>Formule :C26H44N4O14Couleur et forme :SolidMasse moléculaire :636.646TCMDC-136230
<p>TCMDC-136230 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystallisation.</p>Formule :C24H34N4O2SCouleur et forme :SolidMasse moléculaire :442.62Glucosylceramide synthase-IN-3
<p>Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.</p>Formule :C21H20FN3O3Couleur et forme :SolidMasse moléculaire :381.4Epelmycin D
CAS :<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.599hDDAH-1-IN-2 sulfate
<p>hDDAH-1-IN-2: selective oral hDDAH-1 inhibitor with low cell toxicity.</p>Formule :C8H24N4O10S2Couleur et forme :SolidMasse moléculaire :400.43MRS-2339
CAS :<p>MRS-2339 is a P2X receptor activator.</p>Formule :C12H15ClN5O6PCouleur et forme :SolidMasse moléculaire :391.70M-89 MLL inhibitor
CAS :<p>M-89, a potent Menin-MLL blocker: Kd 1.4 nM, IC50 25 nM for MV4;11 cells, 55 nM for MOLM-13, >100x selective over HL-60.</p>Formule :C37H47N5O4SCouleur et forme :SolidMasse moléculaire :657.87Pentacosafluorotridecanoic Acid
CAS :<p>Pentacosafluorotridecanoic Acid (PFTrDA) is a perfluoroalkyl substance (PFAS) that exhibits various biological impacts across different species. In zebrafish embryos, exposure to PFTrDA induces yolk sac edema and increases mRNA expression of thyroid hormone synthesis genes, including tshβ, at concentrations of 0.1 and 0.3 mg/L. At a dosage of 10 mg/kg, PFTrDA reduces serum testosterone and luteinizing hormone levels, as well as palmitic acid, linoleic acid, and oleic acid levels in the testicular interstitial cells of late adolescent rats. In humans, maternal plasma levels of PFTrDA during pregnancy are positively correlated with the development of eczema in female infants (but not male infants), and PFTrDA levels are higher in the livers of cancerous humans compared to non-cancerous ones. Additionally, PFTrDA is found in marine mammals.</p>Formule :C13HF25O2Couleur et forme :SolidMasse moléculaire :664.11STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formule :C17H12N4O4Couleur et forme :SolidMasse moléculaire :336.3Anti-Trypanosoma cruzi agent-1
<p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49Epihygromycin
CAS :<p>Epihygromycin is a glycoside antibiotic with relatively weak activity against Gram-positive bacteria.</p>Formule :C23H29NO12Couleur et forme :SolidMasse moléculaire :511.476MI-1851
CAS :<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formule :C34H53N15O6Couleur et forme :SolidMasse moléculaire :767.88Enpp-1-IN-7
<p>Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)</p>Formule :C18H19N7O4SCouleur et forme :SolidMasse moléculaire :429.45Dinordrin
CAS :Dinordrin is an implantation inhibitor and hormone.Formule :C27H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.57Vps34-IN-3
<p>Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .</p>Formule :C14H20N4O2Couleur et forme :SolidMasse moléculaire :276.33Panosialin wA
CAS :<p>Panosialin wA inhibits α,β-glucosidase and mannosidase enzymes, but does not exhibit inhibitory activity against the influenza virus. However, it has a mild antibacterial effect.</p>Formule :C21H36O5SCouleur et forme :SolidMasse moléculaire :400.57NNC-11-1585
CAS :<p>NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.</p>Formule :C18H19N3OSCouleur et forme :SolidMasse moléculaire :325.43Deoxyfuconojirimycin hydrochloride
CAS :<p>Deoxyfuconojirimycin hydrochloride acts as a specific competitive inhibitor targeting human liver α-L-fucosidase.</p>Formule :C6H14ClNO3Couleur et forme :SolidMasse moléculaire :183.63Darlucin A
CAS :<p>Darlucin A exhibits both antibacterial and antifungal properties, accompanied by mild cytotoxicity.</p>Formule :C19H16N2O3Couleur et forme :SolidMasse moléculaire :320.342PPARα agonist 1
<p>PPARα agonist 1 is a complete and potent PPARα agonist.</p>Formule :C27H34O4Couleur et forme :SolidMasse moléculaire :422.56Pluracidomycin C2
CAS :<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C11H15NO9S2Couleur et forme :SolidMasse moléculaire :369.37LY-2979165
CAS :<p>LY-2979165 is a metabotropic glutamate receptor agonist prodrug.</p>Formule :C13H17N5O5SCouleur et forme :SolidMasse moléculaire :355.37Mycelianamide
CAS :<p>Mycelianamide is an antibiotic effective against Gram-positive bacteria.</p>Formule :C22H28N2O5Couleur et forme :SolidMasse moléculaire :400.4682-PPA
CAS :2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.Formule :C11H10N2Couleur et forme :SolidMasse moléculaire :170.21(-)-Adenophorine
CAS :<p>(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.</p>Formule :C8H17NO4Couleur et forme :SolidMasse moléculaire :191.22Tazide
<p>Tazide is an antitumor agent [1].</p>Formule :C12H16N4OCouleur et forme :SolidMasse moléculaire :232.28Sargachromanol E
CAS :<p>Sargachromanol E is a compound isolated from the marine brown alga, Sargassum horneri. It has been studied for its inhibitory effect on skin ageing.</p>Formule :C27H40O4Couleur et forme :SolidMasse moléculaire :428.6WM382
CAS :<p>WM382, a potent dual PMIX/X inhibitor, has IC50s of 1.4 nM/0.03 nM and effective against various malaria stages.</p>Formule :C29H36N4O4Couleur et forme :SolidMasse moléculaire :504.62Ici D1542
CAS :Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.Formule :C25H30N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :470.51SP inhibitor 1
<p>SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.</p>Formule :C36H38N2O2Couleur et forme :SolidMasse moléculaire :530.7SSTR5 antagonist 2 hydrochloride
<p>SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.</p>Formule :C32H36ClFN2O5Couleur et forme :SolidMasse moléculaire :583.09ETP-47037
CAS :<p>ETP-47037: strong PI3Kα inhibitor (IC50: 0.99 nM), also targets PI3Kβ, δ, γ; may protect telomeres.</p>Formule :C20H27N9O3SCouleur et forme :SolidMasse moléculaire :473.559(S),10(S),13(S)-TriHOME
CAS :<p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>Formule :C18H34O5Couleur et forme :SolidMasse moléculaire :330.46J-104132
CAS :<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Formule :C31H33NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :531.60Lycopodine
CAS :<p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38EBI-907
CAS :<p>EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.</p>Formule :C23H21ClF2N4O3SCouleur et forme :SolidMasse moléculaire :506.95Narbomycin
CAS :<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Formule :C28H47NO7Couleur et forme :SolidMasse moléculaire :509.675AZD2353
CAS :<p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>Formule :C22H19ClFN3O3Couleur et forme :SolidMasse moléculaire :427.86LY 178210
CAS :<p>LY 178210 is a 5-hydroxytryptamine receptor agonist.</p>Formule :C18H25N3OCouleur et forme :SolidMasse moléculaire :299.41Epoformin
CAS :<p>Epoformin is a fungal cyclohexene epoxide that can be isolated from Diplodia quercivora. This compound acts as an antibiotic with mild inhibitory effects on rye seedling sheath growth. Additionally, Epoformin exhibits antifungal properties, effectively inhibiting Phytophthora cinnamomi and Phytophthora plurivora.</p>Formule :C7H8O3Couleur et forme :SolidMasse moléculaire :140.137KCa2 channel modulator 2
Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.Formule :C16H15ClFN5Couleur et forme :SolidMasse moléculaire :331.78Anticancer agent 17
<p>Anticancer agent 17 was effective against HeLa cells (IC50: 0.19 μM) and A2780 cells (IC50: 0.09 μM).</p>Formule :C27H34BrN3OCouleur et forme :SolidMasse moléculaire :496.48TrxR-IN-2
<p>TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.</p>Formule :C22H22N4O4Couleur et forme :SolidMasse moléculaire :406.43P-gp modulator 2
<p>P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.</p>Formule :C22H20BrN3O4Couleur et forme :SolidMasse moléculaire :470.32Anti-inflammatory agent 18
<p>Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.</p>Formule :C30H50O6Couleur et forme :SolidMasse moléculaire :506.71NA 0346
CAS :<p>NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.</p>Formule :C26H22N4O3Couleur et forme :SolidMasse moléculaire :438.48Antileishmanial agent-5
<p>Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.</p>Formule :C17H17ClN4O4Couleur et forme :SolidMasse moléculaire :376.79RSK4-IN-1
CAS :<p>RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.</p>Formule :C19H20F2N4O3Couleur et forme :SolidMasse moléculaire :390.38Unoprostone isopropyl
CAS :<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Formule :C25H44O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.61Methyl 5-thia-6,8,11,14-eicosatetraenoate
CAS :<p>Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.</p>Formule :C20H32O2SCouleur et forme :SolidMasse moléculaire :336.53Vulolisib
CAS :<p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>Formule :C18H19F2N5O3SCouleur et forme :SolidMasse moléculaire :423.44Octacosamicin A
CAS :<p>Octacosamicin A exhibits activity against bacteria, yeast, and filamentous fungi, although its antibacterial effects are relatively weak.</p>Formule :C31H52N4O9Couleur et forme :SolidMasse moléculaire :624.7662-Hydroxy-5-iminoazacyclopent-3-ene
CAS :<p>2-Hydroxy-5-iminoazacyclopent-3-ene is a pyrroline-class antibiotic with mild activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C4H6N2OCouleur et forme :SolidMasse moléculaire :98.103GSK-1264
CAS :<p>GSK-1264: allosteric HIV integrase inhibitor, halts viral replication & abnormal protein multimerization.</p>Formule :C26H28FNO5Couleur et forme :SolidMasse moléculaire :453.5Orvepitant
CAS :<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Formule :C31H35F7N4O2Couleur et forme :SolidMasse moléculaire :628.62IDX-320
CAS :<p>IDX-320 is an HCV protease inhibitor.</p>Formule :C37H43F3N6O7S2Couleur et forme :SolidMasse moléculaire :804.9Quinocycline B
CAS :<p>Quinocycline B is a quinone and other glycoside antibiotic that demonstrates resistance to Gram-positive bacteria.</p>Formule :C33H32N2O10Couleur et forme :SolidMasse moléculaire :616.62α-Prumycin hydrochloride
CAS :<p>α-Prumycin hydrochloride is a carbohydrate antibiotic with antifungal properties and weak antibacterial activity.</p>Formule :C8H19Cl2N3O4Couleur et forme :SolidMasse moléculaire :292.16TIY-7
<p>TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.</p>Couleur et forme :SolidBacithrocin A
CAS :<p>Bacithrocin C is a thrombin inhibitor that also suppresses factor Xa, trypsin, and papain, with IC50 values of 48 μM, 13 μM, 0.65 μM, and 0.02 μM, respectively.</p>Formule :C20H31N5O3Couleur et forme :SolidMasse moléculaire :389.492Polyoxin J
CAS :<p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>Formule :C17H25N5O12Masse moléculaire :491.41Maltophilin
CAS :<p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>Formule :C29H38N2O6Masse moléculaire :510.62De-N-methylpamamycin-593A
CAS :<p>De-N-methylpamamycin-593A is a 16-membered macrocyclic dilactone known for its ability to induce aerial mycelium formation.</p>Formule :C34H59NO7Masse moléculaire :593.84BMS-520
CAS :<p>BMS-520: potent oral S1P1 agonist, effective in rat arthritis and mouse multiple sclerosis model.</p>Formule :C23H17F3N4O4Couleur et forme :SolidMasse moléculaire :470.42-Hydroxygentamicin C2
CAS :<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C20H41N5O8Couleur et forme :SolidMasse moléculaire :479.568Tezampanel hydrate
CAS :<p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>Formule :C13H23N5O3Couleur et forme :SolidMasse moléculaire :297.35Pyrromycin
CAS :<p>Pyrromycin is a monosaccharide anthracycline which can be used to inhibit cellular RNA synthesis.</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.60Ganciclovir monophosphonate
CAS :<p>Ganciclovir monophosphate treats CMV, inhibiting replication in human/animal strains (IC50: 0.01μM).</p>Formule :C10H16N5O6PCouleur et forme :SolidMasse moléculaire :333.24Polyoxin H
CAS :<p>Polyoxin H is a nucleoside antifungal antibiotic that exhibits significant efficacy against rice sheath blight.</p>Formule :C23H32N6O13Couleur et forme :SolidMasse moléculaire :600.53Sannamycin J
CAS :<p>Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C14H30N4O4Couleur et forme :SolidMasse moléculaire :318.41Bacithrocin C
CAS :<p>Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.</p>Formule :C18H27N5O3Couleur et forme :SolidMasse moléculaire :361.439PD-1/PD-L1-IN-30
CAS :<p>PD-1/PD-L1-IN-30: Cancer research inhibitor with 0.018 μM IC50.</p>Formule :C29H28F3NO5Couleur et forme :SolidMasse moléculaire :527.53ODN 2088
CAS :<p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>Couleur et forme :SolidCalphostin I
CAS :<p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>Formule :C44H38O15Couleur et forme :SolidMasse moléculaire :806.76Endophenazine A
CAS :<p>Endophenazine A exhibits activity against Gram-positive bacteria and filamentous fungi such as Mucor and Penicillium, but demonstrates limited herbicidal effect on Lemna.</p>Formule :C18H16N2O2Couleur et forme :SolidMasse moléculaire :292.332Anti-ToCV agent 1
<p>Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.</p>Formule :C22H19FN2O5SCouleur et forme :SolidMasse moléculaire :442.46Neihumicin
CAS :<p>Neihumicin exhibits resistance against the yeast Saccharomyces cerevisiae (ATCC 9763) and the mold Penicillium italicum (Wehmer), but it does not show resistance to bacteria.</p>Formule :C19H16N2O2Couleur et forme :SolidMasse moléculaire :304.342AMPK Activator SC4
CAS :<p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>Formule :C26H18ClN3O4Couleur et forme :SolidMasse moléculaire :471.89U 75875
CAS :<p>U 75875 is a protease inhibitor.</p>Formule :C45H61N7O7Couleur et forme :SolidMasse moléculaire :812.01BMS-986120
CAS :BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.Formule :C23H23N5O5S2Couleur et forme :SolidMasse moléculaire :513.59Pateamine A
CAS :<p>Pateamine A: marine-sourced macrolide from Mycale hentscheli; anticancer, antiviral, and translation inhibitor.</p>Formule :C31H45N3O4SCouleur et forme :SolidMasse moléculaire :555.77Dermostatin A
CAS :<p>Dermostatin A is a polyene antibiotic with antifungal properties suitable for studying fungal infections.</p>Formule :C40H64O11Couleur et forme :SolidMasse moléculaire :720.93Nanaomycin B
CAS :<p>Nanaomycin B is an antibiotic with activity against Gram-positive bacteria, mycobacteria, mycoplasma, and fungi.</p>Formule :C16H16O7Couleur et forme :SolidMasse moléculaire :320.294Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formule :C20H22N2OCouleur et forme :SolidMasse moléculaire :306.4LH secretion antagonist 1
CAS :<p>LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.</p>Formule :C18H24ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.84ZIKV-IN-5
<p>ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.</p>Formule :C36H45NO4SiCouleur et forme :SolidMasse moléculaire :583.83TP-030-2
CAS :<p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>Formule :C23H21BrN4O3Couleur et forme :SolidMasse moléculaire :481.34YKL-05-093
CAS :<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formule :C35H40N6O4Couleur et forme :SolidMasse moléculaire :608.73TLR7/8 antagonist 2
<p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>Formule :C22H26FN5Couleur et forme :SolidMasse moléculaire :379.47ATX inhibitor 22
<p>ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.</p>Formule :C19H17Cl3F2N2O4SCouleur et forme :SolidMasse moléculaire :513.77Calphostin D
CAS :<p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>Formule :C30H30O10Couleur et forme :SolidMasse moléculaire :550.55GSK065
CAS :<p>GSK065 is a potent inhibitor of kynurenine-3-monooxygenase (KMO).</p>Formule :C17H15ClN2O4Couleur et forme :SolidMasse moléculaire :346.77GYKI-53784
CAS :<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Formule :C19H20N4O3Couleur et forme :SolidMasse moléculaire :352.39Feudomycin B
CAS :<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Formule :C28H31NO10Couleur et forme :SolidMasse moléculaire :541.546SLC4011540
<p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>Formule :C24H23ClF3N7OSCouleur et forme :SolidMasse moléculaire :550PF-446687
CAS :<p>PF-446687 is a highly selective MC4 receptor (MC4R) agonist.</p>Formule :C28H37ClF2N2O2Couleur et forme :SolidMasse moléculaire :507.06Xylarianaphthol-1
CAS :<p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>Formule :C16H20BrFN2O2Couleur et forme :SolidMasse moléculaire :371.24Granaticin B
CAS :<p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>Formule :C28H30O12Couleur et forme :SolidMasse moléculaire :558.531SOAT-IN-1
CAS :SOAT-IN-1 (compound 40) is a potent and selective inhibitor targeting the sodium-dependent organic anion transporter (SOAT), exhibiting IC50 values of 1.6 µM for SOAT and 14.3 µM for NTCP.Formule :C20H16ClN3O6SCouleur et forme :SolidMasse moléculaire :461.88
