Autres inhibiteurs
Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.
37921 produits trouvés pour "Autres inhibiteurs"
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YEATS4 binder-1
<p>YEATS4 binder-1(4e) is an effective and selective compound that targets the KAc recognition site within the YEATS structural domain, exhibiting a binding</p>Formule :C23H34N4O3Couleur et forme :SolidMasse moléculaire :414.54Pyrromycin
CAS :<p>Pyrromycin is a monosaccharide anthracycline which can be used to inhibit cellular RNA synthesis.</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.60Griseolic acid C
CAS :<p>Griseolic acid C (Dihydrodeoxygriseolic acid) is an antibiotic found in the Streptomyces griseoaurantiacus SANK43894 strain. This compound is a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase [EC 3.1.4.17], with an IC50 of 0.12 μM (enzyme sourced from rat brain tissue).</p>Formule :C14H15N5O7Couleur et forme :SolidMasse moléculaire :365.298GRPR antagonist-1
<p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>Formule :C29H33F3N4O4Couleur et forme :SolidMasse moléculaire :558.59Epiderstatin
CAS :<p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>Formule :C15H20N2O4Couleur et forme :SolidMasse moléculaire :292.33SCP1-IN-2
<p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>Formule :C19H17F3N2O6S2Couleur et forme :SolidMasse moléculaire :490.47Dihydrokainic acid
CAS :<p>EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake</p>Formule :C10H17NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :215.25Polyoxin H
CAS :<p>Polyoxin H is a nucleoside antifungal antibiotic that exhibits significant efficacy against rice sheath blight.</p>Formule :C23H32N6O13Couleur et forme :SolidMasse moléculaire :600.53Granaticin B
CAS :<p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>Formule :C28H30O12Couleur et forme :SolidMasse moléculaire :558.531Salvinorin A Propionate
CAS :<p>Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.</p>Formule :C24H30O8Couleur et forme :SolidMasse moléculaire :446.49Heme Oxygenase-1-IN-2
<p>Heme Oxygenase-1-IN-2 is a novel inhibitor of heme oxygenase-1 (HO-1), displaying potent antiproliferative activity in vitro, with an IC50 value of 0.95 μM.</p>Formule :C19H18ClN3OCouleur et forme :SolidMasse moléculaire :339.82L-690330 hydrate
<p>L-690330 hydrate inhibits IMPase; Ki: 0.30 μM (human), 0.42 μM (bovine cortex); 0.27 μM (recom. human), 0.19 μM (bovine).</p>Formule :C8H14O9P2Couleur et forme :SolidMasse moléculaire :316.14Calphostin A
CAS :<p>Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.</p>Formule :C44H38O12Couleur et forme :SolidMasse moléculaire :758.77CYP11B1-IN-2
<p>CYP11B1-IN-2 selectively inhibits human and rat CYP11B1 (IC50: 9/25 nM) orally to research cortisol-related diseases.</p>Couleur et forme :SolidPiperazinomycin
CAS :<p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>Formule :C18H20N2O2Couleur et forme :SolidMasse moléculaire :296.36Epithienamycin A
CAS :<p>Epithienamycin A is a carbapenem antibiotic demonstrating activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C13H18N2O5SCouleur et forme :SolidMasse moléculaire :314.357SGK1-IN-3
<p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>Formule :C23H20Cl2N6O3SCouleur et forme :SolidMasse moléculaire :531.41NAZ2329
CAS :<p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>Formule :C21H18F3NO4S3Couleur et forme :SoildMasse moléculaire :501.56Antitumor agent-187
CAS :<p>Antitumor agent-187 (compound I) is an isoflavone derivative with antitumor activity. It exhibits IC50 values of 5.23 μM and 2.63 μM against A2780 and SKOV3 cell lines, respectively.</p>Formule :C24H26N2O7Couleur et forme :SolidMasse moléculaire :454.47p38-α MAPK-IN-5
CAS :<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Formule :C37H49N11O2Couleur et forme :SolidMasse moléculaire :679.86AMG-222 tosylate
CAS :<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Formule :C39H47N9O6SCouleur et forme :SolidMasse moléculaire :769.91Crotocin
CAS :<p>Crotocin exhibits bactericidal activity against Cryptococcus neoformans, Candida albicans, and Saccharomyces cerevisiae (brewer’s yeast), but it can be inactivated by blood.</p>Formule :C19H24O5Couleur et forme :SolidMasse moléculaire :332.391Annonin VI
CAS :<p>Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.</p>Formule :C37H66O7Couleur et forme :SolidMasse moléculaire :622.92GW-597901 cinnamate
CAS :<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formule :C34H46N2O8SCouleur et forme :SolidMasse moléculaire :642.80Sannamycin J
CAS :<p>Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C14H30N4O4Couleur et forme :SolidMasse moléculaire :318.41PPARα/γ agonist 1
<p>PPARα/γ agonist 1 is a potent and dual PPARα/γ partial agonist which is a promising prototype for the research of dyslipidemia and diabetes.</p>Formule :C18H19NO2Couleur et forme :SolidMasse moléculaire :281.35Elaiomycin
CAS :<p>Elaiomycin exhibits activity against Gram-positive bacteria, certain anaerobic bacteria, Eimeria tenella, and Eimeria stiedai.</p>Formule :C13H26N2O3Couleur et forme :SolidMasse moléculaire :258.3571-Deamino-1-hydroxygentamicin C1a
CAS :<p>1-Deamino-1-hydroxygentamicin C1a (AntibioticSU-2) is an aminoglycoside antibiotic effective against both gram-positive and gram-negative bacteria.</p>Formule :C19H38N4O8Couleur et forme :SolidMasse moléculaire :450.527Cytochalasin L
CAS :<p>Cytochalasin L possesses reversible biological activities, including the inhibition of cytoplasmic division, as well as the suppression of both endocytosis and exocytosis in phagocytic macrophages.</p>Formule :C32H37NO7Couleur et forme :SolidMasse moléculaire :547.639Gentamicin A
CAS :<p>Gentamicin A is an antibiotic exhibiting effective antibacterial activity against both Gram-positive and Gram-negative bacteria, and it also demonstrates activity against most methicillin-sensitive staphylococci.</p>Formule :C18H36N4O10Couleur et forme :SolidMasse moléculaire :468.499Plumbemycin B
CAS :<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Formule :C12H21N4O8PCouleur et forme :SolidMasse moléculaire :380.29Napyradiomycin C2
CAS :<p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>Formule :C25H27Cl3O5Couleur et forme :SolidMasse moléculaire :513.838ONO-AE1-259 lysine
CAS :<p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>Formule :C28H49ClN2O6Couleur et forme :SolidMasse moléculaire :545.15Hynapene B
CAS :<p>Hynapene B exhibits an inhibitory minimum inhibitory concentration (MIC) of 34.7 μM against Eimeria tenella.</p>Formule :C18H24O3Couleur et forme :SolidMasse moléculaire :288.381Melithiazole N
CAS :<p>Melithiazol N is an antibiotic. It acts as a β-methoxyacrylate (MOA) inhibitor with potent antidrug activity.</p>Formule :C20H24N2O5S2Couleur et forme :SolidMasse moléculaire :436.545AMPK Activator SC4
CAS :<p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>Formule :C26H18ClN3O4Couleur et forme :SolidMasse moléculaire :471.89PF1070A
CAS :<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Formule :C31H44N4O6Couleur et forme :SolidMasse moléculaire :568.710-Decarbomethoxyaclacinomycin A
CAS :<p>10-Decarbomethoxyaclacinomycin A is an anthracycline antibiotic produced by the mutant strain Streptomyces galilaeus MA144-Mlt KE303. This compound exhibits antibacterial activity.</p>Formule :C40H51NO13Couleur et forme :SolidMasse moléculaire :753.832PF-06815345 hydrochloride
CAS :<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Formule :C27H30Cl2FN9O4Couleur et forme :SolidMasse moléculaire :634.49Pacidamycin D
CAS :<p>Pacidamycin D is an antibiotic of the Pacidamycin class, demonstrating activity against Pseudomonas aeruginosa with a minimum inhibitory concentration (MIC) of 4-16 μg/mL. It shows no efficacy against other Gram-negative or Gram-positive bacteria, nor does it affect drug-resistant strains of Pseudomonas aeruginosa.</p>Formule :C32H41N9O10Couleur et forme :SolidMasse moléculaire :711.722FR-900482
CAS :<p>FR-900482 exhibits high sensitivity to Thermoactinomyces calidolactis strain C 953 and demonstrates activity against cell lines such as P388, B16, EL4, FM3A, L1210, BHK-21, among others.</p>Formule :C14H15N3O6Couleur et forme :SolidMasse moléculaire :321.29Epoxyquinomicin A
CAS :<p>Epoxyquinomicin A is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus with MIC values of 3-12.5 µg/mL. Additionally, it shows cytotoxicity in cancer cells L1210, B16, and S180, with an IC50 of 2-8 µg/mL. Furthermore, Epoxyquinomicin A demonstrates anti-inflammatory effects in collagen-induced arthritis.</p>Formule :C14H10ClNO6Couleur et forme :SolidMasse moléculaire :323.685BAY-850 HCl
<p>BAY-850 is a selective probe targeting Atad2A's bromine domain, displacing acetylated H4 peptides and detaching ATAD2 from chromatin at 1μm.</p>Formule :C38H48Cl5N5O3Couleur et forme :SolidMasse moléculaire :800.08Eupenoxide
CAS :<p>Eupenoxide is an antibiotic with antifungal properties, derived from fungi belonging to the Eupenicillium genus.</p>Formule :C14H22O4Couleur et forme :SolidMasse moléculaire :254.322CGS 22652
CAS :<p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>Formule :C22H29ClN2O4SCouleur et forme :SolidMasse moléculaire :452.99FTI 276 TFA
CAS :<p>FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).</p>Formule :C23H28F3N3O5S2Couleur et forme :SolidMasse moléculaire :547.61Megovalicin G
CAS :<p>Megovalicin G is effective against Bacillus subtilis and Escherichia coli, and it also acts on Pseudomonas aeruginosa.</p>Formule :C35H61NO7Couleur et forme :SolidMasse moléculaire :607.86KT2-962
CAS :<p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>Formule :C23H27ClNNaO5S2Couleur et forme :SolidMasse moléculaire :520.04CU-2010
CAS :<p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>Formule :C37H42N6O6SCouleur et forme :SolidMasse moléculaire :698.833-epi-Deoxynegamycin
CAS :<p>3-epi-Deoxynegamycin exhibits antibacterial activity, primarily effective against most Gram-positive bacteria, while its effectiveness is somewhat reduced against Gram-negative bacteria.</p>Formule :C9H20N4O3Couleur et forme :SolidMasse moléculaire :232.28Anticancer agent 35
<p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>Formule :C15H13N3O3S3Couleur et forme :SolidMasse moléculaire :379.48Enteromycin
CAS :<p>Enteromycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C6H8N2O5Couleur et forme :SolidMasse moléculaire :188.138Kri 1314
CAS :<p>Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.</p>Formule :C38H51N5O7Couleur et forme :SolidMasse moléculaire :689.84Antiviral agent 6
<p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>Formule :C23H27BrN2O3S2Couleur et forme :SolidMasse moléculaire :523.513-Methoxy-2,5-toluquinone
CAS :<p>3-Methoxy-2,5-toluquinone is an antimicrobial agent that exhibits moderate antibacterial and antifungal properties.</p>Formule :C8H8O3Couleur et forme :SolidMasse moléculaire :152.147FR 900452
CAS :<p>FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.</p>Formule :C22H25N3O3SCouleur et forme :SolidMasse moléculaire :411.52Henagliflozin
CAS :<p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>Formule :C22H24ClFO7Couleur et forme :SolidMasse moléculaire :454.87Fumaryl-DL-alanine
CAS :<p>Fumaryl-DL-alanine exhibits activity against Gram-positive bacteria.</p>Formule :C7H9NO5Couleur et forme :SolidMasse moléculaire :187.15Eurystatin A
CAS :<p>Eurystatin A is a prolyl endopeptidase inhibitor, with L-leucine and L-ornithine serving as direct precursors to the L-leucine and L-ornithine components of eurystatins A.</p>Formule :C23H38N4O5Couleur et forme :SolidMasse moléculaire :450.572ATX inhibitor 22
<p>ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.</p>Formule :C19H17Cl3F2N2O4SCouleur et forme :SolidMasse moléculaire :513.77Oncopterin
CAS :<p>Oncopterin is found in urine from patients with solid and blood cancers.</p>Formule :C12H18N6O3Couleur et forme :SolidMasse moléculaire :294.31Juglomycin A
CAS :<p>Juglomycin A exhibits broad-spectrum antibacterial and anti-mycobacterial activity and can inhibit Ehrlich ascites carcinoma in mice.</p>Formule :C14H10O6Couleur et forme :SolidMasse moléculaire :274.226Sucistil
<p>Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].</p>Formule :C9H15NO4SCouleur et forme :SolidMasse moléculaire :233.28iMDK quarterhydrate
<p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>Formule :C21H15FN2O3SCouleur et forme :SolidMasse moléculaire :380.91FTO-IN-1 TFA
<p>FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.</p>Formule :C20H17Cl2F3N4O4Couleur et forme :SolidMasse moléculaire :505.27Transthyretin-IN-1
<p>Transthyretin-IN-1 inhibits TTR fibril formation, aiding Alzheimer’s research.</p>Formule :C10H9Br2NO4Couleur et forme :SolidMasse moléculaire :366.991-Hydroxyoxaunomycin
CAS :<p>1-Hydroxyoxaunomycin is an antibiotic that inhibits the growth of U210 cells as well as the synthesis of DNA and RNA, with IC50 values of 0.0005 μg/mL, 1.00 μg/mL, and 0.76 μg/mL, respectively.</p>Formule :C26H29NO11Couleur et forme :SolidMasse moléculaire :531.509Gentamicin C2
CAS :<p>Gentamicin C2 is an aminoglycoside antibiotic.</p>Formule :C20H41N5O7Couleur et forme :SolidMasse moléculaire :463.569C-di-IMP
CAS :<p>Cyclic-di-IMP (C-di-IMP), a STING agonist, serves as a research tool in tumor studies.</p>Formule :C20H22N8O14P2Couleur et forme :SolidMasse moléculaire :660.38AKR1C3-IN-7
<p>AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.</p>Formule :C24H20N2O4Couleur et forme :SolidMasse moléculaire :400.433-O-Demethylmonensin A
CAS :<p>3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).</p>Formule :C35H60O11Couleur et forme :SolidMasse moléculaire :656.84Bacithrocin B
CAS :<p>Bacithrocin B is a thrombin inhibitor that suppresses the activity of thrombin, Factor Xa, trypsin, and papain, with IC50 values of 84 μM, 17 μM, 1.7 μM, and 0.02 μM, respectively.</p>Formule :C19H29N5O3Couleur et forme :SolidMasse moléculaire :375.465MtDTBS-IN-1
<p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>Formule :C16H16N4O5Couleur et forme :SolidMasse moléculaire :344.32HS-731
CAS :<p>HS-731 is a μ-Opioid Receptor Agonist.</p>Formule :C20H26N2O5Couleur et forme :SolidMasse moléculaire :374.43Oximidine Ⅲ
CAS :<p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>Formule :C23H24N2O6Couleur et forme :SolidMasse moléculaire :424.45GYKI-53784
CAS :<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Formule :C19H20N4O3Couleur et forme :SolidMasse moléculaire :352.39Difeterol
CAS :<p>Difeterol is a biochemical.</p>Formule :C25H29NO2Couleur et forme :SolidMasse moléculaire :375.50Bacithrocin C
CAS :<p>Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.</p>Formule :C18H27N5O3Couleur et forme :SolidMasse moléculaire :361.439Exfoliamycin
CAS :<p>Exfoliamycin is a naphthoquinone antibiotic found in the Streptomyces strain Exfoliamycin Tu 1424, and it exhibits activity against Gram-positive bacteria.</p>Formule :C22H26O9Couleur et forme :SolidMasse moléculaire :434.436Naltrindole
CAS :<p>Naltrindole is a delta opioid receptor antagonist.</p>Formule :C26H26N2O3Couleur et forme :SolidMasse moléculaire :414.5Sovesudil hydrochloride
<p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>Formule :C23H23ClFN3O3Couleur et forme :SolidMasse moléculaire :443.9Trk-IN-7
<p>Trk-IN-7 inhibits TRKA/B/C (IC50: 0.25-10 nM) & EML4-ALK (<15 nM), also targets various ALK mutations (IC50: 5-50 nM).</p>Formule :C18H17FN6O2Couleur et forme :SolidMasse moléculaire :368.36Gepotidacin hydrochloride
CAS :<p>Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.</p>Formule :C24H29ClN6O3Couleur et forme :SolidMasse moléculaire :484.98Xylarianaphthol-1
CAS :<p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>Formule :C16H20BrFN2O2Couleur et forme :SolidMasse moléculaire :371.24Antiangiogenic agent 3
<p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>Formule :C19H20O7Couleur et forme :SolidMasse moléculaire :360.36Citrinin hydrate
CAS :<p>Citrinin hydrate is an inhibitor of human rhinovirus (HRV) 3C protease, with an IC50 of 1.0 mM.</p>Formule :C13H16O6Couleur et forme :SolidMasse moléculaire :268.263Fusarin C
CAS :<p>Fusarin C is a mutagenic compound found in strains of the Fusarium genus.</p>Formule :C23H29NO7Couleur et forme :SolidMasse moléculaire :431.4791-Hydroxy-2-nonyn-4-one
CAS :<p>1-Hydroxy-2-nonyn-4-one is an antibiotic with activity against yeasts, filamentous fungi, tumors, and shows weak efficacy against both Gram-positive and Gram-negative bacteria.</p>Formule :C9H14O2Couleur et forme :SolidMasse moléculaire :154.206Dienomycin B
CAS :<p>Dienomycin B exhibits mild antibacterial activity.</p>Formule :C18H23NO2Couleur et forme :SolidMasse moléculaire :285.38NS2B/NS3-IN-4
CAS :<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Formule :C15H11NO4Couleur et forme :SolidMasse moléculaire :269.25Pyloricidin B
CAS :<p>Pyloricidin B is an antibiotic specifically effective against Helicobacter pylori, showing potent anti-Helicobacter pylori activity. It exhibits no activity against other bacteria or yeast.</p>Formule :C26H42N4O9Couleur et forme :SolidMasse moléculaire :554.63Panosialin wA
CAS :<p>Panosialin wA inhibits α,β-glucosidase and mannosidase enzymes, but does not exhibit inhibitory activity against the influenza virus. However, it has a mild antibacterial effect.</p>Formule :C21H36O5SCouleur et forme :SolidMasse moléculaire :400.57Clavamycin E
CAS :<p>Clavamycin E is a clavulanic acid antibiotic.</p>Formule :C11H17N3O6Couleur et forme :SolidMasse moléculaire :287.269LMD-A
CAS :<p>LMD-A, also known as CCR8 antagonist LMD-A, is a CCR8 antagonist.</p>Formule :C27H32N4O4SCouleur et forme :SolidMasse moléculaire :508.63Endophenazine D
CAS :<p>Endophenazine D is a phenazine-class antibiotic.</p>Formule :C15H12N2O4Couleur et forme :SolidMasse moléculaire :284.27Saframycin D
CAS :<p>Saframycin D exhibits activity against Gram-positive bacteria and shows weaker potency against mycobacteria.</p>Formule :C28H31N3O9Couleur et forme :SolidMasse moléculaire :553.56Canosimibe
CAS :<p>Canosimibe is a cholesterol absorption inhibitor</p>Formule :C44H60FN3O10Couleur et forme :SolidMasse moléculaire :809.96Quinagolide Free Base
CAS :<p>Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.</p>Formule :C20H33N3O3SCouleur et forme :SolidMasse moléculaire :395.56Steroid sulfatase/17β-HSD1-IN-4
<p>Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).</p>Formule :C18H17N3O4S2Couleur et forme :SolidMasse moléculaire :403.48WAY-855
CAS :<p>WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.</p>Formule :C9H11NO4Couleur et forme :SolidMasse moléculaire :197.19Metocurine chloride
CAS :<p>Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.</p>Formule :C40H48Cl2N2O6Couleur et forme :SolidMasse moléculaire :723.72Espinomycin A3
CAS :<p>Espinomycin A3 is a 16-membered macrolide antibiotic (antibiotic) that exhibits activity against Gram-positive bacteria.</p>Formule :C40H65NO15Couleur et forme :SolidMasse moléculaire :799.942Benadrostin
CAS :<p>Benadrostin is a Poly(ADP-ribose) synthetase inhibitor with an IC50 of 35μM.</p>Formule :C8H5NO4Couleur et forme :SolidMasse moléculaire :179.13TEI-9063
CAS :<p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>Formule :C23H38O4Couleur et forme :SolidMasse moléculaire :378.55Carpetimycin C
CAS :<p>Carpetimycin C exhibits strong activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. It also has a powerful inhibitory effect on β-lactamase .</p>Formule :C14H20N2O6SCouleur et forme :SolidMasse moléculaire :344.383Mycelianamide
CAS :<p>Mycelianamide is an antibiotic effective against Gram-positive bacteria.</p>Formule :C22H28N2O5Couleur et forme :SolidMasse moléculaire :400.468Leu-AMS R enantiomer
CAS :<p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>Formule :C16H25N7O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.48Calcipotriol Impurity C
CAS :<p>Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.</p>Formule :C27H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.614Alentemol hydrobromide
CAS :<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formule :C19H26BrNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.32Leucomycin U
CAS :<p>Leucomycin U is a macrolide antibiotic. It demonstrates significant activity against Gram-positive bacteria and also exhibits effects on spirochetes, rickettsiae, and chlamydiae.</p>Formule :C37H61NO14Couleur et forme :SolidMasse moléculaire :743.878Dinordrin I diacetate
CAS :<p>Dinordrin I diacetate is an implantation inhibitor and hormone.</p>Formule :C25H32O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.52Lorajmine
CAS :<p>Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.</p>Formule :C22H27ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.91MEIS-IN-1
CAS :<p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>Formule :C24H21F3N2O4Couleur et forme :SolidMasse moléculaire :458.43EP4 receptor antagonist 2
CAS :<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formule :C27H29N3O5Couleur et forme :SolidMasse moléculaire :475.54Hetrombopag olamine
CAS :<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Formule :C29H36N6O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :580.63FR 901537
CAS :<p>FR 901537 is a new aromatase inhibitor with antitumor effects.</p>Formule :C23H29N3O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.62PF-446687
CAS :<p>PF-446687 is a highly selective MC4 receptor (MC4R) agonist.</p>Formule :C28H37ClF2N2O2Couleur et forme :SolidMasse moléculaire :507.063HKT-IN-1
CAS :<p>3HKT-IN-1 (Compound 17122279) is an inhibitor of Anopheles gambiae 3-hydroxykynurenine transaminase (3HKT) and is utilized in malaria research.</p>Formule :C12H11BrN2O3Couleur et forme :SolidMasse moléculaire :311.131KUSC-5037
<p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>Formule :C18H17F3N6O2Couleur et forme :SolidMasse moléculaire :406.13651DWN-12088 HCl
CAS :<p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>Formule :C15H21Cl4N3OCouleur et forme :SolidMasse moléculaire :401.15Dihydropergillin
CAS :<p>Dihydropergillin is produced by the Aspergillus terreus strain (ATCC 38849) and has the ability to inhibit plant growth.</p>Formule :C15H18O4Masse moléculaire :262.30BMS-748730
CAS :<p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>Formule :C22H26ClN7O3SCouleur et forme :SolidMasse moléculaire :504.01Resorcinomycin A
CAS :<p>Resorcinomycin A is an antibiotic with potent antimycobacterial activity and relatively weaker activity against mycoplasma.</p>Formule :C14H20N4O5Couleur et forme :SolidMasse moléculaire :324.332Glucoallosamidin A
CAS :<p>Glucoallosamidin A is a glycoside antibiotic that inhibits chitinase activity. It effectively suppresses the chitinase enzyme in Candida albicans [ATCC 10231], exhibiting an IC50 of 3.4 μg/mL.</p>Formule :C26H44N4O14Couleur et forme :SolidMasse moléculaire :636.646Eurocidin E
CAS :<p>Eurocidin E is an antibiotic that inhibits degranulation and histamine release from rat mast cells.</p>Formule :C40H61NO14Couleur et forme :SolidMasse moléculaire :779.911RSV-IN-5
CAS :<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Formule :C28H37N7O2Couleur et forme :SolidMasse moléculaire :503.64Lp-PLA2-IN-6
CAS :<p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>Formule :C25H21F5N4O3Couleur et forme :SolidMasse moléculaire :520.45Glaucarubin
CAS :<p>Glaucarubin is a bitter lactone naturally found in the fruits of Simaruba glauca. It is employed as an anti-amebic agent in research focused on amebiasis. The compound exhibits good tolerability, with a median lethal dose (LD50) of 1,600 mg/kg in mice and 6,400 mg/kg in rats.</p>Formule :C25H36O10Masse moléculaire :496.55Porothramycin B
CAS :<p>Porothramycin B is an antibiotic with activity against Gram-positive bacteria and anaerobes.</p>Formule :C19H23N3O4Couleur et forme :SolidMasse moléculaire :357.404Ornoprostil
CAS :<p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>Formule :C23H38O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.54Epelmycin D
CAS :<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Formule :C30H35NO11Couleur et forme :SolidMasse moléculaire :585.599Butaprost
CAS :<p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>Formule :C24H40O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.57Gentamicin C1
CAS :<p>Gentamicin C1 is a broad-spectrum aminoglycoside antibiotic with antibacterial activity.</p>Formule :C21H43N5O7Couleur et forme :SolidMasse moléculaire :477.595Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formule :C20H22N2OCouleur et forme :SolidMasse moléculaire :306.4RS 2135
CAS :<p>RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.</p>Formule :C18H21ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.83Hypercalin B
CAS :<p>Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.</p>Formule :C33H42O5Couleur et forme :SolidMasse moléculaire :518.684Haloquinone
CAS :<p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>Formule :C17H12O5Couleur et forme :SolidMasse moléculaire :296.274P2X receptor-1
<p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>Formule :C14H14ClN3O3S2Couleur et forme :SolidMasse moléculaire :371.86Cbl-b-IN-1
CAS :<p>Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.</p>Formule :C29H34N6O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :498.631BRD-9526
CAS :<p>BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).</p>Formule :C26H31Cl2N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :584.51IDX-320
CAS :<p>IDX-320 is an HCV protease inhibitor.</p>Formule :C37H43F3N6O7S2Couleur et forme :SolidMasse moléculaire :804.9Anti-Trypanosoma cruzi agent-1
<p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>Formule :C23H29N3O5Couleur et forme :SolidMasse moléculaire :427.49L 767679
CAS :<p>L 767679 is an antagonist of the fibrinogen receptors.</p>Formule :C20H24N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :384.43γ-Chloronorvaline
CAS :<p>γ-Chloronorvaline exhibits antimicrobial activity against Pseudomonas aeruginosa, Serratia, Klebsiella pneumoniae, and Bacillus subtilis in synthetic media, while it shows no effect on Escherichia coli.</p>Formule :C5H10ClNO2Couleur et forme :SolidMasse moléculaire :151.591PD-1-IN-17 TFA
<p>PD-1-IN-17 TFA is a potent PD-1 inhibitor, blocking 92% of splenocyte growth at 100 nM.</p>Formule :C15H23F3N6O9Couleur et forme :SolidMasse moléculaire :488.37Harziphilone
CAS :<p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>Formule :C15H18O4Couleur et forme :SolidMasse moléculaire :262.301SSR-182289A (Free)
CAS :<p>SSR-182289A (Free) is a thrombin inhibitor.</p>Formule :C30H33F2N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.68Dinordrin
CAS :<p>Dinordrin is an implantation inhibitor and hormone.</p>Formule :C27H36O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.57Melithiazole A
CAS :<p>Melithiazol A is an antibiotic and a potent β-methoxyacrylate (MOA) inhibitor with antifungal and cytotoxic properties.</p>Formule :C20H26N2O4S2Couleur et forme :SolidMasse moléculaire :422.561Revamilast sodium
CAS :<p>Revamilast sodium, also known as GRC4039 sodium, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritis</p>Formule :C18H8Cl2F2N3NaO4Couleur et forme :SolidMasse moléculaire :462.17GP-1681
CAS :<p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>Formule :C24H30NaO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.48Calphostin I
CAS :<p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>Formule :C44H38O15Couleur et forme :SolidMasse moléculaire :806.76Enpp-1-IN-12
<p>ENPP1-IN-12 is a potent, oral ENPP1 inhibitor with a Ki of 41 nM and anti-tumor properties.</p>Formule :C17H19N5O3SCouleur et forme :SolidMasse moléculaire :373.43OncoFAP
CAS :<p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>Formule :C21H19F2N5O5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :459.40UNC7467
CAS :<p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>Formule :C20H13NO3Degré de pureté :98.28% - 98.64%Couleur et forme :SoildMasse moléculaire :315.32Celesticetin B
CAS :<p>Celesticetin B is an antibiotic primarily exhibiting antibacterial activity against Gram-positive microorganisms.</p>Formule :C21H38N2O8SCouleur et forme :SolidMasse moléculaire :478.6Griseolutein A
CAS :<p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C17H14N2O6Couleur et forme :SolidMasse moléculaire :342.303Anti-inflammatory agent 16
<p>Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.</p>Formule :C21H23N5O3Couleur et forme :SolidMasse moléculaire :393.44De-N-methylpamamycin-593A
CAS :<p>De-N-methylpamamycin-593A is a 16-membered macrocyclic dilactone known for its ability to induce aerial mycelium formation.</p>Formule :C34H59NO7Masse moléculaire :593.84D18
CAS :<p>D18: Dual agonist for TLR7/8, boosts PD-L1, aids tumor sensitivity to PD-1/PD-L1 inhibitors, and is a cytotoxin for ADC HE-S2.</p>Formule :C21H28N6Couleur et forme :SolidMasse moléculaire :364.49Rhamnitol
CAS :<p>Rhamnitol, the reduction product of L-rhamnose, can be observed during the metabolism of rhamnose in the body. Rhamnitol is promising for use in assessing intestinal permeability and studying carbohydrate metabolism.</p>Formule :C6H14O5Couleur et forme :SolidMasse moléculaire :166.17SS-RJW100
<p>SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.</p>Formule :C28H34OCouleur et forme :SolidMasse moléculaire :386.57Pluracidomycin C2
CAS :<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formule :C11H15NO9S2Couleur et forme :SolidMasse moléculaire :369.37Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Formule :C24H26O8Couleur et forme :SolidMasse moléculaire :442.46H 218-54
CAS :<p>H 218-54 is a renin inhibitor.</p>Formule :C37H56N2O5SCouleur et forme :SolidMasse moléculaire :640.92Hydrolyzed Fumonisin B2
CAS :<p>Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.</p>Formule :C22H47NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.61Demethoxyviridin
CAS :<p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>Formule :C19H14O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.31Antibiotic MA 144M1
CAS :<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formule :C42H55NO15Couleur et forme :SolidMasse moléculaire :813.88J-104118
CAS :<p>J-104118 potentially inhibits squalene synthase.</p>Formule :C28H26Cl2FNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :546.41Nemotin
CAS :<p>Nemotin exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while its effectiveness against Gram-negative bacteria is present but relatively weaker.</p>Formule :C11H8O2Couleur et forme :SolidMasse moléculaire :172.18Papyracon D
CAS :<p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>Formule :C14H18O5Masse moléculaire :266.29METTL3-IN-2
CAS :<p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>Formule :C25H26N8OCouleur et forme :SolidMasse moléculaire :454.53MRS2500
CAS :<p>MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.</p>Formule :C13H18IN5O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :561.16PAT-347
CAS :<p>PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.</p>Formule :C28H21ClF2N2O3SCouleur et forme :SolidMasse moléculaire :538.99Oxythiamine diphosphate ammonium
<p>Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).</p>Couleur et forme :SolidYM-355179
CAS :<p>YM-355179 is a novel, selective antagonist of CC chemokine receptor 3 with oral activity.</p>Formule :C33H34FN4O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :617.64SORT1-IN-3
CAS :<p>SORT1-IN-3 (compound 5) is a SORT1 inhibitor characterized by its ability to permeate the blood-brain barrier.</p>Formule :C16H26ClNO3Couleur et forme :SolidMasse moléculaire :315.84ONO-AE1-329
CAS :<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Formule :C22H30O6S2Couleur et forme :SolidMasse moléculaire :454.6L 668750
CAS :<p>L 668750 is an inhibitor of platelet-activating factor.</p>Formule :C25H34O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.6Maltophilin
CAS :<p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>Formule :C29H38N2O6Masse moléculaire :510.62Anticancer agent 12
<p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>Formule :C16H17BrN4O2SCouleur et forme :SolidMasse moléculaire :409.3Polyoxin J
CAS :<p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>Formule :C17H25N5O12Masse moléculaire :491.41PZ-3022
CAS :<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Formule :C20H21N5OCouleur et forme :SolidMasse moléculaire :347.41S39625
CAS :<p>S39625 is a stable, potent topoisomerase I inhibitor with anticancer properties, resistant to efflux transporters, inducing gamma-H2AX at nanomolar levels.</p>Formule :C25H22N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.45Anticancer agent 79
<p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>Formule :C20H12F3NO5Couleur et forme :SolidMasse moléculaire :403.31RIPK1-IN-14
CAS :<p>RIPK1-IN-14 inhibits RIPK1 with 92 nM IC50 and reduces necrotic apoptosis in U937 cells.</p>Couleur et forme :SoildNovokinin
CAS :<p>Angiotensin AT2 receptor agonist</p>Formule :C39H61N11O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :795.97EP-7041 HCl
CAS :<p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>Formule :C19H27ClN4O4Couleur et forme :SolidMasse moléculaire :410.89L-Tyrosyl-L-glutamic acid
CAS :<p>L-Tyrosyl-L-glutamic acid acts as an inhibitor of the amino acid permease GAP1.</p>Formule :C14H18N2O6Couleur et forme :SolidMasse moléculaire :310.3P-gp modulator 3
<p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>Formule :C31H37N3O5Couleur et forme :SolidMasse moléculaire :531.64RTIOX-372
CAS :<p>RTIOX-372 is a potent and selective orexin-1 receptor antagonist.</p>Formule :C30H39N5O3Couleur et forme :SolidMasse moléculaire :517.66GSK3527497
CAS :<p>GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).</p>Formule :C17H16ClFN4O4SCouleur et forme :SolidMasse moléculaire :426.85Antioxidant agent-3
<p>Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.</p>Formule :C18H14O8Couleur et forme :SolidMasse moléculaire :358.3PREP inhibitor-1
CAS :<p>PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.</p>Formule :C22H28N4O2Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :380.48MV151
CAS :<p>MV151 is a fluorescent proteasome inhibitor that targets all active subunits of the proteasome and immunoproteasome in living cells.</p>Formule :C59H91BF2N8O9SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1137.28O-Propargyl-Puromycin
CAS :<p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>Formule :C24H29N7O5Degré de pureté :97.83% - 99.70%Couleur et forme :SolidMasse moléculaire :495.53VCPIP1-IN-1
CAS :<p>VCPIP1-IN-1 is a VCPIP1 inhibitor used in cancer research.</p>Formule :C13H15ClN2O2Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :266.72OB-1
CAS :<p>OB-1 is a STOML3 inhibitor that interferes with the self-association of stomatin, inhibiting fat formation and blocking lipid droplet growth.</p>Formule :C21H17N3O6Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :407.38YTH-IN-1
CAS :<p>YTH-IN-1 is an inhibitor of the five YTH structural domains in the human.The YTH family of proteins is an N 6-methyladenosine (m6A) reader in gene expression.</p>Formule :C18H24N6O3Degré de pureté :98.46% - 99.94%Couleur et forme :SolidMasse moléculaire :372.42Skp2 inhibitor 1
CAS :<p>Skp2 inhibitor 1 is a Skp2-Cks1 interaction inhibitor (IC50: 2.8μM) with antitumor activity and can be used to study cancer.</p>Formule :C23H23ClN4ODegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :406.91
