
Signalisation du cytosquelette
Les inhibiteurs de la signalisation du cytosquelette sont des composés qui perturbent les voies de signalisation régulant le cytosquelette, essentiel pour la forme, la motilité, la division des cellules et le transport intracellulaire. Ces inhibiteurs sont utilisés pour étudier la dynamique des protéines du cytosquelette, telles que l'actine et la tubuline, et leur rôle dans des processus comme la migration cellulaire, l'adhésion et la métastase du cancer. Les inhibiteurs de la signalisation du cytosquelette sont précieux dans la recherche en biologie cellulaire, en cancérologie et en neurobiologie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs de la signalisation du cytosquelette de haute qualité pour soutenir vos recherches dans ces domaines.
1381 produits trouvés pour "Signalisation du cytosquelette"
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XL228
CAS :<p>XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).</p>Formule :C22H31N9ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :437.54Imatinib
CAS :<p>Imatinib (STI571) is a multi-targeted receptor tyrosine kinase inhibitor that selectively inhibits the kinase activities of BCR/ABL, v-Abl, PDGFR, and c-kit</p>Formule :C29H31N7ODegré de pureté :99.42% - 99.94%Couleur et forme :Off White PowderMasse moléculaire :493.6OSU-T315
CAS :<p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>Formule :C30H30F3N5ODegré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :533.59TPPB
CAS :<p>TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).</p>Formule :C27H30F3N3O3Degré de pureté :97.71% - 98.00%Couleur et forme :SolidMasse moléculaire :501.54Ro 31-8220 Mesylate
CAS :<p>Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor, and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β.</p>Formule :C25H23N5O2S·CH4O3SDegré de pureté :98.79% - 99.02%Couleur et forme :SolidMasse moléculaire :553.65Flumatinib mesylate
CAS :<p>Flumatinib mesylate (HHGV678 mesylate) is a selective inhibitor of c-Abl, PDGFRβ and c-Kit, effectively overcomes drug resistance of certain KIT mutants.</p>Formule :C30H33F3N8O4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :658.69D-64131
CAS :<p>D-64131 is a tubulin polymerization inhibitor with an IC50 value of 0.53 μM.</p>Formule :C16H13NO2Degré de pureté :99.48% - 99.67%Couleur et forme :SolidMasse moléculaire :251.28Tirbanibulin
CAS :<p>Tirbanibulin (KX2-391) is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal models of a variety of cancers.</p>Formule :C26H29N3O3Degré de pureté :99.43% - 99.67%Couleur et forme :SolidMasse moléculaire :431.53Procyanidin A1
CAS :<p>Procyanidin A1 (Proanthocyanidin A1) has antiallergic effects, it inhibits degranulation downstream of protein kinase C activation or Ca2+.</p>Formule :C30H24O12Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :576.5Borussertib
CAS :<p>Borussertib is a covalent-allosteric and first-in-class inhibitor of protein kinase Akt(IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt)</p>Formule :C36H32N6O3Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :596.68Ingenol
CAS :<p>Ingenol mebutate treats actinic keratosis, has anticancer properties, and may reactivate latent HIV.</p>Formule :C20H28O5Degré de pureté :99.78% - 99.87%Couleur et forme :SolidMasse moléculaire :348.43BX517
CAS :<p>BX517 (PDK1 inhibitor 2) is a potent and selective inhibitor of PDK1.</p>Formule :C15H14N4O2Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :282.3Monastrol
CAS :<p>Monastrol ((±)-Monastrol) is a potent and cell-permeable inhibitor of the mitotic kinesin Eg5.</p>Formule :C14H16N2O3SDegré de pureté :98.02% - 98.59%Couleur et forme :SolidMasse moléculaire :292.35Sotrastaurin
CAS :<p>Sotrastaurin (AEB071) is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKCα/βI/δ/ε/η/θ).</p>Formule :C25H22N6O2Degré de pureté :98% - 99.70%Couleur et forme :SolidMasse moléculaire :438.48Valrubicin
CAS :<p>Valrubicin (AD-32) (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.</p>Formule :C34H36F3NO13Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :723.64Pep2m, myristoylated acetate
<p>Pep2m, a myristoylated acetate, inhibits GluA2-NSF interaction, reducing AMPA receptor function and expression in neurons.</p>Formule :C65H122N18O16SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :1443.96PF-431396
CAS :<p>PF-431396 is a dual PYK2/FAK inhibitor (IC50: 11/2 nM).</p>Formule :C22H21F3N6O3SDegré de pureté :98.83% - 99.82%Couleur et forme :SolidMasse moléculaire :506.5Vodobatinib
CAS :<p>Vodobatinib (K-0706) is a novel 3rd generation (3G) TKI effective against wild-type and mutated BCR-ABL1 with limited off-target activity.</p>Formule :C27H20ClN3O2Degré de pureté :99.06% - 99.55%Couleur et forme :SolidMasse moléculaire :453.92Decursin
CAS :<p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>Formule :C19H20O5Degré de pureté :97.22% - 99.84%Couleur et forme :SolidMasse moléculaire :328.36Pimitespib
CAS :<p>Pimitespib (TAS-116) is an ATP-competitive and highly specific HSP90α/HSP90β inhibitor (Kis: 34.7 nM and 21.3 nM, respectively).</p>Formule :C25H26N8ODegré de pureté :99.22% - 99.49%Couleur et forme :SolidMasse moléculaire :454.53Ζ-Stat
CAS :<p>ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis in</p>Formule :C10H8O10S3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :384.36Dimethylenastron
CAS :<p>Dimethylenastron, an Eg5 inhibitor, arrests cells with monopolar spindles to which all chromosomes attach in a syntelic manner.</p>Formule :C16H18N2O2SDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :302.39GLPG0187
CAS :<p>GLPG0187, a broad spectrum integrin receptor antagonist, inhibits αvβ1-integrin (IC50: 1.3 nM).</p>Formule :C29H37N7O5SDegré de pureté :99.4% - 99.70%Couleur et forme :SolidMasse moléculaire :595.71Chelerythrine chloride
CAS :<p>Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to</p>Formule :C21H18ClNO4Degré de pureté :95% - 99.19%Couleur et forme :Yellow To Orange SolidMasse moléculaire :383.83T807
CAS :<p>T807 (AV-1451) is a novel tracer of tau positron emission tomography (PET).</p>Formule :C16H10FN3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :263.27LP-261
CAS :<p>LP-261 is a novel tubulin targeting anticancer agent that binds at the colchicine site on tubulin, inducing G2/M arrest.</p>Formule :C22H19N3O4SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :421.47VER-82576
CAS :<p>VER-82576 (NVP-BEP800), a synthetic HSP90β inhibitor (IC50: 58 nM), exhibits >70-fold selectivity against Hsp90 family members Trap-1 and Grp94.</p>Formule :C21H23Cl2N5O2SDegré de pureté :97.31% - 99.85%Couleur et forme :SolidMasse moléculaire :480.41PND-1186
CAS :<p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>Formule :C25H26F3N5O3Degré de pureté :99.14% - 99.75%Couleur et forme :SolidMasse moléculaire :501.5PF-562271 hydrochloride
CAS :<p>PF-562271 hydrochloride (PF-562271 HCl) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK.</p>Formule :C21H20F3N7O3SHClDegré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :543.95R59949
CAS :<p>R59949 is used as a Diacylglycerol kinase (DGK) inhibitor.</p>Formule :C28H25F2N3OSDegré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :489.58Natalizumab
CAS :<p>Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.</p>Degré de pureté :98.00%Couleur et forme :LiquidMasse moléculaire :N/AEmpesertib
CAS :<p>Empesertib (BAY 1161909) is an orally bioavailable and selective inhibitor Mps1(IC50 < 1 nM), with potential antineoplastic activity.</p>Formule :C29H26FN5O4SDegré de pureté :97.45% - 99.4%Couleur et forme :SolidMasse moléculaire :559.61MAP4343
CAS :<p>Map4343, a 3-methyl ether pregnenolone derivative, binds MAP2, boosts tubulin polymerization, spurs neurite growth, and guards neurons.</p>Formule :C22H34O2Degré de pureté :97.024%Couleur et forme :SolidMasse moléculaire :330.5HSF1A
CAS :<p>HSF1A is a cell-permeable activator of HSF1 that protects mammalian cells against stress-induced apoptosis.</p>Formule :C21H19N3O2S2Degré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :409.52Curvulin
CAS :<p>Curvulin is the active metabolite isolated from Paraphoma sp. VIZR 1.46. Curvularin inhibits iNOS expression and microtubule assembly.</p>Formule :C12H14O5Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :238.24TASP0415914
CAS :<p>TASP0415914 is an orally potent inhibitor of phosphoinositide 3-kinase γ (PI3Kγ). T</p>Formule :C13H17N5O3SDegré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :323.37Mavacamten
CAS :<p>Mavacamten (MYK-461) is an orally bioavailable inhibitor of cardiac myosin ATPase,( IC50s of 490, 711 nM for bovine cardiac and human cardiac, respectively)</p>Formule :C15H19N3O2Degré de pureté :99.53% - 99.98%Couleur et forme :SolidMasse moléculaire :273.33Hydroxy-Dynasore
CAS :<p>Hydroxy-Dynasore (Dyngo-4a) , a effective dynamin inhibitor, inhibits withDynI (brain), DynI (rec), and DynII (rec) of IC50 of 0.38 μM, 1.1 μM, and 2.3 μM,</p>Formule :C18H14N2O5Degré de pureté :97.60% - >99.99%Couleur et forme :SolidMasse moléculaire :338.31PKCβ inhibitor 1
CAS :<p>PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,</p>Formule :C24H21N5O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :411.46ARQ 621
CAS :<p>ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. Phase 1.</p>Formule :C28H24Cl2FN5O2Degré de pureté :97.01% - 98.38%Couleur et forme :SolidMasse moléculaire :552.43HM03
CAS :<p>HM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity.</p>Formule :C26H27ClN4O2Degré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :462.97CZC-8004
CAS :<p>CZC-8004 (CZC-00008004) is a pan-kinase(ABL kinase) inhibitor and binds a range of tyrosine kinases.</p>Formule :C17H16FN5Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :309.34Taurolithocholic acid sodium salt
CAS :<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formule :C26H44NNaO5SDegré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :505.69Teduglutide acetate
<p>Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.</p>Formule :C166H256N44O56SDegré de pureté :97.39%Couleur et forme :SoildMasse moléculaire :3812.13BAY1125976
CAS :<p>BAY1125976 is an allosteric inhibitor of Akt1 and Akt2 (IC50s of 5.2 and 18 nM, respectively, in a time-resolved FRET assay)</p>Formule :C23H21N5ODegré de pureté :99.28% - ≥98%Couleur et forme :SolidMasse moléculaire :383.45Desmethylglycitein
CAS :<p>Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which has</p>Formule :C15H10O5Degré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :270.24Hexapeptide-10 Acetate
<p>Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) is a synthetic peptide.</p>Formule :C30H57N7O10Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :675.81KW-2478
CAS :<p>KW-2478 is a non-ansamycin HSP90 inhibitor with IC50 of 3.8 nM.</p>Formule :C30H42N2O9Degré de pureté :98.68% - 99.52%Couleur et forme :SolidMasse moléculaire :574.66LXW7
CAS :<p>LXW7 is an octamer disulfide cyclic peptide and αvβ3 integrin ligand, acts as a potent and specific endothelial progenitor cells (EPCs) and endothelial cells (</p>Formule :C29H48N12O12S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :820.89Multi-kinase inhibitor 1
CAS :<p>Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.</p>Formule :C20H17F3N4O3Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :418.37MMAF
CAS :<p>MMAF (MonoMethyl auristatin F), an antimitotic agent, inhibits cell division by blocking the polymerization of tubulin.</p>Formule :C39H65N5O8Degré de pureté :97.00% - 99.88%Couleur et forme :SolidMasse moléculaire :731.96Ispinesib
CAS :<p>Ispinesib (SB-715992), a selective, effectvie and reversible inhibitor of kinesin spindle protein (KSP), is derived from quinazolinone, with antineoplastic</p>Formule :C30H33ClN4O2Degré de pureté :98% - 99.09%Couleur et forme :SolidMasse moléculaire :517.06Gap 26
CAS :<p>Gap 26 is a mimetic peptide corresponding to the residues 63-75 of connexin 43, which is a gap junction blocker.</p>Formule :C70H107N19O19SDegré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :1550.78Dasatinib N-oxide
CAS :<p>Dasatinib N-oxide is a key metabolite and potential impurity of the kinase inhibitor dasatinib.</p>Formule :C22H26ClN7O3SDegré de pureté :98.54% - 99.94%Couleur et forme :SolidMasse moléculaire :504PF04929113
CAS :<p>PF04929113 (SNX-5422), a synthetic small molecule Hsp90 inhibitor, offers potent efficacy orally for various cancers.</p>Formule :C25H30F3N5O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :521.53XL888
CAS :<p>XL888 is an orally bioavailable Hsp90 inhibitor, blocking cell proliferation and inducing tumor regression with an IC50 of 24 nM.</p>Formule :C29H37N5O3Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :503.64H-Gly-Arg-Gly-Asp-Asn-Pro-OH
CAS :<p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>Formule :C23H38N10O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :614.61PKC ζ pseudosubstrate acetate
<p>PKC ζ pseudosubstrate acetate is an inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide.</p>Formule :C78H132N30O18Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :1778.10ILK-IN-2
CAS :<p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>Formule :C30H30F3N5ODegré de pureté :99.30%Couleur et forme :SolidMasse moléculaire :533.59Fingolimod hydrochloride
CAS :<p>Fingolimod hydrochloride (FTY720) , a novel immune modulator, is a sphingosine 1-phosphate (S1P) antagonist (IC50: 0.033 nM in K562 and NK cells).</p>Formule :C19H34ClNO2Degré de pureté :99.26% - 99.83%Couleur et forme :White SolidMasse moléculaire :343.93HA-100
CAS :<p>HA-100 is an inhibitor of protein kinase</p>Formule :C13H15N3O2SDegré de pureté :99.44%Couleur et forme :Pale Yellow Crystalline SolidMasse moléculaire :277.34TAT-Gap19 acetate
<p>TAT-Gap19 acetate, a Cx43 HC inhibitor, crosses blood-brain barrier, reduces liver fibrosis in mice, and spares Cx43 GJCs.</p>Formule :C119H212N46O26Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :2703.25Plinabulin
CAS :<p>Plinabulin (NPI-2358) (NPI-2358) is a vascular disrupting agent (VDA) against tubulin-depolymerizing tumor cells ( IC50: 9.8-18 nM).</p>Formule :C19H20N4O2Degré de pureté :98.69% - >99.99%Couleur et forme :SolidMasse moléculaire :336.39Hypocrellin A
CAS :<p>Hypocrellin A is a natural PKC inhibitor with light-induced antitumor, antifungal and antiviral activities.Cost-effective and quality-assured.</p>Formule :C30H26O10Degré de pureté :98% - 99.81%Couleur et forme :SolidMasse moléculaire :546.52Nilotinib monohydrochloride monohydrate
CAS :<p>Nilotinib monohydrochloride monohydrate (Nilotinib (monohydrochloride monohydrate)) is significantly potent BCR-ABL against, is a second generation tyrosine</p>Formule :C28H22F3N7O·HCl·H2ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :583.99Soblidotin
CAS :<p>Soblidotin (TZT-1027) (Auristatin PE) is an inhibitor of tubulin polymerization. It is also a novel synthetic Dolastatin 10 derivative.</p>Formule :C39H67N5O6Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :701.98Adaphostin
CAS :<p>Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.</p>Formule :C24H27NO4Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :393.48Protein Kinase C 19-31 acetate
<p>PKC 19-31 acetate, a serine-altered PKCa-derived PKC inhibitor, tests PKC activity.</p>Formule :C69H122N26O18Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1603.9Hypericin
CAS :<p>Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. Cost-effective and quality-assured.</p>Formule :C30H16O8Degré de pureté :99.05% - ≥98%Couleur et forme :Red-Coloured Anthraquinone-DerivativeMasse moléculaire :504.44Gly-Arg-Gly-Asp-Ser acetate(96426-21-0 free base)
<p>Gly-Arg-Gly-Asp-Ser (GRGDS) acetate is a cell binding protein domain derived from the cell-binding region of fibronectin.</p>Formule :C19H34N8O11Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :550.52Lifitegrast
CAS :<p>Lifitegrast (SAR 1118) is a lymphocyte, function-associated antigen-1 antagonist.</p>Formule :C29H24Cl2N2O7SDegré de pureté :99.39% - 99.66%Couleur et forme :SolidMasse moléculaire :615.48PF-562271
CAS :<p>PF-562271 is an effective ATP-competitive, reversible inhibitor of FAK(IC50=1.5 nM) and Pyk2 kinase(IC50=13 nM).</p>Formule :C21H20F3N7O3SDegré de pureté :97.17% - >99.99%Couleur et forme :SolidMasse moléculaire :507.49Bisindolylmaleimide V
CAS :<p>Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.</p>Formule :C21H15N3O2Degré de pureté :90%Couleur et forme :Red SolidMasse moléculaire :341.36Defactinib
CAS :<p>Defactinib (VS-6063) is a second-generation inhibitor of FAK. Defactinib has potential antitumor activity. Cost-effective and quality-assured.</p>Formule :C20H21F3N8O3SDegré de pureté :98% - 99.71%Couleur et forme :SolidMasse moléculaire :510.49PF-AKT400
CAS :<p>PF-AKT400 (AKT protein kinase inhibitor) is a broadly selective and ATP-competitive inhibitor of Akt.</p>Formule :C20H22F2N6ODegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :400.43Estramustine
CAS :<p>Estramustine (LEO-275), a nitrogen mustard-estradiol compound, treats prostate cancer and protects against radiation.</p>Formule :C23H31Cl2NO3Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :440.4ML346
CAS :<p>ML346 is a novel activator of Hsp70.</p>Formule :C14H12N2O4Degré de pureté :97.32% - 99.36%Couleur et forme :SolidMasse moléculaire :272.26PD173955
CAS :<p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>Formule :C21H16Cl2N4OSDegré de pureté :98.52% - 98.99%Couleur et forme :SolidMasse moléculaire :443.35ILK-IN-3
CAS :ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.Formule :C10H12N6ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :232.24Ansamitocin P 3'
CAS :<p>Ansamitocin P 3' (Maytansinol butyrate) is an antibody-drug conjugate cytotoxin with antitumor activity.</p>Formule :C32H43ClN2O9Degré de pureté :98.16% - 99.16%Couleur et forme :SolidMasse moléculaire :635.14AST 487
CAS :<p>AST 487 (NVP-AST 487) is a RET kinase inhibitor, inhibiting RET autophosphorylation and activation of downstream effectors. It also can inhibit Flt-3.</p>Formule :C26H30F3N7O2Degré de pureté :98.17% - 99.56%Couleur et forme :SolidMasse moléculaire :529.56Pamidronate disodium pentahydrate
CAS :<p>Pamidronate disodium pentahydrate strengthens bones and prevents osteoporosis.</p>Formule :C3H21NNa2O12P2Degré de pureté :99.84%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.13roxifiban
CAS :<p>Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.</p>Formule :C21H29N5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.48IM-12
CAS :<p>IM-12, an effective GSK-3β inhibitor(IC50=53 nM), regulates Wnt signalling.</p>Formule :C22H20FN3O2Degré de pureté :99.42% - >99.99%Couleur et forme :SolidMasse moléculaire :377.41Dynamin inhibitory peptide, myristoylated acetate
<p>Myristoylated acetate peptide inhibits DynaMin, blocking amphiphysin binding; myristoylated TFA variant hinders endocytosis.</p>Formule :C63H111N19O16Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :1390.67Olverembatinib
CAS :<p>Olverembatinib (GZD 824) is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM).</p>Formule :C29H27F3N6ODegré de pureté :98.53% - >99.99%Couleur et forme :SolidMasse moléculaire :532.56[Ala107]-MBP (104-118) acetate
<p>[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP).</p>Formule :C59H108N20O21Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :1553.72VER49009
CAS :<p>VER49009 (CCT0129397) is an effective HSP90 inhibitor(IC50 =25 nM, Kd=78 nM).</p>Formule :C19H18ClN3O4Degré de pureté :98.95% - >99.99%Couleur et forme :SolidMasse moléculaire :387.82Cyclo(RADfK)
CAS :<p>Cyclo(RADfK) is a selective α(v)β(3) integrin ligand used in neoangiogenesis research, therapy, and diagnostics; it's a control for RGD peptides.</p>Formule :C28H43N9O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :617.7Trimethyloctadecylammonium bromide
CAS :<p>Trimethyloctadecylammonium bromide is an inhibitor of Dynamin I(IC50 : 1.9 μM) and also inhibits Dynamin Ⅱ.</p>Formule :C21H46N·BrDegré de pureté :99.09%Couleur et forme :Solid SolidMasse moléculaire :392.5E7820
CAS :<p>E7820 (ER68203-00) is an angiogenesis inhibitor by suppressing integrin a2 (a cell adhesion molecule expressed on endothelial cells).</p>Formule :C17H12N4O2SDegré de pureté :98.31% - 99.11%Couleur et forme :SolidMasse moléculaire :336.37CK-636
CAS :<p>CK-636 (CK-0944636), an Arp2/3 complex inhibitor, can inhibit actin polymerization induced by the human, fission yeast and bovine Arp2/3 complex.</p>Formule :C16H16N2OSDegré de pureté :98.1% - 98.88%Couleur et forme :SolidMasse moléculaire :284.38N-Phenylbenzylamine
CAS :<p>A series of N-Phenylbenzylamine (Benzenemethanamine) as potential cytotoxic and antimitotic agents acting by inhibition of tubulin polymerization</p>Formule :C13H13NDegré de pureté :98.75%Couleur et forme :Colorless To Pale Yellow Crystalline PowderMasse moléculaire :183.25Y15
CAS :<p>Y15 (1,2,4,5-Benzenetetramine tetrahydrochlor) is a potent and specificsmall-molecule FAK scaffolding inhibitor that inhibits its autophosphorylation activity,</p>Formule :C6H14Cl4N4Degré de pureté :98% - 99.32%Couleur et forme :Dark Brown CrystalsMasse moléculaire :284.01Tianeptine sodium salt
CAS :<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Formule :C21H24ClN2NaO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :458.93Eptifibatide acetate (148031-34-9 free base)
CAS :<p>Eptifibatide acetate (148031-34-9), a cyclic heptapeptide GP IIb/IIIa inhibitor antiplatelet drug.</p>Formule :C35H49N11O9S2·xC2H4O2Degré de pureté :99.7% - 99.87%Couleur et forme :SolidMasse moléculaire :831.96 (free base)KNK437
CAS :<p>KNK437 (Heat Shock Protein Inhibitor I), a pan-HSP inhibitor, suppresses the synthesis of inducible HSPs(HSP105, HSP72, and HSP40).</p>Formule :C13H11NO4Degré de pureté :98.90%Couleur et forme :SolidMasse moléculaire :245.23TAS-301
CAS :<p>TAS-301, an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon injury to rat carotid arteries.</p>Formule :C23H19NO3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :357.4GNF-7
CAS :<p>GNF-7 is Bcr-Abl WT and Bcr-Abl T315I inhibitor with IC50 of 133 nM and 61 nM, respectively.</p>Formule :C28H24F3N7O2Degré de pureté :97.05% - 99.7%Couleur et forme :SolidMasse moléculaire :547.53Verbascoside
CAS :<p>Verbascoside (Kusaginin) is a protein kinase C inhibitor with antimicrobial, anti-inflammatory activities.</p>Formule :C29H36O15Degré de pureté :97.46% - 99.55%Couleur et forme :SolidMasse moléculaire :624.59
