Signalisation du cytosquelette
Les inhibiteurs de la signalisation du cytosquelette sont des composés qui perturbent les voies de signalisation régulant le cytosquelette, essentiel pour la forme, la motilité, la division des cellules et le transport intracellulaire. Ces inhibiteurs sont utilisés pour étudier la dynamique des protéines du cytosquelette, telles que l'actine et la tubuline, et leur rôle dans des processus comme la migration cellulaire, l'adhésion et la métastase du cancer. Les inhibiteurs de la signalisation du cytosquelette sont précieux dans la recherche en biologie cellulaire, en cancérologie et en neurobiologie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs de la signalisation du cytosquelette de haute qualité pour soutenir vos recherches dans ces domaines.
1382 produits trouvés pour "Signalisation du cytosquelette"
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Pre-084
CAS :<p>Pre-084 is a high affinity, selective σ1 agonist.</p>Formule :C19H28ClNO3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :353.88Shepherdin 79-87 acetate
<p>Shepherdin 79-87 acetate is a peptidomimetic antagonist of the complex between Hsp90 and survivin, another key regulator of tumor cell viability.</p>Formule :C43H68N12O14SDegré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1009.14AZ13705339 hemihydrate
<p>AZ13705339 hemihydrate: potent PAK1 inhibitor (IC50: 0.33 nM), also binds PAK1/2 (Kd: 0.28/0.32 nM), for cancer research.</p>Formule :C33H36FN7O3SH2OCouleur et forme :SolidMasse moléculaire :638.77Bexotegrast
CAS :<p>Bexotegrast (PLN-74809) is an αvβ6 and αvβ1 integrin inhibitor with antifibrotic properties for the study of idiopathic pulmonary fibrosis (IPF).</p>Formule :C27H36N6O3Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :492.61Alvespimycin
CAS :<p>Alvespimycin (17-DMAG) is a potent Hsp90 inhibitor with potential anticancer activity, which acts by binding to Hsp90.</p>Formule :C32H48N4O8Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :616.75FAK activator 1
CAS :<p>ZINC40099027 is a FAK activator that induces gastric mucosal repair in persistent aspirin-associated gastric injury.</p>Formule :C23H26F3N3O3Degré de pureté :99.19%Couleur et forme :SoildMasse moléculaire :449.47RO0270608
CAS :<p>RO0270608 is an α4β1/α4β7 integrin antagonist with anti-inflammatory activity for the study of allergic inflammatory responses.</p>Formule :C24H19Cl3N2O4Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :505.78Muromonab
CAS :<p>Muromonab (OKT3) is a mouse-derived antibody targeting the CD3 receptor, blocking all cytotoxic T cell functions.</p>Degré de pureté :95% - 97.51% (SEC-HPLC)Couleur et forme :LiquidNeurodazine
CAS :<p>Neurodazine is a neural inducer that promotes the differentiation of pluripotent cells into neuronal cells.</p>Formule :C27H21ClN2O3Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :456.92Bosutinib hydrate
CAS :<p>Bosutinib hydrate (SKI-606 hydrate) is a kinase inhibitor of BCR-ABL and Src tyrosine kinases for the study of leukemia.</p>Formule :C26H31Cl2N5O4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :548.46Etaracizumab
CAS :<p>Etaracizumab (LM 609) is a humanized monoclonal antibody targeting integrin αvβ3, inhibiting angiogenesis and melanoma growth, used in the study of melanoma.</p>Degré de pureté :96.77% (SEC-HPLC) - 99.32% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :144.3 (kDa)Vevorisertib trihydrochloride
CAS :<p>Vevorisertib trihydrochloride (ARQ 751 trihydrochloride) is ainhibitor of pan-AKT and AKT1-E17K mutations, inhibiting AKT1, AKT2 and AKT3.</p>Formule :C35H41Cl3N8ODegré de pureté :98.28%Couleur et forme :SolidMasse moléculaire :696.12Ruboxistaurin hydrochloride
CAS :<p>Ruboxistaurin HCl (LY 333531) selectively inhibits PKCβI/II with IC50 of 4.7/5.9 nM; much less effective on other PKC types and ATP-kinases.</p>Formule :C28H28N4O3·HClDegré de pureté :98.44% - 99.22%Couleur et forme :SolidMasse moléculaire :505.01H-Ile-Lys-Val-Ala-Val-OH
CAS :<p>H-Ile-Lys-Val-Ala-Val-OH can induce rapid differentiation of neural progenitor cells into neurons and neurite growth.</p>Formule :C25H48N6O6Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :528.69Arg-Gly-Asp-Ser
CAS :<p>Arg-Gly-Asp-Ser (RGDS peptide) is a conserved tetrapeptide sequence found in fibronectin, and the von Willebrand factor.</p>Formule :C15H27N7O8Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :433.42NQTrp
CAS :<p>NQTrp is an inhibitor of the aggregation of the tau protein with generic anti-amyloidogenic effects.</p>Formule :C21H16N2O4Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :360.36Mps1-IN-2
CAS :<p>Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor.</p>Formule :C26H36N6O3Degré de pureté :96.24% - 99.75%Couleur et forme :SolidMasse moléculaire :480.6WZU-13
CAS :<p>WZU-13 is an inhibitor of carboxylesterase (CES). At a concentration of 100 μM, WZU-13 suppresses 77% of CES activity.</p>Formule :C22H16N2OCouleur et forme :SolidMasse moléculaire :324.38Anti-Mouse CD3ε Antibody (145-2C11)
<p>Anti-Mouse CD3ε Antibody (145-2C11) is an antibody inhibitor targeting CD3ε in Armenian hamsters, in TCR formation and in T lymphocyte activation</p>Degré de pureté :99%Couleur et forme :Odour LiquidST-401
CAS :<p>ST-401, a microtubule-targeting agent (MTA), functions as a brain-penetrant microtubule (MT) assembly inhibitor. It disrupts microtubule (MT) function by gently and reversibly reducing MT assembly, which leads to mitotic delay and interphase cell death. ST-401 demonstrates potent antitumor activity.</p>Formule :C24H20N2OCouleur et forme :SolidMasse moléculaire :352.43Vepsitamab
CAS :<p>Vepsitamab (AMG 199), an anti-MUC17/CD3 BiTE, targets T cells and tumors for cell lysis and T cell activation.</p>Couleur et forme :LiquidPinatuzumab
CAS :<p>Pinatuzumab is a humanised monoclonal antibody targeting CD22, B-cell malignancies non-Hodgkin lymphoma (NHL) and chronic lymphocytic leukaemia (CLL).</p>Degré de pureté :95%Couleur et forme :LiquidPasotuxizumab
CAS :<p>Pasotuxizumab (BAY 2010112) is a BiTE that targets PSMA & CD3 with K D s 47.0 & 9.4 nM, for mCRPC research.</p>Couleur et forme :LiquidTepoditamab
CAS :<p>Tepoditamab (MCLA-117) is a bispecific antibody targeting CLEC12A and CD3, inducing T cell lysis of AML cells.</p>Couleur et forme :LiquidGresonitamab
CAS :<p>Gresonitamab (AMG 910) is an HLE BiTE antibody targeting CD3+ T cells and CLDN18.2+ tumors, for adenocarcinoma research.</p>Couleur et forme :LiquidObrindatamab
CAS :<p>Obrindatamab: a humanized bispecific antibody targeting B7-H3/CD3, enhances CTL-mediated cancer cell killing.</p>Couleur et forme :LiquidEnlimomab
CAS :<p>Enlimomab (BI-RR 0001), a mouse IgG2a antibody, blocks leukocyte binding to ICAM-1, reducing inflammation and used in stroke research.</p>Couleur et forme :LiquidNivatrotamab
<p>Nivatrotamab: Humanized anti-GD2/CD3 bispecific antibody for neuroblastoma research.</p>Couleur et forme :Odour LiquidSemorinemab
CAS :<p>Semorinemab (RG6100) is a humanised monoclonal antibody targeting the N-terminal domain of tau protein with a Kd of 3.8 nM, suitable for Alzheimer's disease.</p>Degré de pureté :95% - 95%Couleur et forme :Liquid4-Desacetylvinblastine hydrazide
CAS :<p>Deacetylvinblastine hydrazide, a cytotoxic vinca alkaloid often conjugated with folic acid to produce EC145, a novel folate-receptor targeted agent.</p>Formule :C43H56N6O7Couleur et forme :SolidMasse moléculaire :768.94Raludotatug
CAS :<p>Raludotatug is a humanized antibody targeting cadherin-6 (CDH6). As part of the ADC Raludotatug deruxtecan, it shows promise in researching platinum-sensitive ovarian cancer.</p>Degré de pureté :95% - 95%Couleur et forme :LiquidGosuranemab
CAS :<p>Gosuranemab (BMS-986168), a humanized IgG4 mAb, targets tau residues 15-22, and may aid in Alzheimer’s research.</p>Degré de pureté :95% - 95%Couleur et forme :LiquidMeclofenamate sodium hydrate
CAS :<p>Meclofenamate sodium: a strong NSAID inhibiting leukocyte function—chemotaxis, degranulation, and radical production.</p>Formule :C14H12Cl2NNaO3Couleur et forme :SolidMasse moléculaire :336.15Posdinemab
CAS :<p>Posdinemab, a humanized IgG1κ antibody, targets the microtubule-associated protein tau (MAPT) [1].</p>Couleur et forme :LiquidPlamotamab
CAS :<p>Plamotamab (XmAb-13676) is a bispecific antibody targeting CD3 and CD20, recruiting T cells to destroy CD20+ tumors and causing mild hematologic reactions.</p>Couleur et forme :LiquidAnti-Mouse IL-1a Antibody (ALF-161)
<p>Anti-Mouse IL-1a Antibody is an IgG1 subtype inhibitor specific to mouse IL-1a, derived from the Armenian Hamster.</p>Degré de pureté :98%Couleur et forme :Odour LiquidUbamatamab
CAS :<p>Ubamatamab (REGN4018), a human bispecific antibody targeting Mucin 16 (MUC16) and CD3, exhibits potent antitumor activity [1].</p>Couleur et forme :LiquidOsemitamab
CAS :<p>Osemitamab (TST001) is a humanised monoclonal antibody targeting claudin-18.2, gastric/gastric-oesophageal junction adenocarcinoma, PDAC, and lung cancer.</p>Degré de pureté :95%Couleur et forme :LiquidVoxalatamab
CAS :<p>Voxalatamab (JNJ-63898081), an IgG4 bispecific antibody targeting PSMA and CD3, demonstrates anti-cancer efficacy in prostate cancer research [1].</p>Couleur et forme :LiquidVonsetamig
CAS :<p>Vonsetamig, a humanized immunoglobulin G4-kappa monoclonal antibody, targets both TNFRSF17 and CD3E. It serves as an antineoplastic agent.</p>Couleur et forme :LiquidFlotetuzumab
CAS :<p>Flotetuzumab (MGD006/S80880) is a CD123/CD3 bispecific DART antibody, reactivating T-cells for AML treatment.</p>Couleur et forme :LiquidPacanalotamab
CAS :<p>Pacanalotamab (AMG 420/BI-836909), a BiTE, directs T-cells to BCMA+ MM cells, causing lysis.</p>Couleur et forme :LiquidVibecotamab
CAS :<p>Vibecotamab, a bispecific antibody, targets CD123/CD3 for T-cell killing of tumors, promising for acute myeloid leukemia.</p>Couleur et forme :LiquidOS-2966
<p>OS-2966 is a humanised de-immunised monoclonal antibody that target Integrin b1/ITGB1/CD29, malignant gliomas, glioblastomas, and astrocytomas.</p>Degré de pureté :95%Couleur et forme :Odour LiquidRovelizumab
CAS :<p>Rovelizumab: humanized anti-CD11/CD18 antibody for MS, hemorrhagic shock, MI, and stroke research.</p>Couleur et forme :LiquidLixudebart
CAS :<p>Lixudebart is a humanised monoclonal antibody targeting CLDN1 (Claudin-1), which can be used to reverse organ fibrosis and reduce initial ALT/AST levels.</p>Degré de pureté :95%Couleur et forme :LiquidVatelizumab
CAS :<p>Vatelizumab is a humanised monoclonal antibody targeting Integrin α2β1 ( VLA-2, CD49b), which enhances the frequency of regulatory T cells multiple sclerosis.</p>Degré de pureté :95%Couleur et forme :LiquidLinvoseltamab
CAS :<p>Linvoseltamab, a bispecific antibody, targets both BCMA (TNFRSF17) and CD3 epsilon, demonstrating a favorable safety profile and promising efficacy in relapsed/</p>Couleur et forme :LiquidCevostamab
CAS :<p>Cevostamab (BFCR4350A, RG6160, RO7187797) is a humanized BsAb IgG1 targeting FcRH5 on MM cells and CD3 on T cells to enhance T-cell-mediated MM cell killing.</p>Couleur et forme :LiquidOdronextamab
CAS :<p>Odronextamab, a fully human, hinge-stabilized IgG4-based bispecific antibody, targets CD3 receptors on T cells and CD20 receptors on B cells [1].</p>Couleur et forme :LiquidPavurutamab
CAS :<p>Pavurutamab (AMG-701) is a bispecific T cell engager targeting CD3 and BCMA with extended half-life, designed to treat MM.</p>Couleur et forme :Liquid17-AEP-GA
CAS :<p>17-AEP-GA is an HSP90 antagonist and a potent inhibitor of glioblastoma cell proliferation, survival, migration and invasion.</p>Formule :C34H50N4O8Degré de pureté :97.77% - 99.56%Couleur et forme :SolidMasse moléculaire :642.78Tubulin polymerization-IN-2
CAS :<p>Tubulin-IN-2, anticancer β-tubulin binder, IC50 0.92 μM, effective against various cancers.</p>Formule :C17H12F2N2O2Couleur et forme :SolidMasse moléculaire :314.29Meclofenamic acid
CAS :<p>Meclofenamic acid: non-selective gap-junction blocker, FTO inhibitor, anti-inflammatory.</p>Formule :C14H11Cl2NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.15SB273005
CAS :<p>SB273005 is a potent integrin inhibitor with Ki of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively.</p>Formule :C22H24F3N3O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :451.44N-Desmethylnefopam
CAS :<p>N-Desmethylnefopam is the main Nefopam metabolite .</p>Formule :C16H17NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.31Ionomycin calcium
CAS :<p>Ionomycin calcium (SQ23377 calcium) is an effective and selective calcium ionophore, exhibiting high specificity for calcium ions. Cost-effective and quality-assured.</p>Formule :C41H70CaO9Degré de pureté :98% - 98.11%Couleur et forme :SolidMasse moléculaire :747.07Phorbol 12,13-dibutyrate
CAS :<p>Phorbol 12,13-dibutyrate (Phorbol dibutyrate) is a PKC activator that induces contraction of isolated rabbit vascular smooth muscle.</p>Formule :C28H40O8Degré de pureté :99.32% - 99.37%Couleur et forme :SolidMasse moléculaire :504.61D-GsMTx4 TFA
<p>D-GsMTx4 TFA, a selective spider venom peptide, is a TRPC1/6 and Piezo2 inhibitor that inhibits cation-permeable mechanosensitive channels (MSCs) belonging to the Piezo and TRP channel families, blocks cation-selective stretch-activated channels (SACs), and attenuates lysophosphatidylcholine (LPC)-induced astrocyte toxicity and microglia reactivity. toxicity and microglia reactivity.D-GsMTx4 TFA prevented myocardial infarction in a mouse model of ischemia/reperfusion and can be used to characterize the role of excitatory MSCs in normal physiology and pathology.</p>Formule :C187H279F3N48O48S6Degré de pureté :99.29% - 99.65%Couleur et forme :SoildMasse moléculaire :4216.93IPA-3
CAS :<p>IPA-3 is a selective non-ATP competitive Pak1 inhibitor with IC50 of 2.5 μM, no inhibition to group II PAKs (PAKs 4-6).</p>Formule :C20H14O2S2Degré de pureté :97.40%Couleur et forme :SolidMasse moléculaire :350.45Tirofiban
CAS :<p>Tirofiban (L700462) (MK-383) is a selective palate GPIIb/IIIa antagonist which inhibits platelet aggregation with IC50 of 9 nM.</p>Formule :C22H36N2O5SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :440.6Auristatin F
CAS :<p>Auristatin F is an effective inhibitor of microtubule and vascular damaging agent. Auristatin F can be used in antibody-drug conjugates.</p>Formule :C40H67N5O8Degré de pureté :98.41% - 99.25%Couleur et forme :SolidMasse moléculaire :745.99Mps1-IN-1
CAS :<p>Mps1-IN-1 is a potent, selective and ATP-competitive inhibitor of Mps1 kinase (IC50 : 367 nM )</p>Formule :C28H33N5O4SDegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :535.66BAY1217389
CAS :<p>BAY 1217389 is an effective and selective inhibitor of the monopolar spindle 1 (MPS1) kinase (IC50<10 nM).</p>Formule :C27H24F5N5O3Degré de pureté :98.14% - 99.42%Couleur et forme :SolidMasse moléculaire :561.5AS1938909
CAS :<p>AS1938909: SHIP2 inhibitor boosts Akt phosphorylation, glucose use, and uptake via GLUT1 in L6 myotubes.</p>Formule :C19H13Cl2F2NO2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.28IQTub4P
CAS :<p>IQTub4P is a potent inhibitor of microtubules. IQTub4P exhibits cytotoxicity in HeLa cells (EC50: 170 nM).</p>Formule :C19H18NNa2O8PCouleur et forme :SolidMasse moléculaire :465.305HSP90-IN-14
CAS :<p>HSP90-IN-14 inhibits Hsp90 (Kd=0.26 μM) and fights influenza A/H3N2, A/H1N1, B with EC50 of 2.6, 3.9, 17 μM in MDCK cells.</p>Formule :C14H8Cl2N4O4SCouleur et forme :SolidMasse moléculaire :399.21Microtubule inhibitor 4
CAS :<p>Microtubule inhibitor 4 (Compound 2) blocks polymerization, toxic to HT-29 cells (IC50: 2.1 nM).</p>Formule :C25H23FN4O3Couleur et forme :SolidMasse moléculaire :446.47NC9 TG2 inhibitor
CAS :<p>NC9 is an irreversible inhibitor of transglutaminase 2 (TG2) and also inhibits Factor XIIIA (FXIIIA).</p>Formule :C35H47N5O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :697.84Antiproliferative agent-30
CAS :<p>Antiproliferative agent-30 (Compound 8g) demonstrates broad-spectrum antiproliferative activity, with IC50 values of 0.054 nM, 0.008 nM, and 0.144 nM against</p>Formule :C24H26N4O4Couleur et forme :SolidMasse moléculaire :434.49Tubulin polymerization-IN-42
CAS :<p>Tubulin polymerization-IN-42 (compound 10j), an indole-substituted furanone, inhibits tubulin polymerization and exhibits anti-cancer properties [1].</p>Formule :C22H21NO5Couleur et forme :SolidMasse moléculaire :379.41CCT251236
CAS :<p>CCT251236 is an orally available Pirin ligand obtained from a heat shock transcription factor 1 (hsf1) phenotypic screen.</p>Formule :C32H32N4O5Degré de pureté :98.82% - 99.89%Couleur et forme :SolidMasse moléculaire :552.62GR 144053 trihydrochloride
CAS :<p>platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonist</p>Formule :C18H30Cl3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.82Alyssin
CAS :<p>Alyssin: sulforaphane analog, antioxidant; boosts Nrf2 and phase II enzymes in cancer cells; lowers PAH metabolism, reducing cancer risk in vitro.</p>Formule :C7H13NOS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :191.31CH5164840
CAS :<p>CH5164840: strong HSP90 blocker; excels in NSCLC treatment; boosts erlotinib efficacy on EGFR-mutant tumors.</p>Formule :C19H23N5O2SCouleur et forme :SolidMasse moléculaire :385.48Tubulozole
CAS :<p>Tubulozole blocks mitosis by inhibiting microtubule dynamics, leading to cell cycle arrest and apoptosis.</p>Formule :C23H23Cl2N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.42SEW84
CAS :<p>SEW84, an Aha1-stimulated Hsp90 inhibitor, has an IC50 of 0.3 μM, aiding protein deposition disease research.</p>Formule :C19H14F4N4OSCouleur et forme :SolidMasse moléculaire :422.4Hsp90-Cdc37-IN-1
CAS :<p>Hsp90-Cdc37-IN-1 is an Hsp90-Cdc37 interaction disruptor (IC50: 140 nM) that inhibit cell migration and reverse drug resistance.</p>Formule :C43H57FN2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :748.99PP2A Cancerous-IN-1
CAS :<p>PP2A Cancerous-IN-1 is a potent inhibitor of CIP2A (Cancerous inhibitor of PP2A) and p-Akt that exhibits potent anti-proliferative effects.</p>Formule :C30H24N4O3Couleur et forme :SolidMasse moléculaire :488.54OXi8007
CAS :<p>OXi8007, a water-soluble prodrug for OXi8006, disrupts vasculature and exhibits strong cytotoxicity against DU-145 cancer cells.</p>Formule :C26H24NNa2O10PCouleur et forme :SolidMasse moléculaire :587.428Hsp90-IN-17
CAS :<p>Hsp90-IN-17 (Example 5) is an inhibitor of HSP90, applicable in researching proliferative diseases, including cancer and neurodegenerative conditions.</p>Formule :C21H20N4O7Couleur et forme :SolidMasse moléculaire :440.41Chrysotobibenzyl
CAS :<p>Chrysotobibenzyl from Dendrobium pulchellum stems may trigger cell death in detached cells and hinder lung cancer growth.</p>Formule :C19H24O5Couleur et forme :SolidMasse moléculaire :332.39Hydromethylthionine HBr
CAS :<p>Hydromethylthionine (LMTM/Leucomethylene Blue) inhibits tau in Alzheimer's/frontotemporal dementia and improves brain function.</p>Formule :C16H21Br2N3SCouleur et forme :SolidMasse moléculaire :447.233CHPG
CAS :<p>CHPG is a selective mGluR5 agonist protects against traumatic brain injury.activates the ERK and Akt pathways, It also alleviates LPS-induced inflammation.</p>Formule :C8H8ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :201.61Heat Shock Protein Inhibitor II
CAS :<p>Hsp inhibitor II, an active benzylidene lactam, blocks inducible Hsp synthesis, reduces tumor thermotolerance, and enhances AmB effects on A. fumigatus.</p>Formule :C12H11NO3Couleur et forme :SolidMasse moléculaire :217.22Tau-aggregation-IN-1
CAS :<p>Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).</p>Formule :C28H37N5O2SCouleur et forme :SolidMasse moléculaire :507.69AK963
CAS :<p>AK963 (40708899) is a powerful PAK1 inhibitor reducing gastric cancer cell growth via the PAK1-NFκB-CyclinB1 pathway.</p>Formule :C16H18N2OCouleur et forme :SolidMasse moléculaire :254.33(R)-TTBK1-IN-1
CAS :<p>(R)-TTBK1-IN-1: potent, selective brain-penetrant TTBK1 inhibitor, studies Alzheimer’s & tauopathies.</p>Formule :C18H19N5O2Couleur et forme :SolidMasse moléculaire :337.38BMS-688521
CAS :<p>BMS-688521 is an LFA-1/ICAM interaction inhibitor, a small molecule antagonist of LFA-1 with potential anti-inflammatory activity.</p>Formule :C26H19Cl2N5O4Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :536.37Syntelin
CAS :<p>Syntelin: a selective CENP-E inhibitor with an IC50 of 160 nM; distinct from GSK923295, effective on resistant mutants.</p>Formule :C21H20N6O2S3Couleur et forme :SolidMasse moléculaire :484.62LS-104
CAS :<p>LS-104 is a JAK2 inhibitor.</p>Formule :C19H16N2O3Couleur et forme :SolidMasse moléculaire :320.34Tubulin polymerization-IN-25
CAS :<p>Tubulin polymerization-IN-25 inhibits tubulin (IC50: 1.11 μM) & FTase (IC50: 0.39 μM), and is cytotoxic to cancer cells, halting growth.</p>Formule :C24H18N2O3SCouleur et forme :SolidMasse moléculaire :414.48AKT-IN-8
CAS :<p>AKT-IN-8 is a potent inhibitor of AKT, acting on AKT1 (IC50: 4.46 nM), AKT2 (IC50: 2.44 nM) and AKT3 (IC50: 9.47 nM).</p>Formule :C22H25ClN6O3Couleur et forme :SolidMasse moléculaire :456.93AKT-IN-5
CAS :<p>AKT-IN-5, an Akt inhibitor, targets Akt1/Akt2 with IC50s: 450/400 nM.</p>Formule :C23H20N4O2Couleur et forme :SolidMasse moléculaire :384.43Zalunfiban
CAS :<p>RUC-4 is an aIIb 3 antagonist. It is also used for prehospital therapy of myocardial infarction.</p>Formule :C16H18N8O2SCouleur et forme :SolidMasse moléculaire :386.43cemadotin free base
CAS :<p>Cemadotin free base(LU103793 free base) is a novel anti-limiting peptide , an analog of Dolastatin 15, a naturally occurring cytotoxic peptide that blocks</p>Formule :C35H56N6O5Degré de pureté :98.70% - 99.64%Couleur et forme :SolidMasse moléculaire :640.86Zarilamide
CAS :<p>Zarilamide disrupts microtubules, inhibiting mitosis in Phytophthora capsici zoospore cysts.</p>Formule :C11H11ClN2O2Couleur et forme :SolidMasse moléculaire :238.67Tubulin polymerization-IN-20
CAS :<p>Tubulin aggregation-IN-20, a potent inhibitor, may be studied for breast and drug-resistant colon cancers.</p>Formule :C25H24FNO5Couleur et forme :SolidMasse moléculaire :437.46Tubulin/MMP-IN-1
<p>Tubulin/MMP-IN-1 inhibits tubulin, MMP, and cancer cell growth; disrupts cell cycles and induces apoptosis.</p>Formule :C38H44NO9PCouleur et forme :SolidMasse moléculaire :689.73HSP90-IN-20
CAS :<p>HSP90-IN-20, a potent inhibitor of HSP90, exhibits an IC50 of ≤10 μM, indicating its potential application in cancer research.</p>Formule :C26H32N4O4Couleur et forme :SolidMasse moléculaire :464.56
