Alpha-bloquants
656 produits trouvés pour "Alpha-bloquants"
5'-Hydroxyphenyl Carvedilol-d5
CAS :Produit contrôléApplications A Labelled metabolite of Carvedilol which is a multiple-action, neurohormonal antagonist that is used in the treatment of hypertension.
References Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 958 (1998).Formule :C24H21D5N2O5Couleur et forme :NeatMasse moléculaire :427.56,7-Dimethoxy-N2,N2-dimethylquinazoline-2,4-diamine
CAS :Produit contrôléFormule :C12H16N4O2Couleur et forme :NeatMasse moléculaire :248.281Tamsulosin Catechol hydrochloride
CAS :Produit contrôléFormule :C18H24N2O5S·ClHCouleur et forme :NeatMasse moléculaire :416.922-(2-Ethoxyphenoxy)ethanamine
CAS :Produit contrôléImpurity Tamsulosin EP Impurity F
Applications 2-(2-Ethoxyphenoxy)ethanamine (Tamsulosin EP Impurity F) is an impurity of Tamsulosin (T006350), a specific α1-adrenoceptor antagonist (1,2). It is used in the treatment of benign prostatic hypertrophy.
References 1. Kawabe, K. et al.: J. Urol. 1990 Oct;144(4):908-11;2. Abrams, P. et al.: Br. J. Urol. 1995 Sep;76(3):325-36.Formule :C10H15NO2Couleur et forme :NeatMasse moléculaire :181.23[3-(9H-Carbazol-4-yloxy)-2-hydroxy]propyl Carvedilol
CAS :Produit contrôléFormule :C39H39N3O6Couleur et forme :NeatMasse moléculaire :645.74R-Mirtazapine
CAS :Produit contrôléApplications R-Mirtazapine is an enantiomer of Mirtazapine (M365000); an antidepressant. R-Mirtazapine showed antinociceptive effects in acute thermal nociception, whereas S-Mirtazapine showed pronociceptive effects.
References Muth-Selbach, Uta., et al.: Brain Res. Bull., 79(1), 63-68 (2009); Smith, Donald F., et al.: Psychopharmacology, 200(2), 273-279 (2008); Freynhagen, Rainer., et al.: Brain Res. Bull., 69(2), 168-173 (2006)Formule :C17H19N3Couleur et forme :NeatMasse moléculaire :265.355’-Hydroxyphenyl Carvedilol
CAS :Applications A metabolite of Carvedilol (C184625). It is used in the treatment of hypertension.
References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),Formule :C24H26N2O5Couleur et forme :NeatMasse moléculaire :422.472-(2-Ethoxyphenoxy)ethyl Bromide
CAS :Formule :C10H13BrO2Couleur et forme :NeatMasse moléculaire :245.11N-Nitroso Tetrahydrofuroylpiprazine
CAS :Produit contrôléFormule :C9H15N3O3Couleur et forme :NeatMasse moléculaire :213.234N-Isopropyl Carvedilol
CAS :Produit contrôléApplications Carvedilol (C184625) derivative.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the packageFormule :C27H32N2O4Couleur et forme :White To Off-WhiteMasse moléculaire :448.555-Acetonyl-2-methoxybenzenesulfonamide
CAS :Produit contrôléFormule :C10H13NO4SCouleur et forme :NeatMasse moléculaire :243.285-Formyl-2-methoxy-benzenesulfonamide
CAS :Produit contrôléImpurity Tamsulosin EP Impurity E
Applications 5-Formyl-2-methoxy-benzenesulfonamide (Tamsulosin EP Impurity E) is an impurity of Tamsulosin (T006350), a specific α1-adrenoceptor antagonist used in the treatment of benign prostatic hypertrophy.
References Kawabe, K., et al.: J. Urol., 144, 908 (1990), Abrams, P., et al.: Br. J. Urol., 76, 325 (1995), Michel, M.C., Expert Opin. Pharmacother., 5, 151 (2004),Formule :C8H9NO4SCouleur et forme :NeatMasse moléculaire :215.23N-Des(2-(2-ethoxy)phenoxy)ethyl), N-(2-(2-ethoxy)phenoxy)acetyl) Tamsulosin
CAS :Produit contrôléApplications Tamsulosin Ether is an impurity of is a Tamsulosin(CAS:106133-20-4) a specific α1-adrenoceptor antagonist. It is used in the treatment of benign prostatic hypertrophy.
References Kawabe, K., et al.: J. Urol., 144, 908 (1990), Abrams, P., et al.: Br. J. Urol., 76, 325 (1995), Michel, M.C., Expert Opin. Pharmacother., 5, 151 (2004),Formule :C20H26N2O6SCouleur et forme :Off-WhiteMasse moléculaire :422.5rac 4-(3-Aminobutyl)phenol
CAS :Produit contrôléApplications A metabolite of the antihypertensive agent, Labetalol (L096500).
References Gal, J., et al.: Res. Comm. Chem. Pathol. Pharmacol., 62, 3 (1988),Formule :C10H15NOCouleur et forme :NeatMasse moléculaire :165.232-(2-Ethoxyphenoxy)ethanamine Hydrochloride
CAS :Produit contrôléFormule :C10H15NO2·ClHCouleur et forme :NeatMasse moléculaire :217.69N2-Methyl alfuzosin-D7 hydrochloride
CAS :N2-Methyl alfuzosin-D7 is a drug product that belongs to the group of alfuzosin, which is a selective inhibitor of the enzyme phosphodiesterase type 5 (PDE5) and is used for the treatment of benign prostatic hyperplasia. It has been designed to reduce the risk of adverse effects associated with other PDE5 inhibitors, such as erectile dysfunction and urinary retention. N2-Methyl alfuzosin-D7 has been shown to be effective in animal studies and in vitro experiments. However, its metabolism remains unknown.Formule :C19H21D7ClN5O4Degré de pureté :Min. 95%Masse moléculaire :432.95 g/mol10-Oxo mirtazapine
CAS :10-Oxo mirtazapine is a metabolite of the antidepressant drug mirtazapine. It is an impurity in the HPLC standard for mirtazapine and has been shown to be pharmacologically active in animal models. 10-Oxo mirtazapine has also been found to be an impurity in other drugs, such as fluoxetine hydrochloride, but it is not known if it has any activity.Formule :C17H17N3ODegré de pureté :Min. 95%Masse moléculaire :279.34 g/mol[4-(4-Amino-6-hydroxy-7-methoxy-2-quinazolinyl)-1-piperazinyl](tetrahydro-2-furanyl)-methanone
CAS :4-(4-Amino-6-hydroxy-7-methoxy-2-quinazolinyl)-1-piperazinyl](tetrahydro-2-furanyl)-methanone (CAS No. 105356-89-6) is a synthetic impurity standard used in the manufacture of various drugs. Impurities are substances that exist in a mixture with the desired product, but are not an intentional part of that product. Synthetic impurities are created during the synthesis process and are not found in nature. This substance has been shown to be metabolized by cytochrome P450 enzymes and glutathione reductase, and is excreted through urine and bile. It also binds to markers expressed at high levels in Mycobacterium tuberculosis strains (e.g., ESX-1 secretion system protein) and inhibits cell growth in culture.Formule :C18H23N5O4Degré de pureté :Min. 95%Masse moléculaire :373.41 g/molN2-Methyl alfuzosin hydrochloride (1:x)
CAS :Alfuzosin is a drug used to treat the signs and symptoms of benign prostatic hyperplasia (BPH). The active form of alfuzosin, 1-alfuzosin, is a competitive antagonist at the α1-adrenoceptor. Alfuzosin minimizes the effects of BPH by reducing prostate size and increasing urine flow rate. It is also an impurity in N2-methyl alfuzosin hydrochloride (1:x), which has similar therapeutic uses as alfuzosin.Degré de pureté :Min. 95%
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