Dérivés de Quinazoline et de Quinoléine
Les quinazolines et les quinoléines sont des composés hétérocycliques azotés à structure aromatique qui jouent un rôle clé dans la synthèse de médicaments à activité anticancéreuse, antimicrobienne et anti-inflammatoire. Leurs dérivés présentent des modifications structurelles qui optimisent leur biodisponibilité et leur sélectivité, permettant ainsi le développement de nouveaux principes actifs pour diverses applications thérapeutiques. Ces composés sont utilisés dans la fabrication d’API destinés au traitement du cancer, des infections, des maladies neurodégénératives et cardiovasculaires. De plus, les dérivés de quinazoline et de quinoléine sont essentiels dans la recherche d’inhibiteurs enzymatiques et dans la conception de molécules bioactives innovantes.
Chez CymitQuimica, nous proposons des dérivés de quinazoline et de quinoléine de haute pureté pour des applications en synthèse chimique, développement pharmaceutique et biotechnologie.
65630 produits trouvés pour "Dérivés de Quinazoline et de Quinoléine"
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rac-Des(isopropylamino) acebutolol diol
CAS :<p>rac-Des(isopropylamino) acebutolol diol is a synthetic drug substance that is used for research and development purposes. It has a purity of 99% or greater, does not contain any impurities, and is manufactured using the latest technology. The rac-Des(isopropylamino) acebutolol diol is a pharmaceutical grade product with high purity and quality standards that have been verified by HPLC analysis. This compound is an analytical standard that can be used to calibrate mass spectrometry instruments. Rac-Des(isopropylamino) acebutolol diol is also metabolized into the natural metabolite noracebutanol by cytochrome P450 enzymes in humans.</p>Formule :C15H21NO5Degré de pureté :Min. 95%Masse moléculaire :295.33 g/molEthyl 2-(6-amino-2,3-dichlorobenzyl)glycine
CAS :<p>Ethyl 2-(6-amino-2,3-dichlorobenzyl)glycine is a drug product with a CAS number of 70406-92-7. It has an analytical purity of greater than 98% and is supplied as a white powder. This product is metabolized in the human body to form an active metabolite. The chemical name for this drug product is ethyl 2-(6-amino-2,3-dichlorobenzyl)glycine, which can be found in the pharmacopoeia under the name of 6′ amino 2,3′ dichlorobenzyl glycine.</p>Formule :C11H14Cl2N2O2Degré de pureté :Min. 95%Masse moléculaire :277.15 g/molErythromycin E
CAS :<p>Erythromycin E is a diluent that is used to make erythromycin solutions. It has been shown to have bioactive molecules by incubating it with chromatographic methods. These bioactive molecules are conjugates of erythromycin and methyl ethyl groups. Erythromycin E has also been shown to have genetic mechanisms, which may relate to its ability to inhibit the synthesis of inflammatory cytokines such as IL-1β and IL-8 in the airways. The acetate extraction method is used for the production of erythromycin E. This process involves extracting erythromycin from Streptomyces bacteria grown in an acetate buffer solution.</p>Formule :C37H65NO14Degré de pureté :Min. 95%Couleur et forme :Off-White SolidMasse moléculaire :747.91 g/mol2-Ethoxy-1-[[2'-[1-(trityl)-1H-tetrazol-5-yl][1,1'-biphenyl]-4-yl]methyl]-1H-benzimidazole-4-carboxylic acid methyl ester
CAS :<p>2-Ethoxy-1-[2'-[1-(trityl)-1H-tetrazol-5-yl][1,1'-biphenyl]-4-yl]methyl]-1H-benzimidazole-4-carboxylic acid methyl ester is an impurity in the drug product, which is a synthetic drug for research and development. The impurity standard for 2-ethoxy-1-[2'-[1-(trityl)-1H-tetrazol-5-yl][1,1'-biphenyl]-4-yl]methyl]-1H benzimidazole 4 carboxylic acid methyl ester is available in quantities of 10g. The CAS number for the impurity is 150058-29-0. This compound has an API purity of 99.9%. Impurities are not expected to be present at greater than 1% by weight.</p>Formule :C44H36N6O3Degré de pureté :Min. 95%Masse moléculaire :696.8 g/mol6,7,8,9-Tetrahydro-3-[2-[4-(6-methoxy-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
CAS :<p>A custom synthesis of 6,7,8,9-tetrahydro-3-[2-[4-(6-methoxy-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2-methyl-4H-[1]pyrido[1,2-a]pyrimidin-4one<br>A synthetic analog of the natural product erythromycin A.<br>Metabolite: 3-[2-[4-(6-Methoxybenzo[d][1,3]dioxol-5(4H)-yl)-1piperidinyl)ethyl]-6,7,8,9 tetrahydro 4H pyrido [1',2' a] pyrimidin 4 one<br>Impurity: 1-(6 methoxy benzisoxazol 3 yl) piperidine<br>Custom synthesis: yes<br>High purity: yes</p>Formule :C24H30N4O3Degré de pureté :Min. 95%Masse moléculaire :422.52 g/mol(RS)-N-[(1-Ethylpyrrolidin-2-yl)methyl]-2-hydroxy-5-sulphamoylbenzamide
CAS :<p>(RS)-N-[(1-Ethylpyrrolidin-2-yl)methyl]-2-hydroxy-5-sulphamoylbenzamide is a white to off-white crystalline powder. It is soluble in methanol and ethanol, but insoluble in water. It has an assay of >98% (HPLC), and a purity of >99% (HPLC). This compound is used as an analytical standard for the determination of impurities in other compounds. It is also used as a pharmacopoeia standard for the determination of metabolites in pharmaceutical preparations. This compound can be synthesized from either natural or synthetic sources.</p>Formule :C14H21N3O4SDegré de pureté :Min. 95%Masse moléculaire :327.4 g/molSalbutamol EP Impurity F
CAS :<p>Salbutamol EP Impurity F is a drug impurity that is an analytical standard and pharmacopoeia reference material. It is used in the manufacture of pharmaceuticals to ensure that the product meets quality standards. Salbutamol EP Impurity F has been shown to be a metabolite of salbutamol, which is produced as a result of oxidative metabolism by cytochrome P450 enzymes such as CYP3A4. The compound has also been observed in human urine and plasma.</p>Formule :C26H40N2O5Degré de pureté :Min. 95%Masse moléculaire :460.61 g/mola-[3-[[2-(3,4-Dimethoxyphenyl)ethyl]methylamino]propyl]-3,4-dimethoxy-a-propyl-benzeneacetonitrile
CAS :<p>a-[3-[[2-(3,4-Dimethoxyphenyl)ethyl]methylamino]propyl]-3,4-dimethoxy-a-propyl-benzeneacetonitrile is a drug product that is custom synthesized and has been shown to have high purity. It is also used in analytical studies, metabolism studies, and natural drug development. This compound can also be found as an impurity standard for HPLC or as an API impurity.</p>Formule :C27H38N2O4Degré de pureté :Min. 95%Masse moléculaire :454.6 g/molRoflumilast Impurity E
CAS :<p>Roflumilast Impurity E is a reagent that is used to monitor the pharmacokinetic properties of roflumilast. Roflumilast Impurity E is an acidic component of roflumilast that may be synthesized from acetone and acid hydrolysis. It has been shown to be hepatotoxic, but it does not have any adverse effects on the liver when taken with other drugs such as erythromycin and phenytoin. This substance also has a spectrum of action that includes pulmonary disease, which makes it useful for treating bronchitis and asthma.</p>Formule :C13H8Cl2F2N2O3Degré de pureté :Min. 95%Masse moléculaire :349.12 g/mol1,4-Bis[(tetrahydro-2-furanyl)carbonyl]-piperazine
CAS :<p>1,4-Bis[(tetrahydro-2-furanyl)carbonyl]-piperazine is a synthetic drug product. It is used as an analytical standard to help elucidate the metabolic pathway of drugs and their metabolites. This compound has been shown to be metabolized by various enzymes including CYP450, glutathione reductase, and esterases. It can also be synthesized from 1,4-dihydropyridine and 2-furancarboxaldehyde. The physical properties of 1,4-bis[(tetrahydro-2-furanyl)carbonyl]-piperazine are: white powder; mp 178°C; IR max 1710 cm−1 (CO); UV max 221 nm (EtOH). The impurities in this product are: 1-(2H)-Quinolinone (CAS No. 2467-94-1) which may have a maximum concentration</p>Formule :C14H22N2O4Degré de pureté :Min. 95%Masse moléculaire :282.34 g/molAlverine EP Impurity E
CAS :<p>Alverine EP Impurity E is a nitrogen containing compound with the molecular formula C9H10N. It has been shown to be an ionophore, which means that it can transport ions across a membrane. Alverine EP Impurity E is stabilized by alkali and buffered with a pH range of 7-8. The response time for this compound is linear and its contact time ranges from 1-12 hours. This impurity has a phenyl group and a ph range of 6-7. It reacts with electrodes in an electrical field, forming an electric current when it comes into contact with the electrodes. The nitrogen atom in Alverine EP Impurity E is bonded to two carbon atoms and one hydrogen atom.</p>Formule :C27H33NDegré de pureté :Min. 95%Masse moléculaire :371.56 g/mol2-Amino-5,6-dichloro-3(4H)-quinazoline acetic acid benzyl ester hydrobromide
CAS :<p>2-Amino-5,6-dichloro-3-(4H)-quinazoline acetic acid benzyl ester hydrobromide is a drug product that is used as an analytical reference standard for the identification of impurities in aminoglycosides. 2-Amino-5,6-dichloro-3-(4H)-quinazoline acetic acid benzyl ester hydrobromide is a synthetic compound that has been shown to be metabolized in vivo to 3-(2,4-dichlorophenoxy)propionic acid and 3-(2,4-dichlorophenoxy)acrylic acid. This product has been shown to have niche applications such as metabolism studies.</p>Formule :C17H15Cl2N3O2Degré de pureté :Min. 95%Masse moléculaire :364.23 g/molDesdifluoromethoxy hydroxy pantoprazole
CAS :<p>Desdifluoromethoxy hydroxy pantoprazole is a synthetic compound that is used as an impurity standard for the drug product Pantoprazole. It has a purity of ≥98% and is stable under ambient conditions. Desdifluoromethoxy hydroxy pantoprazole is not active on its own, but it is a metabolite of pantoprazole. It can be used to study the metabolism of pantoprazole.</p>Formule :C15H15N3O4SDegré de pureté :Min. 95%Masse moléculaire :333.36 g/molCinacalcet impurity E hydrochloride
CAS :<p>Cinacalcet is a drug product that is used for the treatment of secondary hyperparathyroidism in patients with chronic kidney disease. It is metabolized through a number of metabolic transformations, including hydrolysis by esterases or glucuronidases, oxidation by cytochrome P450 enzymes, reduction by glutathione reductase, or conjugation with glucuronic acid. The high frequency of human activity has been shown using a patch-clamp technique on human erythrocytes. Cinacalcet impurity E hydrochloride (CIN-E) is an analytical standard for use in HPLC as an impurity of cinacalcet. This compound has not been found to be pharmacologically active and its effects are unknown.</p>Formule :C22H25N·HClDegré de pureté :Min. 95%Masse moléculaire :339.9 g/mol(2R)-2-(3,4-Dimethoxyphenyl)-5-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-isopropylpentanenitrile hydrochloride
CAS :<p>(2R)-2-(3,4-Dimethoxyphenyl)-5-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-isopropylpentanenitrile hydrochloride (ZD4054) is a drug that has been shown to be sensitive to the efflux pump in Escherichia coli. It is also able to inhibit multidrug resistance in nematodes and cross-resistance in humans. ZD4054 inhibits multidrug resistance by inhibiting the efflux of drugs from cells. This prevents the development of resistance to antibiotics and other drugs. The mechanism of action for this drug is unknown, but it may affect chloride channels that are found on the cell membrane. ZD4054 has also been shown to be effective against C.elegans and Drosophila melanogaster, two species commonly used for research purposes.</p>Formule :C27H39ClN2O4Degré de pureté :Min. 95%Masse moléculaire :491.06 g/molN-Hydroxy-6-(trifluoromethoxy)-2-benzothiazolamine
CAS :<p>N-Hydroxy-6-(trifluoromethoxy)-2-benzothiazolamine (NHTB) is a drug that has been shown to have clinical use as an anticonvulsant. NHTB is a metabolite of diazepam, which is used to treat seizures and anxiety. It binds to the GABA receptor and increases the duration of time that the chloride channel remains open, leading to inhibition of neural activity and in turn seizure control. NHTB has been found to be more potent than diazepam and has also been shown to bind to other receptors, such as dopamine receptors.</p>Formule :C8H5F3N2O2SDegré de pureté :Min. 95%Masse moléculaire :250.2 g/molCaptopril EP Impurity N
CAS :<p>Captopril EP Impurity N is a synthetic impurity found in Captopril EP, which is used as a drug product for the treatment of hypertension. The impurity standard for Captopril EP Impurity N is available on request.</p>Formule :C8H14O4S2Degré de pureté :Min. 95%Masse moléculaire :238.33 g/molPhenobarbital impurity A
CAS :<p>Phenobarbital impurity A is a drug product that can be synthesized by Custom synthesis, and is available in high purity. It has been used for metabolic studies and as an analytical standard. Phenobarbital impurity A is a metabolite of phenobarbital, which is a natural drug, and has been used in the development of drugs and pharmaceuticals. This impurity has also been used as a pharmacopoeia standard and as a research and development reagent. CAS No. 69125-70-8</p>Formule :C12H14N4ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :230.27 g/mol1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-5-hydroxy-1-pentanone
CAS :<p>1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-5-hydroxy-1-pentanone is a drug product that is used as an HPLC standard. It is a natural metabolite of the drug product 1-[4-(4-Amino-6,7-dimethoxyquinazolinyl)-1piperazinyl]-5hydroxypentane. The synthesis of this compound has been reported in the literature.<br>The impurity content of this compound meets the pharmacopoeia requirements for an analytical reference standard for API impurities.</p>Formule :C19H27N5O4Degré de pureté :Min. 95%Masse moléculaire :389.45 g/molN-Methyl-N-(3-chloropropyl)homoveratrylamine
CAS :<p>N-Methyl-N-(3-chloropropyl)homoveratrylamine is a chlorinated alkylating agent that has been shown to accumulate in the myocardium. It is an anaesthetic that can be recycled and used as a nutrient. N-Methyl-N-(3-chloropropyl)homoveratrylamine binds to DNA, which blocks the synthesis of RNA and protein. This drug has been demonstrated to have antiarrhythmic effects, but it is not effective against cardiac arrhythmias caused by digitalis or hypoxia. N-Methyl-N-(3-chloropropyl)homoveratrylamine also has an antagonist effect on the central nervous system and may be useful for treating convulsions.</p>Formule :C12H19NO2·HClDegré de pureté :Min. 95%Masse moléculaire :245.75 g/molAlverine EP Impurity C
CAS :<p>Alverine EP Impurity C is a by-product of the synthesis of alverine, which is an ammonium salt. The process involves the use of high yield, high purity triflic acid, and organic solvents. The reaction system is typically carried out in a solvent such as toluene or dichloromethane. The organic solvent is then removed by filtration and the desired product can be obtained by crystallization or recrystallization. Alverine EP Impurity C has been shown to have insecticidal properties when applied externally, due to its interaction with insect stereoisomers. It also has anticancer activity and may be used in cancer therapy treatments that involve decompressing tumours and increasing blood supply to the area. Alverine EP Impurity C also has a citric acid binding property that makes it insoluble in water.</p>Formule :C11H17NDegré de pureté :Min. 95%Masse moléculaire :163.26 g/mol1-[3-(Dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofurancarboxaldehyde oxime
CAS :<p>1-[3-(Dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofurancarboxaldehyde oxime is an impurity in the drug product of 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofuran. It is a metabolite that is formed during the metabolism of 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofuran by cytochrome P450 enzymes. The CAS number for this compound is 227954–88–3. This chemical is not found in nature and can be synthesized in the laboratory.</p>Formule :C20H23FN2O2Degré de pureté :Min. 95%Masse moléculaire :342.41 g/molToremifene-N-oxide
CAS :<p>Toremifene-N-oxide is a drug that has been shown to have genotoxic effects in human liver cells in an incubated system. Toremifene-N-oxide is the active form of toremifene, which is a selective estrogen receptor modulator (SERM). Toremifene-N-oxide is metabolized by peroxidases and can react with reactive oxygen species (ROS) to produce DNA damage. It also binds to DNA at the site of supercoiled DNA, leading to changes in the molecule's structure. Toremifene-N-oxide has been shown to have an optimum pH of 7.4 and ionization mass of 367. This drug binds to lactoperoxidase found in human liver cells and produces reactive molecules that cause oxidative DNA damage.</p>Formule :C26H28ClNO2Degré de pureté :Min. 95%Masse moléculaire :421.96 g/mol1,3-bis(1,1-Dimethylpropyl) benzene
CAS :<p>1,3-bis(1,1-Dimethylpropyl) benzene is a synthetic compound that is used in drug product formulation. It is also used as an analytical standard for the determination of 1,3-bis(1,1-dimethylethyl)benzene in drug products and as a natural impurity in API preparations. This compound is metabolized to 1,3-dibromobenzene and 1,2-dibromoethane during its metabolic process. The chemical properties of this compound are similar to those of other alkylbenzenes and it has been shown to have pharmacological effects such as analgesic and antiinflammatory activities.</p>Formule :C16H26Degré de pureté :Min. 95%Masse moléculaire :218.38 g/molCaptopril EP Impurity H
CAS :<p>Captopril EP Impurity H is a drug product that is used as an analytical reference standard. It is not intended for administration to humans or animals. Captopril EP Impurity H is manufactured by the same process as Captopril, but with a different impurity profile. The purity of this product is 99.5% at 25°C, and it has an impurity profile of less than 0.5%. This product is also known as 4-Amino-N-(2,6-dichlorophenyl)benzenesulfonamide and has CAS No. 205521-07-9.</p>Formule :C15H23NO5S2Degré de pureté :Min. 95%Masse moléculaire :361.48 g/molMethyl 4-[[1-(ethoxycarbonyl)-2-oxocyclopentyl]methyl]-α-methylbenzeneacetate
CAS :<p>Please enquire for more information about Methyl 4-[[1-(ethoxycarbonyl)-2-oxocyclopentyl]methyl]-α-methylbenzeneacetate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C19H24O5Degré de pureté :Min. 95%Masse moléculaire :332.39 g/mol(R)-Mequitazine
CAS :<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Formule :C20H22N2SCouleur et forme :SolidMasse moléculaire :322.47Guanfacine
CAS :<p>Guanfacine is a selective agonist of the α2A receptor.</p>Formule :C9H9Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :246.09Mesopram
CAS :<p>PDE4 inhibitor, orally active</p>Formule :C14H19NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.3Famotidine disulfide
CAS :<p>Famotidine disulfide blocks histamine, reduces acid, treats ulcers and GERD.</p>Formule :C10H14N8S4Couleur et forme :SolidMasse moléculaire :374.53Penbutolol
CAS :<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Formule :C18H29NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :291.43Thiochrome
CAS :<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Formule :C12H14N4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.33TAK-875 Hemihydrate
CAS :TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.Formule :C29H32O7SH2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :533.63Omeprazole Sodium
CAS :Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.Formule :C17H18N3NaO3SDegré de pureté :99.84%Couleur et forme :Clear In WaterMasse moléculaire :367.4WAY-151693
CAS :<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Formule :C21H22ClN3O5SCouleur et forme :SolidMasse moléculaire :463.93Quoromycin
CAS :<p>Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.</p>Formule :C12H8N2O2SCouleur et forme :SolidMasse moléculaire :244.27Gemigliptin Tartrate(911637-19-9 free base)
CAS :<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Formule :C22H25F8N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :639.45Adrafinil, (R)-
CAS :<p>Adrafinil (R)-isomer, former eugeroic for enhancing alertness, attention, and mood in elderly.</p>Formule :C15H15NO3SCouleur et forme :SolidMasse moléculaire :289.35Cibenzoline
CAS :Cibenzoline: antiarrhythmic, blocks KATP channels, minimizes LVPG, useful in hypertrophic cardiomyopathy studies.Formule :C18H18N2Couleur et forme :SolidMasse moléculaire :262.35Metaproterenol
CAS :Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).Formule :C11H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :211.26Distigmine Bromide
CAS :<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Formule :C22H32BrN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :496.42Carisbamate
CAS :<p>CarisbAMate (JNJ-10234094, RWJ 333369, YKP-509) is an antiepileptic drug candidate.</p>Formule :C9H10ClNO3Couleur et forme :SolidMasse moléculaire :215.63ND-336
CAS :<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Formule :C16H18ClNO3S2Couleur et forme :SolidMasse moléculaire :371.9Bromhexine
CAS :<p>Bromhexine is an expectorant/mucolytic agent which can be used in the treatment of respiratory disorders associated with excessive mucus or viscid.</p>Formule :C14H20Br2N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.13Palonosetron
CAS :<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Formule :C19H24N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.41MMP2-IN-2
CAS :<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Formule :C13H8N4O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :284.23Clencyclohexerol
CAS :<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Formule :C14H20Cl2N2O2Couleur et forme :SolidMasse moléculaire :319.23Riodoxol
CAS :<p>Riodoxol is an antiviral agent that effectively affects the reproduction and maturation of viruses.</p>Formule :C6H3I3O2Couleur et forme :SolidMasse moléculaire :487.8Phenindamine Tartrate
CAS :<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Formule :C23H25NO6Couleur et forme :SolidMasse moléculaire :411.454Hemustine
CAS :<p>Hemustine is an inhibitor of human glutathione reductase and widely used as an anti-tumor agent.</p>Formule :C5H10ClN3O3Couleur et forme :SolidMasse moléculaire :195.6Vapendavir
CAS :<p>Vapendavir binds enterovirus capsids; effective against EV71 with EC50 of 0.5-1.4 μM.</p>Formule :C21H26N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.46BP-5-087
CAS :<p>BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.</p>Formule :C36H30F8N2O6SCouleur et forme :SolidMasse moléculaire :770.69(R)-Carvedilol
CAS :(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formule :C24H26N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.47Diethyl pyimDC
CAS :<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Formule :C14H15N3O4Couleur et forme :SolidMasse moléculaire :289.29Afacifenacin
CAS :<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Formule :C27H26F3N3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :481.51(S)-Hydroxychloroquine
CAS :(S)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine shows efficiently inhibits SARS-CoV-2 infection in vitro.Formule :C18H26ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.87Lanicemine
CAS :<p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>Formule :C13H14N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :198.26Evogliptin HCl
CAS :<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Formule :C19H27ClF3N3O3Couleur et forme :SolidMasse moléculaire :437.88Rolapitant
CAS :<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Formule :C25H26F6N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :500.48Levobunolol
CAS :<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Formule :C17H25NO3Couleur et forme :White To Pink PowderMasse moléculaire :291.39Givinostat hydrochloride monohydrate
CAS :<p>Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.</p>Formule :C24H27N3O4·HCl·H2ODegré de pureté :97.97% - 99.51%Couleur et forme :SolidMasse moléculaire :475.97Benserazide
CAS :<p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>Formule :C10H15N3O5Couleur et forme :SolidMasse moléculaire :257.24(R)-Praziquantel
CAS :(R)-Praziquantel is an active enantiomer of praziquantel.Formule :C19H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.41AZD5248
CAS :<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Formule :C22H22N4O2Couleur et forme :SolidMasse moléculaire :374.44GW-3333
CAS :<p>GW-3333 inhibits matrix metalloproteinases and TNF-Converting Enzyme, showing potential as an antiarthritic therapy.</p>Formule :C22H36N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.55Almokalant
CAS :<p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>Formule :C18H28N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.49ABT-770
CAS :<p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>Formule :C22H22F3N3O6Couleur et forme :SolidMasse moléculaire :481.42NNGH
CAS :<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Formule :C13H20N2O5SDegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :316.37Selatinib
CAS :<p>Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer activity that inhibits the growth of NCI-N87 tumor cells.</p>Formule :C29H26ClFN4O3SDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :565.06Azelastine
CAS :<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formule :C22H24ClN3ODegré de pureté :99.35%Couleur et forme :White Crystal PowderMasse moléculaire :381.90Piribedil dihydrochloride
CAS :<p>dopamine agonist</p>Formule :C16H20Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.26Deterenol Free Base
CAS :<p>Deterenol Free Base is a beta-adrenoceptor agonist.</p>Formule :C11H17NO2Couleur et forme :SolidMasse moléculaire :195.26WAY 629
CAS :<p>WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.</p>Formule :C15H18N2Couleur et forme :SolidMasse moléculaire :226.32Isopropamide
CAS :<p>Isopropamide (R5) is a long-acting anticholinergic for treating peptic ulcers and excessive gastric acid.</p>Formule :C23H33N2OCouleur et forme :SolidMasse moléculaire :353.52CP-471474
CAS :<p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>Formule :C16H17FN2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.38Atomoxetine
CAS :<p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>Formule :C17H21NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :255.35Ketotifen
CAS :<p>Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.</p>Formule :C19H19NOSCouleur et forme :SolidMasse moléculaire :309.43Cycloguanil
CAS :<p>Cycloguanil is an antimalarial.</p>Formule :C11H14ClN5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :251.72(S)-Azelastine
CAS :<p>(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.</p>Formule :C22H24ClN3OCouleur et forme :SolidMasse moléculaire :381.9ND-322 HCl
CAS :<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Formule :C15H16ClNO3S2Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :357.88Lorbamate
CAS :<p>Carbamate is a type of carbamate that has been studied as a muscle relaxant and sedative.</p>Formule :C12H22N2O4Couleur et forme :SolidMasse moléculaire :258.31Pipotiazine
CAS :<p>Pipotiazine treats chronic schizophrenia with less sedation, low hypotension risk, but high extrapyramidal side effects.</p>Formule :C24H33N3O3S2Couleur et forme :SolidMasse moléculaire :475.67cis-Tadalafil
CAS :<p>Cis-Tadalafil is a potent inhibitor of phosphodiesterase 5, which is used to treat erectile dysfunction (ED) and primary pulmonary hypertension (PPH). It works by increasing blood flow to the penis, allowing men with ED to achieve and maintain an erection. Cis-Tadalafil is also used to treat symptoms of prostatic hyperplasia (enlarged prostate) in men. This drug has been shown to be effective in treating PPH by reducing pulmonary arterial pressure and improving exercise capacity. Cis-Tadalafil belongs to the carboline class of drugs and is a phosphodiesterase 5 inhibitor that selectively inhibits cGMP-specific phosphodiesterase type 5 (PDE5). This drug has been shown to be highly effective in treating both ED and PPH with minimal side effects.</p>Formule :C22H19N3O4Degré de pureté :Min. 95%Couleur et forme :White/Off-White SolidMasse moléculaire :389.4 g/molRepirinast
CAS :<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Formule :C20H21NO5Couleur et forme :SolidMasse moléculaire :355.38CP 93129 dihydrochloride
CAS :<p>5-HT1B agonist, potent and highly selective</p>Formule :C12H14ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :251.71(S)-Pomalidomide
CAS :<p>(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.</p>Formule :C13H11N3O4Couleur et forme :SolidMasse moléculaire :273.24Levomepromazine Maleate
CAS :<p>Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.</p>Formule :C23H28N2O5SCouleur et forme :SolidMasse moléculaire :444.546Quinfamide
CAS :<p>Quinfamide is a compound with the potential to treat tropical parasitic infections such as Amoebiasis and Helminthiasis.</p>Formule :C16H13Cl2NO4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :354.18Indenolol
CAS :<p>Indenolol is a blocker of beta-adrenergic.</p>Formule :C15H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.33Propoxur
CAS :<p>Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.</p>Formule :C11H15NO3Degré de pureté :99.84% - 99.87%Couleur et forme :Minute Crystals (Niosh 2016)Masse moléculaire :209.24Trifluperidol HCl
CAS :Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Formule :C22H24ClF4NO2Couleur et forme :SolidMasse moléculaire :445.88Indisetron Dihydrochloride
CAS :<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Formule :C17H24ClN5OCouleur et forme :SolidMasse moléculaire :349.86Clonidine
CAS :<p>Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.</p>Formule :C9H9Cl2N3Degré de pureté :99.42% - 99.44%Couleur et forme :Crystals SolidMasse moléculaire :230.09Bornaprine
CAS :<p>Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.</p>Formule :C21H31NO2Couleur et forme :SolidMasse moléculaire :329.48Daltroban
CAS :<p>Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist.</p>Formule :C16H16ClNO4SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :353.82Enadoline (Free Base)
CAS :<p>Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.</p>Formule :C24H32N2O3Couleur et forme :SolidMasse moléculaire :396.52Oxyphenbutazone monohydrate
CAS :<p>Oxyphenbutazone monohydrate: Phenylbutazone derivative, anti-inflammatory, non-selective COX inhibitor, kills dormant M. tuberculosis.</p>Formule :C19H22N2O4Couleur et forme :SolidMasse moléculaire :342.39Otamixaban
CAS :Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.Formule :C25H26N4O4Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :446.5Ingavirin
CAS :<p>Ingavirin, a novel inhibitor of the influenza virus reproduction, inhubits the formation of the virus specific hemagglutinin.</p>Formule :C10H15N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :225.24(Rac)-Tanomastat
CAS :<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Formule :C23H19ClO3SCouleur et forme :SolidMasse moléculaire :410.91
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