Dérivés des Benzodiazépines
Les benzodiazépines sont des composés organiques dotés d’un noyau bicyclique fusionné de benzodiazépine, largement utilisées dans le développement de médicaments aux propriétés anxiolytiques, sédatives, anticonvulsivantes et myorelaxantes. Leurs dérivés incluent des structures modifiées qui améliorent leur sélectivité et leur profil pharmacocinétique, permettant la création de nouvelles molécules aux applications thérapeutiques avancées. Ces composés sont employés dans la formulation d’APIs pour le traitement des troubles du sommeil, de l’anxiété, de l’épilepsie et des spasmes musculaires. De plus, les dérivés des benzodiazépines sont essentiels dans la recherche de nouveaux agents psychotropes et dans l’optimisation des traitements neurologiques.
Chez CymitQuimica, nous proposons des dérivés de benzodiazépines de haute pureté pour des applications en synthèse chimique, en développement pharmaceutique et en neurosciences.
333 produits trouvés pour "Dérivés des Benzodiazépines"
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9-Nitro-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one
CAS :Formule :C9H9N3O3Degré de pureté :95.0%Masse moléculaire :207.1897-Bromo-2,3,4,5-tetrahydro-1h-1,4-benzodiazepin-5-one
CAS :Degré de pureté :95+%Masse moléculaire :241.08799748-Amino-4-Boc-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C14H21N3O2Degré de pureté :97%Masse moléculaire :263.3417-Fluoro-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione
CAS :Formule :C9H7FN2O2Degré de pureté :97.0%Couleur et forme :SolidMasse moléculaire :194.1654-Boc-2,3,4,5-Tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C14H20N2O2Degré de pureté :97.0%Couleur et forme :SolidMasse moléculaire :248.3264-Boc-9-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C15H22N2O2Degré de pureté :97.0%Masse moléculaire :262.3538-Chloro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C9H11ClN2Degré de pureté :97.0%Couleur et forme :SolidMasse moléculaire :182.653-(Piperidin-4-yl)-1,3,4,5-tetrahydro-2H-benzo[d][1,3]diazepin-2-one
CAS :Degré de pureté :97%Masse moléculaire :245.3260044-Boc-7-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C15H22N2O2Degré de pureté :97.0%Masse moléculaire :262.3532,3,4,5-Tetrahydro-1H-benzo[e][1,4]diazepine
CAS :Formule :C9H12N2Degré de pureté :97.0%Couleur et forme :White to yellow/orange crystalline powderMasse moléculaire :148.2098-Bromo-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one
CAS :Formule :C9H9BrN2ODegré de pureté :97.0%Masse moléculaire :241.0881,2,4,5-Tetrahydro-benzo[e][1,4]diazepin-3-one
CAS :Formule :C9H10N2ODegré de pureté :97.0%Couleur et forme :SolidMasse moléculaire :162.1924-Methyl-2,3,4,5-tetrahydro-1h-benzo[e][1,4]diazepine
CAS :Degré de pureté :95%Masse moléculaire :162.23599242,3,4,5-TETRAHYDRO-1H-BENZO[E][1,4]DIAZEPIN-8-YLAMINE 2HCL
CAS :Formule :C9H15Cl2N3Degré de pureté :97.0%Masse moléculaire :236.143-Amino-4-(2-fluorophenyl)-1-methyl-6-nitroquinolin-2(1H)-one
CAS :Produit contrôléFormule :C16H12FN3O3Couleur et forme :NeatMasse moléculaire :313.283-Methyl Clobazam
CAS :Produit contrôlé<p>Applications 3-Methyl Clobazam is a metabolite of Clobazam (C582500), a benzodiazepine psychotherapeutic agent that has proven efficacy against multiple seizure types. An anxiolytic; anticonvulsant.<br>References Gastaut, H., et al.: Epilepsia, 20, 437 (1979); Guberman, A., et al.: Can J. Neurol. Sci., 17, 311 (1990); Munn, R., et al.: Pediatr. Neurol. 9, 465 (1993)<br></p>Formule :C17H15ClN2O2Couleur et forme :NeatMasse moléculaire :314.773,3-Dimethyl Clobazam
Produit contrôléFormule :C18H17ClN2O2Couleur et forme :NeatMasse moléculaire :328.792-(2-Aminoacetamido)-5-nitro-2'-chlorobenzophenone Hydrochloride (Clonazepam Impurity)
CAS :Produit contrôléFormule :C15H12ClN3O4·ClHCouleur et forme :WhiteMasse moléculaire :370.18747-Aminonorflunitrazepam
CAS :Produit contrôléFormule :C15H12FN3OCouleur et forme :Light YellowMasse moléculaire :269.27N,N-Dimethylformamide Diethyl Acetal
CAS :Produit contrôlé<p>Stability Moisture Sensitive<br>Applications N,N-Dimethylformamide Diethyl Acetal is used as a reagent in the design of EGF-R tyrosine kinase inhibitors. Also used in the synthesis of aminopyridine derivatives.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Traxler, P. et al.: J. Med. Chem., 40, 3601 (1997); Cheikh, N. et al.: Tetrahedron, 69, 1234 (2013);<br></p>Formule :C7H17NO2Couleur et forme :NeatMasse moléculaire :147.22Flumazenil Carboxylic Acid-D3
Produit contrôlé<p>Applications Flumazenil Carboxylic Acid-D3 is an isotope labelled form of Flumazenil Carboxylic Acid (F500455); a derivative of Flumazenil (F500455), a benzodiazepine antagonist that can prevent or abolish (at the receptor level) the effects of a benzodiazepine.<br>References Brogden, R. & Goa, K.: Drugs, 35, 448 (1988); Klotz, U. & Kanto, J.: Clin. Pharmacokinet., 14, 1 (1988)<br></p>Formule :C13H7D3FN3O3Couleur et forme :NeatMasse moléculaire :278.252-Amino-5-nitrobenzophenone
CAS :Produit contrôléFormule :C13H10N2O3Couleur et forme :NeatMasse moléculaire :242.233-Amino-6-chloro-3,4-dihydro-2-methyl-4-phenyl-4-quinazolinol
CAS :Produit contrôléFormule :C15H14ClN3OCouleur et forme :NeatMasse moléculaire :287.742-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine
CAS :Produit contrôlé<p>Applications 2-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine is an impurity of Alprazolam (A575650.<br>References Hester, J.B., et al.: J. Org. Chem., 44, 2688, (1979); Anjaneyulu, Y., et al.: Asian. J. Chem., 19, 3375 (2007);<br></p>Formule :C17H15ClN4OCouleur et forme :White To Off-WhiteMasse moléculaire :326.782-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide
CAS :Produit contrôlé<p>Applications 2-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formule :C14H10Br2N2O2Couleur et forme :NeatMasse moléculaire :398.05N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide
CAS :Produit contrôlé<p>Applications N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formule :C14H10BrClN2O2Couleur et forme :Light Yellow To BeigeMasse moléculaire :353.60Alprazolam 5,6-Epoxide
CAS :Produit contrôlé<p>Applications Alprazolam derivative.<br>References Hester, J. et al., J. of Med. Chem. 23, 643 (1980)<br></p>Formule :C17H13ClN4OCouleur et forme :NeatMasse moléculaire :324.772-(2-Amino-5-bromobenzoyl)pyridine
CAS :<p>2-(2-Amino-5-bromobenzoyl)pyridine (2ABBP) is a chemical compound with the molecular formula C10H7BrN3. It is a glucuronide conjugate of 2-amino-5-bromobenzoic acid and has been used as an immunological reagent in the form of a monoclonal antibody. 2ABBP binds to dryopteris, which is a plant species that contains polyphenols called pteridines. 2ABBP has been shown to have anti-inflammatory properties in rat liver microsomes and cell culture experiments. The mechanism of action may involve inhibition of cyclooxygenase enzymes, which are involved in prostaglandin synthesis. 2ABBP also binds to human serum albumin and chaperones, proteins that bind other proteins or small molecules. The biological activity of 2ABBP may be due to its ability to form coval</p>Formule :C12H9BrN2ODegré de pureté :Min. 95%Masse moléculaire :277.12 g/molClobazam CIV
CAS :Produit contrôléClobazam (inn) and methyprylon (inn)Formule :C16H13ClN2O2Couleur et forme :White Crystalline PowderMasse moléculaire :300.066567-Amino Clonazepam-d4
CAS :Produit contrôlé<p>Applications A labelled major metabolite of Clonazepam (C587080).<br>References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),<br></p>Formule :C152H4H8ClN3OCouleur et forme :NeatMasse moléculaire :289.75
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![2,3,4,5-TETRAHYDRO-1H-BENZO[E][1,4]DIAZEPIN-8-YLAMINE 2HCL](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF304019.webp&w=3840&q=75)
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