
Sels et Dérivés d’API
Les sels des Ingrédients Pharmaceutiques Actifs (API) sont des composés formés par la réaction d’un acide avec une base, aboutissant à un équilibre ionique. Ces sels améliorent souvent la solubilité et la stabilité des API, facilitant ainsi leur absorption par l’organisme. Les dérivés des API sont des variantes chimiques d’un principe actif qui peuvent présenter des propriétés améliorées ou modifiées afin d’optimiser leur efficacité thérapeutique. Les sels d’API sont utilisés dans la formulation de médicaments oraux, injectables et topiques. De plus, les dérivés d’API peuvent améliorer la pharmacocinétique des médicaments, notamment en permettant une libération contrôlée des substances actives.
Chez CymitQuimica, nous proposons des sels et dérivés d’API avec la pureté et la qualité requises pour la recherche et le développement de formulations pharmaceutiques.
79369 produits trouvés pour "Sels et Dérivés d’API"
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TAK-653
CAS :<p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>Formule :C19H23N3O3SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :373.47Codeine N-Oxide CI
CAS :Produit contrôléConcentrates of poppy straw; buprenorphine (inn) codeine, dihydrocodeine (inn), ethylmorphine (inn), etorphine (inn), heroin, hydrococdone (inn), etc.Formule :C18H21NO4Couleur et forme :Brown White PowderMasse moléculaire :315.14706N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide
CAS :<p>N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide is a cavity inhibitor that has inhibitory activity against polymerization. It also reacts with chloride and alkene, which can be used to synthesize an amide. N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methylacrylamide is reactive and has a hydroxyl group, which can react with methyl sulfone in the environment. This agent has been shown to have anticancer activity in cell lines and tumor models.</p>Formule :C12H9F3N2ODegré de pureté :Min. 95%Masse moléculaire :254.21 g/molNaltrexone Related Compound A CII (17-(But-3-en-1-yl)-4,5α-epoxy-3,14-dihydroxymorphinan-6-one hydrochloride)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFormule :C20H23NO4·HClCouleur et forme :Off-White PowderMasse moléculaire :341.16271Noroxymorphone Hydrochloride CII (4,5α-Epoxy-3,14-dihydroxymorphinan-6-one hydrochloride)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFormule :C16H18NO4ClCouleur et forme :Light Brown PowderMasse moléculaire :323.09244AMPA receptor antagonist-2
CAS :<p>AMPA receptor antagonist-2 is an AMPA receptor antagonist.</p>Formule :C18H17N3O4Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :339.35Oxandrolone Related Compound A CIII (17β-hydroxy-17α-methyl-2-oxa-5α-androst-7-en-3-one)
CAS :Produit contrôléLactones nesoiFormule :C19H28O3Couleur et forme :White Crystalline PowderMasse moléculaire :304.20384Trospium Chloride Related Compound A (Benzilic Acid)
CAS :Carboxylic acids w/ alcohol function but w/o other oxygen function and their derivatives, nesoiFormule :C14H12O3Couleur et forme :White PowderMasse moléculaire :228.07864AV-101
CAS :<p>AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.</p>Formule :C10H11ClN2O3Degré de pureté :97.78% - 98.27%Couleur et forme :SolidMasse moléculaire :242.66Mibampator
CAS :<p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>Formule :C21H30N2O4S2Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :438.6ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
CAS :<p>Please enquire for more information about ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C22H22N4O4Degré de pureté :Min. 95%Masse moléculaire :406.43 g/molPSI 7976
CAS :<p>PSI 7976 is an analog of the nucleophilic attack drug, ribavirin. PSI 7976 inhibits the hepatitis C virus (HCV) replicon by inhibiting the function of the NS5B polymerase. In clinical studies, PSI 7976 has been shown to be active against HCV genotype 1 and 3. It has also been shown to inhibit replication of HIV-1 in vitro and to act synergistically with lamivudine against HIV-1 in human cells. PSI 7976 may be useful as a potential antiviral agent for treatment of other viral infections such as hepatitis B virus (HBV), herpes simplex virus type 2 (HSV-2), or cytomegalovirus (CMV).</p>Formule :C22H29FN3O9PDegré de pureté :Min. 95%Masse moléculaire :529.45 g/molDiphenoxylate Related Compound A CI (1-(3-Cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxylic acid)
CAS :Produit contrôléAlfentanil (inn), anileridine (inn), bezitramide (inn), bromazepam (inn), difenoxin (inn), diphenoxylate (inn), dipipanone (inn), fentanyl (inn), etc.Formule :C28H28N2O2Couleur et forme :PowderMasse moléculaire :424.21508Selurampanel
CAS :<p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>Formule :C16H19N5O4SDegré de pureté :99.60% - 99.78%Couleur et forme :SolidMasse moléculaire :377.42Benzaldehyde
CAS :Produit contrôléBenzaldehydeFormule :C7H6OCouleur et forme :Colorless LiquidMasse moléculaire :106.04186Oxymorphone Related Compound A CII (4,5α-Epoxy-3,14-dihydroxy-17-methylmorphinan-6-one N-oxide)
CAS :Produit contrôléConcentrates of poppy straw; buprenorphine (inn) codeine, dihydrocodeine (inn), ethylmorphine (inn), etorphine (inn), heroin, hydrococdone (inn), etc.Formule :C17H19NO5Couleur et forme :Off-White PowderMasse moléculaire :317.126322',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine
CAS :<p>2',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine is a cytosine analog that is used as an industrial chemical. It is prepared by the reaction of 5'-deoxycytidine with acetic anhydride in the presence of sodium bicarbonate, followed by a purification procedure. 2',3'-Di-O-acetyl-5'-deoxy-5-fluorocytidine reacts with toluene and trifluoromethanesulfonic acid to form 2',3'-di-O-acetyl 5'-deoxyfluorocytidine. This compound can be converted to 5'-deoxyfluorocytosine by heating in the presence of sodium tetrachloride. The yield for this process is high.</p>Formule :C13H16FN3O6Degré de pureté :Min. 95%Masse moléculaire :329.29 g/molExemestane Related Compound C CIII (androsta-1,4-diene-3,17-dione)
CAS :Produit contrôléAdrenal cortical hormones and their derivatives nesoiFormule :C19H24O2Couleur et forme :White PowderMasse moléculaire :284.17763Hydromorphone N-Oxide Hydrochloride CII (4,5α-Epoxy-3-hydroxy-17-methylmorphinan-6-one N-oxide, hydrochloride)
CAS :Produit contrôlé<p>Alkaloids of opium and their derivatives, salts thereof</p>Formule :C17H19NO4·HClCouleur et forme :Off-White PowderMasse moléculaire :337.79Clopidogrel EP Impurity B hydrochloride
CAS :<p>Please enquire for more information about Clopidogrel EP Impurity B hydrochloride including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C16H16ClNO2S•HClDegré de pureté :Min. 95%Masse moléculaire :358.28 g/molTAK-137
CAS :<p>TAK-137 is an AMPA receptor enhancer with antidepressant effects. TAK-137 has the ability to improve cognition and could be used to study schizophrenia.</p>Formule :C19H16N2O3SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :352.41Apixaban Impurity 6
CAS :<p>Please enquire for more information about Apixaban Impurity 6 including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C26H26N4O5Degré de pureté :Min. 95%Masse moléculaire :474.51 g/molZolpidem Impurities Mixture CIV
Produit contrôléDiagnostic or lab reagents on a backing, prepared diagnostic or lab reagents whether or not on a backing, whether or not in the form of kits, nesoiCouleur et forme :PowderHydromorphone Related Compound A CII (7,8-didehydro-4,5α-epoxy-3-hydroxy-17-methylmorphinan-6-one perchlorate)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereof, not elsewhere specified or includedFormule :C17H17NO3·HClO4Couleur et forme :Off-White Light Yellow PowderMasse moléculaire :383.07718Edoxaban
CAS :<p>Edoxaban: potent, selective FXa inhibitor; Ki 0.561 nM. Used as an oral anticoagulant for stroke prevention, also inhibits thrombin and FIXa.</p>Formule :C24H30ClN7O4SDegré de pureté :97.67% - 99.71%Couleur et forme :SolidMasse moléculaire :548.06Hydrocodone Related Compound A CII (4-hydroxy-3-methoxy-17-methylmorphinan-6-one)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereofFormule :C18H23NO3Couleur et forme :White PowderMasse moléculaire :301.16779GNE-8324
CAS :<p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>Formule :C18H18FN3OSDegré de pureté :98.68% - 99.34%Couleur et forme :SolidMasse moléculaire :343.42Tropicamide Related Compound D (2-Phenylacetic acid)
CAS :Produit contrôléPhenylacetic acid (alpha-toluic acid) and its saltsFormule :C8H8O2Couleur et forme :Beige PowderMasse moléculaire :136.05243Cathinone Hydrochloride CI (α-Aminopropiophenone hydrochloride)
CAS :Produit contrôléVegetable alkaloids, natural or reproduced by synthesis, their salts and other derivatives, nesoiFormule :C9H11NO·HClCouleur et forme :White PowderMasse moléculaire :149.08406Testosterone Enanthate Related Compound B CIII (Androst-4-en-3-one-17β-yl hexanoate)
CAS :Produit contrôléAdrenal cortical hormones and their derivatives nesoiFormule :C25H38O3Couleur et forme :White PowderMasse moléculaire :386.2821Dextromethorphan Related Compound A CI (3-Methoxy-9α,13α,14α-morphinan hydrochloride)
CAS :Produit contrôléCompounds containing a quinoline or isoquinoline ring-system, whether or not hydrogenated, not further fused, excluding drugs and pesticidesFormule :C17H23NO·HClCouleur et forme :White PowderMasse moléculaire :257.17796Fentanyl Related Compound E CII (N-Phenyl-1-(2-phenylethyl)-4-piperidinamine)
CAS :Produit contrôlé4-anilino-n-phenethylpiperidine (anpp)Formule :C19H24N2Couleur et forme :White Light Brown Crystalline PowderMasse moléculaire :280.19395Oxycodone Related Compound C CII (codeinone)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereofFormule :C18H19NO3Couleur et forme :PowderMasse moléculaire :297.13649Zopiclone R-Isomer CIV ((-)-(5R)-6-(5-Chloropyridin-2-yl)-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-yl 4-methylpiperazine-1-carboxylate)
CAS :Produit contrôléLactams, nesoiFormule :C17H17ClN6O3Couleur et forme :Light Brown SolidMasse moléculaire :388.10507Apixaban Impurity 1
CAS :<p>Apixaban Impurity 1 is an impurity found in Apixaban, a drug used for the prevention of stroke. It is produced by condensation of 2-aminopyridine and 3-hydroxybenzaldehyde in ethanol with sodium hydroxide as a catalyst. The reaction proceeds via amination of the pyridine ring followed by transesterification. The yield of this impurity is low at about 4%.</p>Degré de pureté :Min. 95%Benzphetamine Related Compound A CIII ((R)-N-Benzyl-N-methyl-1-phenylpropan-2-amine hydrochloride)
CAS :Produit contrôlé<p>Aromatic monoamines not elsewhere specified or included and their derivatives, salts therof</p>Formule :C17H21N·HClCouleur et forme :White Off-White PowderMasse moléculaire :275.14408Dextroamphetamine Related Compound B CII (Phenyl acetone)
CAS :Produit contrôléPhenylacetone (phenylpropan-2-one)Formule :C9H10OCouleur et forme :Clear Pale Yellow LiquidMasse moléculaire :134.07316Oxandrolone Related Compound C CIII (17,17-dimethyl-18-nor-2-oxa-5α-androst-13-en-3-one)
Produit contrôléLactones nesoiFormule :C19H28O2Couleur et forme :PowderMasse moléculaire :288.42Delucemine Hydrochloride
CAS :<p>Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.</p>Formule :C16H18ClF2NDegré de pureté :98.49% - 99.30%Couleur et forme :SolidMasse moléculaire :297.77Oxacyclohexane open ring tacrolimus
CAS :<p>Please enquire for more information about Oxacyclohexane open ring tacrolimus including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C44H71NO13Degré de pureté :Min. 95%Masse moléculaire :822.04 g/molCNS-5161 hydrochloride
CAS :<p>CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.</p>Formule :C16H19Cl2N3S2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :388.38Neboglamine hydrochloride
CAS :<p>Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.</p>Formule :C13H25ClN2O3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :292.84-PPBP maleate
CAS :<p>4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.</p>Formule :C25H31NO4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :409.52Oxandrolone Related Compound B CIII (17 β-hydroxy-17 α-methyl-4-oxa-5 α-androsta-3-one)
CAS :Produit contrôléLactones, nesoiFormule :C19H30O3Couleur et forme :Off-White Crystalline PowderMasse moléculaire :306.21949Fentanyl Related Compound G CI (N-(1-Phenethylpiperidin-4-yl)-N-phenylacetamide)
CAS :Produit contrôlé<p>Fentanyls and their derivatives containing an unfused pyrazole ring, whether or not hydrogenated, nesoi</p>Formule :C21H26N2OCouleur et forme :White PowderMasse moléculaire :322.45Morphine Related Compound A CI (7,8-Didehydro-4,5α-epoxy-17-methylmorphinan-3,6α-diol, N-oxide)
CAS :Produit contrôléAlkaloids of opium and their derivatives, salts thereofFormule :C17H19NO4Couleur et forme :Yellow Tan PowderMasse moléculaire :301.13141Ro 25-6981
CAS :<p>Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.</p>Formule :C22H29NO2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :339.47NMDA receptor modulator 4
CAS :<p>NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1].</p>Formule :C13H9F3N2O3SCouleur et forme :SolidMasse moléculaire :330.28NMDA receptor modulator 6
CAS :<p>NMDA receptor regulator 6 (Compound 183) is an effective NMDA receptor regulator and has research value in neurological disorders.</p>Formule :C20H17FN2O4SCouleur et forme :SolidMasse moléculaire :400.42DQP-26
CAS :<p>DQP-26, a potent negative allosteric modulator of NMDA receptors (NMDARs), exhibits IC50 values of 0.77 μM for GluN2C and 0.44 μM for GluN2D subunits,</p>Formule :C28H21Cl2N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.39AMPA receptor modulator-5
CAS :<p>AMPA Receptor Modulator-5 (Example 217) serves as an AMPA receptor modulator, utilized in neurological disease research [1].</p>Formule :C20H12F4N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.34AMPA receptor modulator-6
CAS :<p>AMPA receptor modulator-6, an AMPA receptor positive allosteric modulator (PAM), is utilized in the research of neurological diseases [1].</p>Formule :C24H36N2O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :480.68AMPA receptor modulator-2
CAS :<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Formule :C15H6F6N4OSDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :404.29PF-4778574
CAS :<p>PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).</p>Formule :C19H22N2O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :390.52TCS 46b
CAS :<p>TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.</p>Formule :C22H23N3ODegré de pureté :99.78% - 99.78%Couleur et forme :SolidMasse moléculaire :345.44Dasolampanel etibutil
CAS :<p>Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).</p>Formule :C23H32ClN5O3Couleur et forme :SolidMasse moléculaire :461.98NS1219
CAS :<p>NS1219, an isomer of NS1209, is a selective AMPA antagonist for studying stroke, neuropathic pain, and epilepsy.</p>Formule :C24H28N4O7SCouleur et forme :SolidMasse moléculaire :516.57Zelquistinel
CAS :<p>Zelquistinel, an NMDA receptor agonist, aids research on depression, anxiety, and psychiatric disorders.</p>Formule :C15H25N3O5Couleur et forme :SolidMasse moléculaire :327.38ADCI
CAS :<p>ADCI inhibits voltage-activated sodium and NMDA channels; boosts dopamine metabolism in prefrontal cortex and nucleus accumbens.</p>Formule :C16H14N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :250.3BMS-986169
CAS :<p>BMS-986169 is a high-affinity and selective negative allosteric modulator of the NMDA receptor GluN2B subunit, depression.</p>Formule :C23H27FN2O2Degré de pureté :97.61%Couleur et forme :SolidMasse moléculaire :382.47GNE-0723
CAS :<p>GNE-0723 is a selective positive allosteric modulator of the NMDA receptor, GluN2A.blood-brain barrier (BBB) and Dravet syndrome and Alzheimer's disease (AD).</p>Formule :C16H8ClF6N5OSDegré de pureté :97.29% - 99.91%Couleur et forme :SolidMasse moléculaire :467.78UBP316
CAS :<p>GluR5-containing kainate receptor antagonist</p>Formule :C20H19N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.45NPEC-caged-(S)-AMPA
CAS :<p>AMPA receptor agonist</p>Formule :C16H17N3O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.32Pregnanolone sulfate (pyridinium)
CAS :<p>Pregnanolone sulfate pyridinium, an endogenous neurosteroid, inhibits NMDA receptors and exhibits neuroprotective properties [1].</p>Formule :C26H39NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.66Nevadistinel
CAS :<p>Nevadistinel (NYX-458; NYX-3054) is a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, indicated for mitigating cognitive deficits</p>Formule :C15H18N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :274.32Risevistinel
CAS :<p>Risevistinel (NYX-783), a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, may mitigate cognitive deficits in neurodegenerative</p>Formule :C14H23N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.35Naspm trihydrochloride
CAS :<p>Naspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride) is a synthetic analogue of Joro spider toxin and is an antagonist of calcium permeable AMPA</p>Formule :C22H37Cl3N4ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :479.91p-fin4
CAS :<p>p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.</p>Formule :C39H53N8O18PCouleur et forme :SolidMasse moléculaire :952.85BMT-108908
CAS :<p>BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.</p>Formule :C22H25FN2O2Couleur et forme :SolidMasse moléculaire :368.44AMPA-IN-1
CAS :<p>AMPA-IN-1: Potent AMPA receptor inhibitor; key in regulating brain excitatory transmission and plasticity.</p>Formule :C23H12F2N4O2Couleur et forme :SolidMasse moléculaire :414.36(R)-3,4-DCPG
CAS :<p>AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors</p>Formule :C10H9NO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.18AMPA receptor antagonist-3
CAS :<p>AMPA receptor antagonist-3 is an AMPA receptor antagonist.</p>Formule :C20H19N5O2SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.46Rislenemdaz
CAS :<p>Rislenemdaz (CERC-301) (CERC-301) is an antagonist of the N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B).</p>Formule :C19H23FN4O2Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :358.41AMPA receptor modulator-1
CAS :<p>AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.</p>Formule :C16H11ClF3NO2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :341.71N1-N2-Di-N-Nitroso methyl (2S,5S)-5-methylpiperazine-2-carboxylate
Formule :C7H12N4O4Masse moléculaire :216.2N2-N-Nitroso methyl (2S,5S)-5-methylpiperazine-2-carboxylate
Formule :C7H13N3O3Masse moléculaire :187.2N1-N-Nitroso methyl (2S,5S)-5-methylpiperazine-2-carboxylate
Formule :C7H13N3O3Masse moléculaire :187.22,2'-(Thiobis(2-hydroxy-5,1-phenylene))bis(4H-benzo[e][1,3]oxazin-4-one)
CAS :<p>Please enquire for more information about 2,2'-(Thiobis(2-hydroxy-5,1-phenylene))bis(4H-benzo[e][1,3]oxazin-4-one) including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C28H16N2O6SDegré de pureté :Min. 95%Masse moléculaire :508.5 g/mol13-O-Desmethyl tacrolimus
CAS :<p>Tacrolimus is a macrolide immunosuppressant that is used to prevent organ rejection in transplant patients. It binds to the cytosolic protein, FKBP-12, which prevents calcineurin from dephosphorylating and activating nuclear factor of activated T cells (NFAT). Tacrolimus inhibits the production of IL-2 and other cytokines by T cells, suppressing proliferation. Tacrolimus has been shown to be bioequivalent when administered orally or intravenously. Bioavailability may be increased when taken with food.</p>Formule :C43H67NO12Degré de pureté :90%MinCouleur et forme :PowderMasse moléculaire :789.99 g/molMacitentan (n-butyl analogue)
CAS :<p>Macitentan n-butyl analogue, an oral ETA/ETB receptor blocker, may treat IPF and PAH.</p>Formule :C20H21Br2N5O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :587.29Tamitinol
CAS :<p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>Formule :C12H20N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :240.373-Methoxy PCE hydrochloride
CAS :<p>3-Methoxy PCE (3-MEO PCE) hydrochloride is an arylcyclohexylamine compound that functions as an NMDA receptor antagonist with a pKi value of 7.22.</p>Formule :C15H24ClNOCouleur et forme :SolidMasse moléculaire :269.81EMD-95885
CAS :<p>EMD-95885 is a selective antagonist of NMDA receptors containing NR2B subunits, with an IC50 of 3.9 nM. It does not interact with other sites on the NMDA receptor.</p>Formule :C22H23FN2O3Couleur et forme :SolidMasse moléculaire :382.428PDE2 inhibitor 6
CAS :<p>PDE2 inhibitor6 (Compound 1) is an orally active phosphodiesterase (PDE) inhibitor, effectively inhibiting PDE2A, PDE3B, and PDE10A2 with IC50 values of 0.95 nM, 6.17 μM (pIC50=5.21), and 87.1 nM (pIC50=7.06), respectively. It modulates AMPA receptor activity, enhances synaptic plasticity, and improves learning and memory in rat models. Furthermore, PDE2 inhibitor6 possesses blood-brain barrier permeability.</p>Formule :C20H22F2N6OCouleur et forme :SolidMasse moléculaire :400.425NMDA agonist 1
CAS :<p>NMDA agonist 1 (compound 42d) is a potent NMDA agonist with a Ki value of 96 nM. It acts as a partial agonist of the GluN1/GluN2B complex, exhibiting an EC50 value of 78 nM.</p>Formule :C12H13N3O3SCouleur et forme :SolidMasse moléculaire :279.315DL-AP5 lithium
CAS :<p>DL-AP5 (2-APV) lithium is a competitive antagonist of the NMDA (N-Methyl-D-aspartate) receptor. It exhibits notable analgesic activity and specifically blocks channels in the rabbit retina.</p>Formule :C5H11LiNO5PCouleur et forme :SolidMasse moléculaire :203.06Metaphit methylsulfate
CAS :<p>Metaphit methylsulfate is a specific PCP antagonist and an acylating agent for the [3H] phencyclidine binding site in rat brain homogenate. It inhibits PCP-induced motor activity through a presynaptic mechanism.</p>Formule :C19H28N2O3S2Couleur et forme :SolidMasse moléculaire :396.567BMS-986163
CAS :<p>BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).</p>Formule :C23H28FN2O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :462.45(RS)-AMPA hydrobromide
CAS :<p>AMPAR agonist</p>Formule :C7H11BrN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.08(RS)-AMPA hydrochloride
CAS :<p>(RS)-AMPA ((±)-AMPA) hydrochloride is a glutamate analog and serves as an efficient selective agonist for the excitatory neurotransmitter L-glutamic acid (L-glutamic acid). It does not interfere with the binding sites of alginate or NMDA receptors.</p>Formule :C7H11ClN2O4Couleur et forme :SolidMasse moléculaire :222.63LY 215490
CAS :<p>LY 215490 is a selective AMPA receptor antagonist with neuroprotective properties in rat ischemia.</p>Formule :C13H21N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.34Caged MK801
CAS :<p>Caged MK801 (cMK801) is a selective, noncompetitive, and irreversible blocker of the NMDA receptor open channel. The NVOC cage is compatible in neuropharmacology and does not alter the intrinsic activity of the molecule.</p>Formule :C26H24N2O6Couleur et forme :SolidMasse moléculaire :460.48EU 1622-240
CAS :<p>EU 1622-240 is an allosteric modulator with a preference for GluN2B, GluN2C, and GluN2D, exhibiting EC50 values of 0.57, 0.82, and 1.1 μM, respectively. It possesses favorable physicochemical properties, along with in vitro stability and permeability.</p>Formule :C20H14BrF2N3O2SCouleur et forme :SolidMasse moléculaire :478.31NMDA receptor antagonist-3
<p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>Formule :C13H19N3O6Couleur et forme :SolidMasse moléculaire :313.31NYX-2925
CAS :<p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>Formule :C14H23N3O4Couleur et forme :SolidMasse moléculaire :297.35Lu AF90103
CAS :<p>Lu AF90103 (Compound 42e) is the methyl ester prodrug of compound 42d, capable of crossing the blood-brain barrier. Compound 42d acts as a partial agonist of the GluN1/GluN2B complex, with an efficacy of 24% and an EC50 value of 78 nM. Lu AF90103 plays a significant role in neuropsychiatric disorder research.</p>Formule :C13H15N3O3SCouleur et forme :SolidMasse moléculaire :293.342Antidepressant agent 9
CAS :<p>Antidepressant agent 9 (Compound 24) is an orally active inhibitor of NMDAR and SERT, with IC50 values of 3.50 μM and 1044 nM, respectively. It exhibits good metabolic stability and plasma exposure, and demonstrates antidepressant-like effects in the forced swim test in mice.</p>Formule :C17H24N2Couleur et forme :SolidMasse moléculaire :256.386(3S,6R)-NML
CAS :<p>(3S,6R)-NML is an NMDA receptor antagonist with pIC50 values of 4.8 [GluN1-GluN2A], 4.6 [GluN1-GluN2B], 5.0 [GluN1-GluN2C], and 5.0 [GluN1-GluN2D]. It is applicable in the study of depression.</p>Formule :C20H27NOCouleur et forme :SolidMasse moléculaire :297.435LY503430
CAS :<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formule :C20H25FN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.49YY-23
CAS :<p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>Formule :C33H54O8Couleur et forme :SolidMasse moléculaire :578.777Onfasprodil
CAS :<p>Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)</p>Formule :C20H23FN2O3Couleur et forme :SolidMasse moléculaire :358.41Antidepressant agent 8
CAS :<p>Antidepressant agent 8 (Compound 1f) acts as a selective antagonist for the NMDA receptor GluN1/2A (NMDA receptorGluN1/2A), with an IC50 of 2.94 μmol/L. In a hydrocortisone-induced zebrafish depression model, it demonstrates antidepressant-like effects and shows good blood-brain barrier penetration.</p>Formule :C18H23FN4OS2Couleur et forme :SolidMasse moléculaire :394.53Caramboxin
CAS :<p>Caramboxin, a neurotoxin, can induce acute kidney injury.</p>Formule :C11H13NO6Couleur et forme :SolidMasse moléculaire :255.22(RS)-AMPA
CAS :<p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>Formule :C7H10N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :186.17Perfluoroheptanesulfonic acid
CAS :<p>Perfluoroheptanesulfonic acid (1-Perfluoroheptanesulfonic acid; Perfluoroheptanesulphonic acid) is a perfluoroalkyl substance (PFAS). This compound has been detected in landfill leachate and has been shown to induce deformities in zebrafish larvae (EC50=168.1 μM). Exposure to PFHpS in fetuses can lead to reduced birth weight.</p>Formule :C7HF15O3SCouleur et forme :SolidMasse moléculaire :450.12LY 235959
CAS :<p>LY 235959 is a NMDA receptor antagonist.</p>Formule :C11H20NO5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.25(RS)-AMPA monohydrate
CAS :<p>(RS)-AMPA monohydrate, potent glutamate analogue, selectively activates L-glutamic acid without affecting kainic acid or NMDA receptors.</p>Formule :C7H12N2O5Couleur et forme :SolidMasse moléculaire :204.182Blixeprodil
CAS :<p>Blixeprodil (GM-1020) is an orally active NMDA receptor antagonist with an affinity of Ki = 3.25 µM in rat cortical tissue. It inhibits NR1/2A-NMDAR-mediated currents in HEK293 cells with an IC50 of 1.192 µM. Blixeprodil demonstrates antidepressant effects in rat models and exhibits blood-brain barrier permeability.</p>Formule :C13H16FNOCouleur et forme :SolidMasse moléculaire :221.271LY3130481
CAS :<p>LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.</p>Formule :C19H18N4O3SCouleur et forme :SolidMasse moléculaire :382.44SDZ 220-040
CAS :<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。</p>Formule :C16H16Cl2NO6PDegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :420.18BDZ-g
CAS :<p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>Formule :C21H21N5O2SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.49Veratramine
CAS :Formule :C27H39NO2Degré de pureté :>98.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :409.614,4'-Diethynylbiphenyl
CAS :Formule :C16H10Degré de pureté :>98.0%(GC)Couleur et forme :White to Light yellow to Light orange powder to crystalMasse moléculaire :202.26D-2-Phenylglycine
CAS :Formule :C8H9NO2Degré de pureté :>99.0%(T)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :151.17tert-Butyl Hydrogen Tetradecanedioate
CAS :Formule :C18H34O4Degré de pureté :>95.0%(GC)(T)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :314.47Isobutyryl Chloride
CAS :Formule :C4H7ClODegré de pureté :>98.0%(GC)(T)Couleur et forme :Colorless to Light yellow clear liquidMasse moléculaire :106.554-Maleimidobutyric Acid
CAS :Formule :C8H9NO4Degré de pureté :>98.0%(GC)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :183.16(1E,4E)-1,5-Bis[3,5-bis(methoxymethoxy)phenyl]-1,4-pentadiene-3-one
CAS :Formule :C25H30O9Degré de pureté :>97.0%(HPLC)Couleur et forme :White to Yellow to Green powder to crystalMasse moléculaire :474.51Ethylhexyl Triazone Related Compound A (2-ethylhexyl 4-aminobenzoate) (DISCONTINUED)
CAS :Aromatic amino-acids and their esters, other than thoseFormule :C15H23NO2Couleur et forme :PlatesMasse moléculaire :249.17288Calcitonin Salmon Related Compound B (calcitonin salmon-glycine) (COLD SHIPMENT REQUIRED) (DISCONTINUED)
CAS :Polypeptide, protein and glycoprotein hormones, their derivatives and structural analogues, nesoiFormule :C147H242N44O50S2Couleur et forme :Colorless LiquidMasse moléculaire :3487.71879





