Composés et métabolites pharmaceutiques et vétérinaires
Cette catégorie inclut des composés pharmaceutiques utilisés en médecine humaine et vétérinaire, ainsi que leurs métabolites. Ces composés sont essentiels pour étudier l'efficacité des médicaments, leur métabolisme et leur sécurité. Chez CymitQuimica, nous offrons une variété de composés pharmaceutiques et vétérinaires pour des applications de recherche, garantissant la conformité aux normes réglementaires et soutenant le développement de nouveaux traitements.
2577 produits trouvés pour "Composés et métabolites pharmaceutiques et vétérinaires"
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Lipoxin A5
CAS :<p>LXA5 is made from EPA by leukocytes, contracts guinea pig lungs like LXA4/LXB4, but doesn't dilate aorta.</p>Formule :C20H30O5Couleur et forme :SolidMasse moléculaire :350.45Dioctanoylphosphatidic acid sodium
CAS :<p>Dioctanoylphosphatidic acid sodium serves as a modulator of phagocyte respiratory bursts, a precursor to diacylglycerol and lyso-phosphatidic acid, and influences the phosphorylation of the mammalian target of rapamycin (mTOR). Additionally, it enhances the viability of gallbladder cancer cells inhibited by histone deacetylase inhibitors (HDACI). This compound is derived from glycerophospholipids through the action of phospholipase D.</p>Formule :C19H36NaO8PCouleur et forme :SolidMasse moléculaire :446.45AubipyOMe
CAS :<p>AubipyOMe serves as an effective inhibitor of Tartrate-resistant Acid Phosphatase (TRAP/ACP5), a metalloenzyme identified in activated osteoclasts and macrophages. It exhibits inhibitory IC50 values of 1.3 μM against TRAP5a and 1.8 μM against TRAP5b. Additionally, it effectively suppresses TRAP activity in extracts from mouse macrophages and human lung tissues.</p>Formule :C12H12AuCl2F6N2O2PCouleur et forme :SolidMasse moléculaire :629.077α,24(S)-Dihydroxycholesterol
CAS :<p>7α,24(S)-Dihydroxycholesterol ((3β,7α,24S)-Cholest-5-ene-3,7,24-triol) acts as a ligand for liver X receptors (LXR), specifically binding to the ligand-binding domains of LXRα and LXRβ. This compound is synthesized through the E-α,β-unsaturated ketone process, starting with arsindole and J-secondary-butyl dimethylsiloxy-bis-positive-5-cholestenal as the initial materials. It undergoes a series of transformations to produce 7α,24(S)-dihydroxycholesterol.</p>Formule :C27H46O3Couleur et forme :SolidMasse moléculaire :418.653-Ferrocenylpropionic anhydride
CAS :<p>3-Ferrocenylpropionic anhydride is extensively used in compound synthesis, serving as an intermediary for producing various bioactive compounds. Additionally, by modulating specific enzyme activities, 3-Ferrocenylpropionic anhydride has demonstrated potential anti-tumor properties.</p>Formule :C26H26Fe2O3Couleur et forme :SolidMasse moléculaire :498.17Homomoschatoline
CAS :<p>Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.</p>Formule :C19H15NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.332,4-Dihydroxybutanoic acid
CAS :<p>2,4-Dihydroxybutanoic acid is typically not found in extracts of normal human urine and is present only in trace amounts in newborns, while cases of succinic semialdehyde dehydrogenase deficiency consistently exhibit elevated levels of this metabolite.</p>Formule :C4H8O4Couleur et forme :SolidMasse moléculaire :120.10RBM14C12
CAS :<p>RBM14C12 is a compound known for its cell signaling activity. It plays a crucial role in researching lipid metabolism and cell membrane structure. Additionally, RBM14C12 can be utilized in the development of novel compounds aimed at modulating the biological mechanisms associated with lipid-related diseases.</p>Formule :C26H39NO6Couleur et forme :SolidMasse moléculaire :461.599-cis-β-Carotene
CAS :<p>9-cis-β-Carotene, a precursor of retinal, is cleaved by beta-carotene oxygenase 1 (BCMO1) to produce 9-cis-retinal.</p>Formule :C40H56Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :536.87(-)-Mesembrine
CAS :<p>Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).</p>Formule :C17H23NO3Couleur et forme :SolidMasse moléculaire :289.37Cyclic-di-GMP sodium
<p>c-di-GMP sodium: STING activator, regulates bacteria biofilm, motility, virulence.</p>Formule :C20H24N10NaO14P2Couleur et forme :SolidMasse moléculaire :713.08464Magnesium ionophore III
CAS :<p>Magnesium ionophore III (ETH 4030) is an ion carrier that regulates intracellular magnesium ion concentrations. It enhances cellular functions and metabolic activities by increasing the permeability of cell membranes to magnesium ions. Additionally, Magnesium ionophore III is utilized in research to explore the significance of magnesium ions in biological processes and their impact on cellular physiology.</p>Formule :C30H58N4O4Couleur et forme :SolidMasse moléculaire :538.81Rostratin A
CAS :<p>Rostratin A, a disulfide from Exserohilum rostratum, is cytotoxic to HCT-116 cells with an IC50 of 8.5 μg/mL.</p>Formule :C18H24N2O6S2Couleur et forme :SolidMasse moléculaire :428.52Urobilin hydrochloride
CAS :<p>Urobilin hydrochloride, a metabolic byproduct of Hemoglobin, is excreted through urine and feces in various mammals. It also serves as an indicator of human waste contamination.</p>Formule :C33H43ClN4O6Couleur et forme :SolidMasse moléculaire :627.17S-MTC acetate
CAS :<p>S-MTC acetate (S-Methyl-L-thiocitrulline acetate) serves as a potent inhibitor of inducible nitric oxide synthases and is especially effective in inhibiting the constitutive (neuronal) type rather than the inducible (endothelial) type.</p>Formule :C9H19N3O4SCouleur et forme :SolidMasse moléculaire :265.33Inosine 5′-diphosphate sodium
CAS :<p>Inosine 5'-diphosphate sodium, a purine ribonucleoside diphosphate with inosine as its nucleobase, plays a role in intracellular energy metabolism and signal transduction processes.</p>Formule :C10H13N4Na3O12P2Couleur et forme :SolidMasse moléculaire :512.15(S)-CPP sodium
CAS :<p>(S)-CPP sodium serves as an inhibitor of the branched-chain α-keto acid dehydrogenase complex (BCKDC) kinase, commonly referred to as BDK or keto acid dehydrogenase kinase. As a negative regulator of BCKDC activity, (S)-CPP (IC50 of 6.3 μM) inhibits BDK, which activates the complex, leading to a significant reduction in the levels of leucine/isoleucine and valine in the plasma of wild-type mice.</p>Formule :C9H8ClNaO2Couleur et forme :SolidMasse moléculaire :206.60Diethylumbelliferyl phosphate
CAS :<p>Diethylumbelliferyl phosphate (DEUP) is a potent and selective inhibitor of cholesterol esterase that does not inhibit protein kinase A activity in vitro. It disrupts steroidogenesis by blocking cholesterol transport to mitochondria in steroidogenic cells, with an IC50 of 11.6 μM. This compound may also limit the absorption of dietary cholesterol.</p>Formule :C14H17O6PCouleur et forme :SolidMasse moléculaire :312.25RS 61756-007
CAS :<p>RS 61756-007 is a selective thromboxane receptor (TP) agonist.</p>Formule :C23H28O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :384.476′SLN
CAS :<p>6′SLN is a characteristic glycan found on the surface of cancer-related extracellular vesicles (EVs) and serves as the primary form of protein glycosylation within EVs. Additionally, 6′SLN, a derivative of sialic acid, interacts with hemagglutinins (HAs) from both human and avian influenza strains, making it relevant in the study of anti-influenza drugs.</p>Formule :C25H42N2O19Couleur et forme :SolidMasse moléculaire :674.6
