Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Fludarabine triphosphate trisodium
CAS :<p>Fludarabine triphosphate trisodium is a nucleotide analog, which is a type of chemotherapy agent derived from purine nucleosides. This compound is the active metabolite of fludarabine, sourced from synthetic chemistry designed to mimic naturally occurring nucleotides involved in DNA replication. The mode of action involves its incorporation into the DNA strand during replication, where it effectively inhibits DNA polymerase and ribonucleotide reductase. This disruption impairs DNA synthesis, leading to apoptosis or programmed cell death, particularly in rapidly dividing cancer cells.</p>Formule :C10H15FN5O13P3·Na3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :594.14 g/molMLN 4924
CAS :<p>MLN 4924 is a selective small molecule that acts as an inhibitor of the Nedd8-activating enzyme. This compound is synthetically derived and functions by inhibiting the conjugation of Nedd8 to cullin proteins. By blocking this pathway, MLN 4924 disrupts the activity of the SCF (Skp, Cullin, F-box containing complex) E3 ubiquitin ligase, leading to an accumulation of proteins that can induce apoptosis and cell cycle arrest.</p>Formule :C21H25N5O4SDegré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :443.52 g/molN-Desmethyl ibandronate sodium
CAS :<p>N-Desmethyl ibandronate sodium is a white crystalline solid with a melting point of 238-240 °C. It has versatile building block, complex compound and research chemicals applications. It is an intermediate used in the synthesis of other compounds, such as speciality chemicals, useful intermediates and useful scaffolds. N-Desmethyl ibandronate sodium can be used in reactions that require high quality and high purity products.</p>Formule :C8H20NO7P2·xNaDegré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :327.18 g/molXAV 939
CAS :<p>Inhibits tankyrase (TNKS1 and TNKS2 with IC50 values of 11 and 4 nM respectively), by binding to the catalytic poly-ADP-ribose polymerase (PARP) domain. This stabilizes cytoplasmic protein Axin, mediating β-catenin depletion and thereby suppresses Wnt signalling pathway. XAV 939 has anti-proliferative and pro-apoptotic effects on neuroblastoma and colorectal cancer cells.</p>Formule :C14H11F3N2OSDegré de pureté :Min. 95%Masse moléculaire :312.31 g/molEpacadostat
CAS :<p>Inhibitor of dioxygenase IDO1</p>Formule :C11H13BrFN7O4SDegré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :438.23 g/molXL184
CAS :<p>Pan-tyrosine kinase inhibitor (VEGFR2, c-MET, RET, KIT); anti-neoplastic</p>Formule :C28H24FN3O5Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :501.51 g/molEtoposide - Bio-X ™
CAS :<p>Etoposide is a cytotoxic drug used in cancer chemotherapy. It inhibits DNA replication through inhibition of DNA topoisomerase II, thus catalysing cell cycle arrest and apoptosis. <br>Etoposide is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Formule :C29H32O13Degré de pureté :Min. 98 Area-%Couleur et forme :White PowderMasse moléculaire :588.56 g/molFinasteride - Bio-X ™
CAS :<p>Finasteride is an antiandrogenic drug that belongs to the group of 5-alpha reductase inhibitors, which are used for the treatment of benign prostatic hyperplasia and male pattern baldness. The conversion of testosterone to 5α-dihydrotestosterone (DHT) is blocked by type II 5α-reductase inhibition, which then results in significant increase in prostatic testosterone concentrations and minimal to moderate increases in serum and tissue DHT concentrations. A reduction in DHT concentration will cause a reduction in prostatic volume as DHT appears to be the main androgen responsible for stimulating prostatic growth.</p>Formule :C23H36N2O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :372.54 g/molRofecoxib - Bio-X ™
CAS :Produit contrôlé<p>Rofecoxib is a non-steroidal anti-inflammatory drug that is used to treat osteoarthritis, acute pain and migraine attacks. This drug is also a COX-2 inhibitor. As a result, it reduces inflammation and pain.</p>Formule :C17H14O4SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :314.36 g/molSacubitril sodium
CAS :<p>Inhibitor of metalloendopeptidase neprilysin</p>Formule :C24H28NNaO5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :433.47 g/molIbandronate sodium monohydrate
CAS :<p>Farnesyl pyrophosphate synthase inhibitor</p>Formule :C9H24NNaO8P2Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :359.23 g/molLestaurtinib
CAS :<p>Lestaurtinib is a multitarget tyrosine kinase inhibitor of the JAK, FLT-3 and TrkA families of tyrosine kinases at nanomolar concentrations. It inhibits proliferation and induces apoptosis in vitro. Lestaurtinib is a FDA approved orphan drug for acute myeloid leukemia.</p>Formule :C26H21N3O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :439.46 g/molBL 918
CAS :<p>A potent small-molecule activator of UNC-51-like kinase 1 (ULK1), a serine-threonine kinase involved in autophagy. Promotes cytoprotective autophagy in MPP+-treated SH-SY5Y cells, via the ULK complex. Improves motor dysfunction and reduces loss of dopaminergic neurons, mediated by MPTP, in in vivo models of Parkinson’s disease.</p>Formule :C23H15F8N3OSDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :533.44 g/molRosuvastatin calcium - Bio-X ™
CAS :<p>Rosuvastatin is a drug that belongs to the group of statins. It is used for the treatment of high cholesterol and as an adjunct therapy for patients with coronary heart disease. Rosuvastatin reduces serum cholesterol by inhibiting HMG-CoA reductase, which is the rate-limiting enzyme in the production of cholesterol. Furthermore, this drug has been shown to have anti-inflammatory properties, which may be due to its ability to inhibit prostaglandin synthesis.</p>Formule :C22H27FN3O6SCaDegré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :500.57 g/molCP 671305
CAS :<p>Inhibitor of PDE4 enzyme</p>Formule :C23H19FN2O7Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :454.4 g/molSNS 314 mesylate
CAS :<p>Inhibitor of Aurora kinases A, B and C</p>Formule :C18H15ClN6OS2•CH4O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :527.04 g/molWM 8014
CAS :<p>Selective and potent inhibitor of lysine acetyltransferases KAT6A and KAT6B with IC50 values of 8 nM and 28 nM, respectively. The compound is a reversible competitor of acetyl coenzyme A domain of KAT6A/B enzymes. It inhibits MYST-catalysed histone acetylation and potentiates senescence in vitro and in zebrafish model of hepatocellular carcinoma. The compound opened the door to a new class of cancer therapeutics that could potentially direct the cancer cells in senescence or permanent dormancy.</p>Formule :C20H17FN2O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :384.43 g/molOxaprozin - Bio-X ™
CAS :<p>Oxaprozin is a non-steroidal anti-inflammatory drug (NSAID) used for the treatment of osteoarthritis and rheumatoid arthritis. This drug relieves swelling and inflammation by inhibiting the enzyme cyclooxygenase which in turn inhibits prostaglandin synthesis.</p>Formule :C18H15NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :293.32 g/molKV 37
CAS :<p>Inhibitor of AKR1C3 (type 5 17β-hydroxysteroid dehydrogenase)</p>Formule :C23H25NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :363.45 g/molALW-II-41-27
CAS :<p>LW-II-41-27 is a novel Eph receptor tyrosine kinase inhibitor used for cancer treatment.</p>Formule :C32H32F3N5O2SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :607.69 g/mol
