Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Mirodenafil dihydrochloride - Bio-X ™
CAS :<p>This product is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Formule :C26H37N5O5S•(HCl)2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :604.59 g/molDarapladib - Bio-X ™
CAS :<p>This product is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Formule :C36H38F4N4O2SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :666.77 g/molFlavoxate HCl - Bio-X ™
CAS :<p>Flavoxate is a muscarinic antagonist and spasmolytic drug that is used for the relief of conditions associatied with a lack of muscle control in the bladder such as urine urgency. This drug acts as a direct antagonist on acetylcholine receptors. This action reduces the tonus of smooth muscles in the bladder.</p>Formule :C24H25NO4•HClDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :427.92 g/molAG 490
CAS :<p>A tyrosine kinase inhibitor with potent activity against EGFR, STAT3, JAK3/STAT, JAK3/AP-1 and JAK3/MAPK. Suppresses IL-2 signaling pathway, inhibits T-cell growth and activation of JAK3, AP-1, STAT, MAPK. Has anti-proliferative and anti-invasive effect on cancer cells.</p>Formule :C17H14N2O3Degré de pureté :Min. 95%Couleur et forme :Yellow PowderMasse moléculaire :294.3 g/molGabexate mesylate
CAS :<p>Serine protease inhibitor</p>Formule :C17H27N3O7SDegré de pureté :Min. 95%Masse moléculaire :417.15697SB 61211 hydrochloride
CAS :<p>Nociceptin/orphanin FQ peptide receptor antagonist</p>Formule :C24H29Cl2NO·HClDegré de pureté :Min. 95%Masse moléculaire :454.86 g/molBML 257
CAS :<p>Inhibits Akt translocation by targeting the pleckstrin homology (PH) domain. Inhibits hepatitis C virus NS5B RNA-dependent RNA polymerase (IC50 = 79 µM). Attenuates cannabinoid agonist-mediated proliferation of neural stem/precursor cells.</p>Formule :C21H14N2O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :326.35 g/molRegorafenib
CAS :<p>Multi-kinase inhibitor; inhibits epoxide hydrolase; antineoplastic</p>Formule :C21H15ClF4N4O3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :482.82 g/molSU 3327
CAS :<p>SU 3327, originally introduced as a thiadiazole JNK inhibitor (De et al. 2009) has recently been identified as having antibiotic activity against a broad range of bacteria including drug-resistant gram positive and negative strains (Strokes et al. 2020). This molecule has been given the fictional name ‘Halicin’ inspired by the AI approach used to discover its novel biological activity.</p>Formule :C5H3N5O2S3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :261.31 g/molZofenopril calcium
CAS :<p>Angiotensin-converting enzyme inhibitor; antioxidant</p>Formule :C44H46N2O8S4•CaDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :899.17 g/molMG 132
CAS :<p>MG 132 is a modified tripeptide that acts as proteasomal inhibitor. In 2006, MG 132 has been experimentally tested in in vitro cell-based and in vivo models for to assess its use in the medical treatment of Parkinson's disease.</p>Formule :C26H41N3O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :475.304621-NM-PP1
CAS :<p>1-NM-PP1, also known as 1NM-PP1, is an inhibitor of the Src kinase. Studies have shown that 1-NM-PP1 inhibits analog-sensitive kinases (as-kinases) characterised by a small amino acid as gatekeeper of the ATP binding site. Tested to prevent parasitic infections, 1-NM-PP1 inhibited the Toxoplasma gondii life cycle when used at a higher concentration than 500 nM.</p>Formule :C20H21N5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :331.1797SB 271046 hydrochloride
CAS :<p>5-HT6 serotonin receptor antagonist; anti-convulsant</p>Formule :C20H22CIN3O3S2·HClDegré de pureté :Min. 95%Masse moléculaire :591.91 g/molTiludronic acid disodium
CAS :<p>Farnesyltransferase inhibitor</p>Formule :C7H9ClO6P2S•Na2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :364.59 g/molApatinib
CAS :<p>Apatinib, also known as rivoceranib, is an inhibitor of the vascular endothelial growth factor receptor 2 (VEGFR2) tyrosine kinase. Apatinib targets VEGFR2 with its action and has proven to have strong anti-tumor effects in human cancers. In studies in mice, apatinib acted as an Inhibitor of VEGFR2 and played an antiangiogenic effect. Apatinib has been suggested for the treatment of ischemia-induced proliferative retinopathy and neovascular age-related macular degeneration.</p>Formule :C24H23N5ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :397.47 g/molPitofenone hydrochloride
CAS :<p>Inhibits acetylcholinesterase (AChE); antispasmodic agent</p>Formule :C22H25NO4·ClHDegré de pureté :Min. 95%Masse moléculaire :403.9 g/molA 922500
CAS :<p>Inhibits human and mouse diacylglycerol O-acyltransferase 1 (DGAT-1) with IC50 values of 9 and 22 nM, respectively. Selective for DGAT-1 over DGAT-2 (IC50 = 53 µM), acyl coenzyme A transferase (IC50 = 296 µM) and other acyltransferases. Reduces plasma and liver triglycerides, FFA, chylomicron secretion and increases HDL cholesterol in vivo.</p>Formule :C26H24N2O4Degré de pureté :Min. 95%Masse moléculaire :428.48 g/molStaurosporine
CAS :Produit contrôlé<p>Inhibitor of protein kinases; induces apoptosis; anti-cancer</p>Formule :C28H26N4O3Degré de pureté :Min. 98 Area-%Couleur et forme :Off-White PowderMasse moléculaire :466.53 g/molTolrestat
CAS :<p>Aldose reductase AKR1B10 inhibitor; hepatotoxic</p>Formule :C16H14F3NO3SDegré de pureté :Min. 95%Masse moléculaire :357.35 g/molCyclosporin B
CAS :<p>Cyclosporin B is an antifungal and immunosuppressive cyclic peptide, which is derived from the fungus *Tolypocladium inflatum*. The compound is a member of the cyclosporin family, characterized by cyclic polypeptides with a unique arrangement of amino acids that enable its biological activity. Though its precise mode of action is not completely delineated, it is observed to influence cell growth and viability by potentially disrupting cellular communication or signal transduction pathways.</p>Formule :C61H109N11O12Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :1,188.59 g/mol
