Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Malotilate - Bio-X ™
CAS :<p>Malotilate is a pharmacological agent that is used to treat symptoms of hepatitis, bowel disease, and collagen diseases. This drug reduces collagen synthesis and cell migration activity of fibroblasts in vitro. It also has been shown to facilitate liver regeneration in rats.</p>Formule :C12H16O4S2Degré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :288.39 g/molKenpaullone
CAS :<p>Inhibitor of glycogen synthase 3 (GSK-3) and cyclin-dependent kinases CDK1, CDK2 and CDK5. Kenpaullone can substitute transcription factor Klf4 in reprogramming of fibroblast to induced pluripotent stem cells when using the method of ectopic expression of transcriptional factors. In an in vitro model for Alzheimer’s disease, kenpaullone decreased production of amyloid beta peptides Aβ40 and Aβ42.</p>Formule :C16H11BrN2ODegré de pureté :Min. 95%Couleur et forme :Yellow To Dark Yellow SolidMasse moléculaire :326.00548GSK 2606414
CAS :<p>Inhibitor of EIF2AK3/PERK kinases</p>Formule :C24H20F3N5ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :451.44 g/mol(S)-Mephenytoin - Bio-X ™
CAS :<p>(S)-Mephenytoin is a substrate of cytochrome P450 enzyme CYP2C19 (a hydroxylase). It is an effective anticonvulsant that improves control of seizures in patients. According to studies, the drug exhibits a genetic polymorphism in CYP2C19 that results in reduced metabolism in some individuals.</p>Formule :C12H14N2O2Degré de pureté :Min. 97 Area-%Couleur et forme :White PowderMasse moléculaire :218.25 g/molCA3
CAS :<p>Inhibits YAP/Tead transcriptional activity. Has anti-tumour effects on oesophageal adenocarcinoma with therapeutic potential in combination with 5-FU. Involved in ferroptosis, mediated by iron-dependent ROS.</p>Formule :C23H27N3O5S2Degré de pureté :Min. 95%Couleur et forme :White Off-White PowderMasse moléculaire :489.61 g/molEtimizol
CAS :<p>Analeptic</p>Formule :C9H14N4O2Degré de pureté :Min. 95%Masse moléculaire :210.23 g/molEtodolac - Bio-X ™
CAS :<p>Etodolac is a non-steroidal anti-inflammatory drug (NSAID) used to treat osteoarthritis and rheumatoid arthritis. It is also used to treat acute pain. This drug works by inhibiting prostaglandin synthesis from the inhibition of the enzyme cyclooxygenase.</p>Formule :C17H21NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :287.35 g/molDMAT
CAS :<p>Inhibitor of protein kinase CK2</p>Formule :C9H7Br4N3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :476.79 g/mol6-Thioguanine - Bio-X ™
CAS :<p>6-Thioguanine is a purine analog used in the therapy for leukemia and for remission consolidation in patients with acute nonlymphocytic anemia. This drug also has antimetabolite action. It replaces guanine during DNA replication. This substitution disrupts the accurate pairing of DNA bases, leading to errors in DNA replication and hinders cell division.</p>Formule :C5H5N5SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :167.19 g/molML 210
CAS :<p>Inhibitor of glutathione peroxidase GPX4</p>Formule :C22H20Cl2N4O4Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :475.32 g/molTriptolide
CAS :<p>Inhibits RNAPII-mediated trasncription; immunosuppressant; anti-inflammatory</p>Formule :C20H24O6Degré de pureté :Min. 97 Area-%Couleur et forme :PowderMasse moléculaire :360.4 g/molBRD 6989
CAS :<p>A small molecule inhibitor with high selectivity for CDK8 over CDK19. Increases IL-10 production in stimulated human and murine macrophages and dendritic cells. Modulatory action on inflammatory responses has therapeutic potential.</p>Formule :C16H16N4Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :264.33 g/molA 769662
CAS :<p>Allosteric activator of AMP-activated protein kinase (AMPK) acting on the AMPK-β subunit with therapeutic potential in metabolic disorders such as diabetes, obesity, etc. A769662 also blocks the differentiation of mouse embryonic stem cells (mESCs) and maintains the mESCs in naïve state even in the absence of leukemia inhibitory factor (2i/L).</p>Formule :C20H12N2O3SDegré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :360.39 g/molTacrolimus - Bio-X ™
CAS :<p>Tacrolimus is a calcineurin inhibitor drug that is used for the prevention of rejection after an organ transplant. This drug can also be used in the treatment of severe atopic dermatitis. Tacrolimus’ mechanism of action is not well known however it is understood that this drug inhibits T-lymphocyte activation by binding to an intracellular protein called FKBP-12. This drug also has anti-inflammatory properties.</p>Formule :C44H69NO12Degré de pureté :Min. 95%Couleur et forme :White Off-White PowderMasse moléculaire :804.02 g/molAZD 9291
CAS :<p>A potent inhibitor of EGFR with sensitizing and T790M resistance mutations, selective over the wild-type form of the receptor. Causes tumour regression in EGFR mutant T790M transgenic and xenograft models in vivo.</p>Formule :C28H33N7O2Degré de pureté :Min. 97%Couleur et forme :SolidMasse moléculaire :499.61 g/molRamipril - Bio-X ™
CAS :<p>Ramipril is an angiotensin-converting enzyme (ACE) inhibitor. It is used in the treatment of high blood pressure, congestive heart failure and other cardiovascular diseases. Ramipril inhibits the conversion of angiotensin I to angiotensin II by blocking ACE, which lowers blood pressure and reduces fluid retention.This product is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Formule :C23H32N2O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :416.51 g/molR-Rolipram
CAS :<p>Inhibitor of PDE4 enzyme; anti-inflammatory</p>Formule :C16H21NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :275.34 g/molAcalabrutinib
CAS :<p>Inhibitor of the Bruton tyrosine kinase</p>Formule :C26H23N7O2Degré de pureté :Min. 98 Area-%Couleur et forme :SolidMasse moléculaire :465.51 g/molFeprazone
CAS :<p>Anti-inflammatory; inducer of P450 II B family</p>Formule :C20H20N2O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :320.39 g/molDiacerein - Bio-X ™
CAS :<p>Diacerein is a slow-onset anthraquinone IL-1 inhibitor that is used in the treatment of joint diseases such as osteoarthritis. This drug is also being studied for the treatment of insulin resistance and diabetes mellitus. Diacerein works to decrease inflammation and cartilage destruction by reducing the level of interleukin-1.</p>Formule :C19H12O8Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :368.29 g/mol
