Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Seratrodast - Bio-X ™
CAS :Seratrodast is a thromboxane receptor antagonist that is used to treat asthma. However, this drug does not affect thrombus formation as other thromboxane synthase inhibitors do such as ozagrel.Formule :C22H26O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :354.44 g/molRebamipide - Bio-X ™
CAS :Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.Formule :C19H15ClN2O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :370.79 g/molAminopterin
CAS :Aminopterin is an antineoplastic agent and antifolate, which is a synthetic derivative of pteroylglutamic acid. It functions as a chemotherapeutic agent by inhibiting dihydrofolate reductase, an enzyme crucial in the folic acid pathway, thereby preventing the conversion of dihydrofolate to tetrahydrofolate. This disruption leads to impaired synthesis of purine nucleotides and thymidylate, which are essential for DNA synthesis and cell division.Formule :C19H20N8O5Degré de pureté :Min. 97 Area-%Couleur et forme :Slightly Yellow PowderMasse moléculaire :440.41 g/molFluvastatin sodium
CAS :Fluvastatin is a statin that lowers blood cholesterol and triglycerides by inhibiting HMG-CoA reductase, an enzyme that plays a critical role in the synthesis of cholesterol. Fluvastatin has also been shown to reduce the incidence of myocardial infarction, and to reduce atherosclerotic lesions in animal models, reducing the incidence of cardiovascular disease. Fluvastatin also has been shown to inhibit the activation of toll-like receptor 4 (TLR4) by lipopolysaccharide (LPS), which may be related to its anti-inflammatory effects. Furthermore, through lowering blood cholesterol, Fluvastatin also inhibits tubulointerstitial injury and prevents renal damage caused by high concentrations of the lipid.
Formule :C24H25FNNaO4Degré de pureté :Min. 98%Couleur et forme :Off-White PowderMasse moléculaire :433.45 g/molApixaban - Bio-X ™
CAS :Apixaban is an anticoagulant agent used for the prophylaxis of stroke and deep vein thrombosis leading to pulmonary embolism. This drug is an inhibitor of factor Xa and prothrominase. As a result, this prevents the formation of a thrombus.Formule :C25H25N5O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :459.5 g/molRosuvastatin calcium - Bio-X ™
CAS :Rosuvastatin is a drug that belongs to the group of statins. It is used for the treatment of high cholesterol and as an adjunct therapy for patients with coronary heart disease. Rosuvastatin reduces serum cholesterol by inhibiting HMG-CoA reductase, which is the rate-limiting enzyme in the production of cholesterol. Furthermore, this drug has been shown to have anti-inflammatory properties, which may be due to its ability to inhibit prostaglandin synthesis.Formule :C22H27FN3O6SCaDegré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :500.57 g/molMethotrexate sodium
CAS :Inhibitor of folate synthesis; folic acid analogueFormule :C20H22N8O5•NaxDegré de pureté :Min. 95%Masse moléculaire :476.42 g/molAfatinib - Bio-X ™
CAS :Afatinib is a small molecule that inhibits the activity of cellular kinases that are involved in the progression of cancer. It is an Irreversible inhibitor of three members of the ErbB family. This molecule binds covalently to cysteine 797 residue in HER2 and blocks downstream cellular signalling which inhibits cellular growth and promotes apoptosis. It has been researched for the treatment of non-small cell lung cancer (NSCLC), breast cancer, pancreatic cancer and colorectal cancer.Formule :C24H25ClFN5O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :485.94 g/molTenatoprazole
CAS :H+/K+ ATPase inhibitorFormule :C16H18N4O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :346.41 g/molCamostat mesylate - Bio-X ™
CAS :Camostat is a serine protease inhibitor that is used for the treatment of chronic pancreatitis. This drug has shown to reduce inflammation and pain. Studies have shown that Camostat has also inhibited the entry of SARS-CoV-2 in lung cells by inhibiting the priming process of S-protein, necessary for the viral entry into host cells.Formule :C20H22N4O5•CH4O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :494.52 g/molPentoxifylline
CAS :Produit contrôléPhosphodiesterase inhibitorFormule :C13H18N4O3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :278.31 g/mol3-(4-Phenylbutyl)-4-propyloxetan-2-one
CAS :Cis/trans-form of GK 563 [2351820-19-2]Formule :C16H22O2Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :246.34 g/molMK 4827
CAS :Inhibitor of PARP1 and PARP2 enzymes
Formule :C19H20N4ODegré de pureté :Min. 96 Area-%Couleur et forme :White PowderMasse moléculaire :320.39 g/molRucaparib camsylate
CAS :Inhibitor of poly (ADP-ribose) polymerase enzyme; antineoplasticFormule :C19H18FN3O•C10H16O4SDegré de pureté :Min. 95%Couleur et forme :Off-White To Yellow SolidMasse moléculaire :555.66 g/molDiacerein - Bio-X ™
CAS :Diacerein is a slow-onset anthraquinone IL-1 inhibitor that is used in the treatment of joint diseases such as osteoarthritis. This drug is also being studied for the treatment of insulin resistance and diabetes mellitus. Diacerein works to decrease inflammation and cartilage destruction by reducing the level of interleukin-1.Formule :C19H12O8Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :368.29 g/molCetilistat - Bio-X ™
CAS :Cetilistat is a drug that is used to treat obesity. This drug inhibits the enzyme pancreatic lipase and so it prevents triglycerides from being hydrolyzed into absorbable free fatty acids.Formule :C25H39NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :401.58 g/molBrivanib alaninate
CAS :VEGFR2 a tyrosine kinase receptor inhibitor; antineoplasticFormule :C22H24FN5O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :441.18123SU 0268
CAS :Inhibitor of 8-oxoguanine DNA glycosylase OGG1 with IC50 of 0.059 μM and excellent specificity over other DNA repair enzymes. OGG1 and its substrate 8-oxoguanine are involved in mutagenesis, genotoxicity, inflammation and cancer. The compound can cause accumulation of 8-oxoguanine in DNA in vitro and is a potent tool for the study of OGG1 biology.Formule :C26H25N3O4SDegré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :475.56 g/molArbutin - Synthetic origin
CAS :Inhibitor of tyrosinase in melanocytes: skin whitener
Formule :C12H16O7Degré de pureté :Min. 98 Area-%Couleur et forme :White PowderMasse moléculaire :272.25 g/molAtorvastatin sodium salt - Bio-X ™
CAS :Atorvastatin is an HMG-CoA reductase inhibitor which is used to lower lipid levels and to reduce the risk of cardiovascular disease. This drug belongs to the class of medicines called statins. It lowers abnormal levels of cholesterol and lipids to reduce the risk of cardiovascular disease by inhibiting the enzyme HMG-CoA.Formule :C33H35FN2O5•NaDegré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :581.63 g/mol
