Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Licofelone
CAS :<p>Dual COX/5-LO inhibitor; anti-inflammatory; analgesic</p>Formule :C23H22ClNO2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :379.88 g/molRasagiline mesylate
CAS :Produit contrôlé<p>Monoamine oxidase-B inhibitor; anti-parkinsonian; neuroprotective</p>Formule :C12H13N•CH4O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :267.35 g/molAZD 1152
CAS :<p>AZD 1152 is an Aurora kinase inhibitor, which is a type of small-molecule therapeutic agent. It is derived from the pharmaceutical research conducted by AstraZeneca. Its primary mode of action involves the selective inhibition of Aurora B kinase, an enzyme crucial for the regulation of mitosis. By interfering with this enzyme, AZD 1152 disrupts the normal progression of cell division, leading to the inhibition of proliferation and induction of apoptosis in rapidly dividing cells.</p>Formule :C26H31FN7O6PDegré de pureté :Min. 97 Area-%Couleur et forme :Slightly Yellow PowderMasse moléculaire :587.54 g/molCerivastatin sodium
CAS :<p>An inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase that reduces total cholesterol and low-density lipoprotein (LDL). Cerivastatin is cardioprotective and anti-atherosclerotic. Cerivastatin inhibits the expression of the atherosclerotic genes monocyte chemoattractant protein-1 (MCP-1) and C-C chemokine receptor type 2 (CCR2), whilst inducing the expression of Kruppel-like factor 2 (KLF2).</p>Formule :C26H33FNNaO5Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :481.53 g/molSU 11274
CAS :<p>MET tyrosine kinase inhibitor; anti-proliferative; pro-apoptotic</p>Formule :C28H30ClN5O4SDegré de pureté :Min. 95%Couleur et forme :Yellow To Orange SolidMasse moléculaire :568.09 g/molOmeprazole - Bio-X ™
CAS :<p>Omeprazole is a proton pump inhibitor (PPI) that inhibits the production of gastric acid in the stomach. This is due to Omeprazole binding through a stable disulphide bond to the H+/K+ ATPase enzyme found on parietal cells, and preventing hydrogen ion transport. Consequently, gastric acid secretion is supressed. As a PPI, Omerprazole can be used to treat disorders where gastric acid is over-secreted. Examples of these disorders are gastroesophageal reflux disease (GERD) and peptic ulcer disease.</p>Formule :C17H19N3O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :345.42 g/molAceclofenac - Bio-X ™
CAS :<p>Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.</p>Formule :C16H13Cl2NO4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :354.18 g/molRivastigmine tartrate - Bio-X ™
CAS :Produit contrôlé<p>Rivastigmine is a cholinergic agent that is used in the treatment of dementia in Parkinson’s and Alzheimer’s disease. This drug is a carbamate derivative that binds to and inactivates cholinesterase such as acetylcholinesterase and butyrylcholinesterase. This leads to an increase concentration of acetylcholine at cholinergic synapse.</p>Formule :C14H22N2O2•C4H6O6Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :400.42 g/molTideglusib
CAS :<p>An irreversible GSK-3β inhibitor that reduces phosphorylation of tau proteins, protects from neuronal loss and has cognitive and behavioural benefits in murine models. Studied for its potential as a therapeutic agent in Alzheimer’s disease and other neurodegenerative diseases. Tideglusib was also shown to inhibit the main protease Mpro from the SARS-CoV-2 virus with IC50 of 1.55 μM.</p>Formule :C19H14N2O2SDegré de pureté :Min. 95%Couleur et forme :White To Off-White SolidMasse moléculaire :334.39 g/molChymostatin
CAS :<p>Inhibitor of chymotrypsin</p>Formule :C31H41N7O6Couleur et forme :White To Yellowish SolidMasse moléculaire :607.7 g/molBAY 607550
CAS :<p>A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.</p>Formule :C27H32N4O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :476.24236Zotarolimus
CAS :<p>Inhibitor of immunophilin FKBP12 and mTOR signalling with immunosuppressant activity. Zotarolimus inhibits proliferation of endothelial cells and smooth muscle cells and is employed in vascular interventional therapies.</p>Formule :C52H79N5O12Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :966.21 g/molRebamipide - Bio-X ™
CAS :<p>Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.</p>Formule :C19H15ClN2O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :370.79 g/molAG 120
CAS :<p>Inhibits isocitrate dehydrogenase 1 (IDH-1) harbouring a gain of function mutation at R132, which causes impaired cellular differentiation via epigenetic modulation. By inhibiting mutant IDH1, synthesis of oncometabolite 2-hydroxyglutarate is reduced. This compound therefore has therapeutic potential in solid and haematological malignancies, such as acute myeloid leukemia (AML).</p>Formule :C28H22ClF3N6O3Degré de pureté :Min. 95%Couleur et forme :White To Off-White SolidMasse moléculaire :582.96 g/molGilteritinib
CAS :<p>Inhibitor of FLT3 and AXL tyrosine kinases</p>Formule :C29H44N8O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :552.71 g/molXMU MP 2
CAS :<p>BRK tyrosine kinase (PTK6) inhibitor; anti-proliferative in breast cancer cells</p>Formule :C32H33F3N8O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :618.65 g/molCZC 25146
CAS :<p>Inhibitor of leucine-rich repeat kinase LRRK2Â</p>Formule :C22H25FN6O4SDegré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :488.54 g/molLovastatin - Bio-X ™
CAS :<p>Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.</p>Formule :C24H36O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :404.54 g/molMRK 560
CAS :<p>γ-secretase inhibitor; reduces amyloid-β in brainÂ</p>Formule :C19H17ClF5NO4S2Degré de pureté :Min. 95%Masse moléculaire :517.92 g/molApremilast - Bio-X ™
CAS :<p>Apremilast is the commercial name of a phosphodiesterase-4 (PDE4) inhibitor developed to treat chronic inflammatory disorders. Similarly to thalidomide, the apremilast molecule carries a phthalimide ring, but it lacks however the glutarimide ring needed to bind to cereblon, specifically targeted by thalidomide. As a drug, apremilast is indicated for the treatment of psoriasis and psoriatic arthritis.</p>Formule :C22H24N2O7SDegré de pureté :Min. 99 Area-%Couleur et forme :White/Off-White SolidMasse moléculaire :460.5 g/mol
