Meptazinol

CAS : 54340-58-8

Ref. 3D-ECA34058

Informations sur le produit

• Nom: Meptazinol
• Synonymes: 1-Methyl-3-ethyl-3-(m-hydroxyphenyl)hexahydro-1H-azepine, 259-109-9, 3-(3-Ethyl-1-Methylazepan-3-Yl)Phenol, 3-(3-Ethylhexahydro-1-methyl-1H-azepin-3-yl)phenol, 4-(3-Ethyl-1-Methyl-Azepan-3-Yl)Phenol, 54340-58-8, Meptamizol, phenol, 3-(3-ethylhexahydro-1-methyl-1H-azepin-3-yl)-

Description

Meptazinol is a centrally acting analgesic that inhibits the synthesis of prostaglandins in the central nervous system. It is an ester hydrochloride that has been studied pharmacokinetically and molecularly docked to the cholinergic receptor. Meptazinol has shown to be highly effective in geriatric patients, with a more rapid onset of action than morphine and similar duration of effect. The drug also has a lower incidence of side effects, such as sedation and respiratory depression, which are common with opioid drugs. Meptazinol is chemically stable under acidic conditions, but decomposes at higher pH levels due to its amine group. Biological properties have been determined using the LC-MS/MS method on rat brain tissue samples, showing that meptazinol binds to receptors for opioids with high affinity and selectivity.

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 233.35 g/mol
• Formule: C₁₅H₂₃NO
• Degré de pureté: Min. 95%