6-Bromoimidazo[1,2-a]pyrazine

CAS : 912773-24-1

Ref. 3D-FB140690

Informations sur le produit

• Nom: 6-Bromoimidazo[1,2-a]pyrazine
• Synonymes: 6-Bromoimidazo[1,2-A]Pyrazine

Description

6-Bromoimidazo[1,2-a]pyrazine is a potent inhibitor of the enzyme phosphatidylinositol-3 kinase (PI3K). It has been used in drug development and has shown to be a reversible inhibitor of PI3K. 6-Bromoimidazo[1,2-a]pyrazine binds to the ATP site on the enzyme and prevents phosphorylation by blocking access to this site. The binding of 6-bromoimidazo[1,2-a]pyrazine is reversible due to its ability to dissociate when ATP is removed. This drug has been shown to inhibit the growth of cancer cells in vitro.

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 198.02 g/mol
• Formule: C₆H₄BrN₃
• Degré de pureté: Min. 95%
• InChI: InChI=1S/C6H4BrN3/c7-5-4-10-2-1-8-6(10)3-9-5/h1-4H
• Code InChI: InChIKey=KKMWDXNBIKMCEH-UHFFFAOYSA-N
• SMILES: Brc1cn2ccnc2cn1