Eledoisin acetate salt

CAS : 69-25-0

Ref. 3D-FE108742

Informations sur le produit

• Nom: Eledoisin acetate salt
• Synonymes: Pyr-Pro-Ser-Lys-Asp-Ala-Phe-Ile-Gly-Leu-Met-NH2, 5-Oxoprolylprolylseryllysyl-Alpha-Aspartylalanylphenylalanylisoleucylglycylleucylmethioninamide, 5-oxo-L-prolyl-L-prolyl-L-seryl-L-lysyl-L-alpha-aspartyl-L-alanyl-L-phenylalanyl-L-isoleucylglycyl-L-leucyl-L-methioninamide

Description

Eledoisin acetate salt is a cell-lysing agent that belongs to the group of potent antagonists. It is an inhibitor of neurokinin-1 receptor which regulates the release of substance P and other inflammatory mediators from nerve terminals. Eledoisin acetate salt has shown to inhibit locomotor activity in rats, as well as nucleotide levels in cells. This drug also has been shown to have carcinoid syndrome-like effects, such as weight loss and diarrhea. These symptoms are caused by the inhibition of substance P at its receptors. The tumor necrosis factor (TNF) may be responsible for these effects, since it causes increased production of substance P in cells.

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 1,188.4 g/mol
• Formule: C₅₄H₈₅N₁₃O₁₅S·xC₂H₄O₂
• Degré de pureté: Min. 95%