(-)-9-Hydroxyrisperidone

CAS : 147663-01-2

Ref. 3D-IH24118

Informations sur le produit

• Nom: (-)-9-Hydroxyrisperidone
• Synonymes: (9S)-3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4 -one(S)-9-Paliperidone, R 078544, 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv., 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-, (9S)-, (9S)-3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one

Description

(-)-9-Hydroxyrisperidone is a metabolite of risperidone that is structurally related to the neurotransmitter dopamine. This compound has been found to be a potent antagonist of serotonin and adrenergic receptors, which may contribute to its therapeutic effects in schizophrenia. (-)-9-Hydroxyrisperidone also has been shown to have a high affinity for human liver plasma proteins, which suggests it may be responsible for the long half-life seen with risperidone. The (+) form of the drug has been shown to be more potent than (-)-9-hydroxyrisperidone, while (-)-9-hydroxyrisperidone is more selective in terms of receptor binding.

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 426.48 g/mol
• Formule: C₂₃H₂₇FN₄O₃
• Degré de pureté: Min. 95%
• Couleur/Forme: Powder