(2R)-2-(5-Fluoro-2-hydroxyphenyl)-2-{1-oxo-6-[4-(piperazin-1-yl)phenyl]-1,3-dihydro-2H-isoindol-2-yl}-N-(1,3-thiazol-2-yl)acetamide

CAS : 2060610-53-7

Ref. 3D-KHD61053

Informations sur le produit

• Nom: (2R)-2-(5-Fluoro-2-hydroxyphenyl)-2-{1-oxo-6-[4-(piperazin-1-yl)phenyl]-1,3-dihydro-2H-isoindol-2-yl}-N-(1,3-thiazol-2-yl)acetamide

Description

(2R)-2-(5-Fluoro-2-hydroxyphenyl)-2-{1-oxo-6-[4-(piperazin-1-yl)phenyl]-1,3-dihydro-2H-isoindol-2-yl}-N-(1,3-thiazol-2-yl)acetamide is a peptide that belongs to the class of inhibitors. It has been shown to inhibit ion channels in cells. The compound has an IC50 of about 0.25 μM for the hERG channel and shows no activity against other ion channels tested such as NMDA, GABA A , and Na V 1.8. (2R)-2-(5 -fluoro-- 2 -hydroxyphenyl)-2-[1 -oxo-- 6 - (4-- piperazin-- 1-- ylphenyl)-- 1,3 -dihydro-- 2H

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 543.6 g/mol
• Formule: C₂₉H₂₆FN₅O₃S
• Degré de pureté: Min. 95%