(±)-WS 75624b

CAS : 188048-45-5

Ref. 3D-NHA04845

Informations sur le produit

• Nom: (±)-WS 75624b
• Synonymes: Ws-75624B

Description

(±)-WS 75624b is a potent and selective activator of the human serotonin 5-HT2C receptor. The binding affinity of (±)-WS 75624b to the human serotonin 5-HT2C receptor was determined by measuring the Ki value with radioligand binding assays using [3H]-mesulergine as the radioligand. The Ki value for (±)-WS 75624b was determined to be 0.8 nM, which is in good agreement with the Ki values reported for other serotonin 5-HT2C receptor agonists.

(±)-WS 75624b binds to the serotonin 5-HT2C receptor with high affinity and selectivity, and it has been shown to activate this receptor in a number of cell types. It has been found to inhibit voltage-gated potassium currents in rat dorsal root ganglion neurons and also inhibits glutamate release from cultured rat cortical cells. These properties make

• Marque: Biosynth

Propriétés chimiques

• Masse moléculaire: 380.5 g/mol
• Formule: C₁₈H₂₄N₂O₅S
• Degré de pureté: Min. 95%