N-Methylcytisine

CAS : 486-86-2

Ref. TM-T5S0994

Informations sur le produit

• Nom: N-Methylcytisine
• Synonymes: Caulophylline, (1R)-11-Methyl-7,11-diazatricyclo[7.3.1.0~2,7~]trideca-2,4-dien-6-one, (1R)-3-methyl-1,2,3,4,5,6-hexahydro-8H-1,5-methanopyrido[1,2-a][1,5]diazocin-8-one, (1R,5S)-1,2,3,4,5,6-Hexahydro-3-methyl-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one, (1S,5S)-3-methyl-1,2,3,4,5,6-hexahydro-8H-1,5-methanopyrido[1,2-a][1,5]diazocin-8-one, 1,2,3,4,5,6-Hexahydro-3-methyl-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one, 1,5-Methano-8H-pyrido[1,2-a][1,5]diazocin-8-one, 1,2,3,4,5,6-hexahydro-3-methyl-, (1R,5S)-, 1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one, 1,2,3,4,5,6-hexahydro-3-methyl-, 1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one, 1,2,3,4,5,6-hexahydro-3-methyl-, (1R)-, 3-Methylcytisine, 3-methyl-1,2,3,4,5,6-hexahydro-8H-1,5-methanopyrido[1,2-a][1,5]diazocin-8-one, Caulophyllin, Cytisine, 12-methyl-, Cytisine, N-methyl-, Cytisine, methyl-, N-methylcytisine
• CAS: 486-86-2

Description

1. N-Methylcytisine (Caulophylline)'s nicotinic receptors have high affinity (KD = 5 nM)to nAChR from squid optical ganglia. 2. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).

• Marque: Targetmol

Propriétés chimiques

• Masse moléculaire: 204.27
• Formule: C₁₂H₁₆N₂O
• Degré de pureté: 99.83%
• Couleur/Forme: Solid
• InChI: InChI=1S/C12H16N2O/c1-13-6-9-5-10(8-13)11-3-2-4-12(15)14(11)7-9/h2-4,9-10H,5-8H2,1H3
• Code InChI: InChIKey=CULUKMPMGVXCEI-UHFFFAOYSA-N
• SMILES: CN1CC2CC(C1)c1cccc(=O)n1C2