(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

CAS : 73168-24-8

Ref. TM-TP2136

Informations sur le produit

• Nom: (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
• Synonymes: (d(CH-2)51,Tyr(Me)2,Arg8)-Vasopressin, 3-Mercapto-3-Methyl-Butyryl-Tyr(Me)-Phe-Gln-Asn-Cys-Pro-Arg-Gly-Nh2, Vasopressin, 1-(1-mercaptocyclohexaneacetic acid)-2-(O- methyl-L-tyrosine)-8-L-arginine-, (beta-Mercapto-beta,beta-cyclopentamethylene-propionyl(sup 1),O-Me-Tyr(sup 2),Arg(sup 8))-vasopressin, (d(CH2)5(1)-O-Me-Tyr(2)-arg(8))vasopressin, 1-(beta-Mercapto-beta,beta-cyclopentamethylenepropionic acid)-2-(O-methyl-tyr)-argipressin, 1-(beta-Mercapto-beta,beta-cyclopentamethylenepropionic acid)-2-O-methyltyrosyl-8-arginine vasopressin, Aavp, Avpa, Arginine vasopressin, beta-mercapto-(beta,beta-cyclopentamethylenepropionic acid)(1)-methyl-tyr(2)-, Argipressin, (beta-mercapto)beta,beta-cyclopentamethylenepropionic acid(1)-O-methyl-tyr(2)-, Cgp 25838, Cpg 25838E, Manning compound, Mcppa-avp, Sk&F 100273, Skf 100273, d(CH2)5(Tyr(Me)(2))AVP, d(CH2)5-Tyr(Me)argipressin, d(CH2)5Tyr(Me)AVP, Glycinamide, N-((1-mercaptocyclohexyl)acetyl)-O-methyl-L-tyrosyl-L-phenylalanyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-arginyl-, cyclic (1-5)-disulfide, 1-{[(10S,13S,16S,19R,22S)-13-(2-amino-2-oxoethyl)-16-(3-amino-3-oxopropyl)-19-benzyl-22-(4-methoxybenzyl)-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacos-10-yl]carbonyl}-L-prolyl-N~5~-(diaminomethylidene)ornithylglycinamide
• CAS: 73168-24-8

Description

Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.

• Marque: Targetmol

Propriétés chimiques

• Masse moléculaire: 1151.38
• Formule: C₅₂H₇₄N₁₄O₁₂S₂
• Degré de pureté: 98%
• Couleur/Forme: White Lyophilized Powder