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Se termine le 31 déc.( plus que 10 jours )
HRO761
CAS :HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.Formule :C31H31ClF3N9O5Degré de pureté :98.74% - 99.62%Couleur et forme :SolidMasse moléculaire :702.08Werner syndrome RecQ helicase-IN-2
CAS :Werner syndrome RecQ helicase-IN-2 is a potent Werner syndrome RecQ DNA helicase (WRN) inhibitor, useful in research on colorectal and gastric cancers.Formule :C32H34F3N9O5Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :681.67Werner syndrome RecQ helicase-IN-3
CAS :Potent WRN inhibitor, Werner syndrome RecQ helicase-IN-3, is orally active with 0.06 µM IC50; exhibits antiproliferative and anticancer effects.Formule :C31H30ClF3N8O5Couleur et forme :SolidMasse moléculaire :687.07Tyr-Gly-Gly-Phe-Met-OH
CAS :<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formule :C27H35N5O7SDegré de pureté :≥95%Couleur et forme :White Lyophilised SolidMasse moléculaire :573.66Werner syndrome RecQ helicase-IN-4
CAS :Werner syndrome RecQ helicase-IN-4 is a WRN inhibitor with anticancer and anti-proliferative activity, used in colorectal and gastric cancer research.Formule :C32H33F3N8O5Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :666.65Clozapine N-oxide dihydrochloride
CAS :Clozapine N-oxide dihydrochloride is a derivative of Clozapine and an agonist of DREADDs.Formule :C18H21Cl3N4ODegré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :415.746-Aminocaproic acid hydrochloride
CAS :6-Aminocaproic acid HCl: Potent oral antifibrinolytic; blocks plasminogen binding; used for bleeding disorder research.Formule :C6H14ClNO2Couleur et forme :SolidMasse moléculaire :167.6345-Iminodaunorubicin hydrochloride
CAS :<p>5-Iminodaunorubicin HCl: quinone-modified anthracycline with antitumor properties, induces DNA breaks in cancer cells.</p>Formule :C27H31ClN2O9Couleur et forme :SolidMasse moléculaire :563.004-Chloro Trazodone hydrochloride
CAS :4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Formule :C19H23Cl2N5OCouleur et forme :SolidMasse moléculaire :408.32Delavirdine mesylate
CAS :<p>Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).</p>Formule :C23H32N6O6S2Degré de pureté :99.99%Couleur et forme :Light Brown SolidMasse moléculaire :552.67Guanosine 5'-diphosphate sodium
CAS :Guanosine 5'-diphosphate (GDP) sodium is a nucleoside diphosphate known for activating the adenosine 5'-triphosphate-sensitive K+ channel and serving as aFormule :C10H14N5NaO11P2Couleur et forme :SolidMasse moléculaire :465.18Tetrahydroxyquinone monohydrate
CAS :<p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>Formule :C6H6O7Couleur et forme :SolidMasse moléculaire :190.11Carbonic anhydrase inhibitor 12
CAS :<p>CA Inhibitor 12 strongly blocks CA II (K_i 1.72 nM), also inhibits CA I (271 nM), shows anticancer effects.</p>Formule :C27H22BrN5O5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :640.53Cap-dependent endonuclease-IN-7
CAS :Cap-dependent endonuclease-IN-7, a potent CEN inhibitor, blocks viral mRNA synthesis and virus spread, with research use for influenza A, B, C.Formule :C36H28FN3O7SCouleur et forme :SolidMasse moléculaire :665.69D,L-erythro-PDMP hydrochloride
CAS :D,L-erythro-PDMP hydrochloride, an isomer of PDMP, inhibits rabbit fibroblast growth and glucosyltransferase.Formule :C23H39ClN2O3Couleur et forme :SolidMasse moléculaire :427.02Delavirdine
CAS :<p>Delavirdine, an NNRTI for HIV-1, is used in HAART.</p>Formule :C22H28N6O3SCouleur et forme :SolidMasse moléculaire :456.56Demecarium bromide
CAS :<p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>Formule :C32H52Br2N4O4Degré de pureté :98%Couleur et forme :White Powder SolidMasse moléculaire :716.59Asterriquinol D dimethyl ether
CAS :<p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>Formule :C26H24N2O4Couleur et forme :SolidMasse moléculaire :428.48Anti-Trypanosoma cruzi agent-4
CAS :<p>Anti-Trypanosoma cruzi Agent-4 is a Trypanosoma cruzi inhibitor utilized for the investigation of infections caused by this parasite.</p>Formule :C17H16N2O3Couleur et forme :SolidMasse moléculaire :296.32(1s,4s)-Menin-MLL inhibitor-23
<p>(1s,4s)-Menin-MLL Inhibitor-23, an enantiomer of Menin-MLL Inhibitor-23 (Example 99A), functions as an inhibitor of the menin-MLL interaction [1].</p>Formule :C36H53FN6O4Couleur et forme :SolidMasse moléculaire :652.84Glutaminyl Cyclase Inhibitor 5
Glutaminyl Cyclase Inhibitor 5 is a potent, selective inhibitor of human glutaminyl cyclase (hQC), demonstrating an inhibition concentration half-max (IC 50) ofFormule :C22H30N6OCouleur et forme :SolidMasse moléculaire :394.51Mitochondrial respiration-IN-3
Mitochondrial respiration-IN-3, a cell-permeable fluorine derivative of Dalfopristin, inhibits glioblastoma stem cell translation for cancer research.Formule :C35H51FN4O7SCouleur et forme :SolidMasse moléculaire :690.87Mitochondrial respiration-IN-2
CAS :Mitochondrial respiration-IN-2, a fluorinated Virginiamycin M1, inhibits glioblastoma stem cell mitochondrial translation.Formule :C28H36FN3O6Couleur et forme :SolidMasse moléculaire :529.60TEPP-46
CAS :<p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C17H16N4O2S2Degré de pureté :98.21% - 98.77%Couleur et forme :SolidMasse moléculaire :372.46Ceftobiprole medocaril sodium
CAS :Ceftobiprole medocaril sodium (BAL5788) is a prodrug of broad-spectrum cephalosporin active against MRSA, VRSA, and resistant streptococci.Formule :C26H25N8NaO11S2Couleur et forme :SolidMasse moléculaire :712.64Velagliflozin proline hydrate
CAS :Velagliflozin proline hydrate, an oral SGLT2 inhibitor, reduces blood sugar by inhibiting renal glucose reabsorption.Formule :C28H36N2O8Couleur et forme :SolidMasse moléculaire :528.596-trans-12-epi-Leukotriene B4
CAS :<p>6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47Montelukast dicyclohexylamine
CAS :Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.Formule :C47H59ClN2O3SCouleur et forme :SolidMasse moléculaire :767.5Loxoprofenol-SRS tromethamine
CAS :Loxoprofenol-SRS tromethamine (HR1405-01), a metabolite of Loxoprofen, is a safe IV NSAID with strong anti-inflammatory and pain relief properties.Formule :C19H31NO6Couleur et forme :SolidMasse moléculaire :369.45Phosphoglycolohydroxamic acid
CAS :Phosphoglycolohydroxamic acid inhibits aldolase/triose-phosphate isomerase; used in antibacterial/antifungal research.Formule :C2H6NO6PCouleur et forme :SolidMasse moléculaire :171.05p-Aminophenylmercuric acetate
CAS :<p>p-Aminophenylmercuric acetate (APMA) is an organic mercury compound and thiol-blocking agent commonly employed as an activator of MMPs .</p>Formule :C8H9HgNO2Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :351.75NM107
CAS :NM107, a ribonucleoside, inhibits HCV NS5B polymerase. It has broad antiviral properties with EC50 of 1.85 μM in wild-type cells.Formule :C10H15N3O5Degré de pureté :97.85%Couleur et forme :White To Off-White PowderMasse moléculaire :257.24Eicosapentaenoic Acid sodium
CAS :<p>EPA sodium, an oral omega-3, demethylates DNA, reactivates tumor suppressors, and induces vasodilation.</p>Formule :C20H29NaO2Couleur et forme :SolidMasse moléculaire :324.43Topoisomerase IV inhibitor 1
CAS :<p>Compound 7d: Inhibits TOPO IV (IC50: 0.23 μM), DNA gyrase (IC50: 0.43 μM), antibacterial against S. aureus (MIC: 0.972 μM), E. coli (MIC: 0.608 μM).</p>Formule :C34H32FN7O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :685.72Topoisomerase IV inhibitor 2
CAS :<p>Compound 5d, a potent TOPO IV inhibitor (IC50: 0.35 μM), also inhibits DNA gyrase (IC50: 0.55 μM) and has antibacterial activity.</p>Formule :C33H30FN7O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :671.7(Rac)-3′-Hydroxy simvastatin
CAS :(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.Formule :C25H38O6Couleur et forme :SolidMasse moléculaire :434.57Difluorocyclooctyne-CH2-COOH
CAS :Difluorocyclooctyne-CH2-COOH is a DIFO analogue for live-cell glycan imaging, reacting swiftly with azides sans copper catalysts.Formule :C10H12F2O2Couleur et forme :SolidMasse moléculaire :202.2Topoisomerase II inhibitor 7
CAS :Topoisomerase II inhibitor 7 halts cell division and induces apoptosis, targeting topoisomerase II alpha with a 3.19 μM IC50.Formule :C32H28BrN5O5SCouleur et forme :SolidMasse moléculaire :674.56Mirogabalin
CAS :<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Formule :C12H19NO2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :209.28HIV-1 integrase inhibitor 10
HIV-1 integrase inhibitor 10: oral ALLINI, blocks NLRepRluc virus in MT-2 cells, EC50 of 3-5 nM, used in HIV-1 research.Formule :C40H45N7O4Couleur et forme :SolidMasse moléculaire :687.83Enpp/Carbonic anhydrase-IN-2
Enpp/Carbonic anhydrase-IN-2: A potent inhibitor (IC50: 1.13-0.33 µM) for NPP1-3, CA-IX/XII; anti-cancer, low toxicity, induces apoptosis.Formule :C23H24FNO4SCouleur et forme :SolidMasse moléculaire :429.5Xanthine oxidoreductase-IN-3
CAS :<p>Xanthine oxidoreductase-IN-3, an oral XOR inhibitor with IC50 of 26.3 nM, is useful for acute hyperuricemia research.</p>Formule :C14H10ClN5ODegré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :299.72Xanthine oxidoreductase-IN-5
CAS :Xanthine oxidoreductase-IN-5: oral XOR inhibitor; IC50 55 nM; for acute hyperuricemia research.Formule :C17H17N5O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :323.35Tubulin polymerization-IN-39
<p>Tubulin-IN-39 inhibits polymerization (IC50: 4.9 μM), blocks colchicine site, stops cancer growth.</p>Formule :C21H21N5O5Couleur et forme :SolidMasse moléculaire :423.42Tubulin polymerization-IN-40
CAS :Tubulin Polymerization-IN-40, an acridane inhibitor; IC50 1.5 μM; blocks cell division, induces apoptosis, has anti-cancer and immune-boosting effects.Formule :C24H22FNO5Couleur et forme :SolidMasse moléculaire :423.1482Bexagliflozin
CAS :<p>Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.</p>Formule :C24H29ClO7Degré de pureté :98.99% - 99.89%Couleur et forme :SolidMasse moléculaire :464.94NaV1.2/1.6 channel blocker-1
CAS :<p>NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.</p>Formule :C14H14N2OSDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :258.344,6-O-Ethylidene-α-D-glucose
CAS :<p>4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucose</p>Formule :C8H14O6Couleur et forme :SolidMasse moléculaire :206.19Marbofloxacin hydrochloride
CAS :Marbofloxacin HCl: 3rd-gen oral fluoroquinolone, broad-spectrum antibacterial against Gram-positive/negative and Mycoplasma.Formule :C17H20ClFN4O4Couleur et forme :SolidMasse moléculaire :398.82Oxyphenbutazone monohydrate
CAS :<p>Oxyphenbutazone monohydrate: Phenylbutazone derivative, anti-inflammatory, non-selective COX inhibitor, kills dormant M. tuberculosis.</p>Formule :C19H22N2O4Couleur et forme :SolidMasse moléculaire :342.39Endomorphin 2
CAS :<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Formule :C32H37N5O5Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :571.67Acetyl-CoA Carboxylase-IN-1
CAS :Acetyl-CoA Carboxylase-IN-1 (ACC-IN-1) is a potent acetyl-CoA carboxylase (ACC) inhibitor with antibacterial activity, used in metabolic disease research.Formule :C13H9Br2N5Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :395.05P-CAB agent 2 hydrochloride
CAS :P-CAB agent 2 hydrochloride is a strong oral gastric acid secretion inhibitor with IC50 <100 nM on H+/K+ ATPase and 18.69 µM on hERG channel, non-toxic.Formule :C22H26ClFN2O4SCouleur et forme :SolidMasse moléculaire :468.97Combretastatin A1 phosphate
CAS :Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.Formule :C18H22O12P2Couleur et forme :SolidMasse moléculaire :492.31Tariquidar dihydrochloride
CAS :Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).Formule :C38H40Cl2N4O6Couleur et forme :SolidMasse moléculaire :719.65Nicotinamide Hydrochloride
CAS :<p>Nicotinamide Hydrochloride, a vitamin B3 form, inhibits SIRT2 and melanoma growth, enhancing NAD+, ATP, ROS, and survival in melanoma mice.</p>Formule :C6H7ClN2OCouleur et forme :SolidMasse moléculaire :158.59Flecainide acetate
CAS :<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formule :C19H24F6N2O5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :474.39Trypsin Inhibitor, soybean
CAS :<p>Trypsin Inhibitor, soybean is a trypsin inhibitor extracted from leguminous plants.</p>Couleur et forme :SolidAntiproliferative agent-20
CAS :Antiproliferative agent-20: potent oral anticancer drug with anti-angiogenic properties.Formule :C23H18N2O6Couleur et forme :SolidMasse moléculaire :418.4Octenyl succinic anhydride
CAS :OSA modifies starch into amphiphilic OS-starch, affecting intermolecular interactions.Formule :C12H18O3Couleur et forme :SolidMasse moléculaire :210.27KCa1.1 channel activator-1
A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.Formule :C25H16O10Couleur et forme :SolidMasse moléculaire :476.39KCa1.1 channel activator-2
<p>KCa1.1 channel activator-2, a Quercetin hybrid, selectively stimulates vascular KCa1.1 channel, with strong myorelaxant effects.</p>Formule :C23H22O8S2Couleur et forme :SolidMasse moléculaire :490.55P2X7 receptor antagonist-3
CAS :P2X7 receptor antagonist-3 is a powerful inhibitor of the P2X7 receptor, exhibiting IC50 values of 4.2 nM in humans and 6.8 nM in rats, indicating its highFormule :C17H12ClF3N6OCouleur et forme :SolidMasse moléculaire :408.77Antiproliferative agent-10
Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.Formule :C35H36Cl2N7PRuCouleur et forme :SolidMasse moléculaire :757.66Prohydrojasmon racemate
CAS :<p>Prohydrojasmon racemate (Propyl dihydrojasmonate) is a synthesized plant gowth regulator, which has jasmonic acid activity.</p>Formule :C15H26O3Degré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :254.37Antiproliferative agent-11
Antiproliferative agent-11, a Ruthenium(II) complex, targets multiple cancers with IC50s of 6-10 μM.Formule :C31H34Cl2N6O3P2RuCouleur et forme :SolidMasse moléculaire :772.56Pyridostatin hydrochloride
CAS :Pyridostatin hydrochloride stabilizes G-quadruplex DNA (Kd=490nM), inhibits cancer cell growth, and reduces SRC in breast cancer.Formule :C31H37Cl5N8O5Couleur et forme :SolidMasse moléculaire :778.94Anti-inflammatory agent 33
CAS :Agent 33: potent p38α inhibitor, reduces NO, iNOS, COX-2, p-p38α, p-MK2; shows anti-inflammatory effects.Formule :C22H15N3O5SCouleur et forme :SolidMasse moléculaire :433.44Reverse transcriptase-IN-3
<p>Reverse transcriptase-IN-3, a pyrimidine carboxamide, inhibits HIV-1 including mutant strains.</p>Formule :C28H31N7O4SCouleur et forme :SolidMasse moléculaire :561.66Antiproliferative agent-17
CAS :Antiproliferative Agent-17 exhibits both antimicrobial properties against Gram-positive bacteria and anticancer activity [1].Formule :C26H28N2OSCouleur et forme :SolidMasse moléculaire :416.58Antiproliferative agent-19
Antiproliferative agent-19 induces apoptosis and G2/M cell cycle arrest in lung cancer cells.Formule :C26H23NOCouleur et forme :SolidMasse moléculaire :365.47Reverse transcriptase-IN-4
<p>Reverse transcriptase-IN-4: potent, selective NNRT inhibitor; EC50 = 0.053 μM for HIV-1, 0.26 μM for E138K mutant.</p>Formule :C17H21N5OSCouleur et forme :SolidMasse moléculaire :343.45Larotinib mesylate hydrate
CAS :Larotinib mesylate hydrate is a potent, broad-spectrum, and orally active tyrosine kinase inhibitor (TKI), primarily targeting EGFR with an IC50 value of 0.6 nMFormule :C26H36ClFN4O11S2Couleur et forme :SolidMasse moléculaire :699.171-Dehydro-[10]-gingerdione
CAS :<p>1-Dehydro-[10]-gingerdione blocks IKKβ, curbs IκBα phosphorylation, halts NF-κB activity, and aids inflammation research.</p>Formule :C21H30O4Couleur et forme :SolidMasse moléculaire :346.46(R,R)-Reboxetine mesylate
CAS :<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Formule :C20H27NO6SCouleur et forme :SolidMasse moléculaire :409.5Satraplatin
CAS :Satraplatin (BMS182751) is an orally available antineoplastic platinum(IV) complex.Satraplatin has a favorable toxicity profile and appears to have clinicalFormule :C10H22Cl2N2O4PtDegré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :500.28Sotuletinib hydrochloride
CAS :Sotuletinib hydrochloride (BLZ945 HCl) is a selective, brain-penetrant CSF-1R (c-Fms) inhibitor (IC50=1 nM),for ALS and TNBC.Formule :C20H23ClN4O3SDegré de pureté :98.812%Couleur et forme :SolidMasse moléculaire :434.94Diamthazole hydrochloride
CAS :Diamthazole (Dimazole) hydrochloride, an antifungal agent, is utilized in infection research.Formule :C15H24ClN3OSCouleur et forme :SolidMasse moléculaire :329.89Efonidipine hydrochloride
CAS :Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.Formule :C34H39ClN3O7PCouleur et forme :SolidMasse moléculaire :668.12CTX-0294885 hydrochloride
CTX-0294885 hydrochloride inhibits 235 kinases, affects AKT family, and aids in studying kinome-related diseases.Formule :C22H25Cl2N7OCouleur et forme :SolidMasse moléculaire :474.39Lesogaberan hydrochloride
Lesogaberan (AZD-3355) HCl: selective GABA B agonist, EC50 8.6 nM, K i 5.1 nM (rat GABA B), 1.4 μM (GABA A), reduces esophageal relaxation.Formule :C3H10ClFNO2PCouleur et forme :SolidMasse moléculaire :177.54DPM-1001 trihydrochloride
DPM-1001 trihydrochloride: Potent PTP1B inhibitor, IC50 100 nM, oral, non-competitive, anti-diabetic.Formule :C35H60Cl3N3O3Couleur et forme :SolidMasse moléculaire :677.23Altretamine hydrochloride
CAS :Altretamine hydrochloride is an alkylating antineoplastic agent.Formule :C9H19ClN6Couleur et forme :SolidMasse moléculaire :246.74ATM-3507 trihydrochloride
CAS :ATM-3507 trihydrochloride, a potent inhibitor of tropomyosin, demonstrates inhibition concentration (IC50) values ranging from 3.83 to 6.84 μM across variousFormule :C37H49Cl3FN5O2Couleur et forme :SolidMasse moléculaire :721.17GS-441524
CAS :GS-441524 treatment of cats with naturally occurring feline infectious peritonitis.Formule :C12H13N5O4Degré de pureté :98.78% - 99.75%Couleur et forme :SolidMasse moléculaire :291.26DSP-1053 benzenesulfonate
CAS :DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.Formule :C32H38BrNO7SCouleur et forme :SolidMasse moléculaire :660.62PF-06815345 hydrochloride
CAS :<p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>Formule :C27H30Cl2FN9O4Couleur et forme :SolidMasse moléculaire :634.49Anti-inflammatory agent 7
<p>Anti-inflammatory Agent 7 suppresses proinflammatory cytokines by hindering the NF-κB/MAPK signaling pathway in both LPS-treated RAW 264.7 cells and mice.</p>Formule :C36H40N4O9Couleur et forme :SolidMasse moléculaire :672.72NK1 receptor antagonist 2
CAS :NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.Formule :C31H35F7N4O2Couleur et forme :SolidMasse moléculaire :628.62β2AR/M-receptor agonist-2
CAS :<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formule :C36H49ClN4O7SCouleur et forme :SolidMasse moléculaire :717.31PF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Formule :C36H50Cl2N4O7SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :753.78PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formule :C36H51Cl3N4O7SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :790.24PI3K/Akt/CREB activator 1
CAS :<p>PI3K/Akt/CREB activator 1 (AE-18) is an iNOS inhibitor that can be used to study vascular dementia and Parkinson's.</p>Formule :C19H15F4NO3Couleur et forme :SolidMasse moléculaire :381.32Antitrypanosomal agent 10
Antitrypanosomal agent 10, an antitrypanosomal compound, effectively inhibits Trypanosoma cruzi with an IC50 of 0.28 μM.Formule :C17H9F6N5OCouleur et forme :SolidMasse moléculaire :413.28Antitrypanosomal agent 11
<p>Antitrypanosomal Agent 11 is a chemical compound effective against Trypanosoma cruzi, exhibiting an inhibition concentration (IC 50) of 0.23 μM.</p>Formule :C16H10F6N6OCouleur et forme :SolidMasse moléculaire :416.28Gestrinone
CAS :Gestrinone (R 2323) 是一种合成类固醇激素,能够抑制平滑肌瘤(IC50:43.67 μM),有用于子宫内膜异位症的研究潜力。Formule :C21H24O2Degré de pureté :99.21%Couleur et forme :Light Yellow SolidMasse moléculaire :308.41SARS-CoV-2/MERS Mpro-IN-1
<p>SARS-CoV-2/MERS Mpro-IN-1 is a potent inhibitor of the main proteases in SARS-CoV-2 and MERS, exhibiting IC50 values of 0.10 and 0.06 µM, respectively.</p>Formule :C30H36N4O7Couleur et forme :SolidMasse moléculaire :564.63SARS-CoV-2/MERS Mpro-IN-2
<p>SARS-CoV-2/MERS Mpro-IN-2 is a potent inhibitor of the main proteases of SARS-CoV-2 and MERS, demonstrating IC50 values of 0.21 and 0.07 µM, respectively.</p>Formule :C28H30Cl2N4O6Couleur et forme :SolidMasse moléculaire :589.473β-Hydroxy-hop-22(29)-ene
CAS :3β-Hydroxy-hop-22(29)-ene is a potent antiparasitic compound demonstrating moderate efficacy against Trypanosoma cruzi and Leishmania mexicana.Formule :C30H50OCouleur et forme :SolidMasse moléculaire :426.72Antibacterial synergist 2
CAS :"Antibacterial Synergist 2 inhibits biofilms of S. enterica, S. aureus, P. aeruginosa, and C. albicans."Formule :C6H3Br3O2Couleur et forme :SolidMasse moléculaire :346.8

