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Se termine le 31 déc.( plus que 8 jours )
STAT3-IN-42
<p>STAT3-IN-42 is a ligand for target proteins in PROTACs (Proteolysis Targeting Chimeras). It is utilized in the synthesis of SD-2301.</p>Formule :C34H42N7O11PSCouleur et forme :SolidMasse moléculaire :787.24006Carumonam
CAS :<p>Carumonam, an antibiotic, could enhance the reactivity of Escherichia coli with mono- and polyclonal antisera to rough Escherichia coli J5.</p>Formule :C12H14N6O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :466.40EGFR-IN-162
<p>EGFR-IN-162 (compound 20) is an effective EGFR inhibitor that enhances both early and late apoptosis (EGFR) as well as necrosis (necrosis). It shows potential for use in breast cancer research.</p>Formule :C27H31N3O2Couleur et forme :SolidMasse moléculaire :429.241635-Hydroxypentanoic acid
CAS :5-Hydroxypentanoic acid is a PROTAC linker utilized in the synthesis of PROTAC AR-V7 degrader-1.Formule :C5H10O3Couleur et forme :SolidMasse moléculaire :118.13CS-VIP 8
CS-VIP 8 is a selective allosteric inhibitor of the WDR5 protein (Ki= 0.008 μM). It induces conformational changes in the MLL1 complex, causing the dissociation of MLL1 from the complex and inhibiting MLL1 histone methyltransferase activity, thereby regulating HOX gene expression. CS-VIP 8 shows potential for research in hematological diseases such as leukemia.Formule :C43H52F4N12O7Couleur et forme :SolidMasse moléculaire :924.4018DM-4111
CAS :<p>DM-4111, one of the primary monohydroxy metabolites of Tolvaptan, is an effective vasopressin V2 receptor (vasopressin V2 receptor) inhibitor. By inhibiting water reabsorption in renal tubules, it facilitates the excretion of electrolyte-free water. DM-4111 holds potential for research in cardiovascular diseases.</p>Formule :C26H25ClN2O4Couleur et forme :SolidMasse moléculaire :464.94Aminopeptidase N inhibitor 2
<p>AminopeptidaseN inhibitor 2 is an APN inhibitor (IC50: 4.3 μM) with antitumor properties.</p>Formule :C12H16F2N2O4SCouleur et forme :SolidMasse moléculaire :322.07988Biebrich scarlet
CAS :<p>Biebrich scarlet, a scarlet dye, stains collagen in Masson's trichrome and eosinophils.</p>Formule :C22H16N4Na2O7S2Couleur et forme :Dark Red PowderMasse moléculaire :558.5Alvespimycin TFA
<p>Alvespimycin (17-DMAG) TFA is a potent inhibitor of Hsp90, binding with an EC50 of 62 ± 29 nM.</p>Formule :C34H49F3N4O10Couleur et forme :SolidMasse moléculaire :730.34008CDK9/EZH2-IN-1
CAS :CDK9/EZH2-IN-1 is a dual-target inhibitor of CDK9 and EZH2 with IC50 values of 83.9 nM and 108.6 nM, respectively. It induces apoptosis and causes DNA double-strand breaks (DSB). Additionally, CDK9/EZH2-IN-1 inhibits the proliferation of MKN45, MDA-MB-453, and SW620 cancer cells, with respective IC50 values of 136.3 nM, 171.3 nM, and 315.7 nM.Formule :C47H59N11O4S2Couleur et forme :SolidMasse moléculaire :906.17RNAP-σ interaction inhibitor-1
CAS :<p>RNAP-σ interaction inhibitor-1 (compound 5d) acts as an inhibitor of the interaction between RNA polymerase and the sigma factor. It exhibits activity against Streptococci with a minimum inhibitory concentration (MIC) ranging from 1-2 µg/mL.</p>Formule :C19H11Cl3N2O6S2Couleur et forme :SolidMasse moléculaire :533.79Omadacycline tosylate
CAS :<p>Omadacycline tosylate (PTK 0796 tosylate) is an orally available antibacterial agent and tetracycline antibiotic, broad-spectrum antimicrobial activity.</p>Formule :C36H48N4O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :728.85ADP-β-S trisodium
ADP-β-S (trisodium) is an analog of ADP and acts as a partial agonist. It can induce human platelet aggregation and inhibit PGE1-stimulated adenylate cyclase.Formule :C10H12N5Na3O9P2SCouleur et forme :SolidMasse moléculaire :508.95241CAXII-IN-2
CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.Formule :C16H13FNO4PCouleur et forme :SolidMasse moléculaire :333.05662PD-1/PD-L1-IN-55
CAS :PD-1/PD-L1-IN-55 (compound D6) is a potent PD-1/PD-L1 inhibitor with an IC50 of 4.8 nM. It enhances IFN-γ secretion and decreases the proportion of late apoptosis due to PD-L1.Formule :C25H23ClN2O3Couleur et forme :SolidMasse moléculaire :434.92Androgen receptor antagonist 13
CAS :Androgen receptor antagonist 13 (compound 8a) is an orally active androgen receptor antagonist with an IC50 of 0.20 μM. It is used in prostate cancer research.Formule :C16H15N3O3SCouleur et forme :SolidMasse moléculaire :329.37Mitochondrial-IN-1
CAS :Mitochondrial-IN (C458) is a potent inhibitor of mitochondrial complex I. It offers significant protection against Aβ toxicity, exhibits favorable pharmacokinetic properties, and has minimal off-target effects.Formule :C22H30N2OCouleur et forme :SolidMasse moléculaire :338.49Deltamethrin
CAS :<p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>Formule :C22H19Br2NO3Degré de pureté :99.25% - 99.85%Couleur et forme :White To Off-White Crystals Or PowderMasse moléculaire :505.20CDA-IN-4
CAS :<p>CDA-IN-4 (compound VS-24) is an inhibitor of chitin deacetylase (CDA). At a concentration of 100 μg/mL, CDA-IN-4 provides a protective effect of 61.2% against rice blast disease.</p>Formule :C10H9BrN4O2SCouleur et forme :SolidMasse moléculaire :329.17Trimegestone
CAS :Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation.Formule :C22H30O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :342.47
