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Se termine le 31 déc.( plus que 7 jours )
NLG802 HCl
CAS :NLG802, an oral indoximod prodrug, inhibits IDO enzyme, modulates immune response, and has anti-cancer properties.Formule :C18H26ClN3O3Couleur et forme :SolidMasse moléculaire :367.874MPT0L145
CAS :<p>MPT0L145 is a first-in-class PIK3C3/FGFR inhibitor.</p>Formule :C25H29Cl3N8O3Couleur et forme :SolidMasse moléculaire :595.91Ronopterin
CAS :Ronopterin is a potent Nitric oxide synthase inhibitor and Neuroprotectant.Formule :C9H16N6O2Couleur et forme :SolidMasse moléculaire :240.26SB1-F-78
CAS :SB1-F-78 is an USP30 inhibitor.Formule :C17H16N6OSCouleur et forme :SolidMasse moléculaire :352.41PF-06862309
CAS :PF-06862309 is a PI3K inhibitorFormule :C20H26F3N8O7PCouleur et forme :SolidMasse moléculaire :578.44CGP-78608
CAS :CGP-78608 is a glycine site-specific N-methyl-D-aspartate receptor antagonist prevents activation of the NMDA/NO/CGMP pathway by ammonia.Formule :C11H13BrN3O5PCouleur et forme :SolidMasse moléculaire :378.12Ochromycinone
CAS :<p>Ochromycinone (STA 21) is a selective STAT3 inhibitor.</p>Formule :C19H14O4Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :306.31Delgocitinib EtOH
CAS :Delgocitinib (LEO-124249/JTE052) is a selective JAK inhibitor used for reducing skin inflammation and treating chronic dermatitis.Formule :C18H24N6O2Couleur et forme :SolidMasse moléculaire :356.43BiBET
CAS :BiBET is a potent, selective, bivalent inhibitor of BET bromodomains.Formule :C26H30N10O3Couleur et forme :SolidMasse moléculaire :530.58MK-8666 Tris
CAS :MK-8666, a partial GPCR agonist, targets GPR40 to enhance insulin secretion, potentially treating type 2 diabetes without adverse effects.Formule :C33H42N2O9SCouleur et forme :SolidMasse moléculaire :642.764Fasoracetam monohydrate
CAS :Fasoracetam monohydrate: synthetic, activates glutamate receptors, trialed in Phases I-III for vascular dementia.Formule :C11H21N3O5Couleur et forme :SolidMasse moléculaire :275.31JPI-547 HCl
CAS :JPI-547 (NOV 1402) is an oral anti-cancer drug targeting PARP 1/2 and Tankyrase 1/2, effective alone or with chemo and immunotherapies.Formule :C23H26Cl2N6OCouleur et forme :SolidMasse moléculaire :473.402KR30031
CAS :KR30031 is a novel verapamil-like P-glycoprotein inhibitor with fewer heart side-effects, potentially boosting paclitaxel's efficacy.Formule :C26H34N2O4Couleur et forme :SolidMasse moléculaire :438.56Quoromycin
CAS :Quoromycin, a new antivirulence drug, hinders Vibrio vulnificus by disrupting SmcR in quorum-sensing, reducing virulence in vitro and in vivo.Formule :C12H8N2O2SCouleur et forme :SolidMasse moléculaire :244.27Tofacitinib maleate
CAS :<p>Tofacitinib (tasocitinib, CP-690550) is a JAK inhibitor blocking cytokine signaling and STAT activation.</p>Formule :C16H20N6O·xC4H4O4Couleur et forme :SolidMasse moléculaire :428.449NAS-181 free base
CAS :NAS-181 free base is a 5-HT(1B) receptor antagonist.Formule :C19H26N2O4Couleur et forme :SolidMasse moléculaire :346.42SU 5402
CAS :SU 5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, FGFR1, and PDGF-Rβ, respectively.Formule :C17H16N2O3Degré de pureté :98.91% - 99.64%Couleur et forme :Yellow-Green SolidMasse moléculaire :296.32CJ-15161 hydrochloride
CAS :CJ-15161 hydrochloride is the salt form of CJ-15161 (free base), an opioid κ-receptor agonist, is undergoing development with Pfizer as an analgesic agent.Formule :C23H32ClN3O2Couleur et forme :SolidMasse moléculaire :417.978CJ-15161 (free base)
CAS :<p>CJ-15161 (free base), an opioid κ-receptor agonist, is undergoing development with Pfizer as an analgesic agent.</p>Formule :C23H31N3O2Couleur et forme :SolidMasse moléculaire :381.51IDN-1965
CAS :IDN-1965: potent, irreversible caspase inhibitor; blocks Fas-induced apoptosis; varied administration; promising for liver injury treatment.Formule :C21H26FN3O5Couleur et forme :SolidMasse moléculaire :419.45Bornaprine
CAS :Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.Formule :C21H31NO2Couleur et forme :SolidMasse moléculaire :329.48TP1287
CAS :TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.Formule :C21H21ClNO8PCouleur et forme :SolidMasse moléculaire :481.82Laropiprant analog
CAS :Laropiprant analog is an antagonist of the prostaglandin PGD2 receptor DP1.Formule :C20H18ClFN2O4SCouleur et forme :SolidMasse moléculaire :436.88ML416
CAS :<p>ML416 is an inhibitor of HIV-1.</p>Formule :C14H15FN2OS2Couleur et forme :SolidMasse moléculaire :310.41RWJ-60475
CAS :RWJ-60475 is a novel CD45 phosphatase inhibitor.Formule :C13H11BrNO7PCouleur et forme :SolidMasse moléculaire :404.11SU6656
CAS :SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, 20 nM, 130 nM, and 170 nM for Src, Yes, Lyn, and Fyn, respectively.Formule :C19H21N3O3SDegré de pureté :98.21% - 98.73%Couleur et forme :SolidMasse moléculaire :371.45AZD5718
CAS :AZD5718: potent FLAP inhibitor (IC50=2.0 nM), treats Coronary Artery Disease, >90% leukotriene suppression, safe in animal studies, in phase 2a trial.Formule :C29H34N6O4Couleur et forme :SolidMasse moléculaire :530.62GNF7156
CAS :GNF7156 is a potent and selective DYRK1A inhibitor.Formule :C22H22N6O3Couleur et forme :SolidMasse moléculaire :418.45ONL-1204
CAS :ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Formule :C71H100N18O16Couleur et forme :SolidMasse moléculaire :1461.66PF-04363467 HCl
CAS :<p>PF-04363467 HCl is a selective dopamine D3/D2 receptor antagonist.</p>Formule :C22H30N2O3SCouleur et forme :SolidMasse moléculaire :402.55Phenamil
CAS :Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.Formule :C12H12ClN7ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :305.72Istaroxime oxalate
CAS :<p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>Formule :C23H34N2O7Couleur et forme :SolidMasse moléculaire :450.53WS-691
CAS :WS-691: potent oral ABCB1 modulator; lowers PTX IC50 to 22.02 nM in SW620/Ad300 cells; raises [3H]-PTX uptake; non-toxic in vivo.Formule :C20H16FN7SCouleur et forme :SolidMasse moléculaire :405.45BC-1485
CAS :<p>BC-1485 is a small molecule inhibitor of FIEL1 that inhibits the degradation of PIAS4 and ameliorates fibrosis in a mouse model.</p>Formule :C19H21N5O5SDegré de pureté :97.03% - 97.15%Couleur et forme :SolidMasse moléculaire :431.47Brostallicin HCl
CAS :Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.Formule :C30H36BrClN12O5Couleur et forme :SolidMasse moléculaire :760.04Risvodetinib
CAS :Risvodetinib: potent inhibitor of protein tyrosine kinases c-Abl1, c-Abl2, and c-kit.Formule :C33H34N8O2Couleur et forme :SolidMasse moléculaire :574.68Tedizolid Phosphate
CAS :Tedizolid Phosphate (TR-701FA) is an oxazolidinone-class antibiotic. Tedizolid phosphate is a phosphate ester prodrug of the active compound tedizolid.Formule :C17H16FN6O6PDegré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :450.32XMU-MP-2
CAS :<p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>Formule :C32H33F3N8O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :618.65CRM-51005
CAS :<p>CRM-51005 is a new phospholipase C inhibitor produced by unidentified fungal strain MT51005</p>Formule :C15H20O3Couleur et forme :SolidMasse moléculaire :248.32VPC-16606
CAS :VPC-16606 inhibits ERα cell growth & gene expression, blocking ERα-LBD & SRC-3 binding dose-dependently.Formule :C17H13ClN2O2SCouleur et forme :SolidMasse moléculaire :344.82Ixazomib citrate EtOH
CAS :Ixazomib citrate (MLN9708), a prodrug of Ixazomib, is an oral, next-gen proteasome inhibitor with enhanced anti-cancer properties.Formule :C22H29BCl2N2O10Couleur et forme :SolidMasse moléculaire :563.188Ticalopride
CAS :Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formule :C14H20ClN3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :313.78Lifirafenib HCl
CAS :Lifirafenib (Beigene-283/BGB-283): a potent, selective RAF/EGFR inhibitor effective against B-RAF mutated colorectal cancers.Formule :C26H19ClF3N3O3Couleur et forme :SolidMasse moléculaire :513.9012BMS-955176 HCl
CAS :<p>GSK-3532795: a broader-spectrum HIV-1 maturation inhibitor than bevirimat, effective in vitro and clinically.</p>Formule :C42H62N2O4SCouleur et forme :SolidMasse moléculaire :727.486AMG2504
CAS :AMG2504 is a TRPA1 inhibitor.Formule :C15H10Cl4N2O3SCouleur et forme :SolidMasse moléculaire :440.13Metitepine
CAS :Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formule :C20H24N2S2Couleur et forme :SolidMasse moléculaire :356.55(S)-Pomalidomide
CAS :(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.Formule :C13H11N3O4Couleur et forme :SolidMasse moléculaire :273.24Teneligliptin hydrobromide
CAS :Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.Formule :C22H30N6OSBrHDegré de pureté :97.83% - 99.92%Couleur et forme :SolidMasse moléculaire :628.86Ruboxistaurin mesylate monohydrate
CAS :<p>Ruboxistaurin mesylate monohydrate, a PKC beta inhibitor, may treat diabetic nephropathy and macular edema, reducing oxidative stress and neovascularization.</p>Formule :C29H34N4O7SCouleur et forme :SolidMasse moléculaire :582.67Difenamizole HCl
CAS :Difenamizole HCl, a pyrazolone NSAID with analgesic effects, modulates dopamine and inhibits monoamine oxidase.Formule :C20H23ClN4OCouleur et forme :SolidMasse moléculaire :370.88
