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Se termine le 31 déc.( plus que 8 jours )
5-hydroxy Isatin
CAS :5-hydroxy Isatin inhibits MAO-A and ANP-induced particulate guanylyl cyclase in rat brain/heart.Formule :C8H5NO3Couleur et forme :SolidMasse moléculaire :163.13Moxaverine hydrochloride
CAS :<p>Moxaverine HCL, a papaverine derivative, is in Phase III trials for treating ocular blood flow in macular degeneration and glaucoma.</p>Formule :C20H22ClNO2Couleur et forme :SolidMasse moléculaire :343.85CPD7 HCl
CAS :<p>CPD7 HCl is a novel non-RBD binding modulator to inhibit SARS-CoV-2 by prohibiting the conformational change of the spike (S) protein.</p>Formule :C20H20ClNO3Couleur et forme :SolidMasse moléculaire :357.834TPPU
CAS :<p>TPPU is a potent inhibitor of both human and mouse sEH (IC50 of 3.7 and 2.8 nM, respectively)</p>Formule :C16H20F3N3O3Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :359.34TTA-A8
CAS :<p>TTA-A8 is an antagonist of T-type calcium channel.</p>Formule :C22H21F3N4O2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :430.42PUN-96956
CAS :PUN-96956, a BAM inhibitor lacking a formal name, impacts OMP folding/insertion. Named via MedKoo Nomenclature.Formule :C21H33ClN2Couleur et forme :SolidMasse moléculaire :348.95ML-077
CAS :<p>ML-077/VU0255011: Selective KCC2 antagonist, IC50=537 nM, saline soluble, cell permeable, submicromolar potency for in vitro KCC2 research.</p>Formule :C17H16N4OS2Couleur et forme :SolidMasse moléculaire :356.47PKC-9
CAS :PKC-9 is a PKC-zeta inhibitor 9.Formule :C25H25N7Couleur et forme :SolidMasse moléculaire :423.51Pyrithione Zinc
CAS :Pyrithione Zinc is a novel KMD5A inhibitor.Formule :C5H5NOSCouleur et forme :SolidMasse moléculaire :127.16Decanoyl chloride
CAS :Decanoyl Chloride helps create metalloproteinase inhibitors and reversible analgesics as a synthesis reagent.Formule :C10H19ClOCouleur et forme :SolidMasse moléculaire :190.71VU0621623
CAS :<p>VU0621623 is an arenavirus multiplication inhibitor which blocks lymphocytic choriomeningitis virus (LCMV) cell entry.</p>Formule :C20H21F2N5O3SCouleur et forme :SolidMasse moléculaire :449.47CypD-IN-29
CAS :CypD-IN-29 is a non-peptidic inhibitor of cyclophilin D as a neuroprotective agent in Aβ-induced mitochondrial dysfunction.Formule :C26H20FN5O2SCouleur et forme :SolidMasse moléculaire :485.53673-A
CAS :673-A inhibits ALDH1A, depletes ovarian CSCs, induces necroptosis, and reverses chemo resistance.Formule :C15H13NOCouleur et forme :SolidMasse moléculaire :223.27ZINC09410451
CAS :ZINC09410451 is a potent ebolavirus (EBOV) inhibitor.Formule :C24H27ClN4O3Couleur et forme :SolidMasse moléculaire :454.95TAK-960
CAS :<p>TAK-960 is an orally bioavailable, selective inhibitor of Plks with IC50 values of 0.8, 16.9, and 50.2 nM for Plk1, Plk2, and Plk3, respectively.</p>Formule :C27H34F3N7O3Degré de pureté :97.06%Couleur et forme :SolidMasse moléculaire :561.6N 0840
CAS :N 0840 is a selective, orally active A(1) adenosine receptor antagonist.Formule :C11H15N5Couleur et forme :SolidMasse moléculaire :217.27Carbazomycin C
CAS :Carbazomycin C, from Streptomyces, targets S. aureus, B. anthracis, fungi, P. falciparum, and is cytotoxic to several cancer cells, inhibiting 5-LO.Formule :C16H17NO3Couleur et forme :SolidMasse moléculaire :271.31SKF-104557
CAS :<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Formule :C13H18N2OCouleur et forme :SolidMasse moléculaire :218.29Azumolene sodium anhydrous
CAS :Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Betazole
CAS :Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formule :C5H9N3Couleur et forme :SolidMasse moléculaire :111.15DCAI Hydrochloride
CAS :DCAI hydrochloride is an inhibitor of nucleotide exchange and nucleotide release, by binding to the pocket adjacent to the Ras-SOS interface.Formule :C11H13Cl3N2Couleur et forme :SolidMasse moléculaire :279.59COR167
CAS :<p>COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.</p>Formule :C28H38N2O2Couleur et forme :SolidMasse moléculaire :434.61E09241
CAS :E09241 boosts OPG, doesn't change RANKL, aids osteoblasts, hinders osteoclasts via Wnt/β-catenin pathway.Formule :C11H9ClN2O2Couleur et forme :SolidMasse moléculaire :236.65N-Phenylthiourea
CAS :N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.Formule :C7H8N2SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :152.22Nelociguat
CAS :<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Formule :C19H17FN8O2Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :408.39Dibenzosuberenol
CAS :Dibenzosuberenol is used in oxidations, carboxylic acid/ketone synthesis, NK1 receptor antagonists creation, and catalysis studies.Formule :C15H12OCouleur et forme :SolidMasse moléculaire :208.26CB-892
CAS :<p>CB-892 is a novel inhibitor of hiv-1 gene expression</p>Formule :C15H14N2O4Couleur et forme :SolidMasse moléculaire :286.28HDAC-IN-6
CAS :HDAC-IN-6 is an HDAC inhibitor, targeting HDAC2, HDAC3, HDAC4, HDAC5, HDAC7, HDAC8, and HDAC9.Formule :C28H36F3N5O7Couleur et forme :SolidMasse moléculaire :611.61Epigenetic Multiple Ligand
CAS :Epigenetic Multiple Ligand inhibits many chromatin enzymes like SIRT1/2 and induces apoptosis or differentiation.Formule :C19H12Br4O4Couleur et forme :SolidMasse moléculaire :623.91BZL-HIS-OME 2HCL
CAS :<p>BZL-HIS-OME 2HCL is the dihydrochloride salt of BZL-HIS-OME, a sweet almond and yeast β-glucosidase inhibitor.</p>Formule :C14H19Cl2N3O2Couleur et forme :SolidMasse moléculaire :332.22iST2-1
CAS :<p>iST2-1 is a first-in-class ST2 inhibitor active in vivo.</p>Formule :C22H22N2O4Couleur et forme :SolidMasse moléculaire :378.42ST101036
CAS :MC activators have recently been described as safe and effective vaccine adjuvants. ST101036 exhibited high degranulation potency in both human and mouse MCs.Formule :C18H21F3N4Couleur et forme :SolidMasse moléculaire :350.386(5H)-Phenanthridinone
CAS :<p>6(5H)-Phenanthridinone suppresses PARP1/2, reduces RDM4 cell growth, downregulates pro-inflammatory genes, and alleviates EAE symptoms in rats.</p>Formule :C13H9NOCouleur et forme :SolidMasse moléculaire :195.22MAO-B ligand-1
CAS :MAO-B ligand-1 is a selective MAO-B inhibitor.Formule :C19H19N5O4SCouleur et forme :SolidMasse moléculaire :413.45ZINC32540717
CAS :ZINC32540717 is a potent ebolavirus (EBOV) inhibitor.Formule :C23H26N4O3Couleur et forme :SolidMasse moléculaire :406.48ITE
CAS :ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity.Formule :C14H10N2O3SDegré de pureté :97.91% - 99.14%Couleur et forme :SolidMasse moléculaire :286.31AM6701
CAS :<p>AM6701 is a novel highly potent inhibitor of human alpha/beta hydrolase domain 6 (habhd6)</p>Formule :C17H17N5ODegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :307.357SU 5616
CAS :<p>SU 5616 (WAY-608241) regulates abnormal cell proliferation and modulates tyrosine kinase signaling.</p>Formule :C13H8ClNOSDegré de pureté :98.84%Couleur et forme :SoildMasse moléculaire :261.7311β-HSD1 inibitor 19
CAS :3-chloro-4-sulfonyl-Benzonitrile inhibits hHSD1/mHSD1, IC50: 16nM/10nM.Formule :C19H16ClF4N3O2SDegré de pureté :99.58%Couleur et forme :SoildMasse moléculaire :461.86JB002
CAS :<p>JB002, a myosin II inhibitor, exhibits potent activity with an IC50 of ≤10 μM.</p>Formule :C18H15NO3Degré de pureté :99.74%Couleur et forme :SoildMasse moléculaire :293.32ZIM
CAS :ZIM, from 4-Aminoantipyrine, induces DNA and chromosomal damage, cell death, and phagocytosis, with potential in cancer therapy.Formule :C20H19N3O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :349.38PCSK9-IN-10
CAS :<p>PCSK9-IN-10: potent oral PCSK9 inhibitor (IC50 = 6.4 µM), upregulates LDLR, curbs atherosclerosis, for hyperlipidemia research.</p>Formule :C18H23N5O4Degré de pureté :99.06%Couleur et forme :SoildMasse moléculaire :373.41p53-MDM2-IN-1
CAS :<p>p53-MDM2-IN-1 (Example 30), an inhibitor targeting the p53-MDM2/X protein interaction, exhibits a K i value of 23.35 µM.</p>Formule :C23H20ClN3O3Degré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :421.886-Methyl-3-pyridinecarboxaldehyde
CAS :6-Methyl-3-pyridinecarboxaldehyde (6-Methoxynicotinaldehyde) has partial antitumor activity.Formule :C7H7NO2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :137.142-Quinolinecarboxaldehyde
CAS :<p>2-Quinolinecarboxaldehyde, a small rigid molecule, used in Henry reaction, inhibits AChE (IC50: 13.48 μM).</p>Formule :C10H7NODegré de pureté :99.5%Couleur et forme :Off-White CrystallineMasse moléculaire :157.17CDK8-IN-13
CAS :<p>CDK8-IN-13 is a CDK8 inhibitor (IC50: 51.9 nM) with potent, selective and oral activity.</p>Formule :C14H11N3ODegré de pureté :99.28%Couleur et forme :SoildMasse moléculaire :237.26Oglufanide
CAS :<p>Oglufanide (H-Glu-Trp-OH) is a naturally occurring thymic immunomodulator,and inhibits vascular endothelial growth factor (VEGF).</p>Formule :C16H19N3O5Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :333.346,6'-Dimethyl-2,2'-dipyridyl
CAS :6,6'-Dimethyl-2,2'-dipyridyl (6,6'-Bi-2-picoline) is a novel time-resolved fluorescent immunoassay (TRFIA) chelate with a good bactericidal effect for the studyFormule :C12H12N2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :184.24BI 1015550
CAS :<p>Nerandomilast (BI 1015550) is an orally active PDE4B inhibitor with IC50 of 7.2 nM.Cost-effective and quality-assured.</p>Formule :C20H25ClN6O2SDegré de pureté :98.06% - 99.71%Couleur et forme :SoildMasse moléculaire :448.97PI5P4Ks-IN-2
CAS :<p>PI5P4Ks-IN-2 inhibits PI5P4K isoforms α, β, γ, γ+ with IC50 <4.3, <4.6, 6.2, 0.32 µM, respectively.</p>Formule :C22H23N5Degré de pureté :98.36% - 99.02%Couleur et forme :SoildMasse moléculaire :357.45
