CAS 106266-06-2

Risperidone

Descrizione:

Risperidone è un farmaco antipsicotico atipico utilizzato principalmente per trattare la schizofrenia, il disturbo bipolare e l'irritabilità associata all'autismo. Funziona come un antagonista della serotonina e della dopamina, influenzando l'attività dei neurotrasmettitori nel cervello, in particolare i recettori della serotonina e della dopamina. Risperidone è caratterizzato dalla sua formula chimica C23H27N3O2 e da un peso molecolare di circa 410,48 g/mol. La sostanza appare come una polvere cristallina bianca o bianco sporco ed è tipicamente somministrata per via orale, sebbene siano disponibili anche formulazioni iniettabili. La sua farmacocinetica indica una emivita relativamente lunga, consentendo una somministrazione una volta al giorno in molti casi. Gli effetti collaterali comuni possono includere sedazione, aumento di peso e cambiamenti metabolici, richiedendo monitoraggio durante il trattamento. Il profilo di efficacia e sicurezza di Risperidone lo rende un'opzione ampiamente prescritta nella cura psichiatrica, sebbene sia essenziale adattare il trattamento alle esigenze individuali del paziente e monitorare i potenziali effetti avversi.

Formula: C₂₃H₂₇FN₄O₂

InChI: InChI=1/C23H27FN4O2/c1-15-18(23(29)28-10-3-2-4-21(28)25-15)9-13-27-11-7-16(8-12-27)22-19-6-5-17(24)14-20(19)30-26-22/h5-6,14,16H,2-4,7-13H2,1H3

InChI key: InChIKey=RAPZEAPATHNIPO-UHFFFAOYSA-N

SMILES: FC=1C=C2C(C(=NO2)C3CCN(CCC=4C(=O)N5C(=NC4C)CCCC5)CC3)=CC1

Sinonimi:

• 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
• 3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one
• 3-[2-[4-(6-Fluor-1,2-benzisoxazol-3-yl)piperidino]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on
• 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-
• Apexidone
• Psychodal
• R 64766
• Rbp 7000
• Resperidone
• Ripedon
• Risbiodal
• Rispa
• Rispadal
• Risperdal
• Risperdal Consta
• Risperdine
• Risperid
• Risperid fort
• Risperidal
• Risperidone ACIS
• Risperidone intermediates
• Spiron
• Zophrenal
• Risperidone
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-(9CI)
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one, R-64766, Belivon, Risperdal
• Risoeridone
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-
• Kesperidone
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydropyrido[2,1-b]pyrimidin-4-one
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, R-64766, Belivon, Risperdal
• 4h-pyrido(1,2-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluoro-1,2-benzi
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-
• soxazol-3-yl)-1-piperidinyl)ethyl)-2-methyl-
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2,a]pyrimidin-4-one

Risperidone - Bio-X ™

Prodotto controllato

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs.
Risperidone is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.

Formula: C₂₃H₂₇FN₄O₂

Purezza: Min. 99.0 Area-%

Colore e forma: White Powder

Peso molecolare: 410.48 g/mol

Ref: 3D-BR164349

Risperidone

Prodotto controllato

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs. Consequently leading to hyperprolactinemia, a negative adverse effect when Risperidone is used as a drug. Risperidone has been shown to have cardiac effects, including increasing heart rate and QT interval. It is also metabolized by cytochrome P450 enzymes and can be detected in wastewater after oral administration of a single dose (0.5 mg/kg).

Formula: C₂₃H₂₇FN₄O₂

Purezza: Min. 98.5 Area-%

Colore e forma: White Off-White Powder

Peso molecolare: 410.48 g/mol

Ref: 3D-FR27737

Risperidone

CAS: 106266-06-2

Formula: C₂₃H₂₇FN₄O₂

Purezza: 98%

Colore e forma: Solid, White to off-white powder

Peso molecolare: 410.212

Ref: 10-F036563