CAS 127984-74-1

10-(4-aminobutil)-19-[(2-ammino-3-naftalen-2-il-propanolo)ammino]-N-(1-carbamoil-2-idrossi-propil)-16-[(4-idrossifenil)metil]-13-(1H-indol-3-ilmetil)-6,9,12,15,18-pentaoxo-7-propan-2-il-1,2-ditia-5,8,11,14,17-pentazacicloicosano-4-carbossamide

Descrizione:

La sostanza chimica nota come "10-(4-amminobutil)-19-[(2-amino-3-naftalen-2-il-propanoyl)amino]-N-(1-carbamoil-2-idrossipropil)-16-[(4-idrossifenil)metil]-13-(1H-indol-3-ilmetil)-6,9,12,15,18-pentaoxo-7-propan-2-il-1,2-ditia-5,8,11,14,17-pentazacicloicosano-4-carboxamide" con numero CAS 127984-74-1 è un composto organico complesso caratterizzato da gruppi multifunzionali e complessità strutturale. Presenta uno scheletro di pentazacicloicosano, che contribuisce alla sua unica conformazione tridimensionale e potenziale attività biologica. La presenza di vari gruppi funzionali, tra cui ammine, idrossili e carbonili, suggerisce che questo composto possa mostrare una reattività e solubilità significative in solventi polari. I suoi componenti strutturali, come i moieties di indolo e naftalene, indicano potenziali interazioni con bersagli biologici, rendendolo di interesse nella chimica medicinale. L'ampia funzionalizzazione del composto può anche influenzare le sue proprietà farmacocinetiche, inclusi assorbimento, distribuzione, metabolismo ed escrezione. In generale, questa sostanza rappresenta un'area affascinante di studio per i ricercatori che esplorano nuovi agenti terapeutici.

Formula: C₅₄H₆₉N₁₁O₁₀S₂xC₂H₄O

InChI: InChI=1/C54H69N11O10S2.C2H4O2/c1-29(2)45-54(75)63-44(53(74)65-46(30(3)66)47(57)68)28-77-76-27-43(62-48(69)38(56)23-32-15-18-33-10-4-5-11-34(33)22-32)52(73)60-41(24-31-16-19-36(67)20-17-31)50(71)61-42(25-35-26-58-39-13-7-6-12-37(35)39)51(72)59-40(49(70)64-45)14-8-9-21-55;1-2(3)4/h4-7,10-13,15-20,22,26,29-30,38,40-46,58,66-67H,8-9,14,21,23-25,27-28,55-56H2,1-3H3,(H2,57,68)(H,59,72)(H,60,73)(H,61,71)(H,62,69)(H,63,75)(H,64,70)(H,65,74);1H3,(H,3,4)

SMILES: CC(C)C1C(=NC(CSSCC(C(=NC(Cc2ccc(cc2)O)C(=NC(Cc2c[nH]c3ccccc23)C(=NC(CCCCN)C(=N1)O)O)O)O)N=C(C(Cc1ccc2ccccc2c1)N)O)C(=NC(C(C)O)C(=N)O)O)O.CC(=O)O

Sinonimi:

• Lanreotide Acetate
• 10-(4-Aminobutyl)-19-[(2-Amino-3-Naphthalen-2-Yl-Propanoyl)Amino]-N-(1-Carbamoyl-2-Hydroxy-Propyl)-16-[(4-Hydroxyphenyl)Methyl]-13-(1H-Indol-3-Ylmethyl)-6,9,12,15,18-Pentaoxo-7-Propan-2-Yl-1,2-Dithia-5,8,11,14,17-Pentazacycloicosane-4-Carboxamide

Lanreotide acetate

CAS: 127984-74-1

Formula: C₅₄H₆₉N₁₁O₁₀S₂·xC₂H₄O₂

Purezza: ≥ 98.0%

Colore e forma: White to off-white solid

Peso molecolare: 1096.32 (free base)

Ref: 7W-GK2805

Lanreotide Acetate

CAS: 127984-74-1

Formula: C₅₄H₆₉N₁₁O₁₀S₂

Purezza: 95%~99%

Colore e forma: White to Off-white Powder

Peso molecolare: 1096.33

Ref: BP-BPPG043

Lanreotide Acetate

Prodotto controllato

CAS: 127984-74-1

Applications Lanreotide Acetate is a drug used in the control and prevention of glycemia and hypoglycemic brain damage without surgery in patients diagnosed with congenital hyperinsulinism. It improves outcomes in patients suffering from acromegalyresulting from invasive pituitary macroadenoma.
References Kuehnen, P. et al.: Horm. Res. Paediat., 78, 106 (2012); Li, Z. et al.: J. Int. Med. Res., 40, 517 (2012);

Formula: C₅₄H₆₉N₁₁O₁₀S₂·C₂H₄O₂

Colore e forma: Neat

Peso molecolare: 1156.38

Ref: TR-L174600

Lanreotide acetate

CAS: 127984-74-1

Lanreotide Acetate is a synthetic cyclic peptide with anti-cancer properties and is used for the treatment of carcinoid syndrome. It binds to somatostatin receptors and inhibits the release of hormones such as gastrin, secretin, vasoactive intestinal peptide, and pancreatic polypeptide. Lanreotide Acetate is used in the treatment of symptoms that are typical for carcinoid syndrome and can also be used in combination with goserelin acetate or triptorelin acetate for patients who do not respond to lanreotide alone. The drug has been shown to be well tolerated in clinical trials and does not show any significant toxicity.

Formula: C₅₄H₆₉N₁₁O₁₀S₂•(C₂H₄O₂)x

Purezza: Min. 95%

Colore e forma: Powder

Peso molecolare: 1,156.4 g/mol

Ref: 3D-CFA98474

Lanreotide acetate - Bio-X ™

Prodotto controllato

CAS: 127984-74-1

Lanreotide is a somatostatin analog that is used for the treatment of tumors and acromegaly. This drug inhibits the growth hormone in the brain and induces apoptosis. Lanreotide also has antiproliferative properties as it blocks production that leads to tumor growth.

Formula: C₅₆H₇₃N₁₁O₁₂S₂

Purezza: Min. 95%

Colore e forma: Powder

Peso molecolare: 1,156.4 g/mol

Ref: 3D-DVD11472